KR20050026535A - Ｖｅｇｆｒ-2 및 ｖｅｇｆｒ-3 억제성 안트라닐아미도피리딘 - Google Patents

Ｖｅｇｆｒ-2 및 ｖｅｇｆｒ-3 억제성 안트라닐아미도피리딘 Download PDF

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KR20050026535A
KR20050026535A KR1020057001611A KR20057001611A KR20050026535A KR 20050026535 A KR20050026535 A KR 20050026535A KR 1020057001611 A KR1020057001611 A KR 1020057001611A KR 20057001611 A KR20057001611 A KR 20057001611A KR 20050026535 A KR20050026535 A KR 20050026535A
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alkyl
alkoxy
halo
group
differently
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KR1020057001611A
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Korean (ko)
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안드레아스 후쓰
마틴 크뤼거
루비그 조른
스튜어트 인세
칼-헤인즈 티에라우츠
안드레아스 멘라드
마틴 하베리
홀거 헤스-스텀프
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쉐링 악티엔게젤샤프트
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Priority claimed from DE10235690A external-priority patent/DE10235690A1/de
Priority claimed from DE10328036A external-priority patent/DE10328036A1/de
Application filed by 쉐링 악티엔게젤샤프트 filed Critical 쉐링 악티엔게젤샤프트
Publication of KR20050026535A publication Critical patent/KR20050026535A/ko

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
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  • Rheumatology (AREA)
  • Oncology (AREA)
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  • Emergency Medicine (AREA)
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KR1020057001611A 2002-07-31 2003-07-22 Ｖｅｇｆｒ-2 및 ｖｅｇｆｒ-3 억제성 안트라닐아미도피리딘 KR20050026535A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE10235690.4 2002-07-31
DE10235690A DE10235690A1 (de) 2002-07-31 2002-07-31 VEGFR-2 und VEGFR-3 inhibitorische Anthranylamidpyridinamide
DE10328036A DE10328036A1 (de) 2003-06-19 2003-06-19 VEGFR-2 und VEGFR-3 inhibitorische Anthranylamidpyridine
DE10328036.7 2003-06-19

Publications (1)

Publication Number Publication Date
KR20050026535A true KR20050026535A (ko) 2005-03-15

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KR1020057001611A KR20050026535A (ko) 2002-07-31 2003-07-22 Ｖｅｇｆｒ-2 및 ｖｅｇｆｒ-3 억제성 안트라닐아미도피리딘

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EP (1) EP1594841A1 (xx)
JP (2) JP4777648B2 (xx)
KR (1) KR20050026535A (xx)
CN (1) CN1671666A (xx)
AU (1) AU2003281855A1 (xx)
BR (1) BR0313122A (xx)
CA (1) CA2493026C (xx)
CO (1) CO5720998A2 (xx)
CR (1) CR7673A (xx)
EC (1) ECSP055631A (xx)
HR (1) HRP20050187A2 (xx)
IL (1) IL166377A0 (xx)
MX (1) MXPA04012948A (xx)
NO (1) NO20051035L (xx)
PL (1) PL374610A1 (xx)
RS (1) RS20050084A (xx)
RU (1) RU2005105683A (xx)
WO (1) WO2004013102A1 (xx)

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GB0229022D0 (en) * 2002-12-12 2003-01-15 Novartis Ag Organic Compounds
MXPA05007513A (es) 2003-01-14 2005-09-21 Cytokinetics Inc Compuestos, composiciones y metodos.
DE102004009238A1 (de) * 2004-02-26 2005-09-08 Merck Patent Gmbh Arylamid-Derivate
BRPI0512193B8 (pt) 2004-06-17 2021-05-25 Cytokinetics Inc composto ou sal farmaceuticamente aceitável, composição farmacêutica, e, uso do composto ou sal
US7176222B2 (en) 2004-07-27 2007-02-13 Cytokinetics, Inc. Syntheses of ureas
US7906533B2 (en) 2004-11-03 2011-03-15 Bayer Schering Pharma Ag Nicotinamide pyridinureas as vascular endothelial growth factor (VEGF) receptor kinase inhibitors
EP1655295A1 (en) 2004-11-03 2006-05-10 Schering Aktiengesellschaft Anthranilamide pyridinureas as VEGF receptor kinase inhibitors
EP1657241A1 (en) * 2004-11-03 2006-05-17 Schering Aktiengesellschaft Novel anthranilamide pyridinureas as VEGF receptor kinase inhibitors
EP1655297A1 (en) * 2004-11-03 2006-05-10 Schering Aktiengesellschaft Nicotinamide pyridinureas as vascular endothelial growth factor (VEGF) receptor kinase inhibitors
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