KR920018038A - 2,2-디메틸-2,3-디하이드로벤조푸란-7-카복실산의 제조방법 및 그의 중간체 - Google Patents
2,2-디메틸-2,3-디하이드로벤조푸란-7-카복실산의 제조방법 및 그의 중간체 Download PDFInfo
- Publication number
- KR920018038A KR920018038A KR1019920003610A KR920003610A KR920018038A KR 920018038 A KR920018038 A KR 920018038A KR 1019920003610 A KR1019920003610 A KR 1019920003610A KR 920003610 A KR920003610 A KR 920003610A KR 920018038 A KR920018038 A KR 920018038A
- Authority
- KR
- South Korea
- Prior art keywords
- methyl
- compound
- preparing
- propenyl
- dihydrobenzofuran
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
- C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
- C07C69/88—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring with esterified carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
- C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
- C07C69/92—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring with etherified hydroxyl groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Furan Compounds (AREA)
- Cosmetics (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
내용 없음
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
Claims (7)
- 유기산의 존재하에서 하기 일반식(Ⅱ)의 페놀을 가열시킴을 포함하는, 하기 일반식(Ⅰ)화합물의 제조방법.상기 식에서, R1은 수소, 메틸, 할로, C1-C3알콕시, (C1-C3알킬)-S(O)t, 트리플루오로메틸 또는 (CH3)2NSO2-이고, t는 0,1또는 2이다.
- 제 1항에 있어서, 유기산이 포름산인 방법.
- 제 1항에 있어서, 일반식(Ⅱ)의 화합물이 5-클로로-2-하이드록시-3-(2-메틸-2-프로페닐)벤조산 2-메틸-2-프로페닐 에스테르인 방법.
- 하기 일반식(Ⅱ)의 화합물.상기 식에서, R1은 수소, 메틸, 할로, C1-C3알콕시, (C1-C3알킬)-S(O)t, 트리플루오로메틸 또는 (CH3)2NSO2-이고, t는 0,1 또는 2이다.
- 제4항에있어서,5-클로로-2-하이드록시-3-(2-메틸-2-프로페닐)벤조산2-메틸-2-프로페닐에 스테르인 화합물.
- 하기 일반식(Ⅲ)의 화합물.상기 식에서, R1은 수소, 메틸, 할로, C1-C3알콕시, (C1-C3알킬)-S(O)t, 트리플루오로메틸 또는 (CH3)2NSO2-이고, t는 0,1 또는 2이다.
- 제6항에 있어서, 5-클로로-2-[(2-메틸-2-프로페닐)옥시]벤조산 2-메틸-2-프로페닐 에스테르인 화합물.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US07/666,279 US5142069A (en) | 1991-03-07 | 1991-03-07 | Process of preparing 2,2-dimethyl-2,3-dihydrobenzofuran-7-carboxylic acids |
US666,279 | 1991-03-07 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR920018038A true KR920018038A (ko) | 1992-10-21 |
KR100193973B1 KR100193973B1 (ko) | 1999-06-15 |
Family
ID=24673565
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR1019920003610A KR100193973B1 (ko) | 1991-03-07 | 1992-03-05 | 2,2-디메틸-2,3-디하이드로벤조푸란-7-카복실산의 제조방법 및 그의 중간체 |
Country Status (16)
Country | Link |
---|---|
US (1) | US5142069A (ko) |
EP (1) | EP0502735B1 (ko) |
JP (1) | JPH04338381A (ko) |
KR (1) | KR100193973B1 (ko) |
AT (1) | ATE127461T1 (ko) |
BR (1) | BR9200768A (ko) |
CA (1) | CA2062329A1 (ko) |
DE (1) | DE69204497T2 (ko) |
DK (1) | DK0502735T3 (ko) |
ES (1) | ES2078652T3 (ko) |
GR (1) | GR3017875T3 (ko) |
HU (1) | HU212786B (ko) |
IE (1) | IE67382B1 (ko) |
IL (1) | IL101149A (ko) |
MX (1) | MX9200962A (ko) |
TW (1) | TW198014B (ko) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5723103A (en) * | 1994-12-09 | 1998-03-03 | Vanderbilt University | Substituted benzamides and radioligand analogs and methods of use |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3860619A (en) * | 1969-05-09 | 1975-01-14 | Novo Terapeutisk Labor As | Sulphonylurea derivatives |
EP0135545A1 (en) * | 1983-02-19 | 1985-04-03 | Beecham Group Plc | Azabicycloalkyl benzamide and anilide derivatives |
CA1297877C (en) * | 1983-12-22 | 1992-03-24 | Daniel Lednicer | Benzofurancarboxamides useful as antiemetic or antipsychotic agents |
US4888353A (en) * | 1986-02-28 | 1989-12-19 | Erbamont, Inc. | Carboxamides useful as antiemetic or antipsychotic agents |
US4921982A (en) * | 1988-07-21 | 1990-05-01 | Eli Lilly And Company | 5-halo-2,3-dihydro-2,2-dimethylbenzofuran-7-carboxylic acids useful as intermediates for 5-HT3 antagonists |
-
1991
- 1991-03-07 US US07/666,279 patent/US5142069A/en not_active Expired - Fee Related
- 1991-09-27 TW TW080107670A patent/TW198014B/zh active
-
1992
- 1992-03-05 MX MX9200962A patent/MX9200962A/es not_active IP Right Cessation
- 1992-03-05 CA CA002062329A patent/CA2062329A1/en not_active Abandoned
- 1992-03-05 ES ES92301904T patent/ES2078652T3/es not_active Expired - Lifetime
- 1992-03-05 HU HU9200745A patent/HU212786B/hu not_active IP Right Cessation
- 1992-03-05 DE DE69204497T patent/DE69204497T2/de not_active Expired - Fee Related
- 1992-03-05 KR KR1019920003610A patent/KR100193973B1/ko not_active IP Right Cessation
- 1992-03-05 EP EP92301904A patent/EP0502735B1/en not_active Expired - Lifetime
- 1992-03-05 DK DK92301904.6T patent/DK0502735T3/da active
- 1992-03-05 IL IL10114992A patent/IL101149A/en not_active IP Right Cessation
- 1992-03-05 AT AT92301904T patent/ATE127461T1/de not_active IP Right Cessation
- 1992-03-06 IE IE920737A patent/IE67382B1/en not_active IP Right Cessation
- 1992-03-06 JP JP4049416A patent/JPH04338381A/ja active Pending
- 1992-03-06 BR BR929200768A patent/BR9200768A/pt not_active IP Right Cessation
-
1995
- 1995-10-25 GR GR950402980T patent/GR3017875T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
EP0502735A1 (en) | 1992-09-09 |
EP0502735B1 (en) | 1995-09-06 |
IL101149A0 (en) | 1992-11-15 |
KR100193973B1 (ko) | 1999-06-15 |
HU9200745D0 (en) | 1992-05-28 |
IE67382B1 (en) | 1996-03-20 |
BR9200768A (pt) | 1992-11-17 |
IL101149A (en) | 1996-09-12 |
MX9200962A (es) | 1992-09-01 |
DE69204497D1 (de) | 1995-10-12 |
HUT61008A (en) | 1992-11-30 |
TW198014B (ko) | 1993-01-11 |
IE920737A1 (en) | 1992-09-09 |
ATE127461T1 (de) | 1995-09-15 |
CA2062329A1 (en) | 1992-09-08 |
DK0502735T3 (da) | 1996-04-09 |
ES2078652T3 (es) | 1995-12-16 |
JPH04338381A (ja) | 1992-11-25 |
US5142069A (en) | 1992-08-25 |
GR3017875T3 (en) | 1996-01-31 |
DE69204497T2 (de) | 1996-03-21 |
HU212786B (en) | 1996-11-28 |
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