LTC1663240I2 - Pirimidino deriniai, turintys nnrti su rt slopikliais - Google Patents

Pirimidino deriniai, turintys nnrti su rt slopikliais

Info

Publication number: LTC1663240I2
Authority: LT; Lithuania
Prior art keywords: pyrimidine; inhibitors; combinations containing; nnrti; containing nnrti
Prior art date: 2003-09-03

Application number

LTPA2015035C

Other languages

English (en)

Original Assignee

Janssen Sciences Ireland Uc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-09-03

Filing date

2016-12-20

Publication date

2022-05-25

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34280181&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LTC1663240(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2016-12-20 Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc

2017-01-10 Publication of LTPA2016044I1 publication Critical patent/LTPA2016044I1/lt

2022-05-25 Publication of LTC1663240I2 publication Critical patent/LTC1663240I2/lt

Links

CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical compound C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 title 1
239000003112 inhibitor Substances 0.000 title 1
239000002726 nonnucleoside reverse transcriptase inhibitor Substances 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Immunology (AREA)
Organic Chemistry (AREA)
Virology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Tropical Medicine & Parasitology (AREA)
Molecular Biology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
AIDS & HIV (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Plural Heterocyclic Compounds (AREA)

LTPA2015035C 2003-09-03 2016-12-20 Pirimidino deriniai, turintys nnrti su rt slopikliais LTC1663240I2 (lt)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
US49977103P	2003-09-03	2003-09-03
EP03103275		2003-09-03
EP03103319		2003-09-08
EP03103335		2003-09-10
EP03103668		2003-10-02
US50848603P	2003-10-03	2003-10-03
EP04787096.9A EP1663240B2 (en)	2003-09-03	2004-09-03	Combinations of a pyrimidine containing nnrti with rt inhibitors
PCT/EP2004/052028 WO2005021001A1 (en)	2003-09-03	2004-09-03	Combinations of a pyrimidine containing nnrti with rt inhibitors

Publications (2)

Publication Number	Publication Date
LTPA2016044I1 LTPA2016044I1 (lt)	2017-01-10
LTC1663240I2 true LTC1663240I2 (lt)	2022-05-25

Family

ID=34280181

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
LTPA2016045C LTPA2016045I1 (lt)	2003-09-03	2016-12-20	Pirimidino deriniai, turintys NNRTI su RT slopikliais
LTPA2015035C LTC1663240I2 (lt)	2003-09-03	2016-12-20	Pirimidino deriniai, turintys nnrti su rt slopikliais

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
LTPA2016045C LTPA2016045I1 (lt)	2003-09-03	2016-12-20	Pirimidino deriniai, turintys NNRTI su RT slopikliais

Country Status (25)

Country	Link
US (9)	US20080200435A1 (lt)
EP (1)	EP1663240B2 (lt)
JP (3)	JP5507791B2 (lt)
KR (1)	KR20060090658A (lt)
CN (1)	CN101060844B (lt)
AP (1)	AP2109A (lt)
AU (5)	AU2004268390B2 (lt)
BE (1)	BE2015C053I2 (lt)
CA (1)	CA2537095C (lt)
CY (5)	CY2015038I2 (lt)
FI (1)	FI1663240T4 (lt)
FR (3)	FR15C0072I2 (lt)
HK (1)	HK1092698A1 (lt)
HR (1)	HRP20150798T4 (lt)
HU (5)	HUS1500053I1 (lt)
IL (2)	IL173438A (lt)
LT (2)	LTPA2016045I1 (lt)
LU (3)	LU92853I2 (lt)
MX (1)	MXPA06002437A (lt)
MY (1)	MY169670A (lt)
NL (2)	NL300781I2 (lt)
NO (5)	NO334877B1 (lt)
NZ (1)	NZ545306A (lt)
PL (1)	PL1663240T5 (lt)
WO (1)	WO2005021001A1 (lt)

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2004
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2009
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Also Published As

Publication number	Publication date
NO2014032I1 (no)	2015-01-05
FR15C0073I2 (fr)	2016-02-12
HUS1500053I1 (hu)	2016-03-29
US20140349971A1 (en)	2014-11-27
LU92853I2 (fr)	2015-12-21
AU2014203484A1 (en)	2014-07-17
NO2014031I1 (no)	2015-01-05
CY2015040I2 (el)	2016-08-31
AU2004268390A1 (en)	2005-03-10
CY2015039I1 (el)	2016-08-31
AU2011201123A1 (en)	2011-04-07
AU2019200813A1 (en)	2019-02-28
US20220008417A1 (en)	2022-01-13
IL213104A (en)	2016-02-29
AU2011201123B2 (en)	2013-10-10
PL1663240T5 (pl)	2024-02-26
NL300781I1 (lt)	2016-04-19
JP5507791B2 (ja)	2014-05-28
HUS1500052I1 (hu)	2016-03-29
FR15C0072I1 (lt)	2015-04-12
HRP20150798T1 (hr)	2015-09-11
FR15C0071I2 (fr)	2016-02-12
AU2014203484B2 (en)	2016-09-29
US8841310B2 (en)	2014-09-23
NO334877B1 (no)	2014-06-23
NZ545306A (en)	2009-11-27
LTPA2016045I1 (lt)	2017-01-10
BE2015C053I2 (lt)	2023-12-14
CY2015038I1 (el)	2016-08-31
CA2537095A1 (en)	2005-03-10
NO2014031I2 (no)	2014-12-18
EP1663240B1 (en)	2015-04-22
US20190216807A1 (en)	2019-07-18
LU92855I2 (fr)	2015-12-21
FR15C0073I1 (lt)	2015-04-12
HUS1600059I1 (hu)	2017-02-28
FR15C0071I1 (lt)	2015-04-12
LU92854I2 (fr)	2015-12-21
JP2007520443A (ja)	2007-07-26
US20200171027A1 (en)	2020-06-04
AU2016210733A1 (en)	2016-08-25
HRP20150798T4 (hr)	2023-06-09
NO2014030I1 (no)	2015-01-05
CN101060844A (zh)	2007-10-24
US20180228800A1 (en)	2018-08-16
IL173438A (en)	2012-03-29
AP2006003551A0 (en)	2006-04-30
MXPA06002437A (es)	2006-06-20
NO20061374L (no)	2006-03-27
CY2016048I2 (el)	2017-07-12
CN101060844B (zh)	2012-01-04
IL213104A0 (en)	2011-07-31
AU2016210733B2 (en)	2018-11-08
PL1663240T3 (pl)	2015-10-30
FR15C0072I2 (fr)	2019-05-17
US20100029591A1 (en)	2010-02-04
NL300781I2 (lt)	2016-04-19
US20080200435A1 (en)	2008-08-21
CY2016048I1 (el)	2017-07-12
CY2015038I2 (el)	2016-08-31
US20170100398A1 (en)	2017-04-13
NO2016025I1 (lt)	2016-12-20
AP2109A (en)	2010-02-26
US20150283135A1 (en)	2015-10-08
CY2016049I2 (el)	2017-07-12
HK1092698A1 (en)	2007-02-16
CA2537095C (en)	2012-05-29
EP1663240B2 (en)	2023-03-01
CY2015039I2 (el)	2016-08-31
NO2014032I2 (no)	2014-12-18
FI1663240T4 (fi)	2023-04-25
HUS1500054I1 (hu)	2016-03-29
CY2016049I1 (el)	2017-07-12
EP1663240A1 (en)	2006-06-07
LTPA2016044I1 (lt)	2017-01-10
JP5820045B2 (ja)	2015-11-24
JP2015044839A (ja)	2015-03-12
NL300768I1 (lt)	2015-12-16
KR20060090658A (ko)	2006-08-14
JP2012051915A (ja)	2012-03-15
AU2004268390B2 (en)	2011-03-31
WO2005021001A1 (en)	2005-03-10
MY169670A (en)	2019-05-08
IL173438A0 (en)	2006-06-11
CY2015040I1 (el)	2016-08-31
NO2014030I2 (no)	2014-12-18
HUS1600058I1 (hu)	2017-02-28
NL300768I2 (nl)	2023-08-09

Publication	Publication Date	Title
LTC1663240I2 (lt)	2022-05-25	Pirimidino deriniai, turintys nnrti su rt slopikliais
NL2000323A1 (nl)	2007-06-21	Pyrimidine-derivaten.
DK1761505T3 (da)	2011-12-05	Pyrimidin-urinstof-derivater som kinaseinhibitorer
DE60313872D1 (de)	2007-06-28	Pyrazoloä1,5-aüpyrimidine als hemmstoffe cyclin-abhängiger kinasen
ATE512960T1 (de)	2011-07-15	Pyrimidinderivate
DK1487805T3 (da)	2012-10-15	Pyrimidinderivater
DE602004012154D1 (de)	2008-04-10	Pyridoä2,3-düpyrimidin-2,4-diamine als pde-2-inhibitoren
NO20055023D0 (no)	2005-10-28	Hurtigskytende vapen
DK1544379T3 (da)	2014-07-07	Klemindretning
DE502004002049D1 (de)	2007-01-04	Halteeinrichtung
DE112004001801D2 (de)	2006-06-01	Haltevorrichtung
FI5917U1 (fi)	2003-08-27	Pidin
ES1059189Y (es)	2005-07-01	Bolsillo.
AT500804B8 (de)	2007-02-15	Abstandhalter
DE602004004185D1 (de)	2007-02-22	Klammer
ES1058704Y (es)	2005-05-16	Antirrobo porta-esquies.
ES1058346Y (es)	2005-03-16	Porta-boligrafos.
ES1053882Y (es)	2003-09-01	Hamaca colgante.
SE0400584D0 (sv)	2004-03-09	NNRTI Antivirals II
ITBO20040669A1 (it)	2005-01-28	Supporto portapane con oliera
SE0301098D0 (sv)	2003-04-11	Dubbelhållare
SE0400585D0 (sv)	2004-03-09	NNRTI Antivirals
ITPD20030088A1 (it)	2004-11-03	Piedino strutturale reggicartello.
UA9581S (uk)	2004-11-15	Тримач
FI20040331A0 (fi)	2004-03-02	Pidike