JPS56142280A - Piperidine compound - Google Patents
Piperidine compoundInfo
- Publication number
- JPS56142280A JPS56142280A JP4650480A JP4650480A JPS56142280A JP S56142280 A JPS56142280 A JP S56142280A JP 4650480 A JP4650480 A JP 4650480A JP 4650480 A JP4650480 A JP 4650480A JP S56142280 A JPS56142280 A JP S56142280A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- group
- alkylene
- lower alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Abstract
NEW MATERIAL:A compound of formula I [R1 is group of formula II (X1 and X2 are H, halogen, lower alkyl, lower alkoxyl, etc.; Y is N, =C=CH-, etc., Z1 and Z2 are H or together link to form single bond, methylene, ethylene, etc.); group of formula III (X3 is H or amino, etc.); R2 is H, lower alkyl, etc.; A is lower alkylene, etc.; B is alkylene or alkylidene].
EXAMPLE: 1-[ 1-[3-( 10,11-Dihydro-5H-dibenz[b,f]azepin-5-yl )propyl]-4-piperidinyl]hydrouracil hydrochloride.
USE: A tranquilizer useful for the remedy of schizophrenia, manic-depressive psychosis, etc.
PROCESS: A compound of formula IV (Q is Cl, Br, etc.) is reacted with a compound of formula V in an inert solvent, e.g. methanol, if necessary in the presence of a deacidifying agent, e.g. Na2CO3, at 0°C to the boiling point of the solvent to give the compound of formula I.
COPYRIGHT: (C)1981,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP4650480A JPS56142280A (en) | 1980-04-08 | 1980-04-08 | Piperidine compound |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP4650480A JPS56142280A (en) | 1980-04-08 | 1980-04-08 | Piperidine compound |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS56142280A true JPS56142280A (en) | 1981-11-06 |
JPS6258357B2 JPS6258357B2 (en) | 1987-12-05 |
Family
ID=12749070
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP4650480A Granted JPS56142280A (en) | 1980-04-08 | 1980-04-08 | Piperidine compound |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS56142280A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0677516A1 (en) * | 1990-06-15 | 1995-10-18 | Eisai Co., Ltd. | Cyclic amide derivatives |
JP2003513088A (en) * | 1999-10-29 | 2003-04-08 | ベーリンガー インゲルハイム ファルマ コマンディトゲゼルシャフト | Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and methods for their preparation |
-
1980
- 1980-04-08 JP JP4650480A patent/JPS56142280A/en active Granted
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0677516A1 (en) * | 1990-06-15 | 1995-10-18 | Eisai Co., Ltd. | Cyclic amide derivatives |
US5521182A (en) * | 1990-06-15 | 1996-05-28 | Eisai Co., Ltd. | 1,2,3,4 tetrahydropteridinone cyclic amide derivatives |
US5620976A (en) * | 1990-06-15 | 1997-04-15 | Eisai Co., Ltd. | Benzoxazine derivatives |
US5654308A (en) * | 1990-06-15 | 1997-08-05 | Eisai Co., Ltd. | Bicyclic amide derivatives, compositions and methods of treatment |
US5919778A (en) * | 1990-06-15 | 1999-07-06 | Eisai Co., Ltd. | Cyclic amide derivatives |
JP2003513088A (en) * | 1999-10-29 | 2003-04-08 | ベーリンガー インゲルハイム ファルマ コマンディトゲゼルシャフト | Arylalkanes, arylalkenes and aryl-azaalkanes, pharmaceutical compositions containing these compounds and methods for their preparation |
Also Published As
Publication number | Publication date |
---|---|
JPS6258357B2 (en) | 1987-12-05 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
GR68522B (en) | ||
ES8705412A1 (en) | Furan derivatives having anti-ulcer activity. | |
JPS56115769A (en) | Piperazine derivative and its preparation | |
EP0555480A4 (en) | Novel thiazole derivative | |
JPS56142280A (en) | Piperidine compound | |
JPS5692884A (en) | Novel piperidine derivative and its preparation | |
JPS54160371A (en) | Novel piperidine derivative and hypotensive agents comprising it | |
JPS56122356A (en) | Carbostyril derivative | |
JPS5649364A (en) | Carbostyril derivative | |
JPS5583749A (en) | Quinolone derivative | |
JPS55104264A (en) | Bezyl ketal derivative | |
YU175484A (en) | Process for obtaining novel in position 5 substituted 5,10-dihydro-11h-dibenzo | |
JPS5524127A (en) | 3,6-endomethylene-delta4-1,2,3,6-tetrahydrophtalimide derivative | |
JPS5714590A (en) | 2-benzyl-5-alkyl-tetrahydro-benzo(b)-1,6-naphthyridin-10-one derivative and its preparation | |
JPS56120686A (en) | Tetrahydrothiopyrano 3,2-b indole derivative | |
JPS56156263A (en) | Carbostyril derivative | |
JPS5459287A (en) | Preparation of 2,2,6,6-tetramethylpiperidne derivative | |
JPS57106663A (en) | 1,4-disubstituted piperazine derivative and its preparation | |
JPS54128583A (en) | Thiosemicarbazone derivative | |
JPS5653654A (en) | Preparation of novel aniline derivative | |
JPS56164183A (en) | Novel piperidine derivative | |
JPS57136561A (en) | Benzenesulfonamide derivative | |
JPS57212174A (en) | Thiazolidine compound | |
JPS56161386A (en) | Novel piperidine derivative | |
HUT36126A (en) | Process for producing new 2,6.dioxa-bicyclo/2.2.2/octan-7-yl-acetaldehyde derivatives |