KR870010007A - 피라졸 유도체, 그의 제조방법 및 농원예용 살균제 - Google Patents

피라졸 유도체, 그의 제조방법 및 농원예용 살균제 Download PDF

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KR870010007A
KR870010007A KR870003952A KR870003952A KR870010007A KR 870010007 A KR870010007 A KR 870010007A KR 870003952 A KR870003952 A KR 870003952A KR 870003952 A KR870003952 A KR 870003952A KR 870010007 A KR870010007 A KR 870010007A
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South Korea
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group
alkyl
phenyl group
formula
haloalkenyl
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KR870003952A
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KR900001196B1 (ko
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히도시 시모도리
쓰도무 이시이
히데오 야마자끼
도시아끼 구와쓰까
유우지 야나세
요시노리 다나까
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도쯔까 야스아끼
미쯔이도아쯔가가꾸 가부시기가이샤
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Electromechanical Clocks (AREA)

Abstract

내용 없음

Description

파라졸 유도체, 그의 제조방법 및 농원예용 살균제
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (8)

  1. 하기 일반식(Ⅰ)로 표시됨을 특징으로 하는 피라졸 유도체.
    상기 식에서,
    R1은 알킬기, 할로알킬, 알케닐, 할로알케닐 또는 페닐기를 나타내고;
    R2및 R3는 각각 수소 또는 할로겐 원자, 또는 알킬, 할로알킬, 알콕시, 알콕시알킬, 또는 페닐기를 나타내며:
    R4는 알킬, 알케닐, 할로알케닐 또는 페닐기, 또는 적어도 1개 이상의 산소, 질소 또는 황원자를 함유하며 치환 또는 비치환된 북소환상 방향족기를 나타낸다.
  2. 제1항에 있어서,
    일반식(Ⅰ)중 R1및 R2가 저급알킬기이고, R3가 수소원자이며, R4가 메틸기 또는 할로겐 원자로 치환 또는 비치환된 2-푸릴, 3-푸릴, 2-티에닐, 3-티에닐 또는 2-피롤릴기임을 특징으로 하는 피라졸 유도체.
  3. 제2항에 있어서,
    일반식(Ⅰ)중 R4가 2-푸릴, 3-푸릴, 2-티에닐 또는 3-티에닐기임을 특징으로 하는 피라졸 유도체.
  4. 제1항에 있어서,
    일반식(Ⅰ)중 R1및 R2가 저급알킬기이고, R3가 수소원자이며, R4가 2-메틸프로펜-1-일기임을 특징으로 하는 피라졸 유도체.
  5. 제1항에 있어서,
    하기 일반식(Ⅱ)로 표시됨을 특징으로 하는 피라졸 유도체.
    상기 식에서,
    R1및 R2는 저급알킬기이고;
    R3는 수소원자이며:
    R4는 2-푸릴, 3-푸릴, 2-티에닐 또는 3-티에닐기이다.
  6. 제5항에 있어서,
    일반식(Ⅱ)중 R4가 2-메틸프로펜-1-일기임을 특징으로 하는 피라졸 유도체.
  7. 하기 일반식(Ⅲ)의 화합물과 하기 일반식(Ⅳ)의 1아미노아세토니트릴 또는 그의 염을 반응시킴을 특징으로 하는 하기 일반식(Ⅰ)의 피라졸 유도체의 제조방법.
    상기 식들에 있어서,
    R1은 알킬기, 할로알킬, 알케닐, 할로알케닐 또는 페닐기를 나타내고:
    R2및 R3는 각각 수소 또는 할로겐 원자, 또는 알킬, 할로알킬, 알콕시, 알콕시알킬, 또는 페닐기를 나타내며:
    R4는 알킬, 알케닐, 할로알케닐 또는 페닐기, 또는 적어도 1개 이상의 산소, 질소 또는 황원자를 함유하며 치환 또는 비치환된 복소환상 방향족기를 나타내며:
    X는 할로겐 원자를 나타낸다.
  8. 하기 일반식(Ⅰ)의 피라졸 유도체를 활성성분으로 함유함을 특징으로 하는 농원예용 살균제.
    상기식에서,
    R1은 알킬기, 할로알킬, 알케닐, 할로알케닐 또는 페닐기를 나타내고:
    R2및 R3는 각각 수소 또는 할로겐 원자, 또는 알킬, 할로알킬, 알콕시, 알콕시알킬, 또는 페닐기를 나타내며:
    R4는 알킬, 알케닐, 할로알케닐 또는 페닐기, 또는 적어도 1개 이상의 산소, 질소 또는 황원자를 함유하며 치환 또는 비치환된 복소환상 방향족기를 나타낸다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019870003952A 1986-04-24 1987-04-24 피라졸 유도체의 제조방법 KR900001196B1 (ko)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
JP61-93328 1986-04-24
JP93328 1986-04-24
JP9332886 1986-04-24
JP61-139981 1986-06-18
JP13998186 1986-06-18
JP139981 1986-06-18
JP26201886 1986-11-05
JP61-262018 1986-11-05
JP262018 1986-11-05

Publications (2)

Publication Number Publication Date
KR870010007A true KR870010007A (ko) 1987-11-30
KR900001196B1 KR900001196B1 (ko) 1990-02-28

Family

ID=27307266

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Application Number Title Priority Date Filing Date
KR1019870003952A KR900001196B1 (ko) 1986-04-24 1987-04-24 피라졸 유도체의 제조방법

Country Status (16)

Country Link
US (1) US4792565A (ko)
KR (1) KR900001196B1 (ko)
AU (1) AU597054B2 (ko)
BR (1) BR8701936A (ko)
CA (1) CA1322759C (ko)
CH (1) CH668771A5 (ko)
DE (1) DE3713774C2 (ko)
ES (1) ES2005186A6 (ko)
FR (1) FR2597866B1 (ko)
GB (1) GB2190375B (ko)
GR (1) GR870626B (ko)
HU (1) HU200080B (ko)
IT (1) IT1203975B (ko)
NL (1) NL8700976A (ko)
PL (2) PL154298B1 (ko)
RO (2) RO100209B1 (ko)

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* Cited by examiner, † Cited by third party
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DE3633840A1 (de) * 1986-10-04 1988-04-14 Hoechst Ag Phenylpyrazolcarbonsaeurederivate, ihre herstellung und verwendung als pflanzenwachstumsregulatoren und safener
EP0268892A3 (en) * 1986-11-06 1990-10-10 Nissan Chemical Industries Ltd. Substituted-amido derivatives, method for preparation of the same and phytopathogenic fungicides containing the same
ES2061556T3 (es) * 1987-05-26 1994-12-16 Sumitomo Chemical Co Derivados amida y su produccion y fungicidas agricolas que los contienen.
IL91418A (en) * 1988-09-01 1997-11-20 Rhone Poulenc Agrochimie (hetero) cyclic amide derivatives, process for their preparation and fungicidal compositions containing them
AU622330B2 (en) * 1989-06-23 1992-04-02 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
FR2665898B1 (fr) * 1990-08-20 1994-03-11 Sanofi Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2682379B1 (fr) * 1991-10-09 1994-02-11 Rhone Poulenc Agrochimie Nouveaux phenylpyrazoles fongicides.
FR2690440B1 (fr) * 1992-04-27 1995-05-19 Rhone Poulenc Agrochimie Arylpyrazoles fongicides.
DE19544800A1 (de) * 1995-12-01 1997-06-05 Bayer Ag Verfahren zur Herstellung von 1,3-Dimethyl-5-fluor-pyrazol-4-carboxaniliden
WO2001023358A1 (fr) * 1999-09-27 2001-04-05 Sagami Chemical Research Center Derives pyrazole, intermediaires pour la preparation de ces derives, procedes de preparation des derives et intermediaires, et herbicides dont ces derives sont le principe actif
BRPI0610459A2 (pt) * 2005-04-05 2010-06-22 Hoffmann La Roche composto, processo para a sua preparação, composições farmacêuticas que o compreendem, método para o tratamento terapêutico e/ou profilático de enfermidades que são moduladas por inibidores de deidrogenase de hidroxiesteróides-11b e utilização do composto
DK1999114T3 (en) 2006-03-22 2015-08-03 Hoffmann La Roche Pyrazoles AS 11-BETA-HSD-1
DE102007002674A1 (de) * 2007-01-18 2008-07-24 Bayer Cropscience Ag Verfahren zum Herstellen von substituierten Pyrazolcarbonsäurechloriden
CN101007772B (zh) * 2007-01-29 2010-05-26 浙江大学 一种手性正缬氨酸的合成方法
JP2010534717A (ja) * 2007-07-31 2010-11-11 バイエル・クロツプサイエンス・エス・アー 殺真菌剤ｎ−５員縮合ヘテロアリール−メチレン−ｎ−シクロアルキル−カルボキサミド誘導体
WO2019016069A1 (de) 2017-07-18 2019-01-24 Bayer Cropscience Aktiengesellschaft Substituierte 5-(het-)arylpyrazolamide sowie deren salze und ihre verwendung als herbizide wirkstoffe

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JPS59122488A (ja) * 1982-12-28 1984-07-14 Nissan Chem Ind Ltd ピラゾ−ルスルホニルウレア誘導体、その製法および該誘導体を含有する除草剤
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EP0268892A3 (en) * 1986-11-06 1990-10-10 Nissan Chemical Industries Ltd. Substituted-amido derivatives, method for preparation of the same and phytopathogenic fungicides containing the same

Also Published As

Publication number Publication date
DE3713774C2 (de) 1993-10-07
KR900001196B1 (ko) 1990-02-28
PL265359A1 (en) 1988-09-01
IT8720267A0 (it) 1987-04-24
FR2597866A1 (fr) 1987-10-30
GB8709654D0 (en) 1987-05-28
RO100209B1 (en) 1992-03-24
US4792565A (en) 1988-12-20
PL152292B1 (en) 1990-12-31
HUT43936A (en) 1988-01-28
AU7196187A (en) 1987-10-29
CA1322759C (en) 1993-10-05
BR8701936A (pt) 1988-02-02
FR2597866B1 (fr) 1990-03-02
HU200080B (en) 1990-04-28
GB2190375B (en) 1990-05-02
GR870626B (en) 1987-08-28
NL8700976A (nl) 1987-11-16
CH668771A5 (de) 1989-01-31
PL154298B1 (en) 1991-07-31
RO100208B1 (en) 1992-03-17
ES2005186A6 (es) 1989-03-01
AU597054B2 (en) 1990-05-24
GB2190375A (en) 1987-11-18
DE3713774A1 (de) 1987-10-29
IT1203975B (it) 1989-02-23

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