KR101582910B1 - 스핑고신 포스페이트 수용체의 신규한 모듈레이터 - Google Patents

스핑고신 포스페이트 수용체의 신규한 모듈레이터 Download PDF

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Publication number
KR101582910B1
KR101582910B1 KR1020107028062A KR20107028062A KR101582910B1 KR 101582910 B1 KR101582910 B1 KR 101582910B1 KR 1020107028062 A KR1020107028062 A KR 1020107028062A KR 20107028062 A KR20107028062 A KR 20107028062A KR 101582910 B1 KR101582910 B1 KR 101582910B1
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South Korea
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delete delete
compound
heteroaryl
alkyl
heterocyclyl
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KR1020107028062A
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English (en)
Korean (ko)
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KR20110010777A (ko
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에드워드 로버츠
휴 로젠
스티븐 브라운
미구엘 에이. 게레로
수에메이 펭
라물루 포두토리
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더 스크립스 리서치 인스티튜트
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Publication of KR20110010777A publication Critical patent/KR20110010777A/ko
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Publication of KR101582910B1 publication Critical patent/KR101582910B1/ko

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Health & Medical Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
KR1020107028062A 2008-05-14 2009-05-14 스핑고신 포스페이트 수용체의 신규한 모듈레이터 KR101582910B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12760308P 2008-05-14 2008-05-14
US61/127,603 2008-05-14

Related Child Applications (1)

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KR1020157013971A Division KR20150064245A (ko) 2008-05-14 2009-05-14 스핑고신 포스페이트 수용체의 신규한 모듈레이터

Publications (2)

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KR20110010777A KR20110010777A (ko) 2011-02-07
KR101582910B1 true KR101582910B1 (ko) 2016-01-08

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KR1020107028062A KR101582910B1 (ko) 2008-05-14 2009-05-14 스핑고신 포스페이트 수용체의 신규한 모듈레이터
KR1020157013971A KR20150064245A (ko) 2008-05-14 2009-05-14 스핑고신 포스페이트 수용체의 신규한 모듈레이터

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KR1020157013971A KR20150064245A (ko) 2008-05-14 2009-05-14 스핑고신 포스페이트 수용체의 신규한 모듈레이터

Country Status (12)

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KR (2) KR101582910B1 (es)
CN (1) CN102118972B (es)
BR (1) BRPI0912545B1 (es)
CA (1) CA2723904C (es)
DK (1) DK2913326T3 (es)
HR (1) HRP20201316T1 (es)
HU (1) HUE050411T2 (es)
IL (1) IL209306A (es)
LT (1) LT2913326T (es)
MX (1) MX2010012461A (es)
SI (1) SI2913326T1 (es)
ZA (1) ZA201007804B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA021672B1 (ru) 2008-05-14 2015-08-31 Дзе Скриппс Рисёч Инститьют Модуляторы рецепторов сфингозин-1-фосфата и их применение
JP6615876B2 (ja) * 2014-06-26 2019-12-04 モナシュ ユニヴァーシティ 酵素相互作用薬剤
US11111223B2 (en) 2016-06-14 2021-09-07 Receptos Llc Crystalline forms of ozanimod and ozanimod hydrochloride, and processes for preparation thereof
WO2018033149A1 (zh) * 2016-08-19 2018-02-22 苏州科睿思制药有限公司 奥扎莫德的晶型及其制备方法
WO2018049632A1 (zh) 2016-09-14 2018-03-22 杭州领业医药科技有限公司 奥扎莫德的晶型、其制备方法及药物组合物
CN109640982A (zh) 2016-09-14 2019-04-16 苏州科睿思制药有限公司 奥扎莫德盐酸盐的晶型及其制备方法
CN106749213B (zh) * 2016-11-25 2019-07-02 济南大学 一种具有1,2,4-恶二唑结构的吲哚衍生物及制备方法和在制备抗菌药物中的应用
US11117876B2 (en) 2017-08-31 2021-09-14 Receptos Llc Crystalline form of ozanimod hydrochloride, and processes for preparation thereof
CN107827837B (zh) * 2017-11-21 2021-09-24 苏州朗科生物技术股份有限公司 鞘氨醇-1-磷酸受体调节剂化合物及其制备方法与应用

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007116866A1 (ja) 2006-04-03 2007-10-18 Astellas Pharma Inc. ヘテロ化合物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4516430B2 (ja) * 2002-12-20 2010-08-04 メルク・シャープ・エンド・ドーム・コーポレイション １−（アミノ）インダン並びに（１，２−ジヒドロ−３−アミノ）−ベンゾフラン、ベンゾチオフェン及びインドール

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007116866A1 (ja) 2006-04-03 2007-10-18 Astellas Pharma Inc. ヘテロ化合物

Also Published As

Publication number Publication date
CA2723904C (en) 2017-03-14
DK2913326T3 (da) 2020-08-17
IL209306A (en) 2017-02-28
CA2723904A1 (en) 2009-12-17
ZA201007804B (en) 2012-01-25
LT2913326T (lt) 2020-09-10
IL209306A0 (en) 2011-01-31
BRPI0912545B1 (pt) 2022-02-01
KR20150064245A (ko) 2015-06-10
MX2010012461A (es) 2013-07-02
KR20110010777A (ko) 2011-02-07
BRPI0912545A2 (pt) 2021-04-13
HUE050411T2 (hu) 2020-12-28
HRP20201316T1 (hr) 2020-11-27
CN102118972A (zh) 2011-07-06
SI2913326T1 (sl) 2020-11-30
CN102118972B (zh) 2015-06-10

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