BE868893A - Nouveaux derives solubles de 2,4-diaminopyrimidines, leur preparation et leur utilisation en tant que medicaments - Google Patents

Nouveaux derives solubles de 2,4-diaminopyrimidines, leur preparation et leur utilisation en tant que medicaments

Info

Publication number
BE868893A
BE868893A BE2057136A BE2057136A BE868893A BE 868893 A BE868893 A BE 868893A BE 2057136 A BE2057136 A BE 2057136A BE 2057136 A BE2057136 A BE 2057136A BE 868893 A BE868893 A BE 868893A
Authority
BE
Belgium
Prior art keywords
preparation
medicinal products
new soluble
diaminopyrimidine derivatives
diaminopyrimidine
Prior art date
Application number
BE2057136A
Other languages
English (en)
Original Assignee
Dick Pierre R G
Rombi Max Andre
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dick Pierre R G, Rombi Max Andre filed Critical Dick Pierre R G
Publication of BE868893A publication Critical patent/BE868893A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
BE2057136A 1977-07-11 1978-07-11 Nouveaux derives solubles de 2,4-diaminopyrimidines, leur preparation et leur utilisation en tant que medicaments BE868893A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7722323A FR2397407A2 (fr) 1977-07-11 1977-07-11 Derives de 2,4-diamino pyrimidines et leur mise en solution en association avec des sulfamides

Publications (1)

Publication Number Publication Date
BE868893A true BE868893A (fr) 1979-01-11

Family

ID=9193583

Family Applications (1)

Application Number Title Priority Date Filing Date
BE2057136A BE868893A (fr) 1977-07-11 1978-07-11 Nouveaux derives solubles de 2,4-diaminopyrimidines, leur preparation et leur utilisation en tant que medicaments

Country Status (13)

Country Link
US (1) US4232023A (fr)
JP (1) JPS5448776A (fr)
AT (1) AT362381B (fr)
AU (1) AU3793378A (fr)
BE (1) BE868893A (fr)
DE (1) DE2829820A1 (fr)
FR (1) FR2397407A2 (fr)
GB (1) GB2001965B (fr)
IE (1) IE47232B1 (fr)
IT (1) IT1096690B (fr)
LU (1) LU79949A1 (fr)
NL (1) NL7807440A (fr)
ZA (1) ZA783957B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2502152A1 (fr) * 1981-03-20 1982-09-24 Panmedica Laboratoires Nouveaux derives solubles n2 substitues de la diamino-2,4-benzyl-5-pyrimidines, leur procede de preparation et medicaments les contenant
US6583148B1 (en) 1999-04-08 2003-06-24 Krenitsky Pharmaceuticals, Inc. Neurotrophic substituted pyrimidines
EP1303495B1 (fr) 2000-07-24 2010-05-26 Krenitsky Pharmaceuticals, Inc. 5-alkynyle pyrimidines substituees avec activite neurotrophique
DK1725540T5 (da) 2004-03-05 2012-10-22 Hoffmann La Roche Diaminopyrimidiner som p2x3- og p2x2/3-antagonister
EP1924566B1 (fr) * 2005-09-01 2016-01-13 F.Hoffmann-La Roche Ag Diaminopyrimidines comme modulateurs p2x3 et p2x2/3
CA2619919C (fr) * 2005-09-01 2014-04-01 F. Hoffmann-La Roche Ag Diaminopyrimidines en tant que modulateurs de p2x3 et p2x2/3
CN101253159B (zh) * 2005-09-01 2011-12-07 弗·哈夫曼-拉罗切有限公司 作为p2x3和p2x2/3调节剂的二氨基嘧啶类化合物
CN101820879B (zh) * 2007-10-08 2013-01-02 疟疾药物投资公司 具有柔性侧链的抗疟用化合物
US9000003B2 (en) * 2011-03-10 2015-04-07 National Science And Technology Development Agency Anti-folate antimalarials with dual-binding modes and their preparation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2287071A (en) * 1938-08-08 1942-06-23 Parke Davis & Co Organic amine derivatives and method of obtaining same
US2374791A (en) * 1942-06-22 1945-05-01 Parke Davis & Co Organic amine derivatives and method of obtaining same
US3111521A (en) * 1962-04-25 1963-11-19 Parke Davis & Co 2-aryl-nu-(polyamino-5-pyrimidinyl)-glycinonitriles
GB1375162A (fr) * 1970-10-22 1974-11-27
BE791627A (fr) * 1971-11-20 1973-05-21 Knapsack Ag Procede pour l'oxydation du monoxyde de carbone et des hydrocarbures

Also Published As

Publication number Publication date
AU3793378A (en) 1980-01-17
IE781377L (en) 1979-01-11
US4232023A (en) 1980-11-04
ZA783957B (en) 1979-09-26
ATA496978A (de) 1980-10-15
GB2001965A (en) 1979-02-14
IT7825569A0 (it) 1978-07-11
JPS5448776A (en) 1979-04-17
IT1096690B (it) 1985-08-26
GB2001965B (en) 1982-03-10
FR2397407A2 (fr) 1979-02-09
IE47232B1 (en) 1984-01-25
LU79949A1 (fr) 1979-04-09
AT362381B (de) 1981-05-11
DE2829820A1 (de) 1979-02-01
FR2397407B2 (fr) 1980-01-04
NL7807440A (nl) 1979-01-15

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