JP2014015447A - Pyrazole derivative and pest control agent - Google Patents

Abstract

PROBLEM TO BE SOLVED: To provide a novel pest control agent, particularly an insecticide or a miticide.SOLUTION: There are provided: a pyrazole derivative represented by formula (1) [In the formula, Arepresents -N(O)or -CR, R, R, R, and Reach represent a hydrogen atom, a halogen atom, cyano, C- Calkyl, C- Chaloalkyl, or the like, and Arepresents -C(R)=NOH, -C(R)=NOR, -C≡CR, or -C(R)=C(R)R.]; and a pest control agent.

Description

本発明は、新規なピラゾール誘導体及びそれらの塩、並びに該化合物を有効成分として含有することを特徴とする有害生物防除剤に関するものである。本発明における有害生物防除剤とは、農園芸分野又は畜産・衛生分野（家畜や愛玩動物としての哺乳動物又は鳥類に対する内部寄生虫・外部寄生虫や家庭用及び業務用の衛生害虫・不快害虫）等における有害な節足動物を対象とした害虫防除剤を意味する。また、本発明における農薬とは、農園芸分野における殺虫・殺ダニ剤、殺線虫剤、除草剤及び殺菌剤等を意味する。   The present invention relates to a novel pyrazole derivative and a salt thereof, and a pest control agent containing the compound as an active ingredient. The pest control agent in the present invention is the field of agriculture and horticulture or the field of livestock and hygiene (internal parasites / external parasites for domestic animals and pets, hygiene pests and unpleasant pests for domestic and commercial use) It means a pest control agent for harmful arthropods such as The agrochemical in the present invention means an insecticide / acaricide, nematicide, herbicide, fungicide, etc. in the field of agriculture and horticulture.

例えば特許文献１〜３にピラゾール誘導体が開示されているが、本発明に係るピラゾール誘導体に関しては何ら開示されていない。さらに、その有害生物防除剤、特に殺虫・殺ダニ剤及び哺乳動物又は鳥類の内部もしくは外部寄生虫防除剤としての有用性も全く知られていない。   For example, Patent Documents 1 to 3 disclose pyrazole derivatives, but nothing is disclosed about the pyrazole derivative according to the present invention. Furthermore, its usefulness as a pest control agent, particularly an insecticide / acaricide, and an internal or ectoparasite control agent for mammals or birds is not known at all.

国際公開第２０１０／０３４８３８号International Publication No. 2010/034838 国際公開第２０１０／０１７０４７号International Publication No. 2010/017047 米国特許出願公開第２００７／２１９２１８号US Patent Application Publication No. 2007/219218

農園芸病害虫、森林病害虫、或いは衛生病害虫等、各種病害虫の防除を目的とする有害生物防除剤の開発が進み、多種多様な薬剤が今日まで実用に供されてきた。   The development of pest control agents for the purpose of controlling various pests such as agricultural and horticultural pests, forest pests, and hygiene pests has progressed, and a wide variety of drugs have been put to practical use to date.

しかしながら、こうした薬剤の長年にわたる使用により、近年、病害虫が薬剤抵抗性を獲得し、従来用いられてきた既存の殺虫剤や殺菌剤による防除が困難となる場面が増えてきている。また、既存の有害生物防除剤の一部のものは毒性が高く、或いはあるものは環境中に長期間残留することにより、生態系を攪乱するという問題も顕在化しつつある。このような状況下、高度な有害生物防除活性を有するのみならず、低毒性且つ低残留性の新規な有害生物防除剤の開発が常に期待されている。   However, due to the long-term use of such drugs, in recent years, pests have acquired drug resistance, making it difficult to control with existing insecticides and fungicides that have been used. In addition, some existing pest control agents are highly toxic, or some of them remain in the environment for a long time, and the problem of disturbing the ecosystem is becoming apparent. Under such circumstances, development of a novel pest control agent having not only high pest control activity but also low toxicity and low persistence is always expected.

本発明者らは、上記の課題解決を目標に鋭意研究を重ねた結果、本発明に係る下記式（１）で表される新規なピラゾール誘導体が優れた有害生物防除活性、特に殺虫・殺ダニ活性を示し、且つ、ホ乳動物、魚類及び益虫等の非標的生物に対してほとんど悪影響の無い、極めて有用な化合物であることを見い出し、本発明を完成した。   As a result of intensive studies aimed at solving the above problems, the present inventors have found that the novel pyrazole derivative represented by the following formula (1) according to the present invention has excellent pest control activity, particularly insecticide / miticide. The present invention has been completed by finding it to be an extremely useful compound that exhibits activity and has almost no adverse effects on non-target organisms such as mammals, fish and beneficial insects.

すなわち、本発明は下記〔１〕〜〔１０〕に関するものである。   That is, the present invention relates to the following [1] to [10].

〔１〕
式（１）： [1]
Formula (1):

〔式中、Ａ^１は、−Ｎ（−Ｏ）_ｍ２又は−ＣＲ^１を表し、
Ｒ^１、Ｒ^３及びＲ^４は、各々独立して水素原子、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、Ｃ_１〜Ｃ_６アルキル、Ｒ^２８ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_３〜Ｃ_８ハロシクロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６ハロアルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルチオカルボニル、Ｃ_１〜Ｃ_６アルコキシチオカルボニル、Ｃ_１〜Ｃ_６アルキルジチオカルボニル、Ｃ_１〜Ｃ₆アルキルアミノカルボニル、Ｃ_１〜Ｃ₆ハロアルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノカルボニル、トリ（Ｃ_１〜Ｃ_６アルキル）シリル、Ｃ_１〜Ｃ₆アルキルアミノスルホニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、Ｃ_１〜Ｃ_６アルキルスルホニルオキシ、Ｃ_１〜Ｃ_６ハロアルキルスルホニルオキシ、Ｃ_１〜Ｃ_６アルキルアミノ、ジ（Ｃ_１〜Ｃ_６アルキル）アミノ、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^２は、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、Ｃ_１〜Ｃ_６アルキル、Ｒ^２８ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_３〜Ｃ_８ハロシクロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６ハロアルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルチオカルボニル、Ｃ_１〜Ｃ_６アルコキシチオカルボニル、Ｃ_１〜Ｃ_６アルキルジチオカルボニル、Ｃ_１〜Ｃ₆アルキルアミノカルボニル、Ｃ_１〜Ｃ₆ハロアルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノカルボニル、トリ（Ｃ_１〜Ｃ_６アルキル）シリル、Ｃ_１〜Ｃ₆アルキルアミノスルホニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、Ｃ_１〜Ｃ_６アルキルスルホニルオキシ、Ｃ_１〜Ｃ_６ハロアルキルスルホニルオキシ、Ｃ_１〜Ｃ_６アルキルアミノ、ジ（Ｃ_１〜Ｃ_６アルキル）アミノ、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、ｎが２以上の整数を表すとき、各々のＲ^２は互いに同一であっても又は互いに相異なってもよく、
Ａ^２は、−Ｃ（Ｒ^ａ）＝ＮＯＨ、−Ｃ（Ｒ^ａ）＝ＮＯＲ^ｂ、−Ｃ≡ＣＲ^ｃ、−Ｃ（Ｒ^ｄ）＝Ｃ（Ｒ^ｅ）Ｒ^ｆ又は−Ｃ（Ｒ^ａ）＝ＮＮ（Ｒ^ｇ）Ｒ^ｇ２を表し、
Ｒ^ａは、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、或いは、Ｒ^ａはＲ^３と一緒になってＣ_２〜Ｃ_５のアルキレン鎖又はＣ_２〜Ｃ_５アルケニレン鎖を形成することにより、Ｒ^ａが結合する炭素原子及びＲ^３が結合する炭素原子と共に５〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１又は２個含んでもよく、且つハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−ＯＨ，−ＯＲ^１１、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１１、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^ｂは、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^ｃは、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^ｄは、水素原子、ハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ又は−Ｃ（Ｏ）Ｒ^７を表し、
Ｒ^ｅ及びＲ^ｆは、各々独立して水素原子、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、或いは、Ｒ^ｅはＲ^ｆと一緒になってＣ_２〜Ｃ_７のアルキレン鎖を形成することにより、Ｒ^ｅ及びＲ^ｆが結合する炭素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖は酸素原子、硫黄原子又は窒素原子を１又は２個個含んでもよく、且つハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−ＯＨ，−ＯＲ^１１、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１１、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^ｇ及びＲ^ｇ２は、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^５は、ハロゲン原子、シアノ、Ｃ_３〜Ｃ_８シクロアルキル、−ＯＨ、−ＯＲ^１１、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１１、−Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｃ（Ｏ）ＯＲ^１１ａ、−Ｃ（Ｓ）ＯＲ^１１ａ、−Ｃ（Ｏ）ＳＲ^１１ａ、−Ｃ（Ｓ）ＳＲ^１１ａ、−Ｃ（Ｏ）Ｒ^１２、−Ｃ（Ｓ）Ｒ^１２、−Ｃ（Ｏ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｃ（Ｓ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｓ（Ｏ）_ｒＮ（Ｒ^１３ａ）Ｒ^１３、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^６及びＲ^６ａは、各々独立してＣ_１〜Ｃ_６アルキル又はＲ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^７は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^８及びＲ^８ａは、各々独立して水素原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−Ｓ（Ｏ）_ｒＲ^１１、−Ｃ（Ｏ）ＯＲ^１１ａ、−Ｃ（Ｓ）ＯＲ^１１ａ、−Ｃ（Ｏ）ＳＲ^１１ａ、−Ｃ（Ｓ）ＳＲ^１１ａ、−Ｃ（Ｏ）Ｒ^１２、−Ｃ（Ｓ）Ｒ^１２、−Ｃ（Ｏ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｃ（Ｓ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｓ（Ｏ）_ｒＮ（Ｒ^１３ａ）Ｒ^１３、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、、或いは、Ｒ^８はＲ^８ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^８及びＲ^８ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、且つハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、フェニル、（Ｚ^２）_ｑ２によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^９、Ｒ^９ａ及びＲ^９ｂは、各々独立してＣ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６アルコキシ又はフェニルを表し、
Ｒ^１１は、−Ｓ（Ｏ）_２Ｒ^１５ａ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１１ａ及びＲ^１２は、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１３及びＲ^１３ａは、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、、或いは、Ｒ^１３はＲ^１３ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^１３及びＲ^１３ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、且つハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、フェニル、（Ｚ^２）_ｑ２によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^１４及びＲ^１４ａは、各々独立してハロゲン原子、シアノ、ニトロ、Ｃ_３〜Ｃ_８シクロアルキル、Ｃ_３〜Ｃ_８ハロシクロアルキル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｃ_３〜Ｃ_８ハロシクロアルケニル、−ＯＨ、−ＯＲ^１５、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１５、−Ｎ（Ｒ^１７ａ）Ｒ^１７、−Ｃ（Ｏ）ＯＲ^１５、−Ｃ（Ｏ）ＳＲ^１５、−Ｃ（Ｓ）ＯＲ^１５、−Ｃ（Ｓ）ＳＲ^１５、−Ｃ（Ｏ）Ｒ^１６、−Ｃ（Ｏ）Ｎ（Ｒ^１７ａ）Ｒ^１７、−Ｃ（Ｓ）Ｎ（Ｒ^１７ａ）Ｒ^１７、−Ｓ（Ｏ）_ｒＮ（Ｒ^１７ａ）Ｒ^１７、−Ｃ（＝ＮＲ^１７）ＯＲ^１５、−Ｃ（＝ＮＲ^１７）Ｓ（Ｏ）_ｒＲ^１５、−Ｃ（＝ＮＲ^１７）Ｒ^１６、−Ｃ（＝ＮＯＨ）Ｒ^１６、−Ｃ（＝ＮＯＲ^１５）Ｒ^１６、−Ｃ｛＝ＮＮ（Ｒ^１７ａ）Ｒ^１７｝Ｒ^１６、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、を表し、
Ｒ^１５及びＲ^１５ａは、各々独立してＣ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１６は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１７及びＲ^１７ａは、各々独立して水素原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、或いは、Ｒ^１７はＲ^１７ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^１７及びＲ^１７ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、且つハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、フェニル、（Ｚ^２）_ｑ２によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^１８は、ハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｄ２−１〜Ｄ２−１０２は、それぞれ下記の構造式で表される環を表し、 [Wherein, A ¹ represents —N (—O) _{m 2} or —CR ¹ ;
R ¹ , R ³ and R ⁴ are each independently optionally substituted with a hydrogen atom, a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , C ₁ -C ₆ alkyl, R ^28a ( C ₁ -C ₆ ) alkyl, C ₃ -C ₈ cycloalkyl, optionally substituted with R ^28a (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ alkenyl, optionally substituted with R ^28a ( C ₂ -C _{6) alkenyl,} C 3 -C ₈ ^{cycloalkenyl,} substituted optionally substituted with ^{R 28a} _(C 3 ~C _{8) cycloalkenyl,} C 2 -C ₆ ^alkynyl, optionally with ^{R 28a} ( C ₂ -C _{6) alkynyl,} C 1 -C _{6 alkoxy,} C 1 -C _{6 haloalkoxy,} C 2 -C _{6 alkenyloxy,} C 1 -C _{6 alkylthio,} C 1 -C _{6 alkylsulfinyl, C} 1 ~ _{6 alkylsulfonyl,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 haloalkylsulfonyl,} C 1 -C _{6 alkylcarbonyl,} C 3 -C _{8 cycloalkylcarbonyl,} C 1 -C _{6 haloalkylcarbonyl,} C 3 -C ₈ halocycloalkyl _carbonyl, C 1 -C _{6 alkoxycarbonyl,} C 1 -C _{6 haloalkoxycarbonyl,} C 1 -C _{6 alkylthiocarbonyl,} C 1 -C _{6 alkoxythiocarbonyl, C} 1 ~ C ₆ alkyldithiocarbonyl, C ₁ -C ₆ alkylaminocarbonyl, C ₁ -C ₆ haloalkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, tri (C ₁ -C ₆ alkyl) silyl, C _1- C ₆ alkylaminosulfonyl, di _(C 1 ~ ₆ alkyl) _{aminosulfonyl,} C 1 -C _{6 alkylcarbonyloxy,} C 1 -C _{6 alkylsulfonyloxy,} C 1 -C _{6 haloalkylsulfonyloxy,} C 1 -C ₆ alkylamino, di _(C 1 -C ₆ alkyl) represents amino, phenyl, ^naphthyl, phenyl substituted with (Z _{2) ^q2,} naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ² is a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^28a , C ₃ -C _8. ^cycloalkyl, substituted optionally substituted with ^{R 28a} _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ ^alkenyl, optionally with ^{R 28a} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ ^{cycloalkenyl,} optionally substituted with ^{R 28a} _(C 3 ~C _{8) cycloalkenyl,} C 2 -C ₆ ^alkynyl, which is optionally substituted with ^{R 28a} _(C 2 ~C _{6) alkynyl,} C 1 -C _{6 alkoxy,} C 1 -C _{6 haloalkoxy,} C 2 -C _{6 alkenyloxy,} C 1 -C _{6 alkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ C _{Roarukiruchio,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 haloalkylsulfonyl,} C 1 -C _{6 alkylcarbonyl,} C 3 -C _{8 cycloalkylcarbonyl,} C 1 -C _{6 haloalkylcarbonyl,} C 3 -C ₈ halo Cycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, C ₁ -C ₆ alkylthiocarbonyl, C ₁ -C ₆ alkoxythiocarbonyl, C ₁ -C ₆ alkyldithiocarbonyl, C _1- C _{6 alkylaminocarbonyl,} C 1 -C ₆ haloalkylcarbonyl aminocarbonyl, di _(C 1 -C ₆ alkyl) aminocarbonyl, tri _(C 1 -C ₆ alkyl) _silyl, C 1 -C ₆ alkylaminosulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, _{C 1} C _{6 alkylcarbonyloxy,} C 1 -C _{6 alkylsulfonyloxy,} C 1 -C _{6 haloalkylsulfonyloxy,} C 1 -C ₆ alkylamino, di _(C 1 -C ₆ alkyl) amino, phenyl, naphthyl, ^{(Z 2} ) Represents a phenyl substituted with _q2 , (Z ² ) a naphthyl substituted with _q2 , or D2-1 to D2-102, and when n represents an integer of 2 or more, each R ² may be the same as each other Or they may be different from each other,
A ² is —C (R ^a ) = NOH, —C (R ^a ) = NOR ^b , —C≡CR ^c , —C (R ^d ) = C (R ^e ) R ^f or —C (R ^a ) = NN (R ^g ) R ^g2 ,
R ^a is a hydrogen _atom, C 1 -C ₆ alkyl, optionally substituted with ^{R 5} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ cycloalkyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkyl,} C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkenyl,} C 2 -C ₆ alkynyl, optionally substituted with ^{R 5} _(C 2 ~C ₆₎ ^{alkynyl, -OH, -OR 6, -SH,} -S (O) r R 6, ^{-N (R 8a) R 8,} -C (O) OR 6a, -C (O) SR 6a, -C (S) OR 6a, -C (S) SR 6a, -C (O) R 7, - ^{C (S) R 7, -C} (O) N (R 8a) R 8, -C (S) N (R 8a) R 8, - _{^{(O) r N (R 8a}} ) R 8, -Si (R 9a) (R 9b) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, naphthyl substituted with (Z _{2) q2} or represents a D2-1～D2-102, or, ^{R a} is by forming an alkylene chain or _C 2 -C ₅ alkenylene chain of _C 2 -C ₅ taken together with ^{R 3, R a} is a bond And a carbon atom to which R ³ is bonded may form a 5- to 8-membered ring, in which case the alkylene chain or alkenylene chain may contain one or two oxygen atoms, sulfur atoms or nitrogen atoms, and halogen atoms, cyano, _nitro, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 14} _(C 1 ~C ₆₎ ^{alkyl, -OH, -OR 11, -SH,} -S (O) r R 11 Oxo group or thioxo Optionally substituted by a group,
R ^b _is, C 1 -C ₆ alkyl, optionally substituted with ^{R 5} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ cycloalkyl, optionally substituted with ^{R 5} _(C 3 ~C ₈ ) _cycloalkyl, C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally substituted with ^{R 5} _(C 3 ~C ₈ ) _{cycloalkenyl,} substituted C 2 -C ₆ alkynyl, optionally with ^{R 5} _(C 2 ~C _{6) ^{alkynyl, -S (O) r R 6}} , -C (O) OR 6a, -C (O) ^{SR 6a, -C (S) OR} 6a, -C (S) SR 6a, -C (O) R 7, -C (S) R 7, -C (O) N (R 8a) R 8, -C _{^{(S) N (R 8a)}} R 8, -S (O) r N (R 8a) R 8, -Si (R 9a) (R 9b) ⁹ represents phenyl, ^naphthyl, phenyl substituted with (Z _{2) ^q2,} naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ^c is hydrogen _atom, C 1 -C ₆ alkyl, optionally substituted with ^{R 5} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ cycloalkyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkyl,} C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkenyl,} C 2 -C ₆ alkynyl, optionally substituted with ^{R 5} _(C 2 ~C ₆₎ ^{alkynyl, -OH, -OR 6, -SH,} -S (O) r R 6, ^{-N (R 8a) R 8,} -C (O) OR 6a, -C (O) SR 6a, -C (S) OR 6a, -C (S) SR 6a, -C (O) R 7, - ^{C (S) R 7, -C} (O) N (R 8a) R 8, -C (S) N (R 8a) R 8, - _{^{(O) r N (R 8a}} ) R 8, -Si (R 9a) (R 9b) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, naphthyl substituted with (Z _{2) q2} Or D2-1 to D2-102,
R ^d is a hydrogen atom, a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ , —OH, —OR ⁶ , —SH, —S _(O) represents the ^{r R 6, -N (R 8a} ) R 8, -C (O) oR 6a or -C (O) ^{R 7,}
R ^e and R ^f are each independently a hydrogen atom, —OH, —OR ⁶ , —SH, —S (O) _r R ⁶ , —N (R ^8a ) R ⁸ , —C (O) OR ^6a , ^{-C (O) SR 6a, -C} (S) OR 6a, -C (S) SR 6a, -C (O) R 7, -C (S) R 7, -C (O) N (R 8a) _{^{R 8, -C (S) N}} (R 8a) R 8, -S (O) r N (R 8a) R 8, -Si (R 9a) (R 9b) R 9, phenyl, naphthyl, ^{(Z 2} ) Represents phenyl substituted with _q2 , (Z ² ) naphthyl substituted with _q2 or D2-1 to D2-102, or R ^e together with R ^f represents a C _{2 to} C ₇ alkylene chain by forming, they may form a 3-8 membered ring together with the carbon atom to which R ^e and R ^f are bonded, this time the alkylene chain oxygen Hara May contain 1 or 2 individual sulfur atom or a nitrogen atom, and a halogen atom, cyano, _nitro, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 14} _(C 1 ~C ₆₎ alkyl, -OH , —OR ¹¹ , —SH, —S (O) _r R ¹¹ , an oxo group or a thioxo group,
R ^g and R ^g2 are each independently a hydrogen atom, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ , C ₃ -C ₈ cycloalkyl, optional with R ⁵ substituted in _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally ^{R 5} (C ₃ -C ₈ ) cycloalkenyl, C ₂ -C ₆ alkynyl, (C ₂ -C ₆ ) alkynyl optionally substituted with R ⁵ , —S (O) _r R ⁶ , —C ( O) OR ^6a , —C (O) SR ^6a , —C (S) OR ^6a , —C (S) SR ^6a , —C (O) R ⁷ , —C (S) R ⁷ , —C (O) ^{N (R 8a) R 8,} -C (S) N (R 8a) R 8, -S (O) r N (R 8a) R ^{, -Si (R 9a) (R} 9b) R 9, represents phenyl, ^naphthyl, phenyl substituted with (Z _{2) ^q2,} naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ⁵ is a halogen atom, cyano, C ₃ -C ₈ cycloalkyl, —OH, —OR ¹¹ , —SH, —S (O) _r R ¹¹ , —N (R ^13a ) R ¹³ , —C (O). OR ^11a , -C (S) OR ^11a , -C (O) SR ^11a , -C (S) SR ^11a , -C (O) R ¹² , -C (S) R ¹² , -C (O) N ( ^{R 13a) R 13, -C (} S) N (R 13a) R 13, -S (O) r N (R 13a) R 13, -Si (R 9a) (R 9b) R 9, phenyl, naphthyl, ^(Z ₂₎ phenyl substituted with ^_q2, represents naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ⁶ and R ^6a each independently represent C ₁ -C ₆ alkyl or (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ ;
R ⁷ is a hydrogen _atom, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 14} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ ^cycloalkyl, optionally substituted with ^{R 14} _{(C 3} -C _{8) cycloalkyl,} C 2 -C ₆ ^alkenyl, optionally substituted with ^{R 14} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ ^{cycloalkenyl,} optionally substituted with ^{R 14} _{(C 3} -C _{8) cycloalkenyl,} optionally substituted with C 2 -C _{6 ^{alkynyl, R 14 (C 2 ~C 6}} ) alkynyl, phenyl, ^naphthyl, phenyl substituted with ^{_{(Z 2) q2, (Z}} 2) represents naphthyl or D2-1 to D2-102 substituted with _q2 ,
R ⁸ and R ^8a are each independently a hydrogen atom, cyano, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ , C ₃ -C ₈ cycloalkyl, R ^14. optionally substituted _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ ^alkenyl, optionally substituted with ^{R 14} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl ^{in, R 14} optionally substituted _(C 3 ~C _{8) cycloalkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14} _(C 2 ~C ₆₎ alkynyl, -S _(O) ^{r R 11} in, - C (O) OR ^11a , -C (S) OR ^11a , -C (O) SR ^11a , -C (S) SR ^11a , -C (O) R ¹² , -C (S) R ¹² , -C ( O) N (R ^13a ) R ¹³ , —C (S) N (R ^13a ) _{^{R 13, -S (O) r}} N (R 13a) R 13, -Si (R 9a) (R 9b) R 9, phenyl, ^naphthyl, phenyl substituted with ^{_{(Z 2) q2, (Z}} 2) q2 in or represents naphthyl or D2-1~D2-102 substituted ,, Alternatively, ^{R 8} forms a alkenylene chain alkylene chain or _C 2 -C ₇ of _C 2 -C ₇ together with ^{R 8a} In this case, a 3- to 8-membered ring may be formed together with the nitrogen atom to which R ⁸ and R ^8a are bonded, and this alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, And a halogen atom, cyano, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ , C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ Alkylthio, ₁ -C _{6 haloalkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ haloalkylsulfonyl, ^phenyl, substituted by (Z _{2) q2} Optionally substituted by a phenyl, oxo group or thioxo group,
R ⁹ , R ^9a and R ^9b each independently represent C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxy or phenyl;
R ¹¹ _is, -S ^{(O) 2} R 15a _substituent, C 1 -C ₆ ^alkyl, which is optionally substituted with ^{R 14a} _(C 1 ~C _{6) alkyl,} C 2 -C ₆ ^alkenyl, optionally with ^{R 14a} been _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14a} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally substituted with ^{R 14a} (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ cycloalkenyl, optionally substituted with (C ₂ -C ₆ ) cycloalkenyl, phenyl, naphthyl, (Z ² ) _q ² optionally substituted with R ^14a Represents phenyl, (Z ² ) _q2 substituted naphthyl or D2-1 to D2-102;
R ^11a and R ¹² are each independently a hydrogen atom, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a , C ₂ -C ₆ alkenyl, optionally with R ^14a substituted substituted _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14a} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally in ^{R 14a} (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ cycloalkenyl, (C ₂ -C ₆ ) cycloalkenyl optionally substituted with R ^14a , phenyl, naphthyl, substituted with (Z ² ) _q ² Naphthyl substituted with phenyl, (Z ² ) _q2 or D2-1 to D2-102,
R ¹³ and R ^13a are each independently a hydrogen atom, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a , C ₂ -C ₆ alkenyl, optionally R ^14a substituted substituted _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14a} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally in ^{R 14a} (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ cycloalkenyl, (C ₂ -C ₆ ) cycloalkenyl optionally substituted with R ^14a , phenyl, naphthyl, substituted with (Z ² ) _q ^{2 phenyl,} (Z ₂₎ ,, or or represents naphthyl or D2-1~D2-102 substituted with ^{_q2, R 13} is an alkylene chain or _C 2 ~ of _C 2 -C ₇ together with ^{R 13a} C Of by forming the alkenylene chain may form a 3-8 membered ring together with the nitrogen atom to which R ¹³ and R ^13a are attached, this time the alkylene chain or alkenylene chain oxygen atom, a sulfur atom or a nitrogen atom One (1) and halogen atom, cyano, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a , C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy , _C 1 -C _{6 alkylthio,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ haloalkylsulfonyl, phenyl, (Z ² ) optionally substituted by a phenyl, oxo group or thioxo group substituted by _q2 ,
R ¹⁴ and ^{R 14a} are each independently a halogen atom, cyano, _nitro, C 3 -C _{8 cycloalkyl,} C 3 -C _{8 halocycloalkyl,} C 3 -C _{8 cycloalkenyl,} C 3 -C ₈ Haroshikuro Alkenyl, —OH, —OR ¹⁵ , —SH, —S (O) _r R ¹⁵ , —N (R ^17a ) R ¹⁷ , —C (O) OR ¹⁵ , —C (O) SR ¹⁵ , —C (S ^{) OR 15, -C (S)} SR 15, -C (O) R 16, -C (O) N (R 17a) R 17, -C (S) N (R 17a) R 17, -S (O _{^{) r N (R 17a) R}} 17, -C (= NR 17) OR 15, -C (= NR 17) S (O) r R 15, -C (= NR 17) R 16, -C (= NOH ^{) R 16, -C (= NOR} 15) R 16, -C {= NN (R 17a) R 1 ^{} R 16, -Si (R 9b} ) (R 9a) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, (Z ₂₎ is substituted with _q2 naphthyl or D2-1~D2-102 Represents, represents,
R ¹⁵ and ^{R 15a} have been replaced each independently _C 1 -C ₆ ^alkyl, optionally substituted with ^{R 18} _(C 1 ~C _{6) alkyl,} C 2 -C ₆ ^alkenyl, optionally with ^{R 18} _(C 2 _{~C 6) alkenyl,} optionally substituted with C 2 -C ₆ ^alkynyl, which is optionally substituted with ^{R 18} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^{cycloalkyl, R 18} ( C ₃ -C _{8) cycloalkyl,} C 2 -C ₆ ^{cycloalkenyl,} optionally substituted with ^{R 18} _(C 2 ~C ₆₎ ^{cycloalkenyl, -Si (R 9b) (R} 9a) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, (Z ₂₎ naphthyl or D2-1~D2-102 substituted with _q2 represent,
R ¹⁶ is a hydrogen _atom, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 18} _(C 1 ~C _{6) alkyl,} C 2 -C ₆ ^alkenyl, optionally substituted with ^{R 18} _(C 2 ~ C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 18} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally substituted with ^{R 18} _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ ^{cycloalkenyl,} optionally substituted with ^{R 18} _(C 2 ~C ₆₎ ^{cycloalkenyl, -Si (R 9b) (R} 9a) R 9, phenyl, naphthyl, (Z phenyl substituted with ^{2) _q2,} the (Z ₂₎ naphthyl or D2-1~D2-102 substituted with _q2 represent,
R ¹⁷ and R ^17a are each independently a hydrogen atom, cyano, nitro, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁸ , C ₂ -C ₆ alkenyl, R optionally substituted with ¹⁸ _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 18} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^{cycloalkyl, R 18} (C ₃ -C ₈ ) cycloalkyl optionally substituted with, C ₂ -C ₆ cycloalkenyl, (C ₂ -C ₆ ) cycloalkenyl optionally substituted with R ¹⁸ , —Si (R ^9b ) (R ^{9a) R 9,} phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, or represents (Z ₂₎ naphthyl or D2-1~D2-102 substituted with _q2, ^{or, R 17} is a ^{R 17a} Together By forming the alkylene chain or alkenylene chain of _C 2 -C ₇ for ₂ -C ^_7, may form a 3-8 membered ring together with the nitrogen atom ^{to which R 17} and ^{R 17a} are attached, this time the alkylene chain Alternatively, the alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and (C ₁ -C ₆ ) alkyl optionally substituted with a halogen atom, cyano, C ₁ -C ₆ alkyl, R ¹⁸ , C ₁ -C _{6 alkoxy,} C 1 -C _{6 haloalkoxy,} C 1 -C _{6 alkylthio,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ haloalkylsulfonyl, ^phenyl, (Z ₂₎ phenyl substituted by _q2, oxo group or thioxo group Thus it may be optionally substituted,
R ¹⁸ is a halogen atom, cyano, nitro, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C 1 ₁ -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ ^{haloalkylsulfonyl, -Si (R 9b) (R} 9a) R 9, phenyl, ^naphthyl, phenyl substituted with (Z _{2) q2} , (Z ² ) naphthyl substituted with _q2 or D2-1 to D2-102,
D2-1 to D2-102 each represent a ring represented by the following structural formula;

Ｘ^２は、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、−Ｃ（Ｏ）ＮＨ_２、−Ｃ（Ｓ）ＮＨ_２、−Ｓ（Ｏ）_２ＮＨ_２又はＲ^２０を表し、ｔ１、ｔ２又はｔ４が２以上の整数を表すとき、各々のＸ^２は互いに同一であっても又は互いに異なってもよく、更に、２つのＸ^２が隣接する場合には、隣接する２つのＸ^２は、−ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＯＣＨ_２−，−ＯＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２Ｓ−，−ＣＨ_２ＳＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２ＯＣＨ_２−，−ＣＨ_２ＯＣＨ_２Ｏ−，−ＯＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２ＣＨ_２Ｓ−又は−ＯＣＨ_２ＣＨ_２Ｓ−を形成することにより、それぞれのＸ^２が結合する炭素原子と共に５員環又は６員環を形成してもよく、このとき環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル基、Ｃ_１〜Ｃ_６ハロアルキル基、Ｃ_１〜Ｃ_６アルコキシ基、Ｃ_１〜Ｃ_６アルキルチオ基、Ｃ_１〜Ｃ_６アルキルスルフィニル基又はＣ_１〜Ｃ_６アルキルスルホニル基によって任意に置換されてもよく、
Ｘ^２ａは、水素原子、シアノ、−ＯＨ、−ＮＨ_２、−ＣＨＯ又はＲ^２０を表し、Ｘ^２ａの隣接位にＸ^２が存在する場合には、隣接するＸ^２ａとＸ^２は、−ＣＨ_２ＣＨ_２ＣＨ_２ＣＨ_２−、−ＣＨ＝ＣＨＣＨ＝ＣＨ−、−Ｎ＝ＣＨＣＨ＝ＣＨ−、−ＣＨ＝Ｎ−ＣＨ＝ＣＨ−、−ＣＨ＝ＣＨ−Ｎ＝ＣＨ−又は−ＣＨ＝ＣＨ−ＣＨ＝Ｎ−を形成することにより、Ｘ^２ａ及びＸ^２のそれぞれが結合する原子と共に６員環を形成してもよく、このとき、環を形成する各々の炭素原子に結合する水素原子は、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル基、Ｃ_１〜Ｃ_６ハロアルキル基、Ｃ_１〜Ｃ_６アルコキシ基、Ｃ_１〜Ｃ_６アルキルチオ基、Ｃ_１〜Ｃ_６アルキルスルフィニル基又はＣ_１〜Ｃ_６アルキルスルホニル基によって任意に置換されてもよく、
Ｘ^２ｂは、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、−Ｃ（Ｏ）ＮＨ_２、−Ｃ（Ｓ）ＮＨ_２、−Ｓ（Ｏ）_２ＮＨ_２、−ＣＨＯ又はＲ^２０を表し、ｕ１、ｕ２、ｕ４、ｕ５、ｕ６、ｕ７、ｕ８又はｕ９が２以上の整数を表すとき、各々のＸ^２ｂは互いに同一であっても、又は互いに相異なってもよく、更に、２つのＸ^２ｂが同一の炭素上に置換している場合、２つのＸ^２ｂは一緒になってオキソ、チオキソ、イミノ、Ｃ_１〜Ｃ_６アルキルイミノ、Ｃ_１〜Ｃ_６アルコキシイミノ又はＣ_１〜Ｃ_６アルキリデンを形成してもよく、
Ｚ^２は、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、−Ｃ（Ｏ）ＮＨ_２、−Ｃ（Ｓ）ＮＨ_２、−Ｓ（Ｏ）_２ＮＨ_２又はＲ^２０を表し、ｑ２が２以上の整数を表すとき、各々のＺ^２は互いに同一であっても又は互いに異なってもよく、更に、２つのＺ^２が隣接する場合には、隣接する２つのＺ^２は−ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＯＣＨ_２−，−ＯＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２Ｓ−，−ＣＨ_２ＳＣＨ_２−，−ＣＨ_２ＣＨ_２Ｎ（Ｘ^２ａ）−，−ＣＨ_２Ｎ（Ｘ^２ａ）ＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２ＯＣＨ_２−，−ＣＨ_２ＯＣＨ_２Ｏ−，−ＯＣＨ_２ＣＨ_２Ｏ−，−ＯＣＨ_２ＣＨ_２Ｓ−，−ＣＨ_２ＣＨ＝ＣＨ−，−ＯＣＨ＝ＣＨ−，−ＳＣＨ＝ＣＨ−，−Ｎ（Ｘ^２ａ）ＣＨ＝ＣＨ−，−ＯＣＨ＝Ｎ−，−ＳＣＨ＝Ｎ−，−Ｎ（Ｘ^２ａ）ＣＨ＝Ｎ−，−Ｎ（Ｘ^２ａ）Ｎ＝ＣＨ−，−ＯＣＨ_２ＣＨ＝ＣＨ−，−Ｎ＝ＣＨＣＨ＝ＣＨ−，−ＣＨ＝ＮＣＨ＝ＣＨ−，−Ｎ＝ＮＣＨ＝ＣＨ−，−ＣＨ＝ＮＮ＝ＣＨ−，−Ｎ＝ＣＨＣＨ＝Ｎ−又は−Ｎ＝ＣＨＮ＝ＣＨ−を形成することにより、それぞれのＺ^２が結合する炭素原子と共に５員環又は６員環を形成してもよく、このとき、環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル基、Ｃ_１〜Ｃ_６ハロアルキル基、Ｃ_１〜Ｃ_６アルコキシ基、Ｃ_１〜Ｃ_６アルキルチオ基、Ｃ_１〜Ｃ_６アルキルスルフィニル基又はＣ_１〜Ｃ_６アルキルスルホニル基によって任意に置換されてもよく、
Ｒ^２０は、Ｃ_１〜Ｃ_６アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^２８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｒ^２８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｒ^２８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｒ^２８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｒ^２８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、−ＯＲ^２５、−Ｓ（Ｏ）_ｒＲ^２５、−Ｃ（Ｏ）ＯＲ^２５、−Ｃ（Ｏ）Ｒ^２６、−Ｎ（Ｒ^２７ａ）Ｒ^２７、−Ｃ（Ｏ）Ｎ（Ｒ^２７ａ）Ｒ^２７、−Ｃ（Ｓ）Ｎ（Ｒ^２７ａ）Ｒ^２７、−Ｓ（Ｏ）_ｒＮ（Ｒ^２７ａ）Ｒ^２７、フェニル、Ｃ_１〜Ｃ_６アルキル又はハロゲン原子で任意に置換されたフェニルを表し、
Ｒ^２５、Ｒ^２６及びＲ^２７ａは、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６ハロアルキル又はＣ_３〜Ｃ_８シクロアルキルを表し、
Ｒ^２７は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６ハロアルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル又はＣ_１〜Ｃ_６ハロアルコキシカルボニルを表し、
Ｒ^２８及びＲ^２８ａは、各々独立してハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_３〜Ｃ_８ハロシクロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６ハロアルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルチオカルボニル、Ｃ_１〜Ｃ_６アルコキシチオカルボニル、Ｃ_１〜Ｃ_６アルキルジチオカルボニル、Ｃ_１〜Ｃ₆アルキルアミノカルボニル、Ｃ_１〜Ｃ₆ハロアルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノカルボニル、トリ（Ｃ_１〜Ｃ_６アルキル）シリル、Ｃ_１〜Ｃ₆アルキルアミノスルホニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、Ｃ_１〜Ｃ_６アルキルスルホニルオキシ、Ｃ_１〜Ｃ_６ハロアルキルスルホニルオキシ、Ｃ_１〜Ｃ_６アルキルアミノ又はジ（Ｃ_１〜Ｃ_６アルキル）アミノを表し、
ｎ、ｔ１及びｕ１は、各々独立して０、１、２又は３の整数を表し、
ｔ２及びｕ２は、各々独立して０、１又は２の整数を表し、
ｔ３は、０又は１の整数を表し、
ｔ４及びｕ４は、各々独立して０、１、２、３又は４の整数を表し、
ｕ５は、０、１、２、３、４又は５の整数を表し、
ｕ６は、各々独立して０、１、２、３、４、５又は６の整数を表し、
ｕ７は、各々独立して０、１、２、３、４、５、６又は７の整数を表し、
ｕ８は、０、１、２、３、４、５、６、７又は８の整数を表し、
ｕ９は、０、１、２、３、４、５、６、７、８又は９の整数を表し、
ｑ２は、１、２、３、４又は５の整数を表し、
ｍ１、ｍ２及びｍ４は、各々独立して０又は１の整数を表し、
ｒ、ｒ２及びｒ３は、各々独立して０、１又は２の整数を表す〕で表されるピラゾール誘導体又はその塩。 X ² represents a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , —C (O) NH ₂ , —C (S) NH ₂ , —S (O) ₂ NH ₂ or R ²⁰ . , T1, t2 or t4 each represents an integer of 2 or more, each X ² may be the same as or different from each other. Further, when two X ² are adjacent, X ² represents —CH ₂ CH ₂ CH ₂ —, —CH ₂ CH ₂ O—, —CH ₂ OCH ₂ —, —OCH ₂ O—, —CH ₂ CH ₂ S—, —CH ₂ SCH ₂ —, — CH ₂ CH ₂ CH ₂ CH ₂ —, —CH ₂ CH ₂ CH ₂ O—, —CH ₂ CH ₂ OCH ₂ —, —CH ₂ OCH ₂ O—, —OCH ₂ CH ₂ O—, —CH ₂ CH ₂ by CH ₂ S- or form a -OCH ₂ CH ₂ S-, it A 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each X ² is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is a halogen atom, C _{1 to} C _6. alkyl _group, C 1 -C ₆ haloalkyl _group, C 1 -C ₆ alkoxy _group, C 1 -C ₆ alkylthio _group, optionally substituted by C 1 -C ₆ alkylsulfinyl group or a _C 1 -C ₆ alkylsulfonyl group Well,
X ^2a is a hydrogen atom, cyano, _-OH, an -NH 2, -CHO or ^{R 20, when X 2} is present at the adjacent position to ^{X 2a} is, ^{X 2a} and ^{X 2} the adjacent, -CH ₂ CH ₂ CH ₂ CH ₂ —, —CH═CHCH═CH—, —N═CHCH═CH—, —CH═N—CH═CH—, —CH═CH—N═CH— or —CH═CH— By forming CH═N—, a 6-membered ring may be formed together with the atom to which each of X ^2a and X ² is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is halogen _atom, C 1 -C ₆ alkyl _group, C 1 -C ₆ haloalkyl _group, C 1 -C ₆ alkoxy _group, C 1 -C ₆ alkylthio _group, C 1 -C ₆ alkylsulfinyl group or a _C 1 -C ₆ alkyl Optionally substituted by a sulfonyl group It may be,
X ^2b is a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , —C (O) NH ₂ , —C (S) NH ₂ , —S (O) ₂ NH ₂ , —CHO or R ^When u1, u2, u4, u5, u6, u7, u8 or u9 represent an integer of 2 or more, each X ^2b may be the same as or different from each other, When two X ^2b are substituted on the same carbon, the two X ^2b together are oxo, thioxo, imino, C ₁ -C ₆ alkylimino, C ₁ -C ₆ alkoxyimino or C _1- C ₆ alkylidene may be formed,
Z ² represents a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , —C (O) NH ₂ , —C (S) NH ₂ , —S (O) ₂ NH ₂ or R ²⁰ . , Q2 represents an integer of 2 or more, each Z ² may be the same as or different from each other, and when two Z ² are adjacent, the two adjacent Z ² are − _{CH 2 CH 2 CH 2 -,} - CH 2 CH 2 O -, - CH 2 OCH 2 -, - OCH 2 O -, - CH 2 CH 2 S -, - CH 2 SCH 2 -, - CH 2 CH 2 N _{^{(X 2a) -, - CH}} 2 N (X 2a) CH 2 -, - CH 2 CH 2 CH 2 CH 2 -, - CH 2 CH 2 CH 2 O -, - CH 2 CH 2 OCH 2 -, - CH ₂ OCH ₂ O—, —OCH ₂ CH ₂ O—, —OCH ₂ CH ₂ S—, —C _{H 2 CH = CH -, -} OCH = CH -, - SCH = CH -, - N (X 2a) CH = CH -, - OCH = N -, - SCH = N -, - N (X 2a) CH = _{^{N -, - N (X 2a}} ) N = CH -, - OCH 2 CH = CH -, - N = CHCH = CH -, - CH = NCH = CH -, - N = NCH = CH -, - CH = NN By forming ═CH—, —N═CHCH═N— or —N═CHN═CH—, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each Z ² is bonded. when the hydrogen atoms bonded to each carbon atom forming the ring, a halogen _atom, C 1 -C ₆ alkyl _group, C 1 -C ₆ haloalkyl _group, C 1 -C ₆ alkoxy _group, C 1 -C ₆ alkylthio _group, C 1 -C ₆ alkylsulfinyl group or a _C 1 -C ₆ Arukirusu It may be optionally substituted by Honiru group,
R ²⁰ is C ₁ -C ₆ alkyl, C ₂ -C ₆ alkenyl, C ₂ -C ₆ alkynyl, C ₃ -C ₈ cycloalkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ²⁸ , optionally substituted with R ²⁸ _(C 2 ~C ₆₎ ^alkenyl, optionally substituted with ^{R 28} _(C 2 ^~C ₆₎ ^alkynyl, optionally substituted with ^{R 28} _(C 3 ^~C ₈₎ cycloalkyl (C ₃ -C ₈ ) cycloalkenyl optionally substituted with alkyl, R ²⁸ , —OR ²⁵ , —S (O) _r R ²⁵ , —C (O) OR ²⁵ , —C (O) R ²⁶ , — ^{N (R 27a) R 27,} -C (O) N (R 27a) R 27, -C (S) N (R 27a) R 27, -S (O) r N (R 27a) R 27, phenyl, phenyl optionally substituted with C ₁ -C ₆ alkyl or halogen atom It represents,
R ²⁵ , R ²⁶ and R ^27a each independently represent a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl or C ₃ -C ₈ cycloalkyl,
R ²⁷ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₁ -C ₆ alkylcarbonyl, C ₃ -C ₈ cycloalkylcarbonyl, C ₁ -C Represents ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl or C ₁ -C ₆ haloalkoxycarbonyl,
R ²⁸ and R ^28a are each independently a halogen atom, cyano, nitro, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₂ -C ₆ alkenyloxy, C ₁ -C ₆ alkylthio, C ₁ -C _{6 alkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 haloalkylsulfonyl,} C 1 -C _{6 alkylcarbonyl,} C 3 -C ₈ cycloalkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₃ -C ₈ halocycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, C ₁ -C ₆ alkylthiocarbonyl, C ₁ -C _{6 alkoxythiocarbonyl,} C 1 -C ₆ alkyl dithio months _Boniru, C 1 -C _{6 alkylaminocarbonyl,} C 1 -C ₆ haloalkylcarbonyl aminocarbonyl, di _(C 1 -C ₆ alkyl) aminocarbonyl, tri _(C 1 -C ₆ alkyl) _silyl, C 1 -C ₆ alkylamino Sulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, C ₁ -C ₆ alkylcarbonyloxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylamino or di _(C 1 -C ₆ alkyl) an amino,
n, t1, and u1 each independently represents an integer of 0, 1, 2, or 3;
t2 and u2 each independently represent an integer of 0, 1 or 2;
t3 represents an integer of 0 or 1,
t4 and u4 each independently represent an integer of 0, 1, 2, 3 or 4;
u5 represents an integer of 0, 1, 2, 3, 4 or 5;
u6 each independently represents an integer of 0, 1, 2, 3, 4, 5 or 6;
u7 each independently represents an integer of 0, 1, 2, 3, 4, 5, 6 or 7;
u8 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7 or 8;
u9 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7, 8 or 9,
q2 represents an integer of 1, 2, 3, 4 or 5,
m1, m2 and m4 each independently represents an integer of 0 or 1,
r, r2 and r3 each independently represents an integer of 0, 1 or 2] or a salt thereof.

〔２〕
Ａ^１は、−ＣＲ^１を表し、
Ｒ^１、Ｒ^３及びＲ^４は、各々独立して水素原子、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^２は、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表す上記〔１〕記載のピラゾール誘導体又はその塩。 [2]
A ¹ represents -CR ¹
R ¹ , R ³ and R ⁴ each independently represents a hydrogen atom, a halogen atom or C ₁ -C ₆ alkyl;
R ² represents a pyrazole derivative or a salt thereof according to the above [1], wherein R ² represents a halogen atom or C ₁ -C ₆ alkyl.

〔３〕
Ａ^１は、−Ｎ（−Ｏ）_ｍ２を表し、
Ｒ^２は、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^３及びＲ^４は、各々独立して水素原子、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表す上記〔１〕記載のピラゾール誘導体又はその塩。 [3]
A ¹ represents -N (-O) _m2 ,
R ² represents a halogen atom or C ₁ -C ₆ alkyl,
R ³ and R ⁴ each independently represents a hydrogen atom, a halogen atom, or a C ₁ -C ₆ alkyl, the pyrazole derivative according to the above [1] or a salt thereof.

〔４〕
Ｒ^１及びＲ^４は、水素原子を表し、
Ａ^２は、−Ｃ（Ｒ^ａ）＝ＮＯＲ^ｂ、−Ｃ≡ＣＲ^ｃ、−Ｃ（Ｒ^ｄ）＝Ｃ（Ｒ^ｅ）Ｒ^ｆ又は−Ｃ（Ｒ^ａ）＝ＮＮ（Ｒ^ｇ）Ｒ^ｇ２を表し、
Ｒ^ａは、水素原子、Ｃ_１〜Ｃ_６アルキル、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｎ（Ｒ^８ａ）Ｒ^８又はＤ２−７を表すか、或いは、Ｒ^ａはＲ^３と一緒になってＣ_３のアルキレン鎖を形成することにより、Ｒ^ａが結合する炭素原子及びＲ^３が結合する炭素原子と共に６員環を形成してもよく、
Ｒ^ｂは、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^ｃは、水素原子、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９又はＤ２−３２を表し、
Ｒ^ｄ及びＲ^ｅは、水素原子を表し、
Ｒ^ｆは、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｎ（Ｒ^８ａ）Ｒ^８、フェニル、（Ｚ^２）_ｑ２で置換されたフェニル又はＤ２−７を表すか、或いは、Ｒ^ｅはＲ^ｆと一緒になってＣ_４のアルキレン鎖を形成することにより、Ｒ^ｅ及びＲ^ｆが結合する炭素原子と共に５員環を形成し、このときこのアルキレン鎖は窒素原子を１個含み、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、オキソ基によって任意に置換されてもよく、
Ｒ^ｇは、−Ｃ（Ｏ）Ｒ^７を表し、
Ｒ^ｇ２は、Ｃ_１〜Ｃ_６アルキルを表し、
Ｒ^５は、ハロゲン原子、−ＯＨ、−ＯＲ^１１、−Ｓ（Ｏ）_ｒＲ^１１又はＤ２−３２又はＤ２−３４を表し、
Ｒ^６及びＲ^６ａは、各々独立してＣ_１〜Ｃ_６アルキルを表し、
Ｒ^７は、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^８は、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−Ｃ（Ｏ）ＯＲ^１１ａ又は−Ｃ（Ｏ）Ｒ^１２を表し、
Ｒ^８ａは、水素原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^１１は、−Ｓ（Ｏ）_２Ｒ^１５ａ又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^１１ａは、Ｃ_１〜Ｃ_６アルキルを表し、
Ｒ^１２は、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^１４は、ハロゲン原子又は−Ｓ（Ｏ）_ｒＲ^１５を表し、
Ｒ^１４ａは、−Ｓ（Ｏ）_ｒＲ^１５を表し、
Ｒ^１５及びＲ^１５ａは、各々独立してＣ_１〜Ｃ_６アルキルを表し、
Ｘ^２及びＺ^２は、各々独立してＣ_１〜Ｃ_６ハロアルキルを表し、
ｑ２は、０又は１の整数を表し、
ｔ１は、１の整数を表し、
ｔ４は、０又は１の整数を表し、
ｎ、ｍ１及びｍ２は、０を表し、
ｒは、０、１又は２の整数を表す上記〔２〕記載のピラゾール誘導体又はその塩。 [4]
R ¹ and R ⁴ represent a hydrogen atom,
A ² represents —C (R ^a ) = NOR ^b , —C≡CR ^c , —C (R ^d ) = C (R ^e ) R ^f or —C (R ^a ) = NN (R ^g ) R ^g2 Represent,
R ^a represents a hydrogen atom, C ₁ -C ₆ alkyl, —C (O) OR ^6a , —C (O) N (R ^8a ) R ⁸ , —N (R ^8a ) R ⁸ or D 2-7. Alternatively, R ^a may form a C ₃ alkylene chain together with R ³ to form a 6-membered ring together with the carbon atom to which R ^a is bonded and the carbon atom to which R ³ is bonded;
R ^b represents C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ ;
R ^c is a hydrogen atom, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ , —S (O) _r R ⁶ , —C (O) SR ^6a , —C (O) N (R ^{8a ) R 8, -Si (R 9a} ) ( represents R 9b) ^{R 9} or D2-32,
R ^d and R ^e represent a hydrogen atom,
R ^{f _{is, -S (O) r R 6}} , -C (O) OR 6a, -C (O) N (R 8a) R 8, -N (R 8a) R 8, ^phenyl, (Z _{2) q2} Represents phenyl or D2-7 substituted with R 5, or R ^e together with R ^f forms a C ₄ alkylene chain to form a 5-membered ring together with the carbon atom to which R ^e and R ^f are bonded. Wherein the alkylene chain contains one nitrogen atom and may be optionally substituted by a (C ₁ -C ₆ ) alkyl, oxo group optionally substituted with R ¹⁴ ,
R ^g represents —C (O) R ⁷ ,
R ^g2 represents C ₁ -C ₆ alkyl,
R ⁵ represents a halogen atom, —OH, —OR ¹¹ , —S (O) _r R ¹¹ or D2-32 or D2-34;
R ⁶ and R ^6a each independently represent C ₁ -C ₆ alkyl,
R ⁷ represents (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ ;
R ⁸ represents C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ , —C (O) OR ^11a or —C (O) R ¹² ,
R ^8a represents a hydrogen atom or C ₁ -C ₆ alkyl;
R ¹¹ represents —S (O) ₂ R ^15a or C ₁ -C ₆ alkyl;
R ^11a represents C ₁ -C ₆ alkyl;
R ¹² represents (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a ,
R ¹⁴ represents a halogen atom or —S (O) _r R ¹⁵ ;
R ^14a represents -S (O) _r R ¹⁵ ;
R ¹⁵ and R ^15a each independently represent C ₁ -C ₆ alkyl;
X ² and Z ² each independently represent C ₁ -C ₆ haloalkyl,
q2 represents an integer of 0 or 1,
t1 represents an integer of 1,
t4 represents an integer of 0 or 1,
n, m1 and m2 represent 0;
The pyrazole derivative or the salt thereof according to the above [2], wherein r represents an integer of 0, 1 or 2.

〔５〕
上記〔１〕〜〔４〕記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する有害生物防除剤。 [5]
A pest control agent containing one or more selected from the pyrazole derivatives described in [1] to [4] above and salts thereof as an active ingredient.

〔６〕
上記〔１〕〜〔４〕記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する農薬。 [6]
An agrochemical containing one or more selected from the pyrazole derivatives according to the above [1] to [4] and salts thereof as an active ingredient.

〔７〕
上記〔１〕〜〔４〕記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する哺乳動物又は鳥類の内部もしくは外部寄生虫防除剤。 [7]
A mammal or bird internal or ectoparasite control agent comprising one or more selected from the pyrazole derivatives and salts thereof described in [1] to [4] as active ingredients.

〔８〕
上記〔１〕〜〔４〕記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する殺虫剤又は殺ダニ剤。 [8]
An insecticide or acaricide containing as an active ingredient one or more selected from the pyrazole derivatives described in [1] to [4] above and salts thereof.

〔９〕
上記〔１〕〜〔４〕記載のピラゾール誘導体及びそれらの塩から選ばれる１種又は２種以上を有効成分として含有する土壌処理剤。 [9]
A soil treatment agent containing one or more selected from the pyrazole derivatives according to the above [1] to [4] and salts thereof as an active ingredient.

〔１０〕
土壌処理方法が土壌潅注処理である上記〔９〕記載の土壌処理剤。 [10]
The soil treatment agent according to the above [9], wherein the soil treatment method is soil irrigation treatment.

本発明化合物は多くの農業害虫、ハダニ類、哺乳動物又は鳥類の内部もしくは外部寄生虫に対して優れた殺虫・殺ダニ活性を有し、既存の殺虫剤に対して抵抗性を獲得した害虫に対しても十分な防除効果を発揮する。さらに、ホ乳類、魚類及び益虫に対してほとんど悪影響を及ぼさず、低残留性で環境に対する負荷も軽い。   The compound of the present invention has excellent insecticidal / miticidal activity against many agricultural pests, spider mites, mammals or birds, or against insects that have acquired resistance to existing insecticides. Even against this, it exhibits a sufficient control effect. Furthermore, it has little adverse effect on mammals, fish and beneficial insects, has low persistence, and has a light environmental impact.

従って、本発明は有用な新規有害生物防除剤を提供することができる。   Therefore, the present invention can provide a useful novel pest control agent.

本発明に包含される化合物には、置換基の種類によってはＥ−体及びＺ−体の幾何異性体が存在する場合があるが、本発明はこれらＥ−体、Ｚ−体又はＥ−体及びＺ−体を任意の割合で含む混合物を包含するものである。また、本発明に包含される化合物は、１個又は２個以上の不斉炭素原子の存在に起因する光学活性体が存在するが、本発明は全ての光学活性体又はラセミ体を包含する。   The compounds included in the present invention may have geometrical isomers of E-form and Z-form depending on the type of substituent, and the present invention is not limited to these E-form, Z-form or E-form. And a mixture containing the Z-form in an arbitrary ratio. In addition, the compounds included in the present invention include optically active substances resulting from the presence of one or more asymmetric carbon atoms, but the present invention includes all optically active substances or racemates.

本発明に包含される化合物のうちで、常法に従って酸付加塩にすることができるものは、例えば、フッ化水素酸、塩酸、臭化水素酸、沃化水素酸等のハロゲン化水素酸の塩、硝酸、硫酸、燐酸、塩素酸、過塩素酸等の無機酸の塩、メタンスルホン酸、エタンスルホン酸、トリフルオロメタンスルホン酸、ベンゼンスルホン酸、ｐ−トルエンスルホン酸等のスルホン酸の塩、ギ酸、酢酸、プロピオン酸、トリフルオロ酢酸、フマール酸、酒石酸、蓚酸、マレイン酸、リンゴ酸、コハク酸、安息香酸、マンデル酸、アスコルビン酸、乳酸、グルコン酸、クエン酸等のカルボン酸の塩又はグルタミン酸、アスパラギン酸等のアミノ酸の塩とすることができる。   Among the compounds included in the present invention, those that can be converted into acid addition salts according to a conventional method include, for example, hydrohalic acids such as hydrofluoric acid, hydrochloric acid, hydrobromic acid, hydroiodic acid, and the like. Salts of inorganic acids such as salts, nitric acid, sulfuric acid, phosphoric acid, chloric acid, perchloric acid, salts of sulfonic acids such as methanesulfonic acid, ethanesulfonic acid, trifluoromethanesulfonic acid, benzenesulfonic acid, p-toluenesulfonic acid, Salts of carboxylic acids such as formic acid, acetic acid, propionic acid, trifluoroacetic acid, fumaric acid, tartaric acid, succinic acid, maleic acid, malic acid, succinic acid, benzoic acid, mandelic acid, ascorbic acid, lactic acid, gluconic acid, citric acid, etc. A salt of an amino acid such as glutamic acid or aspartic acid can be used.

或いは、本発明に包含される化合物のうちで、常法に従って金属塩にすることができるものは、例えば、リチウム、ナトリウム、カリウムといったアルカリ金属の塩、カルシウム、バリウム、マグネシウムといったアルカリ土類金属の塩又はアルミニウムの塩とすることができる。   Alternatively, among the compounds included in the present invention, those that can be converted into a metal salt according to a conventional method include, for example, alkali metal salts such as lithium, sodium, and potassium, and alkaline earth metals such as calcium, barium, and magnesium. It can be a salt or a salt of aluminum.

次に、本明細書において示した各置換基の具体例を以下に示す。ここで、ｎ−はノルマル、ｉ−はイソ、ｓ−はセカンダリー及びｔｅｒｔ−はターシャリーを各々意味し、Ｐｈはフェニルを意味する。   Next, specific examples of each substituent shown in the present specification are shown below. Here, n- represents normal, i- represents iso, s- represents secondary, and tert- represents tertiary, and Ph represents phenyl.

本発明化合物におけるハロゲン原子としては、フッ素原子、塩素原子、臭素原子及びヨウ素原子が挙げられる。尚、本明細書中「ハロ」の表記もこれらのハロゲン原子を表す。   As a halogen atom in this invention compound, a fluorine atom, a chlorine atom, a bromine atom, and an iodine atom are mentioned. In the present specification, the notation “halo” also represents these halogen atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状の炭化水素基を表し、例えばメチル基、エチル基、ｎ−プロピル基、ｉ−プロピル基、ｎ−ブチル基、ｉ−ブチル基、ｓ−ブチル基、ｔｅｒｔ−ブチル基、ｎ−ペンチル基、１，１−ジメチルプロピル基、ｎ−ヘキシル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkyl in the present specification represents a linear or branched hydrocarbon group having a carbon number of _a to _b , for example, methyl group, ethyl group, n-propyl group, Specific examples include i-propyl group, n-butyl group, i-butyl group, s-butyl group, tert-butyl group, n-pentyl group, 1,1-dimethylpropyl group, n-hexyl group, and the like. Each selected range of carbon atoms is selected.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状の炭化水素基を表し、このとき、２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えばフルオロメチル基、クロロメチル基、ブロモメチル基、ヨードメチル基、ジフルオロメチル基、ジクロロメチル基、トリフルオロメチル基、クロロジフルオロメチル基、トリクロロメチル基、ブロモジフルオロメチル基、２−フルオロエチル基、２−クロロエチル基、２−ブロモエチル基、２，２−ジフルオロエチル基、２，２，２−トリフルオロエチル基、２−クロロ−２，２−ジフルオロエチル基、２，２，２−トリクロロエチル基、１，１，２，２−テトラフルオロエチル基、２−クロロ−１，１，２−トリフルオロエチル基、ペンタフルオロエチル基、３，３，３−トリフルオロプロピル基、２，２，３，３，３−ペンタフルオロプロピル基、１，１，２，３，３，３−ヘキサフルオロプロピル基、ヘプタフルオロプロピル基、２，２，２−トリフルオロ−１−（トリフルオロメチル）エチル基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチル基、２，２，３，３，４，４，４−ヘプタフルオロブチル基、ノナフルオロブチル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b haloalkyl is represented by a linear or branched chain having _a to _b carbon atoms in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. Represents a hydrocarbon group, and when substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, fluoromethyl group, chloromethyl group, bromomethyl group, iodomethyl group, difluoromethyl group, dichloromethyl group, trifluoromethyl group, chlorodifluoromethyl group, trichloromethyl group, bromodifluoromethyl group, 2-fluoroethyl group, 2- Chloroethyl group, 2-bromoethyl group, 2,2-difluoroethyl group, 2,2,2-trifluoroethyl group, 2-chloro-2,2-difluoroethyl group, 2,2,2-trichloroethyl group, 1 , 1,2,2-tetrafluoroethyl group, 2-chloro-1,1,2-trifluoroethyl group, pentafluoroethyl group, 3,3,3-trifluoropropyl group, 2,2,3,3 , 3-pentafluoropropyl group, 1,1,2,3,3,3-hexafluoropropyl group, heptafluoropropyl group 2,2,2-trifluoro-1- (trifluoromethyl) ethyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethyl group, 2,2,3,3,4, Specific examples include 4,4-heptafluorobutyl group, nonafluorobutyl group and the like, and each is selected within the range of the number of carbon atoms designated.

本明細書におけるＣ_ａ〜Ｃ_ｂシクロアルキルの表記は、炭素原子数がａ〜ｂ個よりなる環状の炭化水素基を表し、３員環から６員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよい。例えばシクロプロピル基、１−メチルシクロプロピル基、２−メチルシクロプロピル基、２，２−ジメチルシクロプロピル基、シクロブチル基、シクロペンチル基、シクロヘキシル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b cycloalkyl represents a cyclic hydrocarbon group having a carbon number of _a to _b , and forms a monocyclic or complex ring structure having 3 to 6 members. I can do it. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms. Specific examples include, for example, cyclopropyl group, 1-methylcyclopropyl group, 2-methylcyclopropyl group, 2,2-dimethylcyclopropyl group, cyclobutyl group, cyclopentyl group, cyclohexyl group and the like. Selected in a range of numbers.

本明細書におけるＣ_ａ〜Ｃ_ｂハロシクロアルキルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる環状の炭化水素基を表し、３員環から６員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよく、ハロゲン原子による置換は環構造部分であっても、側鎖部分であっても、或いはそれらの両方であってもよく、さらに、２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていてもよい。例えば２，２−ジフルオロシクロプロピル基、２，２−ジクロロシクロプロピル基、２，２−ジブロモシクロプロピル基、２，２−ジフルオロ−１−メチルシクロプロピル基、２，２−ジクロロ−１−メチルシクロプロピル基、２，２−ジブロモ−１−メチルシクロプロピル基、２，２，３，３−テトラフルオロシクロブチル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b halocycloalkyl is a cyclic hydrocarbon group having a carbon number of _a to _b in which a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom. And can form monocyclic or complex ring structures from 3 to 6-membered rings. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the substitution with a halogen atom may be a ring structure part, a side chain part, They may be both, and when they are substituted by two or more halogen atoms, the halogen atoms may be the same as or different from each other. For example, 2,2-difluorocyclopropyl group, 2,2-dichlorocyclopropyl group, 2,2-dibromocyclopropyl group, 2,2-difluoro-1-methylcyclopropyl group, 2,2-dichloro-1-methyl Specific examples include cyclopropyl group, 2,2-dibromo-1-methylcyclopropyl group, 2,2,3,3-tetrafluorocyclobutyl group, and the like, and each is selected within the range of the designated number of carbon atoms. The

本明細書におけるＣ_ａ〜Ｃ_ｂアルケニルの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、且つ分子内に１個又は２個以上の二重結合を有する不飽和炭化水素基を表し、例えばビニル基、１−プロペニル基、２−プロペニル基、１−メチルエテニル基、２−ブテニル基、２−メチル−２−プロペニル基、３−メチル−２−ブテニル基、１，１−ジメチル−２−プロペニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b alkenyl is a linear or branched chain composed of _a to _b carbon atoms and has one or more double bonds in the molecule. Represents a saturated hydrocarbon group, for example, vinyl group, 1-propenyl group, 2-propenyl group, 1-methylethenyl group, 2-butenyl group, 2-methyl-2-propenyl group, 3-methyl-2-butenyl group, 1 , 1-dimethyl-2-propenyl group and the like are listed as specific examples, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂシクロアルケニルの表記は、炭素原子数がａ〜ｂ個よりなる環状の、且つ１個又は２個以上の二重結合を有する不飽和炭化水素基を表し、３員環から６員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよく、さらに、二重結合はｅｎｄｏ−又はｅｘｏ−のどちらの形式であってもよい。例えば１−シクロペンテン−１−イル基、２−シクロペンテン−１−イル基、１−シクロヘキセン−１−イル基、２−シクロヘキセン−１−イル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b cycloalkenyl in the present specification represents a cyclic unsaturated hydrocarbon group having 1 to 2 carbon atoms and having 1 or 2 or more double bonds. A monocyclic or complex ring structure from a member ring to a 6-member ring can be formed. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the double bond may be either endo- or exo-. Specific examples include 1-cyclopenten-1-yl group, 2-cyclopenten-1-yl group, 1-cyclohexen-1-yl group, 2-cyclohexen-1-yl group, and the like. Selected in a range of numbers.

本明細書におけるＣ_ａ〜Ｃ_ｂハロシクロアルケニルの表記は、炭素原子に結合した水素原子が、ハロゲン原子によって任意に置換された、炭素原子数がａ〜ｂ個よりなる環状の、且つ１個又は２個以上の二重結合を有する不飽和炭化水素基を表し、３員環から６員環までの単環又は複合環構造を形成することが出来る。また、各々の環は指定の炭素原子数の範囲でアルキル基によって任意に置換されていてもよく、さらに、二重結合はｅｎｄｏ−又はｅｘｏ−のどちらの形式であってもよい。また、ハロゲン原子による置換は環構造部分であっても、側鎖部分であっても、或いはそれらの両方であってもよく、２個以上のハロゲン原子によって置換されている場合、それらのハロゲン原子は互いに同一でも、又は互いに相異なっていても良い。例えば２−フルオロ−１−シクロペンテニル基、２−クロロ−１−シクロペンテニル基、３−クロロ−２−シクロペンテニル基、２−フルオロ−１−シクロヘキセニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b halocycloalkenyl has the following notation: a hydrogen atom bonded to a carbon atom is optionally substituted with a halogen atom, a cyclic one having 1 to b carbon atoms, and one Alternatively, it represents an unsaturated hydrocarbon group having two or more double bonds, and can form a monocyclic or complex ring structure having 3 to 6 members. Each ring may be optionally substituted with an alkyl group within the range of the specified number of carbon atoms, and the double bond may be either endo- or exo-. In addition, the substitution by a halogen atom may be a ring structure part, a side chain part or both of them, and when substituted by two or more halogen atoms, those halogen atoms May be the same as or different from each other. For example, 2-fluoro-1-cyclopentenyl group, 2-chloro-1-cyclopentenyl group, 3-chloro-2-cyclopentenyl group, 2-fluoro-1-cyclohexenyl group and the like can be mentioned as specific examples. Selected within the specified number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキリデンの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、二重結合によって結合した炭化水素基を表し、例えばメチリデン基、エチリデン基、プロピリデン基、１−メチルエチリデン基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b alkylidene represents a linear or branched hydrocarbon group having a carbon number of _a to _b and bonded by a double bond, such as methylidene group, ethylidene Specific examples include a group, a propylidene group, a 1-methylethylidene group, and the like, and each group is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキニルの表記は、炭素原子数がａ〜ｂ個よりなる直鎖状又は分岐鎖状で、且つ分子内に１個又は２個以上の三重結合を有する不飽和炭化水素基を表し、例えばエチニル基、１−プロピニル基、２−プロピニル基、１−ブチニル基、２−ブチニル基、３−ブチニル基、１，１−ジメチル−２−プロピニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b alkynyl is a linear or branched chain composed of _a to _b carbon atoms and has one or more triple bonds in the molecule. Represents a hydrocarbon group, for example, ethynyl group, 1-propynyl group, 2-propynyl group, 1-butynyl group, 2-butynyl group, 3-butynyl group, 1,1-dimethyl-2-propynyl group, etc. Each of which is selected for each specified number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルコキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｏ−基を表し、例えばメトキシ基、エトキシ基、ｎ−プロピルオキシ基、ｉ−プロピルオキシ基、ｎ−ブチルオキシ基、ｉ−ブチルオキシ基、ｓ−ブチルオキシ基、ｔｅｒｔ−ブチルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkoxy in the present specification represents an alkyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methoxy group, ethoxy group, n-propyloxy group, Specific examples include an i-propyloxy group, an n-butyloxy group, an i-butyloxy group, an s-butyloxy group, a tert-butyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルコキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｏ−基を表し、例えばジフルオロメトキシ基、トリフルオロメトキシ基、クロロジフルオロメトキシ基、ブロモジフルオロメトキシ基、２−フルオロエトキシ基、２−クロロエトキシ基、２，２，２−トリフルオロエトキシ基、１，１，２，２，−テトラフルオロエトキシ基、２−クロロ−１，１，２−トリフルオロエトキシ基、１，１，２，３，３，３−ヘキサフルオロプロピルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkoxy in the present specification represents a haloalkyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethoxy group, trifluoromethoxy group, chlorodifluoro Methoxy group, bromodifluoromethoxy group, 2-fluoroethoxy group, 2-chloroethoxy group, 2,2,2-trifluoroethoxy group, 1,1,2,2, -tetrafluoroethoxy group, 2-chloro-1 Specific examples include 1,2,2-trifluoroethoxy group, 1,1,2,3,3,3-hexafluoropropyloxy group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルケニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル−Ｏ−基を表し、例えば２−プロペニルオキシ基、２−ブテニルオキシ基、２−メチル−２−プロペニルオキシ基、３−メチル−２−ブテニルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkenyloxy in the present specification represents an alkenyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, 2-propenyloxy group, 2-butenyloxy group, Specific examples include 2-methyl-2-propenyloxy group, 3-methyl-2-butenyloxy group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルチオの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ−基を表し、例えばメチルチオ基、エチルチオ基、ｎ−プロピルチオ基、ｉ−プロピルチオ基、ｎ−ブチルチオ基、ｉ−ブチルチオ基、ｓ−ブチルチオ基、ｔｅｒｔ−ブチルチオ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylthio in the present specification represents an alkyl-S-group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylthio group, ethylthio group, n-propylthio group, i Specific examples include -propylthio group, n-butylthio group, i-butylthio group, s-butylthio group, tert-butylthio group and the like, which are selected within the range of the number of carbon atoms specified.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルチオの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｓ−基を表し、例えばジフルオロメチルチオ基、トリフルオロメチルチオ基、クロロジフルオロメチルチオ基、ブロモジフルオロメチルチオ基、２，２，２−トリフルオロエチルチオ基、１，１，２，２−テトラフルオロエチルチオ基、２−クロロ−１，１，２−トリフルオロエチルチオ基、ペンタフルオロエチルチオ基、１，１，２，３，３，３−ヘキサフルオロプロピルチオ基、ヘプタフルオロプロピルチオ基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチルチオ基、ノナフルオロブチルチオ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkylthio in the present specification represents a haloalkyl-S-group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethylthio group, trifluoromethylthio group, chlorodifluoro Methylthio group, bromodifluoromethylthio group, 2,2,2-trifluoroethylthio group, 1,1,2,2-tetrafluoroethylthio group, 2-chloro-1,1,2-trifluoroethylthio group, Pentafluoroethylthio group, 1,1,2,3,3,3-hexafluoropropylthio group, heptafluoropropylthio group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylthio group , Nonafluorobutylthio group and the like are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルスルフィニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ（Ｏ）−基を表し、例えばメチルスルフィニル基、エチルスルフィニル基、ｎ−プロピルスルフィニル基、ｉ−プロピルスルフィニル基、ｎ−ブチルスルフィニル基、ｉ−ブチルスルフィニル基、ｓ−ブチルスルフィニル基、ｔｅｒｔ−ブチルスルフィニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylsulfinyl in the present specification represents an alkyl-S (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylsulfinyl group, ethylsulfinyl group, Specific examples include n-propylsulfinyl group, i-propylsulfinyl group, n-butylsulfinyl group, i-butylsulfinyl group, s-butylsulfinyl group, tert-butylsulfinyl group and the like. The range is selected.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルスルフィニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｓ（Ｏ）−基を表し、例えばジフルオロメチルスルフィニル基、トリフルオロメチルスルフィニル基、クロロジフルオロメチルスルフィニル基、ブロモジフルオロメチルスルフィニル基、２，２，２−トリフルオロエチルスルフィニル基、１，２，２，２−テトラフルオロ−１−（トリフルオロメチル）エチルスルフィニル基、ノナフルオロブチルスルフィニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkylsulfinyl in the present specification represents a haloalkyl-S (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethylsulfinyl group, trifluoromethyl Sulfinyl group, chlorodifluoromethylsulfinyl group, bromodifluoromethylsulfinyl group, 2,2,2-trifluoroethylsulfinyl group, 1,2,2,2-tetrafluoro-1- (trifluoromethyl) ethylsulfinyl group, nona Specific examples include a fluorobutylsulfinyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルスルホニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−ＳＯ_２−基を表し、例えばメチルスルホニル基、エチルスルホニル基、ｎ−プロピルスルホニル基、ｉ−プロピルスルホニル基、ｎ−ブチルスルホニル基、ｉ−ブチルスルホニル基、ｓ−ブチルスルホニル基、ｔｅｒｔ−ブチルスルホニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylsulfonyl in the present specification represents an alkyl-SO ₂ -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylsulfonyl group, ethylsulfonyl group, n- Specific examples include a propylsulfonyl group, an i-propylsulfonyl group, an n-butylsulfonyl group, an i-butylsulfonyl group, an s-butylsulfonyl group, a tert-butylsulfonyl group, and the range of each designated number of carbon atoms. Selected.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルスルホニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−ＳＯ_２−基を表し、例えばジフルオロメチルスルホニル基、トリフルオロメチルスルホニル基、クロロジフルオロメチルスルホニル基、ブロモジフルオロメチルスルホニル基、２，２，２−トリフルオロエチルスルホニル基、１，１，２，２−テトラフルオロエチルスルホニル基、２−クロロ−１，１，２−トリフルオロエチルスルホニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkylsulfonyl in the present specification represents a haloalkyl-SO ₂ -group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a difluoromethylsulfonyl group or a trifluoromethylsulfonyl group. Chlorodifluoromethylsulfonyl group, bromodifluoromethylsulfonyl group, 2,2,2-trifluoroethylsulfonyl group, 1,1,2,2-tetrafluoroethylsulfonyl group, 2-chloro-1,1,2-trimethyl Specific examples include a fluoroethylsulfonyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルアミノの表記は、水素原子の一方が炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたアミノ基を表し、例えばメチルアミノ基、エチルアミノ基、ｎ−プロピルアミノ基、ｉ−プロピルアミノ基、ｎ−ブチルアミノ基、ｉ−ブチルアミノ基、ｔｅｒｔ−ブチルアミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylamino in the present specification represents an amino group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, a methylamino group , Ethylamino group, n-propylamino group, i-propylamino group, n-butylamino group, i-butylamino group, tert-butylamino group and the like. Selected by range.

本明細書におけるジ（Ｃ_ａ〜Ｃ_ｂアルキル）アミノの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたアミノ基を表し、例えばジメチルアミノ基、エチル（メチル）アミノ基、ジエチルアミノ基、ｎ−プロピル（メチル）アミノ基、ｉ−プロピル（メチル）アミノ基、ジ（ｎ−プロピル）アミノ基、ジ（ｎ−ブチル）アミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of di (C _a -C _b alkyl) amino has the above-mentioned meaning that the number of carbon atoms which may be the same or different from each other is ab. Represents an amino group substituted by an alkyl group, such as dimethylamino group, ethyl (methyl) amino group, diethylamino group, n-propyl (methyl) amino group, i-propyl (methyl) amino group, di (n-propyl) Specific examples include an amino group, a di (n-butyl) amino group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルイミノの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｎ＝基を表し、例えばメチルイミノ基、エチルイミノ基、ｎ−プロピルイミノ基、ｉ−プロピルイミノ基、ｎ−ブチルイミノ基、ｉ−ブチルイミノ基、ｓ−ブチルイミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylimino in the present specification represents an alkyl-N = group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylimino group, ethylimino group, n-propylimino group. Specific examples include i-propylimino group, n-butylimino group, i-butylimino group, s-butylimino group, and the like, and each is selected within the range of the number of carbon atoms designated.

本明細書におけるＣ_ａ〜Ｃ_ｂアルコキシイミノの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルコキシ−Ｎ＝基を表し、例えばメトキシイミノ基、エトキシイミノ基、ｎ−プロピルオキシイミノ基、ｉ−プロピルオキシイミノ基、ｎ−ブチルオキシイミノ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkoxyimino in the present specification represents an alkoxy-N = group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methoxyimino group, ethoxyimino group, n-propyl. Specific examples include an oxyimino group, an i-propyloxyimino group, an n-butyloxyimino group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｃ（Ｏ）−基を表し、例えばアセチル基、プロピオニル基、ブチリル基、イソブチリル基、バレリル基、イソバレリル基、２−メチルブタノイル基、ピバロイル基、ヘキサノイル基、ヘプタノイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylcarbonyl in the present specification represents an alkyl-C (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, acetyl group, propionyl group, butyryl group. , Isobutyryl group, valeryl group, isovaleryl group, 2-methylbutanoyl group, pivaloyl group, hexanoyl group, heptanoyl group, and the like, and specific examples thereof are selected within the range of the number of carbon atoms designated.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｃ（Ｏ）−基を表し、例えばフルオロアセチル基、クロロアセチル基、ジフルオロアセチル基、ジクロロアセチル基、トリフルオロアセチル基、クロロジフルオロアセチル基、ブロモジフルオロアセチル基、トリクロロアセチル基、ペンタフルオロプロピオニル基、ヘプタフルオロブタノイル基、３−クロロ−２，２−ジメチルプロパノイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkylcarbonyl in the present specification represents a haloalkyl-C (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a fluoroacetyl group, a chloroacetyl group, Difluoroacetyl group, dichloroacetyl group, trifluoroacetyl group, chlorodifluoroacetyl group, bromodifluoroacetyl group, trichloroacetyl group, pentafluoropropionyl group, heptafluorobutanoyl group, 3-chloro-2,2-dimethylpropanoyl group Etc. are given as specific examples, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂシクロアルキルカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるシクロアルキル−Ｃ（Ｏ）−基を表し、例えばシクロプロピルカルボニル基、２−メチルシクロプロピルカルボニル基、シクロブチルカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b cycloalkylcarbonyl in the present specification represents a cycloalkyl-C (O) -group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as cyclopropylcarbonyl group, 2 Specific examples include -methylcyclopropylcarbonyl group, cyclobutylcarbonyl group, etc., and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂハロシクロアルキルカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロシクロアルキル−Ｃ（Ｏ）−基を表し、例えば２，２−ジクロロシクロプロピルカルボニル基、２，２−ジクロロ−１−メチルシクロプロピルカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C _a -C _b halocycloalkylcarbonyl represents a halocycloalkyl-C (O) — group having the above-mentioned meaning consisting of _a to _b carbon atoms. Specific examples include a dichlorocyclopropylcarbonyl group, a 2,2-dichloro-1-methylcyclopropylcarbonyl group, and the like, which are selected in the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルコキシカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｏ−Ｃ（Ｏ）−基を表し、例えばメトキシカルボニル基、エトキシカルボニル基、ｎ−プロピルオキシカルボニル基、ｉ−プロピルオキシカルボニル基、ｎ−ブトキシカルボニル基、ｉ−ブトキシカルボニル基、ｔｅｒｔ−ブトキシカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkoxycarbonyl in the present specification represents an alkyl-O—C (O) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methoxycarbonyl group, ethoxycarbonyl Group, n-propyloxycarbonyl group, i-propyloxycarbonyl group, n-butoxycarbonyl group, i-butoxycarbonyl group, tert-butoxycarbonyl group and the like, and specific ranges of the number of carbon atoms are designated. Selected.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルコキシカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキル−Ｏ−Ｃ（Ｏ）−基を表し、例えばクロロメトキシカルボニル基、２−クロロエトキシカルボニル基、２，２−ジフルオロエトキシカルボニル基、２，２，２−トリフルオロエトキシカルボニル基、２，２，２−トリクロロエトキシカルボニル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkoxycarbonyl in the present specification represents a haloalkyl-O—C (O) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, such as a chloromethoxycarbonyl group, Specific examples include 2-chloroethoxycarbonyl group, 2,2-difluoroethoxycarbonyl group, 2,2,2-trifluoroethoxycarbonyl group, 2,2,2-trichloroethoxycarbonyl group, and the like. Selected in the range of the number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルチオカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ−Ｃ（Ｏ）−基を表し、例えばメチルチオ−Ｃ（Ｏ）−基、エチルチオ−Ｃ（Ｏ）−基、ｎ−プロピルチオ−Ｃ（Ｏ）−基、ｉ−プロピルチオ−Ｃ（Ｏ）−基、ｎ−ブチルチオ−Ｃ（Ｏ）−基、ｉ−ブチルチオ−Ｃ（Ｏ）−基、ｔｅｒｔ−ブチルチオ−Ｃ（Ｏ）−基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylthiocarbonyl in the present specification represents an alkyl-S—C (O) — group having the above meaning consisting of _a to _b carbon atoms, for example, methylthio-C (O) -Group, ethylthio-C (O)-group, n-propylthio-C (O)-group, i-propylthio-C (O)-group, n-butylthio-C (O)-group, i-butylthio-C Specific examples include (O) -group, tert-butylthio-C (O) -group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルコキシチオカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｏ−Ｃ（Ｓ）−基を表し、例えばメトキシ−Ｃ（Ｓ）−基、エトキシ−Ｃ（Ｓ）−基、ｎ−プロピルオキシ−Ｃ（Ｓ）−基、ｉ−プロピルオキシ−Ｃ（Ｓ）−基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C _a -C _b alkoxythiocarbonyl represents an alkyl-O—C (S) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methoxy-C (S ) -Group, ethoxy-C (S) -group, n-propyloxy-C (S) -group, i-propyloxy-C (S) -group, etc. Selected in a range of numbers.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルジチオカルボニルの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル−Ｓ−Ｃ（Ｓ）−基を表し、例えばメチルチオ−Ｃ（Ｓ）−基、エチルチオ−Ｃ（Ｓ）−基、ｎ−プロピルチオ−Ｃ（Ｓ）−基、ｉ−プロピルチオ−Ｃ（Ｓ）−基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkyldithiocarbonyl in the present specification represents an alkyl-S—C (S) — group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylthio-C (S ) -Group, ethylthio-C (S) -group, n-propylthio-C (S) -group, i-propylthio-C (S) -group and the like. Selected by range.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルアミノカルボニルの表記は、水素原子の一方が炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたカルバモイル基を表し、例えばメチルカルバモイル基、エチルカルバモイル基、ｎ−プロピルカルバモイル基、ｉ−プロピルカルバモイル基、ｎ−ブチルカルバモイル基、ｉ−ブチルカルバモイル基、ｓ−ブチルカルバモイル基、ｔｅｒｔ−ブチルカルバモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylaminocarbonyl in the present specification represents a carbamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylcarbamoyl Group, ethylcarbamoyl group, n-propylcarbamoyl group, i-propylcarbamoyl group, n-butylcarbamoyl group, i-butylcarbamoyl group, s-butylcarbamoyl group, tert-butylcarbamoyl group, etc. Is selected within the range of the specified number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルアミノカルボニルの表記は、水素原子の一方が炭素原子数ａ〜ｂ個よりなる前記の意味であるハロアルキル基によって置換されたカルバモイル基を表し、例えば２−フルオロエチルカルバモイル基、２−クロロエチルカルバモイル基、２，２−ジフルオロエチルカルバモイル基、２，２，２−トリフルオロエチルカルバモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the expression C _a -C _b haloalkylaminocarbonyl represents a carbamoyl group in which one of the hydrogen atoms is substituted with a haloalkyl group having the above-described meaning consisting of _a to _b carbon atoms, for example, 2-fluoro Specific examples include ethylcarbamoyl group, 2-chloroethylcarbamoyl group, 2,2-difluoroethylcarbamoyl group, 2,2,2-trifluoroethylcarbamoyl group, etc. Is done.

本明細書におけるジ（Ｃ_ａ〜Ｃ_ｂアルキル）アミノカルボニルの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたカルバモイル基を表し、例えばＮ，Ｎ−ジメチルカルバモイル基、Ｎ−エチル−Ｎ−メチルカルバモイル基、Ｎ，Ｎ−ジエチルカルバモイル基、Ｎ，Ｎ−ジ（ｎ−プロピル）カルバモイル基、Ｎ，Ｎ−ジ（ｎ−ブチル）カルバモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of di (C _a -C _b alkyl) aminocarbonyl means in the above meaning that the number of carbon atoms which may be the same or different from each other is _a to _b. Represents a carbamoyl group substituted by an alkyl group, such as N, N-dimethylcarbamoyl group, N-ethyl-N-methylcarbamoyl group, N, N-diethylcarbamoyl group, N, N-di (n-propyl) carbamoyl Specific examples include a group, an N, N-di (n-butyl) carbamoyl group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルアミノスルホニルの表記は、水素原子の一方が炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたスルファモイル基を表し、例えばメチルスルファモイル基、エチルスルファモイル基、ｎ−プロピルスルファモイル基、ｉ−プロピルスルファモイル基、ｎ−ブチルスルファモイル基、ｉ−ブチルスルファモイル基、ｓ−ブチルスルファモイル基、ｔｅｒｔ−ブチルスルファモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, C _a -C _b alkylaminosulfonyl represents a sulfamoyl group in which one of the hydrogen atoms is substituted with an alkyl group having the above-mentioned meaning consisting of _a to _b carbon atoms. Famoyl group, ethylsulfamoyl group, n-propylsulfamoyl group, i-propylsulfamoyl group, n-butylsulfamoyl group, i-butylsulfamoyl group, s-butylsulfamoyl group, Specific examples include a tert-butylsulfamoyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるジ（Ｃ_ａ〜Ｃ_ｂアルキル）アミノスルホニルの表記は、水素原子が両方とも、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたスルファモイル基を表し、例えばＮ，Ｎ−ジメチルスルファモイル基、Ｎ−エチル−Ｎ−メチルスルファモイル基、Ｎ，Ｎ−ジエチルスルファモイル基、Ｎ，Ｎ−ジ（ｎ−プロピル）スルファモイル基、Ｎ，Ｎ−ジ（ｎ−ブチル）スルファモイル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of di (C _a -C _b alkyl) aminosulfonyl means in the above meaning that the number of carbon atoms which may be the same or different from each other is _a to _b. Represents a sulfamoyl group substituted by an alkyl group, such as N, N-dimethylsulfamoyl group, N-ethyl-N-methylsulfamoyl group, N, N-diethylsulfamoyl group, N, N-di- Specific examples include (n-propyl) sulfamoyl group, N, N-di (n-butyl) sulfamoyl group and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるトリ（Ｃ_ａ〜Ｃ_ｂアルキル）シリルの表記は、それぞれ同一でも又は互いに相異なっていてもよい炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基によって置換されたシリル基を表し、例えばトリメチルシリル基、トリエチルシリル基、トリ（ｎ−プロピル）シリル基、エチルジメチルシリル基、ｎ−プロピルジメチルシリル基、ｎ−ブチルジメチルシリル基、ｉ−ブチルジメチルシリル基、ｔｅｒｔ−ブチルジメチルシリル基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 In the present specification, the notation of tri (C _a -C _b alkyl) silyl is substituted by an alkyl group having the above-mentioned meanings, each having the same or different number of carbon atoms. Represents a silyl group, for example, trimethylsilyl group, triethylsilyl group, tri (n-propyl) silyl group, ethyldimethylsilyl group, n-propyldimethylsilyl group, n-butyldimethylsilyl group, i-butyldimethylsilyl group, tert- Specific examples include a butyldimethylsilyl group and the like, and each butyldimethylsilyl group is selected within a range of each designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルカルボニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキルカルボニル−Ｏ−基を表し、例えばアセトキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylcarbonyloxy in the present specification represents an alkylcarbonyl-O-group having the above-mentioned meaning consisting of _a to _b carbon atoms, and examples thereof include an acetoxy group and the like. , Each selected range of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂアルキルスルホニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキルスルホニル−Ｏ−基を表し、例えばメチルスルホニルオキシ基、エチルスルホニルオキシ基、ｎ−プロピルスルホニルオキシ基、ｉ−プロピルスルホニルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b alkylsulfonyloxy in the present specification represents an alkylsulfonyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, methylsulfonyloxy group, ethylsulfonyloxy group Specific examples include an n-propylsulfonyloxy group, an i-propylsulfonyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＣ_ａ〜Ｃ_ｂハロアルキルスルホニルオキシの表記は、炭素原子数がａ〜ｂ個よりなる前記の意味であるハロアルキルスルホニル−Ｏ−基を表し、例えばジフルオロメチルスルホニルオキシ基、トリフルオロメチルスルホニルオキシ基、クロロジフルオロメチルスルホニルオキシ基、ブロモジフルオロメチルスルホニルオキシ基等が具体例として挙げられ、各々の指定の炭素原子数の範囲で選択される。 The notation of C _a -C _b haloalkylsulfonyloxy in the present specification represents a haloalkylsulfonyl-O— group having the above-mentioned meaning consisting of _a to _b carbon atoms, for example, difluoromethylsulfonyloxy group, trifluoromethyl Specific examples include a sulfonyloxy group, a chlorodifluoromethylsulfonyloxy group, a bromodifluoromethylsulfonyloxy group, and the like, and each is selected within the range of the designated number of carbon atoms.

本明細書におけるＲ^５で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル、Ｒ^１４で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル、Ｒ^１４ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル、Ｒ^１８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル、Ｒ^２８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル又はＲ^２８ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキル等の表記は、任意のＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキル基上の置換基Ｒ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａが２個以上存在するとき、それぞれのＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａは互いに同一でも異なってもよい。 Herein optionally substituted with ^{R 5} _(C a ^~C _b) ^alkyl, optionally substituted with ^{R 14} _(C a ^~C _b) ^alkyl, optionally substituted with ^{R 14a} _(C ^a ~ C _b) ^alkyl, optionally substituted with ^{R 18} _(C a ^~C _b) ^alkyl, optionally substituted with ^{R 28} _(C a ^~C _b) alkyl or optionally substituted with ^{R 28a} _{(C a} -C _b) notation alkyl or the like, any of ^{R 5, R 14, R 14a} , by R ^{18, R 28} or ^{R 28a,} carbon atoms bonded to hydrogen atoms are optionally substituted carbon atoms a~ It represents an alkyl group as defined above consisting of b, and is selected in the range of the respective designated number of carbon atoms. At this time, when two or more substituents R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a on each (C _a -C _b ) alkyl group are present, each R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a may be the same as or different from each other.

本明細書におけるＲ^５で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル、Ｒ^１４で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル、Ｒ^２８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル又はＲ^２８ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル等の表記は、任意のＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がａ〜ｂ個よりなる前記の意味であるシクロアルキル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの（Ｃ_ａ〜Ｃ_ｂ）シクロアルキル基上の置換基Ｒ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａが２個以上存在するとき、それぞれのＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａは互いに同一でも異なってもよく、さらに置換位置は環構造部分であっても、側鎖部分であっても、或いはそれらの両方にあってもよい。 Herein optionally substituted with ^{R 5} _(C a ^~C _b) ^cycloalkyl, optionally substituted with ^{R 14} _(C a ^~C _b) ^cycloalkyl, optionally substituted with ^{R 14a} (C _a -C _b) ^cycloalkyl, substituted optionally substituted with ^{R 18} _(C a ~C _b) ^cycloalkyl, optionally in optionally substituted with ^{R 28} _(C a ~C _b) cycloalkyl or ^{R 28a} The notation of (C _a -C _b ) cycloalkyl, etc., is optionally substituted with a hydrogen atom bonded to a carbon atom by any R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a It represents a cycloalkyl group having the above-mentioned meaning consisting of a to b carbon atoms, and is selected in the range of each designated number of carbon atoms. At this time, when two or more substituents R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a on each (C _a -C _b ) cycloalkyl group are present, each R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a may be the same or different from each other, and the substitution position may be a ring structure part, a side chain part or both of them. Good.

本明細書におけるＲ^５で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル、Ｒ^１４で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル、Ｒ^１８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル、Ｒ^２８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル又はＲ^２８ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルケニル等の表記は、任意のＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がａ〜ｂ個よりなる前記の意味であるアルケニル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルケニル基上の置換基Ｒ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａが２個以上存在するとき、それぞれのＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａは互いに同一でも異なってもよい。 Herein optionally substituted with ^{R 5} _(C a ^~C _b) ^alkenyl, optionally substituted with ^{R 14} _(C a ^~C _b) ^alkenyl, optionally substituted with ^{R 14a} _(C ^a ~ C _b) ^alkenyl, optionally substituted with ^{R 18} _(C a ^~C _b) ^alkenyl, optionally substituted with ^{R 28} _(C a ^~C _b) alkenyl or optionally substituted with ^{R 28a} _{(C a} -C _b) notation alkenyl or the like, any of ^{R 5, R 14, R 14a} , by R ^{18, R 28} or ^{R 28a,} carbon atoms bonded to hydrogen atoms are optionally substituted carbon atoms a~ It represents an alkenyl group having the above meaning consisting of b, and is selected within the range of each designated number of carbon atoms. At this time, when two or more substituents R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a on each (C _a -C _b ) alkenyl group are present, each R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a may be the same as or different from each other.

本明細書におけるＲ^５で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル、Ｒ^１４で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル、Ｒ^２８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル又はＲ^２８ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル等の表記は、任意のＲ^５、Ｒ^１４、Ｒ^１８、Ｒ^２８又はＲ^２８ａによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がａ〜ｂ個よりなる前記の意味であるシクロアルケニル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの（Ｃ_ａ〜Ｃ_ｂ）シクロアルケニル基上の置換基Ｒ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａが２個以上存在するとき、それぞれのＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａは互いに同一でも異なってもよく、さらに置換位置は環構造部分であっても、側鎖部分であっても、或いはそれらの両方にあってもよい。 Herein optionally substituted with ^{R 5} _(C a ^~C _b) ^{cycloalkenyl,} optionally substituted with ^{R 14} _(C a ^~C _b) ^{cycloalkenyl,} optionally substituted with ^{R 14a} (C _a -C _b) substituted ^{cycloalkenyl,} optionally substituted with ^{R 18} _(C a ~C _b) ^{cycloalkenyl,} optionally in optionally substituted with ^{R 28} _(C a ~C _b) cycloalkenyl or ^{R 28a} The notation such as (C _a -C _b ) cycloalkenyl is the number of carbon atoms in which the hydrogen atom bonded to the carbon atom is optionally substituted by any R ⁵ , R ¹⁴ , R ¹⁸ , R ²⁸ or R ^28a Represents a cycloalkenyl group having the above-mentioned meaning consisting of a to b, and is selected in the range of each designated number of carbon atoms. At this time, when two or more substituents R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a on each (C _a -C _b ) cycloalkenyl group are present, each R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a may be the same or different from each other, and the substitution position may be a ring structure part, a side chain part or both of them. Good.

本明細書におけるＲ^５で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル、Ｒ^１４で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル、Ｒ^１４ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル、Ｒ^１８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル、Ｒ^２８で任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル又はＲ^２８ａで任意に置換された（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル等の表記は、任意のＲ^５、Ｒ^５ｂ、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａによって、炭素原子に結合した水素原子が任意に置換された炭素原子数がａ〜ｂ個よりなる前記の意味であるアルキ二ル基を表し、各々の指定の炭素原子数の範囲で選択される。このとき、それぞれの（Ｃ_ａ〜Ｃ_ｂ）アルキ二ル基上の置換基Ｒ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａが２個以上存在するとき、それぞれのＲ^５、Ｒ^１４、Ｒ^１４ａ、Ｒ^１８、Ｒ^２８又はＲ^２８ａは互いに同一でも異なってもよい。 Herein optionally substituted with ^{R 5} _(C a ^~C _b) alkynylene ^Le, optionally substituted with ^{R 14} _(C a ^~C _b) alkynylene ^Le, optionally substituted with ^{R 14a} _(C a ~C _b) alkynylene ^Le, optionally substituted with ^{R 18} _(C a _{~C b)} alkynylene ^Le, optionally substituted with ^{R 28} _(C a _{~C b)} alkynylene le or R optionally substituted with ^28a _(C ^{a ~C} _b) notation alkynylene Le etc., any ^{R 5, R 5b, R 14} , R 14a, by R ^{18, R 28} or ^{R 28a,} attached to a carbon atom Represents an alkynyl group as defined above, wherein the number of carbon atoms optionally substituted with hydrogen atoms is a to b, and is selected within the range of the respective designated number of carbon atoms. At this time, when two or more substituents R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a on each (C _a -C _b ) alkynyl group are present, each R ⁵ , R ¹⁴ , R ^14a , R ¹⁸ , R ²⁸ or R ^28a may be the same as or different from each other.

本明細書における
〔Ｒ^８はＲ^８ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^８及びＲ^８ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、〕
〔Ｒ^１３はＲ^１３ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^１３及びＲ^１３ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、〕
〔Ｒ^１７はＲ^１７ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^１７及びＲ^１７ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、〕
等の表記の具体例として、例えばアジリジン、アゼチジン、アゼチジン−２−オン、ピロリジン、ピロリジン−２−オン、オキサゾリジン、オキサゾリジン−２−オン、オキサゾリジン−２−チオン、チアゾリジン、チアゾリジン−２−オン、チアゾリジン−２−チオン、イミダゾリジン、イミダゾリジン−２−オン、イミダゾリジン−２−チオン、ピペリジン、ピペリジン−２−オン、ピペリジン−２−チオン、２Ｈ−３，４，５，６−テトラヒドロ−１，３−オキサジン−２−オン、２Ｈ−３，４，５，６−テトラヒドロ−１，３−オキサジン−２−チオン、モルホリン、２Ｈ−３，４，５，６−テトラヒドロ−１，３−チアジン−２−オン、２Ｈ−３，４，５，６−テトラヒドロ−１，３−チアジン−２−チオン、チオモルホリン、ペルヒドロピリミジン−２−オン、ピペラジン、ホモピペリジン、ホモピペリジン−２−オン、ヘプタメチレンイミン等が挙げられ、各々の指定の原子数の範囲で選択される。 In the present specification, [R ⁸ together with R ^8a forms a C _{2 to} C ₇ alkylene chain or a C _{2 to} C ₇ alkenylene chain, whereby 3 together with the nitrogen atom to which R ⁸ and R ^8a are bonded. An 8-membered ring may be formed, in which case the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom.]
^{[R 13} is by forming a alkenylene chain alkylene chain or _C 2 -C ₇ of _C 2 -C ₇ together with ^{R 13a,} 3 to 8-membered ring together with the nitrogen atom ^{to which R 13} and ^{R 13a} are attached Wherein the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom,
^{[R 17} is by forming alkenylene chain alkylene chain or _C 2 -C ₇ of _C 2 -C ₇ together with ^{R 17a,} 3 to 8-membered ring together with the nitrogen atom ^{to which R 17} and ^{R 17a} are attached Wherein the alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom,
Specific examples of notation such as aziridine, azetidine, azetidin-2-one, pyrrolidine, pyrrolidin-2-one, oxazolidine, oxazolidine-2-one, oxazolidine-2-thione, thiazolidine, thiazolidine-2-one, thiazolidine -2-thione, imidazolidine, imidazolidine-2-one, imidazolidine-2-thione, piperidine, piperidin-2-one, piperidine-2-thione, 2H-3,4,5,6-tetrahydro-1, 3-Oxazin-2-one, 2H-3,4,5,6-tetrahydro-1,3-oxazine-2-thione, morpholine, 2H-3,4,5,6-tetrahydro-1,3-thiazine- 2-one, 2H-3,4,5,6-tetrahydro-1,3-thiazine-2-thione, thiomorpholine, pe Tetrahydropyrimidine-2-one, piperazine, homopiperidine, homopiperidine-2-one, heptamethyleneimine, and the like, may be selected from the range of the number of each of the specified atoms.

本発明化合物は、以下の方法で製造することができる。   The compound of the present invention can be produced by the following method.

製造法Ａ   Manufacturing method A

式（２）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ａ及びｎは前記と同じ意味を表す。］で表される化合物を、式（３）［式中Ｒ^ｂは前記と同じ意味を表す。］で表される化合物と反応させることにより、式（４）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ａ、Ｒ^ｂ及びｎは前記と同じ意味を表す。］で表される本発明化合物を合成することができる。 Formula (2) [wherein A ¹ , R ² , R ³ , R ⁴ , R ^a and n represent the same meaning as described above. The compound represented by formula (3) [wherein R ^b represents the same meaning as described above. In the formula (4), A ¹ , R ² , R ³ , R ⁴ , R ^a , R ^b and n have the same meaning as described above. This invention compound represented by this can be synthesize | combined.

本反応では式（２）で表される化合物１当量に対して、式（３）で表される化合物は、０．５〜５０当量の範囲で用いることができる。   In this reaction, the compound represented by the formula (3) can be used in the range of 0.5 to 50 equivalents with respect to 1 equivalent of the compound represented by the formula (2).

必要ならば、炭酸カリウム、トリエチルアミン、ピリジン、４−（ジメチルアミノ）ピリジン等の塩基又は塩酸、硫酸、ｐ−トルエンスルホン酸等の酸を使用することができる。   If necessary, a base such as potassium carbonate, triethylamine, pyridine and 4- (dimethylamino) pyridine or an acid such as hydrochloric acid, sulfuric acid and p-toluenesulfonic acid can be used.

本反応は、無溶媒で実施してもよいが、溶媒を用いてもよく、例えば、Ｎ，Ｎ−ジメチルホルムアミド、Ｎ，Ｎ−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、１，３−ジメチル−２−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、２−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、ｎ−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の２種類以上を混合して用いてもよい。   This reaction may be carried out without solvent, but a solvent may be used, for example, N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2- Polar solvents such as imidazolinone and water, alcohols such as methanol, ethanol, propanol, 2-propanol and ethylene glycol, ethers such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, Halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, and aliphatic hydrocarbons such as pentane and n-hexane. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−６０℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常５分から１００時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

式（３）で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて容易に合成することができる。   Some of the compounds represented by formula (3) are known compounds, and some of them are commercially available. Others can be easily synthesized according to known methods described in the literature.

製造法Ｂ   Manufacturing method B

式（５）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４及びｎは前記と同じ意味を表し、Ｊ^１はハロゲン原子、−ＯＳＯ_２ＣＨ_３、−ＯＳＯ_２ＣＦ_３等の脱離基を表す。］で表される化合物は、文献既知の公知の方法、例えばジャーナル オブ ヘテロサイクリック ケミストリー １９８１年，１８巻，９頁等に記載の方法に準じて容易に製造することができる。 Formula (5) [wherein A ¹ , R ² , R ³ , R ⁴ and n represent the same meaning as described above, J ¹ represents a halogen atom, a leaving group such as —OSO ₂ CH ₃ , —OSO ₂ CF _3, etc. Represents. ] Can be easily produced according to a known method known in the literature, for example, the method described in Journal of Heterocyclic Chemistry 1981, Vol. 18, p.

また、式（６）で表される化合物［式中Ｒ^ｃは前記と同じ意味を表す。］の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて容易に合成することができる。 Further, a compound represented by formula (6) [wherein R ^c represents the same meaning as described above. ] Are known compounds, some of which are commercially available. Others can be easily synthesized according to known methods described in the literature.

式（５）で表される化合物と、式（６）で表される化合物とを、触媒及び塩基の存在下で反応させることにより、式（７）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ｃ及びｎは前記と同じ意味を表す。］で表される本発明化合物を合成することができる。 By reacting the compound represented by the formula (5) with the compound represented by the formula (6) in the presence of a catalyst and a base, the compound represented by the formula (7) [A ¹ , R ² , R ^{3 in the} formula] , R ⁴ , R ^c and n represent the same meaning as described above. This invention compound represented by this can be synthesize | combined.

式（６）で表される化合物の量は、式（５）で表される化合物１当量に対して０．８〜５当量の範囲で、用いることができる。   The amount of the compound represented by the formula (6) can be used in the range of 0.8 to 5 equivalents relative to 1 equivalent of the compound represented by the formula (5).

本反応で使用できる触媒としては、例えば、パラジウム−炭素、塩化パラジウム、酢酸パラジウム、ビス（トリフェニルホスフィン）パラジウムジクロリド、テトラキス（トリフェニルホスフィン）パラジウム等のパラジウム触媒又は金属銅、酢酸銅（Ｉ）、酢酸銅（ＩＩ）、酸化銅（Ｉ）、酸化銅（ＩＩ）、ヨウ化銅等の銅触媒が挙げられる。触媒の使用量は、式（１０）で表される化合物１当量に対して０．００１〜１．０当量で、用いることができる。   Examples of the catalyst that can be used in this reaction include palladium catalysts such as palladium-carbon, palladium chloride, palladium acetate, bis (triphenylphosphine) palladium dichloride, tetrakis (triphenylphosphine) palladium, or copper metal, copper acetate (I). And copper catalysts such as copper (II) acetate, copper (I) oxide, copper (II) oxide and copper iodide. The usage-amount of a catalyst can be used with 0.001-1.0 equivalent with respect to 1 equivalent of compounds represented by Formula (10).

使用する塩基としては、例えば、ピリジン、ジイソプロピルエチルアミン、トリエチルアミン等の三級アミン化合物、例えば水酸化ナトリウム水酸化カリウム、炭酸ナトリウム、炭酸カリウム、炭酸セシウム、炭酸水素ナトリウム等の無機塩基等が挙げられる。塩基の使用量は、式（１０）で表される化合物１当量に対して０．１〜５０当量の範囲で用いることができる。   Examples of the base to be used include tertiary amine compounds such as pyridine, diisopropylethylamine, and triethylamine, and inorganic bases such as sodium hydroxide, sodium carbonate, potassium carbonate, cesium carbonate, and sodium bicarbonate. The usage-amount of a base can be used in 0.1-50 equivalent with respect to 1 equivalent of compounds represented by Formula (10).

本反応は、無溶媒も実施することができるが、溶媒を用いてもよい。例えば、Ｎ，Ｎ−ジメチルホルムアミド、Ｎ，Ｎ−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、１，３−ジメチル−２−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、２−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、ｎ−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の２種類以上を混合して用いてもよい。   This reaction can be carried out without a solvent, but a solvent may be used. For example, polar solvent such as N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2-imidazolinone, water, methanol, ethanol, propanol, 2-propanol, ethylene glycol Alcohols such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, pentane and n-hexane And aliphatic hydrocarbons. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−６０℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常５分から１００時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

製造法Ｃ   Manufacturing method C

式（５）で表される化合物と式（８）［式中Ｒ^ｄ、Ｒ^ｅ及びＲ^ｆは前記と同じ意味を表し、Ｌ^２は水素原子又はＢ（ＯＲ^５０）_２｛式中Ｒ^５０は水素原子又は同一又は異なってもよくＣ_１〜Ｃ_６アルキルを表すか、或いは、２つのＲ^５０が一緒になって−ＣＨ_２ＣＨ_２−又は−Ｃ（ＣＨ_３）_２Ｃ（ＣＨ_３）_２−を形成してもよい。｝を表す。］で表される化合物を反応させて、式（９）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ｄ、Ｒ^ｅ、Ｒ^ｆ及びｎは前記と同じ意味を表す。］で表される本発明化合物を製造法Ｂと同様の方法を用いて合成することができる。 Compound represented by formula (5) and formula (8) [wherein R ^d , R ^e and R ^f represent the same meaning as described above, L ² represents a hydrogen atom or B (OR ⁵⁰ ) ₂ {where R ⁵⁰ May be the same or different and may represent the same or different C ₁ -C ₆ alkyl, or two R ⁵⁰ together represent —CH ₂ CH ₂ — or —C (CH ₃ ) ₂ C (CH ₃ ). _2- may be formed. }. The compound represented by formula (9) [wherein A ¹ , R ² , R ³ , R ⁴ , R ^d , R ^e , R ^f and n represent the same meaning as described above] is reacted. The compound of the present invention represented by the formula can be synthesized using the same method as in Production Method B.

式（８）で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて容易に合成することができる。   Some of the compounds represented by formula (8) are known compounds, and some of them are commercially available. Others can be easily synthesized according to known methods described in the literature.

製造法Ｄ   Manufacturing method D

式（２）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ａ及びｎは前記と同じ意味を表す。］で表される化合物を、式（１０）［式中Ｒ^ｇ及びＲ^ｇ２は前記と同じ意味を表す。］で表される化合物と反応させることにより、式（１１）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ａ、Ｒ^ｇ、Ｒ^ｇ２及びｎは前記と同じ意味を表す。］で表される本発明化合物を合成することができる。 Formula (2) [wherein A ¹ , R ² , R ³ , R ⁴ , R ^a and n represent the same meaning as described above. A compound represented by formula (10): wherein R ^g and R ^g2 represent the same meaning as described above. In the formula (11), A ¹ , R ² , R ³ , R ⁴ , R ^a , R ^g , R ^g2 and n have the same meaning as described above. This invention compound represented by this can be synthesize | combined.

本反応では式（２）で表される化合物１当量に対して、式（１０）で表される化合物は、０．５〜５０当量の範囲で用いることができる。   In this reaction, the compound represented by the formula (10) can be used in the range of 0.5 to 50 equivalents with respect to 1 equivalent of the compound represented by the formula (2).

必要ならば、炭酸カリウム、トリエチルアミン、ピリジン、４−（ジメチルアミノ）ピリジン等の塩基又は塩酸、硫酸、ｐ−トルエンスルホン酸等の酸を使用することができる。   If necessary, a base such as potassium carbonate, triethylamine, pyridine and 4- (dimethylamino) pyridine or an acid such as hydrochloric acid, sulfuric acid and p-toluenesulfonic acid can be used.

本反応は、無溶媒で実施してもよいが、溶媒を用いてもよく、例えば、Ｎ，Ｎ−ジメチルホルムアミド、Ｎ，Ｎ−ジメチルアセトアミド、アセトニトリル、ジメチルスルホキシド、１，３−ジメチル−２−イミダゾリノン、水等の極性溶媒、メタノール、エタノール、プロパノール、２−プロパノール、エチレングリコール等のアルコール類、ジエチルエーテル、テトラヒドロフラン、ジフェニルエーテル等のエーテル類、ベンゼン、トルエン、キシレン等の芳香族炭化水素類、塩化メチレン、クロロホルム、四塩化炭素等のハロゲン化炭化水素類、ペンタン、ｎ−ヘキサン等の脂肪族炭化水素類が挙げられる。これらの溶媒は単独で用いても、これらの内の２種類以上を混合して用いてもよい。   This reaction may be carried out without solvent, but a solvent may be used, for example, N, N-dimethylformamide, N, N-dimethylacetamide, acetonitrile, dimethyl sulfoxide, 1,3-dimethyl-2- Polar solvents such as imidazolinone and water, alcohols such as methanol, ethanol, propanol, 2-propanol and ethylene glycol, ethers such as diethyl ether, tetrahydrofuran and diphenyl ether, aromatic hydrocarbons such as benzene, toluene and xylene, Halogenated hydrocarbons such as methylene chloride, chloroform and carbon tetrachloride, and aliphatic hydrocarbons such as pentane and n-hexane. These solvents may be used alone or as a mixture of two or more thereof.

反応温度は、−６０℃から反応混合物の還流温度までの任意の温度を設定することができ、反応時間は、反応基質の濃度、反応温度によって変化するが、通常５分から１００時間の範囲で任意に設定できる。   The reaction temperature can be set to any temperature from −60 ° C. to the reflux temperature of the reaction mixture, and the reaction time varies depending on the concentration of the reaction substrate and the reaction temperature, but is usually arbitrary in the range of 5 minutes to 100 hours. Can be set.

式（１０）で表される化合物の或るものは公知化合物であり、一部は市販品として入手できる。また、それ以外のものも文献記載の公知の方法に準じて容易に合成することができる。   Some of the compounds represented by formula (10) are known compounds, and some of them are commercially available. Others can be easily synthesized according to known methods described in the literature.

製造法Ａ乃至製造法Ｄの反応において、反応終了後の反応混合物は、直接濃縮、又は有機溶媒に溶解し、水洗後濃縮、又は氷水に投入、有機溶媒抽出後濃縮といった通常の後処理を行ない、目的の本発明化合物を得ることができる。また、精製の必要が生じたときには、再結晶、カラムクロマトグラフ、薄層クロマトグラフ、液体クロマトグラフ分取等の任意の精製方法によって分離、精製することができる。   In the reaction of production method A to production method D, the reaction mixture after completion of the reaction is directly concentrated, or dissolved in an organic solvent, concentrated after washing with water, or poured into ice water and concentrated after extraction with an organic solvent, followed by normal post-treatment. The objective compound of the present invention can be obtained. Moreover, when the necessity for purification arises, it can be separated and purified by any purification method such as recrystallization, column chromatograph, thin layer chromatograph, liquid chromatographic fractionation and the like.

製造法Ａで用いられる式（２）で表される化合物は、例えば以下のようにして合成することが出来る。   The compound represented by the formula (2) used in the production method A can be synthesized, for example, as follows.

反応式１   Reaction formula 1

すなわち、式（２−１）［式中Ｒ^３、Ｒ^ａ及びＲ^４は前記と同じ意味を表す。］で表される化合物を、文献既知の公知の方法、例えばジャーナル ヘテロサイクリック ケミストリー １９８６年，２３巻，２７５頁等に記載の方法に準じて、公知の式（２−２）［式中Ａ^１、Ｒ^２及びｎは前記と同じ意味を表し、Ｌ_１はフッ素原子、塩素原子、臭素原子、ヨウ素原子、−Ｂ（ＯＨ）_２基又は−Ｂ（ＯＲ^５０）_２基（式中Ｒ^５０は、水素原子又は、同一又は異なってもよいＣ_１〜Ｃ_６アルキルを表し、或いは、２つのＧが一緒になって−ＣＨ_２ＣＨ_２−又は−Ｃ（ＣＨ_３）_２Ｃ（ＣＨ_３）_２−を形成してもよい）を表す。］で表される化合物と、パラジウムなどの遷移金属触媒及び塩基の存在下で反応させることにより、式（２）［式中Ａ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^ａ及びｎは前記と同じ意味を表す。］の化合物を容易に製造することができる。 That is, formula (2-1) [wherein R ³ , R ^a and R ⁴ represent the same meaning as described above. In accordance with a known method known in the literature, for example, the method described in Journal Heterocyclic Chemistry 1986, Vol. 23, page 275, etc., the known formula (2-2) [in the formula A ¹ , R ² and n represent the same meaning as described above, and L ₁ represents a fluorine atom, a chlorine atom, a bromine atom, an iodine atom, —B (OH) ₂ group or —B (OR ⁵⁰ ) ₂ group (wherein R ⁵⁰ Represents a hydrogen atom or C _{1 to} C ₆ alkyl which may be the same or different, or two G together represent —CH ₂ CH ₂ — or —C (CH ₃ ) ₂ C (CH ₃ ). _2- may be formed). ] In the presence of a transition metal catalyst such as palladium and a base, wherein A ¹ , R ² , R ³ , R ⁴ , R ^a and n are as defined above. Means the same. ] Can be easily produced.

本発明に包含される活性化合物としては、具体的に例えば第１表乃至第６表に示す化合物が挙げられる。但し、第１表乃至第３表に記載された化合物は例示のためのものであって、本発明はこれらのみに限定されるものではない。尚、表中、Ｍｅと記載される置換基はメチル基を表し、以下、Ｅｔとの記載はエチル基を表し、ｎ−Ｐｒ及びＰｒ−ｎはノルマルプロピル基を、ｉ−Ｐｒ及びＰｒ−ｉはイソプロピル基を、ｃ−Ｐｒ及びＰｒ−ｃはシクロプロピル基を、ｎ−Ｂｕ及びＢｕ−ｎノルマルブチル基を、ｓ−Ｂｕ及びＢｕ−ｓはセカンダリーブチル基を、ｉ−Ｂｕ及びＢｕ−ｉはイソブチル基を、ｔ−Ｂｕ及びＢｕ−ｔはターシャリーブチル基を、ｃ−Ｂｕ及びＢｕ−ｃはシクロブチル基を、ｎ−Ｐｅｎ及びＰｅｎ−ｎはノルマルペンチル基を、ｃ−Ｐｅｎ及びＰｅｎ−ｃはシクロペンチル基を、ｎ−Ｈｅｘ及びＨｅｘ−ｎはノルマルヘキシル基を、ｃ−Ｈｅｘ及びＨｅｘ−ｃはシクロヘキシル基を、Ｈｅｐｔはヘプチル基を、Ｏｃｔはオクチル基を、Ｐｈはフェニル基をそれぞれ表す。   Specific examples of the active compound included in the present invention include compounds shown in Tables 1 to 6. However, the compounds described in Tables 1 to 3 are for illustrative purposes, and the present invention is not limited thereto. In the table, the substituent described as Me represents a methyl group, hereinafter, Et represents an ethyl group, n-Pr and Pr-n represent normal propyl groups, i-Pr and Pr-i. Is an isopropyl group, c-Pr and Pr-c are cyclopropyl groups, n-Bu and Bu-n normal butyl groups, s-Bu and Bu-s are secondary butyl groups, i-Bu and Bu-i. Is an isobutyl group, t-Bu and Bu-t are tertiary butyl groups, c-Bu and Bu-c are cyclobutyl groups, n-Pen and Pen-n are normal pentyl groups, c-Pen and Pen- c is a cyclopentyl group, n-Hex and Hex-n are normal hexyl groups, c-Hex and Hex-c are cyclohexyl groups, Hept is a heptyl group, Oct is an octyl group, and Ph is a fethyl group. It represents Le group, respectively.

また、表中Ｄ２−１ａ〜Ｄ２−１０８ｂは下記の構造式を表し、Ｄ２−１ｃ、Ｄ２−１ｄ、Ｄ２−２ｃ、Ｄ２−２ｄ、Ｄ２−３ｂ、Ｄ２−４ｃ、Ｄ２−４ｄ、Ｄ２−５ｄ、Ｄ２−５ｅ、Ｄ２−５ｆ、Ｄ２−６ｄ、Ｄ２−６ｅ、Ｄ２−６ｆ、Ｄ２−７ｂ、Ｄ２−８ｄ、Ｄ２−８ｅ、Ｄ２−８ｆ、Ｄ２−９ｄ、Ｄ２−９ｅ、Ｄ２−９ｆ、Ｄ２−１０ｄ、Ｄ２−１０ｅ、Ｄ２−１０ｆ、Ｄ２−１１ｂ、Ｄ２−１２ｄ、Ｄ２−１２ｅ、Ｄ２−１２ｆ、Ｄ２−２０ｂ、Ｄ２−２２ｂ、Ｄ２−２４ｂ、Ｄ２−２６ｂ、Ｄ２−３２ｂ、Ｄ２−３３ｂ、Ｄ２−３４ｂ、Ｄ２−３５ｃ、Ｄ２−３５ｄ、Ｄ２−３６ｂ、Ｄ２−３７ｂ、Ｄ２−３８ｂ、Ｄ２−３９ｂの各構造式に記された番号は、Ｘ^２の置換位置を表し、Ｄ２−１０８ｂの構造式に記された番号は、Ｚ^２の置換位置を表す。 In the table, D2-1a to D2-108b represent the following structural formulas: D2-1c, D2-1d, D2-2c, D2-2d, D2-3b, D2-4c, D2-4d, D2-5d D2-5e, D2-5f, D2-6d, D2-6e, D2-6f, D2-7b, D2-8d, D2-8e, D2-8f, D2-9d, D2-9e, D2-9f, D2 -10d, D2-10e, D2-10f, D2-11b, D2-12d, D2-12e, D2-12f, D2-20b, D2-22b, D2-24b, D2-26b, D2-32b, D2-33b , D2-34b, D2-35c, D2-35d, D2-36b , D2-37b, D2-38b, numbers written in the structural formula of D2-39b represents the substitution position of ^{X 2,} D2-108b The number written in the structural formula of It represents the substitution position of Z ^2.

〔第１表〕 [Table 1]

第１表
--------------------------------------
R^a R^b
--------------------------------------
H H
H Me
H Et
H Pr-n
H Pr-i
H Pr-c
H Bu-n
H Bu-i
H Bu-c
H Bu-s
H Bu-t
H Pen-n
H Pen-c
H Hex-n
H Hex-c
H CH₂Pr-c
H CH₂Bu-c
H CH₂Pen-c
H CH₂Hex-c
H CH₂CH=CH₂
H CH₂CH=C(Cl)₂
H CH₂C≡CH
H CH₂CN
H CH₂CF₃
H CH₂OMe
H CH₂OCF₃
H CH₂SMe
H CH₂S(O)Me
H CH₂S(O)₂Me
H CH₂SCF₃
H CH₂S(O)CF₃
H CH₂S(O)₂CF₃
H CH₂CH(OMe)₂
H CH₂CH(SMe)₂
H CH₂C(O)Me
H CH₂C(O)CF₃
H CH₂C(O)OMe
H CH₂(D2-32a)
H CH₂(D2-33a)
H CH₂(D2-34a)
H CH₂(D2-37a)
H CH₂(D2-81a)
H CH₂(D2-82a)
H CH₂(D2-84a)
H CH₂(D2-85a)
H CH₂(D2-87a)
H CH₂(D2-92a)
H CH₂(D2-93a)
H CH₂(D2-95a)
H CH₂(D2-96a)
H CH₂(D2-98a)
H CH₂(D2-108a)
H CH₂(D2-108b,Z²=2-Cl)
H CH₂(D2-108b,Z²=3-Me)
H CH₂(D2-108b,Z²=4-OMe)
H CH₂(D2-108b,Z²=2-SMe)
H CH₂(D2-108b,Z²=3-CF₃)
H CH₂(D2-108b,Z²=4-OCF₃)
H CH₂(D2-108b,Z²=2-SCF₃)
H CH₂CH₂CN
H CH₂CH₂CF₃
H CH₂CH₂OMe
H CH₂CH₂SMe
H CH₂CH₂S(O)Me
H CH₂CH₂S(O)₂Me
H D2-32a
H D2-33a
H D2-34a
H D2-37a
H D2-81a
H D2-82a
H D2-84a
H D2-85a
H D2-87a
H D2-92a
H D2-93a
H D2-95a
H D2-96a
H D2-98a
H D2-108a
H D2-108b(Z²=2-Cl)
H D2-108b(Z²=3-Me)
H D2-108b(Z²=4-OMe)
H D2-108b(Z²=2-SMe)
H D2-108b(Z²=3-CF₃)
H D2-108b(Z²=4-OCF₃)
H D2-108b(Z²=2-SCF₃)
H C(O)Me
H C(O)CF₃
H C(O)OMe
CF₃ Me
CF₃ Et
CF₃ Pr-n
CF₃ Pr-i
CF₃ Pr-c
CF₃ Bu-n
CF₃ Bu-i
CF₃ Bu-c
CF₃ Bu-s
CF₃ Bu-t
CF₃ Pen-n
CF₃ Pen-c
CF₃ Hex-n
CF₃ Hex-c
CF₃ CH₂Pr-c
CF₃ CH₂Bu-c
CF₃ CH₂Pen-c
CF₃ CH₂Hex-c
CF₃ CH₂CH=CH₂
CF₃ CH₂CH=C(Cl)₂
CF₃ CH₂C≡CH
CF₃ CH₂CN
CF₃ CH₂CF₃
CF₃ CH₂OMe
CF₃ CH₂OCF₃
CF₃ CH₂SMe
CF₃ CH₂S(O)Me
CF₃ CH₂S(O)₂Me
CF₃ CH₂SCF₃
CF₃ CH₂S(O)CF₃
CF₃ CH₂S(O)₂CF₃
CF₃ CH₂CH(OMe)₂
CF₃ CH₂CH(SMe)₂
CF₃ CH₂C(O)Me
CF₃ CH₂C(O)CF₃
CF₃ CH₂C(O)OMe
CF₃ CH₂(D2-32a)
CF₃ CH₂(D2-33a)
CF₃ CH₂(D2-34a)
CF₃ CH₂(D2-37a)
CF₃ CH₂(D2-81a)
CF₃ CH₂(D2-82a)
CF₃ CH₂(D2-84a)
CF₃ CH₂(D2-85a)
CF₃ CH₂(D2-87a)
CF₃ CH₂(D2-92a)
CF₃ CH₂(D2-93a)
CF₃ CH₂(D2-95a)
CF₃ CH₂(D2-96a)
CF₃ CH₂(D2-98a)
CF₃ CH₂(D2-108a)
CF₃ CH₂(D2-108b,Z²=2-Cl)
CF₃ CH₂(D2-108b,Z²=3-Me)
CF₃ CH₂(D2-108b,Z²=4-OMe)
CF₃ CH₂(D2-108b,Z²=2-SMe)
CF₃ CH₂(D2-108b,Z²=3-CF₃)
CF₃ CH₂(D2-108b,Z²=4-OCF₃)
CF₃ CH₂(D2-108b,Z²=2-SCF₃)
CF₃ CH₂CH₂CN
CF₃ CH₂CH₂CF₃
CF₃ CH₂CH₂OMe
CF₃ CH₂CH₂SMe
CF₃ CH₂CH₂S(O)Me
CF₃ CH₂CH₂S(O)₂Me
CF₃ D2-32a
CF₃ D2-33a
CF₃ D2-34a
CF₃ D2-37a
CF₃ D2-81a
CF₃ D2-82a
CF₃ D2-84a
CF₃ D2-85a
CF₃ D2-87a
CF₃ D2-92a
CF₃ D2-93a
CF₃ D2-95a
CF₃ D2-96a
CF₃ D2-98a
CF₃ D2-108a
CF₃ D2-108b(Z²=2-Cl)
CF₃ D2-108b(Z²=3-Me)
CF₃ D2-108b(Z²=4-OMe)
CF₃ D2-108b(Z²=2-SMe)
CF₃ D2-108b(Z²=3-CF₃)
CF₃ D2-108b(Z²=4-OCF₃)
CF₃ D2-108b(Z²=2-SCF₃)
CF₃ C(O)Me
CF₃ C(O)CF₃
CF₃ C(O)OMe
Me Me
Me Et
Me Pr-n
Me Pr-i
Me Pr-c
Me Bu-n
Me Bu-i
Me Bu-c
Me Bu-s
Me Bu-t
Me Pen-n
Me Pen-c
Me Hex-n
Me Hex-c
Me CH₂Pr-c
Me CH₂Bu-c
Me CH₂Pen-c
Me CH₂Hex-c
Me CH₂CH=CH₂
Me CH₂CH=C(Cl)₂
Me CH₂C≡CH
Me CH₂CN
Me CH₂CF₃
Me CH₂OMe
Me CH₂OCF₃
Me CH₂SMe
Me CH₂S(O)Me
Me CH₂S(O)₂Me
Me CH₂SCF₃
Me CH₂S(O)CF₃
Me CH₂S(O)₂CF₃
Me CH₂CH(OMe)₂
Me CH₂CH(SMe)₂
Me CH₂C(O)Me
Me CH₂C(O)CF₃
Me CH₂C(O)OMe
Me CH₂(D2-32a)
Me CH₂(D2-33a)
Me CH₂(D2-34a)
Me CH₂(D2-37a)
Me CH₂(D2-81a)
Me CH₂(D2-82a)
Me CH₂(D2-84a)
Me CH₂(D2-85a)
Me CH₂(D2-87a)
Me CH₂(D2-92a)
Me CH₂(D2-93a)
Me CH₂(D2-95a)
Me CH₂(D2-96a)
Me CH₂(D2-98a)
Me CH₂(D2-108a)
Me CH₂(D2-108b,Z²=2-Cl)
Me CH₂(D2-108b,Z²=3-Me)
Me CH₂(D2-108b,Z²=4-OMe)
Me CH₂(D2-108b,Z²=2-SMe)
Me CH₂(D2-108b,Z²=3-CF₃)
Me CH₂(D2-108b,Z²=4-OCF₃)
Me CH₂(D2-108b,Z²=2-SCF₃)
Me CH₂CH₂CN
Me CH₂CH₂CF₃
Me CH₂CH₂OMe
Me CH₂CH₂SMe
Me CH₂CH₂S(O)Me
Me CH₂CH₂S(O)₂Me
Me D2-32a
Me D2-33a
Me D2-34a
Me D2-37a
Me D2-81a
Me D2-82a
Me D2-84a
Me D2-85a
Me D2-87a
Me D2-92a
Me D2-93a
Me D2-95a
Me D2-96a
Me D2-98a
Me D2-108a
Me D2-108b(Z²=2-Cl)
Me D2-108b(Z²=3-Me)
Me D2-108b(Z²=4-OMe)
Me D2-108b(Z²=2-SMe)
Me D2-108b(Z²=3-CF₃)
Me D2-108b(Z²=4-OCF₃)
Me D2-108b(Z²=2-SCF₃)
Me C(O)Me
Me C(O)CF₃
Me C(O)OMe
OMe Me
OMe Et
OMe Pr-n
OMe Pr-i
OMe Pr-c
OMe Bu-n
OMe Bu-i
OMe Bu-c
OMe Bu-s
OMe Bu-t
OMe Pen-n
OMe Pen-c
OMe Hex-n
OMe Hex-c
OMe CH₂Pr-c
OMe CH₂Bu-c
OMe CH₂Pen-c
OMe CH₂Hex-c
OMe CH₂CH=CH₂
OMe CH₂CH=C(Cl)₂
OMe CH₂C≡CH
OMe CH₂CN
OMe CH₂CF₃
OMe CH₂OMe
OMe CH₂OCF₃
OMe CH₂SMe
OMe CH₂S(O)Me
OMe CH₂S(O)₂Me
OMe CH₂SCF₃
OMe CH₂S(O)CF₃
OMe CH₂S(O)₂CF₃
OMe CH₂CH(OMe)₂
OMe CH₂CH(SMe)₂
OMe CH₂C(O)Me
OMe CH₂C(O)CF₃
OMe CH₂C(O)OMe
OMe CH₂(D2-32a)
OMe CH₂(D2-33a)
OMe CH₂(D2-34a)
OMe CH₂(D2-37a)
OMe CH₂(D2-81a)
OMe CH₂(D2-82a)
OMe CH₂(D2-84a)
OMe CH₂(D2-85a)
OMe CH₂(D2-87a)
OMe CH₂(D2-92a)
OMe CH₂(D2-93a)
OMe CH₂(D2-95a)
OMe CH₂(D2-96a)
OMe CH₂(D2-98a)
OMe CH₂(D2-108a)
OMe CH₂(D2-108b,Z²=2-Cl)
OMe CH₂(D2-108b,Z²=3-Me)
OMe CH₂(D2-108b,Z²=4-OMe)
OMe CH₂(D2-108b,Z²=2-SMe)
OMe CH₂(D2-108b,Z²=3-CF₃)
OMe CH₂(D2-108b,Z²=4-OCF₃)
OMe CH₂(D2-108b,Z²=2-SCF₃)
OMe CH₂CH₂CN
OMe CH₂CH₂CF₃
OMe CH₂CH₂OMe
OMe CH₂CH₂SMe
OMe CH₂CH₂S(O)Me
OMe CH₂CH₂S(O)₂Me
OMe D2-32a
OMe D2-33a
OMe D2-34a
OMe D2-37a
OMe D2-81a
OMe D2-82a
OMe D2-84a
OMe D2-85a
OMe D2-87a
OMe D2-92a
OMe D2-93a
OMe D2-95a
OMe D2-96a
OMe D2-98a
OMe D2-108a
OMe D2-108b(Z²=2-Cl)
OMe D2-108b(Z²=3-Me)
OMe D2-108b(Z²=4-OMe)
OMe D2-108b(Z²=2-SMe)
OMe D2-108b(Z²=3-CF₃)
OMe D2-108b(Z²=4-OCF₃)
OMe D2-108b(Z²=2-SCF₃)
OMe C(O)Me
OMe C(O)CF₃
OMe C(O)OMe
SMe Me
SMe Et
SMe Pr-n
SMe Pr-i
SMe Pr-c
SMe Bu-n
SMe Bu-i
SMe Bu-c
SMe Bu-s
SMe Bu-t
SMe Pen-n
SMe Pen-c
SMe Hex-n
SMe Hex-c
SMe CH₂Pr-c
SMe CH₂Bu-c
SMe CH₂Pen-c
SMe CH₂Hex-c
SMe CH₂CH=CH₂
SMe CH₂CH=C(Cl)₂
SMe CH₂C≡CH
SMe CH₂CN
SMe CH₂CF₃
SMe CH₂OMe
SMe CH₂OCF₃
SMe CH₂SMe
SMe CH₂S(O)Me
SMe CH₂S(O)₂Me
SMe CH₂SCF₃
SMe CH₂S(O)CF₃
SMe CH₂S(O)₂CF₃
SMe CH₂CH(OMe)₂
SMe CH₂CH(SMe)₂
SMe CH₂C(O)Me
SMe CH₂C(O)CF₃
SMe CH₂C(O)OMe
SMe CH₂(D2-32a)
SMe CH₂(D2-33a)
SMe CH₂(D2-34a)
SMe CH₂(D2-37a)
SMe CH₂(D2-81a)
SMe CH₂(D2-82a)
SMe CH₂(D2-84a)
SMe CH₂(D2-85a)
SMe CH₂(D2-87a)
SMe CH₂(D2-92a)
SMe CH₂(D2-93a)
SMe CH₂(D2-95a)
SMe CH₂(D2-96a)
SMe CH₂(D2-98a)
SMe CH₂(D2-108a)
SMe CH₂(D2-108b,Z²=2-Cl)
SMe CH₂(D2-108b,Z²=3-Me)
SMe CH₂(D2-108b,Z²=4-OMe)
SMe CH₂(D2-108b,Z²=2-SMe)
SMe CH₂(D2-108b,Z²=3-CF₃)
SMe CH₂(D2-108b,Z²=4-OCF₃)
SMe CH₂(D2-108b,Z²=2-SCF₃)
SMe CH₂CH₂CN
SMe CH₂CH₂CF₃
SMe CH₂CH₂OMe
SMe CH₂CH₂SMe
SMe CH₂CH₂S(O)Me
SMe CH₂CH₂S(O)₂Me
SMe D2-32a
SMe D2-33a
SMe D2-34a
SMe D2-37a
SMe D2-81a
SMe D2-82a
SMe D2-84a
SMe D2-85a
SMe D2-87a
SMe D2-92a
SMe D2-93a
SMe D2-95a
SMe D2-96a
SMe D2-98a
SMe D2-108a
SMe D2-108b(Z²=2-Cl)
SMe D2-108b(Z²=3-Me)
SMe D2-108b(Z²=4-OMe)
SMe D2-108b(Z²=2-SMe)
SMe D2-108b(Z²=3-CF₃)
SMe D2-108b(Z²=4-OCF₃)
SMe D2-108b(Z²=2-SCF₃)
SMe C(O)Me
SMe C(O)CF₃
SMe C(O)OMe
CH₂OMe Me
CH₂OMe Et
CH₂OMe Pr-n
CH₂OMe Pr-i
CH₂OMe Pr-c
CH₂OMe Bu-n
CH₂OMe Bu-i
CH₂OMe Bu-c
CH₂OMe Bu-s
CH₂OMe Bu-t
CH₂OMe Pen-n
CH₂OMe Pen-c
CH₂OMe Hex-n
CH₂OMe Hex-c
CH₂OMe CH₂Pr-c
CH₂OMe CH₂Bu-c
CH₂OMe CH₂Pen-c
CH₂OMe CH₂Hex-c
CH₂OMe CH₂CH=CH₂
CH₂OMe CH₂CH=C(Cl)₂
CH₂OMe CH₂C≡CH
CH₂OMe CH₂CN
CH₂OMe CH₂CF₃
CH₂OMe CH₂OMe
CH₂OMe CH₂OCF₃
CH₂OMe CH₂SMe
CH₂OMe CH₂S(O)Me
CH₂OMe CH₂S(O)₂Me
CH₂OMe CH₂SCF₃
CH₂OMe CH₂S(O)CF₃
CH₂OMe CH₂S(O)₂CF₃
CH₂OMe CH₂CH(OMe)₂
CH₂OMe CH₂CH(SMe)₂
CH₂OMe CH₂C(O)Me
CH₂OMe CH₂C(O)CF₃
CH₂OMe CH₂C(O)OMe
CH₂OMe CH₂(D2-32a)
CH₂OMe CH₂(D2-33a)
CH₂OMe CH₂(D2-34a)
CH₂OMe CH₂(D2-37a)
CH₂OMe CH₂(D2-81a)
CH₂OMe CH₂(D2-82a)
CH₂OMe CH₂(D2-84a)
CH₂OMe CH₂(D2-85a)
CH₂OMe CH₂(D2-87a)
CH₂OMe CH₂(D2-92a)
CH₂OMe CH₂(D2-93a)
CH₂OMe CH₂(D2-95a)
CH₂OMe CH₂(D2-96a)
CH₂OMe CH₂(D2-98a)
CH₂OMe CH₂(D2-108a)
CH₂OMe CH₂(D2-108b,Z²=2-Cl)
CH₂OMe CH₂(D2-108b,Z²=3-Me)
CH₂OMe CH₂(D2-108b,Z²=4-OMe)
CH₂OMe CH₂(D2-108b,Z²=2-SMe)
CH₂OMe CH₂(D2-108b,Z²=3-CF₃)
CH₂OMe CH₂(D2-108b,Z²=4-OCF₃)
CH₂OMe CH₂(D2-108b,Z²=2-SCF₃)
CH₂OMe CH₂CH₂CN
CH₂OMe CH₂CH₂CF₃
CH₂OMe CH₂CH₂OMe
CH₂OMe CH₂CH₂SMe
CH₂OMe CH₂CH₂S(O)Me
CH₂OMe CH₂CH₂S(O)₂Me
CH₂OMe D2-32a
CH₂OMe D2-33a
CH₂OMe D2-34a
CH₂OMe D2-37a
CH₂OMe D2-81a
CH₂OMe D2-82a
CH₂OMe D2-84a
CH₂OMe D2-85a
CH₂OMe D2-87a
CH₂OMe D2-92a
CH₂OMe D2-93a
CH₂OMe D2-95a
CH₂OMe D2-96a
CH₂OMe D2-98a
CH₂OMe D2-108a
CH₂OMe D2-108b(Z²=2-Cl)
CH₂OMe D2-108b(Z²=3-Me)
CH₂OMe D2-108b(Z²=4-OMe)
CH₂OMe D2-108b(Z²=2-SMe)
CH₂OMe D2-108b(Z²=3-CF₃)
CH₂OMe D2-108b(Z²=4-OCF₃)
CH₂OMe D2-108b(Z²=2-SCF₃)
CH₂OMe C(O)Me
CH₂OMe C(O)CF₃
CH₂OMe C(O)OMe
CH₂SMe Me
CH₂SMe Et
CH₂SMe Pr-n
CH₂SMe Pr-i
CH₂SMe Pr-c
CH₂SMe Bu-n
CH₂SMe Bu-i
CH₂SMe Bu-c
CH₂SMe Bu-s
CH₂SMe Bu-t
CH₂SMe Pen-n
CH₂SMe Pen-c
CH₂SMe Hex-n
CH₂SMe Hex-c
CH₂SMe CH₂Pr-c
CH₂SMe CH₂Bu-c
CH₂SMe CH₂Pen-c
CH₂SMe CH₂Hex-c
CH₂SMe CH₂CH=CH₂
CH₂SMe CH₂CH=C(Cl)₂
CH₂SMe CH₂C≡CH
CH₂SMe CH₂CN
CH₂SMe CH₂CF₃
CH₂SMe CH₂OMe
CH₂SMe CH₂OCF₃
CH₂SMe CH₂SMe
CH₂SMe CH₂S(O)Me
CH₂SMe CH₂S(O)₂Me
CH₂SMe CH₂SCF₃
CH₂SMe CH₂S(O)CF₃
CH₂SMe CH₂S(O)₂CF₃
CH₂SMe CH₂CH(OMe)₂
CH₂SMe CH₂CH(SMe)₂
CH₂SMe CH₂C(O)Me
CH₂SMe CH₂C(O)CF₃
CH₂SMe CH₂C(O)OMe
CH₂SMe CH₂(D2-32a)
CH₂SMe CH₂(D2-33a)
CH₂SMe CH₂(D2-34a)
CH₂SMe CH₂(D2-37a)
CH₂SMe CH₂(D2-81a)
CH₂SMe CH₂(D2-82a)
CH₂SMe CH₂(D2-84a)
CH₂SMe CH₂(D2-85a)
CH₂SMe CH₂(D2-87a)
CH₂SMe CH₂(D2-92a)
CH₂SMe CH₂(D2-93a)
CH₂SMe CH₂(D2-95a)
CH₂SMe CH₂(D2-96a)
CH₂SMe CH₂(D2-98a)
CH₂SMe CH₂(D2-108a)
CH₂SMe CH₂(D2-108b,Z²=2-Cl)
CH₂SMe CH₂(D2-108b,Z²=3-Me)
CH₂SMe CH₂(D2-108b,Z²=4-OMe)
CH₂SMe CH₂(D2-108b,Z²=2-SMe)
CH₂SMe CH₂(D2-108b,Z²=3-CF₃)
CH₂SMe CH₂(D2-108b,Z²=4-OCF₃)
CH₂SMe CH₂(D2-108b,Z²=2-SCF₃)
CH₂SMe CH₂CH₂CN
CH₂SMe CH₂CH₂CF₃
CH₂SMe CH₂CH₂OMe
CH₂SMe CH₂CH₂SMe
CH₂SMe CH₂CH₂S(O)Me
CH₂SMe CH₂CH₂S(O)₂Me
CH₂SMe D2-32a
CH₂SMe D2-33a
CH₂SMe D2-34a
CH₂SMe D2-37a
CH₂SMe D2-81a
CH₂SMe D2-82a
CH₂SMe D2-84a
CH₂SMe D2-85a
CH₂SMe D2-87a
CH₂SMe D2-92a
CH₂SMe D2-93a
CH₂SMe D2-95a
CH₂SMe D2-96a
CH₂SMe D2-98a
CH₂SMe D2-108a
CH₂SMe D2-108b(Z²=2-Cl)
CH₂SMe D2-108b(Z²=3-Me)
CH₂SMe D2-108b(Z²=4-OMe)
CH₂SMe D2-108b(Z²=2-SMe)
CH₂SMe D2-108b(Z²=3-CF₃)
CH₂SMe D2-108b(Z²=4-OCF₃)
CH₂SMe D2-108b(Z²=2-SCF₃)
CH₂SMe C(O)Me
CH₂SMe C(O)CF₃
CH₂SMe C(O)OMe
CH₂S(O)Me Me
CH₂S(O)Me Et
CH₂S(O)Me Pr-n
CH₂S(O)Me Pr-i
CH₂S(O)Me Pr-c
CH₂S(O)Me Bu-n
CH₂S(O)Me Bu-i
CH₂S(O)Me Bu-c
CH₂S(O)Me Bu-s
CH₂S(O)Me Bu-t
CH₂S(O)Me Pen-n
CH₂S(O)Me Pen-c
CH₂S(O)Me Hex-n
CH₂S(O)Me Hex-c
CH₂S(O)Me CH₂Pr-c
CH₂S(O)Me CH₂Bu-c
CH₂S(O)Me CH₂Pen-c
CH₂S(O)Me CH₂Hex-c
CH₂S(O)Me CH₂CH=CH₂
CH₂S(O)Me CH₂CH=C(Cl)₂
CH₂S(O)Me CH₂C≡CH
CH₂S(O)Me CH₂CN
CH₂S(O)Me CH₂CF₃
CH₂S(O)Me CH₂OMe
CH₂S(O)Me CH₂OCF₃
CH₂S(O)Me CH₂SMe
CH₂S(O)Me CH₂S(O)Me
CH₂S(O)Me CH₂S(O)₂Me
CH₂S(O)Me CH₂SCF₃
CH₂S(O)Me CH₂S(O)CF₃
CH₂S(O)Me CH₂S(O)₂CF₃
CH₂S(O)Me CH₂CH(OMe)₂
CH₂S(O)Me CH₂CH(SMe)₂
CH₂S(O)Me CH₂C(O)Me
CH₂S(O)Me CH₂C(O)CF₃
CH₂S(O)Me CH₂C(O)OMe
CH₂S(O)Me CH₂(D2-32a)
CH₂S(O)Me CH₂(D2-33a)
CH₂S(O)Me CH₂(D2-34a)
CH₂S(O)Me CH₂(D2-37a)
CH₂S(O)Me CH₂(D2-81a)
CH₂S(O)Me CH₂(D2-82a)
CH₂S(O)Me CH₂(D2-84a)
CH₂S(O)Me CH₂(D2-85a)
CH₂S(O)Me CH₂(D2-87a)
CH₂S(O)Me CH₂(D2-92a)
CH₂S(O)Me CH₂(D2-93a)
CH₂S(O)Me CH₂(D2-95a)
CH₂S(O)Me CH₂(D2-96a)
CH₂S(O)Me CH₂(D2-98a)
CH₂S(O)Me CH₂(D2-108a)
CH₂S(O)Me CH₂(D2-108b,Z²=2-Cl)
CH₂S(O)Me CH₂(D2-108b,Z²=3-Me)
CH₂S(O)Me CH₂(D2-108b,Z²=4-OMe)
CH₂S(O)Me CH₂(D2-108b,Z²=2-SMe)
CH₂S(O)Me CH₂(D2-108b,Z²=3-CF₃)
CH₂S(O)Me CH₂(D2-108b,Z²=4-OCF₃)
CH₂S(O)Me CH₂(D2-108b,Z²=2-SCF₃)
CH₂S(O)Me CH₂CH₂CN
CH₂S(O)Me CH₂CH₂CF₃
CH₂S(O)Me CH₂CH₂OMe
CH₂S(O)Me CH₂CH₂SMe
CH₂S(O)Me CH₂CH₂S(O)Me
CH₂S(O)Me CH₂CH₂S(O)₂Me
CH₂S(O)Me D2-32a
CH₂S(O)Me D2-33a
CH₂S(O)Me D2-34a
CH₂S(O)Me D2-37a
CH₂S(O)Me D2-81a
CH₂S(O)Me D2-82a
CH₂S(O)Me D2-84a
CH₂S(O)Me D2-85a
CH₂S(O)Me D2-87a
CH₂S(O)Me D2-92a
CH₂S(O)Me D2-93a
CH₂S(O)Me D2-95a
CH₂S(O)Me D2-96a
CH₂S(O)Me D2-98a
CH₂S(O)Me D2-108a
CH₂S(O)Me D2-108b(Z²=2-Cl)
CH₂S(O)Me D2-108b(Z²=3-Me)
CH₂S(O)Me D2-108b(Z²=4-OMe)
CH₂S(O)Me D2-108b(Z²=2-SMe)
CH₂S(O)Me D2-108b(Z²=3-CF₃)
CH₂S(O)Me D2-108b(Z²=4-OCF₃)
CH₂S(O)Me D2-108b(Z²=2-SCF₃)
CH₂S(O)Me C(O)Me
CH₂S(O)Me C(O)CF₃
CH₂S(O)Me C(O)OMe
CH₂S(O)₂Me Me
CH₂S(O)₂Me Et
CH₂S(O)₂Me Pr-n
CH₂S(O)₂Me Pr-i
CH₂S(O)₂Me Pr-c
CH₂S(O)₂Me Bu-n
CH₂S(O)₂Me Bu-i
CH₂S(O)₂Me Bu-c
CH₂S(O)₂Me Bu-s
CH₂S(O)₂Me Bu-t
CH₂S(O)₂Me Pen-n
CH₂S(O)₂Me Pen-c
CH₂S(O)₂Me Hex-n
CH₂S(O)₂Me Hex-c
CH₂S(O)₂Me CH₂Pr-c
CH₂S(O)₂Me CH₂Bu-c
CH₂S(O)₂Me CH₂Pen-c
CH₂S(O)₂Me CH₂Hex-c
CH₂S(O)₂Me CH₂CH=CH₂
CH₂S(O)₂Me CH₂CH=C(Cl)₂
CH₂S(O)₂Me CH₂C≡CH
CH₂S(O)₂Me CH₂CN
CH₂S(O)₂Me CH₂CF₃
CH₂S(O)₂Me CH₂OMe
CH₂S(O)₂Me CH₂OCF₃
CH₂S(O)₂Me CH₂SMe
CH₂S(O)₂Me CH₂S(O)Me
CH₂S(O)₂Me CH₂S(O)₂Me
CH₂S(O)₂Me CH₂SCF₃
CH₂S(O)₂Me CH₂S(O)CF₃
CH₂S(O)₂Me CH₂S(O)₂CF₃
CH₂S(O)₂Me CH₂CH(OMe)₂
CH₂S(O)₂Me CH₂CH(SMe)₂
CH₂S(O)₂Me CH₂C(O)Me
CH₂S(O)₂Me CH₂C(O)CF₃
CH₂S(O)₂Me CH₂C(O)OMe
CH₂S(O)₂Me CH₂(D2-32a)
CH₂S(O)₂Me CH₂(D2-33a)
CH₂S(O)₂Me CH₂(D2-34a)
CH₂S(O)₂Me CH₂(D2-37a)
CH₂S(O)₂Me CH₂(D2-81a)
CH₂S(O)₂Me CH₂(D2-82a)
CH₂S(O)₂Me CH₂(D2-84a)
CH₂S(O)₂Me CH₂(D2-85a)
CH₂S(O)₂Me CH₂(D2-87a)
CH₂S(O)₂Me CH₂(D2-92a)
CH₂S(O)₂Me CH₂(D2-93a)
CH₂S(O)₂Me CH₂(D2-95a)
CH₂S(O)₂Me CH₂(D2-96a)
CH₂S(O)₂Me CH₂(D2-98a)
CH₂S(O)₂Me CH₂(D2-108a)
CH₂S(O)₂Me CH₂(D2-108b,Z²=2-Cl)
CH₂S(O)₂Me CH₂(D2-108b,Z²=3-Me)
CH₂S(O)₂Me CH₂(D2-108b,Z²=4-OMe)
CH₂S(O)₂Me CH₂(D2-108b,Z²=2-SMe)
CH₂S(O)₂Me CH₂(D2-108b,Z²=3-CF₃)
CH₂S(O)₂Me CH₂(D2-108b,Z²=4-OCF₃)
CH₂S(O)₂Me CH₂(D2-108b,Z²=2-SCF₃)
CH₂S(O)₂Me CH₂CH₂CN
CH₂S(O)₂Me CH₂CH₂CF₃
CH₂S(O)₂Me CH₂CH₂OMe
CH₂S(O)₂Me CH₂CH₂SMe
CH₂S(O)₂Me CH₂CH₂S(O)Me
CH₂S(O)₂Me CH₂CH₂S(O)₂Me
CH₂S(O)₂Me D2-32a
CH₂S(O)₂Me D2-33a
CH₂S(O)₂Me D2-34a
CH₂S(O)₂Me D2-37a
CH₂S(O)₂Me D2-81a
CH₂S(O)₂Me D2-82a
CH₂S(O)₂Me D2-84a
CH₂S(O)₂Me D2-85a
CH₂S(O)₂Me D2-87a
CH₂S(O)₂Me D2-92a
CH₂S(O)₂Me D2-93a
CH₂S(O)₂Me D2-95a
CH₂S(O)₂Me D2-96a
CH₂S(O)₂Me D2-98a
CH₂S(O)₂Me D2-108a
CH₂S(O)₂Me D2-108b(Z²=2-Cl)
CH₂S(O)₂Me D2-108b(Z²=3-Me)
CH₂S(O)₂Me D2-108b(Z²=4-OMe)
CH₂S(O)₂Me D2-108b(Z²=2-SMe)
CH₂S(O)₂Me D2-108b(Z²=3-CF₃)
CH₂S(O)₂Me D2-108b(Z²=4-OCF₃)
CH₂S(O)₂Me D2-108b(Z²=2-SCF₃)
CH₂S(O)₂Me C(O)Me
CH₂S(O)₂Me C(O)CF₃
CH₂S(O)₂Me C(O)OMe
CH₂SCF₃ Me
CH₂SCF₃ Et
CH₂SCF₃ Pr-n
CH₂SCF₃ Pr-i
CH₂SCF₃ Pr-c
CH₂SCF₃ Bu-n
CH₂SCF₃ Bu-i
CH₂SCF₃ Bu-c
CH₂SCF₃ Bu-s
CH₂SCF₃ Bu-t
CH₂SCF₃ Pen-n
CH₂SCF₃ Pen-c
CH₂SCF₃ Hex-n
CH₂SCF₃ Hex-c
CH₂SCF₃ CH₂Pr-c
CH₂SCF₃ CH₂Bu-c
CH₂SCF₃ CH₂Pen-c
CH₂SCF₃ CH₂Hex-c
CH₂SCF₃ CH₂CH=CH₂
CH₂SCF₃ CH₂CH=C(Cl)₂
CH₂SCF₃ CH₂C≡CH
CH₂SCF₃ CH₂CN
CH₂SCF₃ CH₂CF₃
CH₂SCF₃ CH₂OMe
CH₂SCF₃ CH₂OCF₃
CH₂SCF₃ CH₂SMe
CH₂SCF₃ CH₂S(O)Me
CH₂SCF₃ CH₂S(O)₂Me
CH₂SCF₃ CH₂SCF₃
CH₂SCF₃ CH₂S(O)CF₃
CH₂SCF₃ CH₂S(O)₂CF₃
CH₂SCF₃ CH₂CH(OMe)₂
CH₂SCF₃ CH₂CH(SMe)₂
CH₂SCF₃ CH₂C(O)Me
CH₂SCF₃ CH₂C(O)CF₃
CH₂SCF₃ CH₂C(O)OMe
CH₂SCF₃ CH₂(D2-32a)
CH₂SCF₃ CH₂(D2-33a)
CH₂SCF₃ CH₂(D2-34a)
CH₂SCF₃ CH₂(D2-37a)
CH₂SCF₃ CH₂(D2-81a)
CH₂SCF₃ CH₂(D2-82a)
CH₂SCF₃ CH₂(D2-84a)
CH₂SCF₃ CH₂(D2-85a)
CH₂SCF₃ CH₂(D2-87a)
CH₂SCF₃ CH₂(D2-92a)
CH₂SCF₃ CH₂(D2-93a)
CH₂SCF₃ CH₂(D2-95a)
CH₂SCF₃ CH₂(D2-96a)
CH₂SCF₃ CH₂(D2-98a)
CH₂SCF₃ CH₂(D2-108a)
CH₂SCF₃ CH₂(D2-108b,Z²=2-Cl)
CH₂SCF₃ CH₂(D2-108b,Z²=3-Me)
CH₂SCF₃ CH₂(D2-108b,Z²=4-OMe)
CH₂SCF₃ CH₂(D2-108b,Z²=2-SMe)
CH₂SCF₃ CH₂(D2-108b,Z²=3-CF₃)
CH₂SCF₃ CH₂(D2-108b,Z²=4-OCF₃)
CH₂SCF₃ CH₂(D2-108b,Z²=2-SCF₃)
CH₂SCF₃ CH₂CH₂CN
CH₂SCF₃ CH₂CH₂CF₃
CH₂SCF₃ CH₂CH₂OMe
CH₂SCF₃ CH₂CH₂SMe
CH₂SCF₃ CH₂CH₂S(O)Me
CH₂SCF₃ CH₂CH₂S(O)₂Me
CH₂SCF₃ D2-32a
CH₂SCF₃ D2-33a
CH₂SCF₃ D2-34a
CH₂SCF₃ D2-37a
CH₂SCF₃ D2-81a
CH₂SCF₃ D2-82a
CH₂SCF₃ D2-84a
CH₂SCF₃ D2-85a
CH₂SCF₃ D2-87a
CH₂SCF₃ D2-92a
CH₂SCF₃ D2-93a
CH₂SCF₃ D2-95a
CH₂SCF₃ D2-96a
CH₂SCF₃ D2-98a
CH₂SCF₃ D2-108a
CH₂SCF₃ D2-108b(Z²=2-Cl)
CH₂SCF₃ D2-108b(Z²=3-Me)
CH₂SCF₃ D2-108b(Z²=4-OMe)
CH₂SCF₃ D2-108b(Z²=2-SMe)
CH₂SCF₃ D2-108b(Z²=3-CF₃)
CH₂SCF₃ D2-108b(Z²=4-OCF₃)
CH₂SCF₃ D2-108b(Z²=2-SCF₃)
CH₂SCF₃ C(O)Me
CH₂SCF₃ C(O)CF₃
CH₂SCF₃ C(O)OMe
CH₂S(O)CF₃ Me
CH₂S(O)CF₃ Et
CH₂S(O)CF₃ Pr-n
CH₂S(O)CF₃ Pr-i
CH₂S(O)CF₃ Pr-c
CH₂S(O)CF₃ Bu-n
CH₂S(O)CF₃ Bu-i
CH₂S(O)CF₃ Bu-c
CH₂S(O)CF₃ Bu-s
CH₂S(O)CF₃ Bu-t
CH₂S(O)CF₃ Pen-n
CH₂S(O)CF₃ Pen-c
CH₂S(O)CF₃ Hex-n
CH₂S(O)CF₃ Hex-c
CH₂S(O)CF₃ CH₂Pr-c
CH₂S(O)CF₃ CH₂Bu-c
CH₂S(O)CF₃ CH₂Pen-c
CH₂S(O)CF₃ CH₂Hex-c
CH₂S(O)CF₃ CH₂CH=CH₂
CH₂S(O)CF₃ CH₂CH=C(Cl)₂
CH₂S(O)CF₃ CH₂C≡CH
CH₂S(O)CF₃ CH₂CN
CH₂S(O)CF₃ CH₂CF₃
CH₂S(O)CF₃ CH₂OMe
CH₂S(O)CF₃ CH₂OCF₃
CH₂S(O)CF₃ CH₂SMe
CH₂S(O)CF₃ CH₂S(O)Me
CH₂S(O)CF₃ CH₂S(O)₂Me
CH₂S(O)CF₃ CH₂SCF₃
CH₂S(O)CF₃ CH₂S(O)CF₃
CH₂S(O)CF₃ CH₂S(O)₂CF₃
CH₂S(O)CF₃ CH₂CH(OMe)₂
CH₂S(O)CF₃ CH₂CH(SMe)₂
CH₂S(O)CF₃ CH₂C(O)Me
CH₂S(O)CF₃ CH₂C(O)CF₃
CH₂S(O)CF₃ CH₂C(O)OMe
CH₂S(O)CF₃ CH₂(D2-32a)
CH₂S(O)CF₃ CH₂(D2-33a)
CH₂S(O)CF₃ CH₂(D2-34a)
CH₂S(O)CF₃ CH₂(D2-37a)
CH₂S(O)CF₃ CH₂(D2-81a)
CH₂S(O)CF₃ CH₂(D2-82a)
CH₂S(O)CF₃ CH₂(D2-84a)
CH₂S(O)CF₃ CH₂(D2-85a)
CH₂S(O)CF₃ CH₂(D2-87a)
CH₂S(O)CF₃ CH₂(D2-92a)
CH₂S(O)CF₃ CH₂(D2-93a)
CH₂S(O)CF₃ CH₂(D2-95a)
CH₂S(O)CF₃ CH₂(D2-96a)
CH₂S(O)CF₃ CH₂(D2-98a)
CH₂S(O)CF₃ CH₂(D2-108a)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=2-Cl)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=3-Me)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=4-OMe)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=2-SMe)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=3-CF₃)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=4-OCF₃)
CH₂S(O)CF₃ CH₂(D2-108b,Z²=2-SCF₃)
CH₂S(O)CF₃ CH₂CH₂CN
CH₂S(O)CF₃ CH₂CH₂CF₃
CH₂S(O)CF₃ CH₂CH₂OMe
CH₂S(O)CF₃ CH₂CH₂SMe
CH₂S(O)CF₃ CH₂CH₂S(O)Me
CH₂S(O)CF₃ CH₂CH₂S(O)₂Me
CH₂S(O)CF₃ D2-32a
CH₂S(O)CF₃ D2-33a
CH₂S(O)CF₃ D2-34a
CH₂S(O)CF₃ D2-37a
CH₂S(O)CF₃ D2-81a
CH₂S(O)CF₃ D2-82a
CH₂S(O)CF₃ D2-84a
CH₂S(O)CF₃ D2-85a
CH₂S(O)CF₃ D2-87a
CH₂S(O)CF₃ D2-92a
CH₂S(O)CF₃ D2-93a
CH₂S(O)CF₃ D2-95a
CH₂S(O)CF₃ D2-96a
CH₂S(O)CF₃ D2-98a
CH₂S(O)CF₃ D2-108a
CH₂S(O)CF₃ D2-108b(Z²=2-Cl)
CH₂S(O)CF₃ D2-108b(Z²=3-Me)
CH₂S(O)CF₃ D2-108b(Z²=4-OMe)
CH₂S(O)CF₃ D2-108b(Z²=2-SMe)
CH₂S(O)CF₃ D2-108b(Z²=3-CF₃)
CH₂S(O)CF₃ D2-108b(Z²=4-OCF₃)
CH₂S(O)CF₃ D2-108b(Z²=2-SCF₃)
CH₂S(O)CF₃ C(O)Me
CH₂S(O)CF₃ C(O)CF₃
CH₂S(O)CF₃ C(O)OMe
CH₂S(O)₂CF₃ Me
CH₂S(O)₂CF₃ Et
CH₂S(O)₂CF₃ Pr-n
CH₂S(O)₂CF₃ Pr-i
CH₂S(O)₂CF₃ Pr-c
CH₂S(O)₂CF₃ Bu-n
CH₂S(O)₂CF₃ Bu-i
CH₂S(O)₂CF₃ Bu-c
CH₂S(O)₂CF₃ Bu-s
CH₂S(O)₂CF₃ Bu-t
CH₂S(O)₂CF₃ Pen-n
CH₂S(O)₂CF₃ Pen-c
CH₂S(O)₂CF₃ Hex-n
CH₂S(O)₂CF₃ Hex-c
CH₂S(O)₂CF₃ CH₂Pr-c
CH₂S(O)₂CF₃ CH₂Bu-c
CH₂S(O)₂CF₃ CH₂Pen-c
CH₂S(O)₂CF₃ CH₂Hex-c
CH₂S(O)₂CF₃ CH₂CH=CH₂
CH₂S(O)₂CF₃ CH₂CH=C(Cl)₂
CH₂S(O)₂CF₃ CH₂C≡CH
CH₂S(O)₂CF₃ CH₂CN
CH₂S(O)₂CF₃ CH₂CF₃
CH₂S(O)₂CF₃ CH₂OMe
CH₂S(O)₂CF₃ CH₂OCF₃
CH₂S(O)₂CF₃ CH₂SMe
CH₂S(O)₂CF₃ CH₂S(O)Me
CH₂S(O)₂CF₃ CH₂S(O)₂Me
CH₂S(O)₂CF₃ CH₂SCF₃
CH₂S(O)₂CF₃ CH₂S(O)CF₃
CH₂S(O)₂CF₃ CH₂S(O)₂CF₃
CH₂S(O)₂CF₃ CH₂CH(OMe)₂
CH₂S(O)₂CF₃ CH₂CH(SMe)₂
CH₂S(O)₂CF₃ CH₂C(O)Me
CH₂S(O)₂CF₃ CH₂C(O)CF₃
CH₂S(O)₂CF₃ CH₂C(O)OMe
CH₂S(O)₂CF₃ CH₂(D2-32a)
CH₂S(O)₂CF₃ CH₂(D2-33a)
CH₂S(O)₂CF₃ CH₂(D2-34a)
CH₂S(O)₂CF₃ CH₂(D2-37a)
CH₂S(O)₂CF₃ CH₂(D2-81a)
CH₂S(O)₂CF₃ CH₂(D2-82a)
CH₂S(O)₂CF₃ CH₂(D2-84a)
CH₂S(O)₂CF₃ CH₂(D2-85a)
CH₂S(O)₂CF₃ CH₂(D2-87a)
CH₂S(O)₂CF₃ CH₂(D2-92a)
CH₂S(O)₂CF₃ CH₂(D2-93a)
CH₂S(O)₂CF₃ CH₂(D2-95a)
CH₂S(O)₂CF₃ CH₂(D2-96a)
CH₂S(O)₂CF₃ CH₂(D2-98a)
CH₂S(O)₂CF₃ CH₂(D2-108a)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=2-Cl)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=3-Me)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=4-OMe)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=2-SMe)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=3-CF₃)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=4-OCF₃)
CH₂S(O)₂CF₃ CH₂(D2-108b,Z²=2-SCF₃)
CH₂S(O)₂CF₃ CH₂CH₂CN
CH₂S(O)₂CF₃ CH₂CH₂CF₃
CH₂S(O)₂CF₃ CH₂CH₂OMe
CH₂S(O)₂CF₃ CH₂CH₂SMe
CH₂S(O)₂CF₃ CH₂CH₂S(O)Me
CH₂S(O)₂CF₃ CH₂CH₂S(O)₂Me
CH₂S(O)₂CF₃ D2-32a
CH₂S(O)₂CF₃ D2-33a
CH₂S(O)₂CF₃ D2-34a
CH₂S(O)₂CF₃ D2-37a
CH₂S(O)₂CF₃ D2-81a
CH₂S(O)₂CF₃ D2-82a
CH₂S(O)₂CF₃ D2-84a
CH₂S(O)₂CF₃ D2-85a
CH₂S(O)₂CF₃ D2-87a
CH₂S(O)₂CF₃ D2-92a
CH₂S(O)₂CF₃ D2-93a
CH₂S(O)₂CF₃ D2-95a
CH₂S(O)₂CF₃ D2-96a
CH₂S(O)₂CF₃ D2-98a
CH₂S(O)₂CF₃ D2-108a
CH₂S(O)₂CF₃ D2-108b(Z²=2-Cl)
CH₂S(O)₂CF₃ D2-108b(Z²=3-Me)
CH₂S(O)₂CF₃ D2-108b(Z²=4-OMe)
CH₂S(O)₂CF₃ D2-108b(Z²=2-SMe)
CH₂S(O)₂CF₃ D2-108b(Z²=3-CF₃)
CH₂S(O)₂CF₃ D2-108b(Z²=4-OCF₃)
CH₂S(O)₂CF₃ D2-108b(Z²=2-SCF₃)
CH₂S(O)₂CF₃ C(O)Me
CH₂S(O)₂CF₃ C(O)CF₃
CH₂S(O)₂CF₃ C(O)OMe
D2-32a Me
D2-32a Et
D2-32a Pr-n
D2-32a Pr-i
D2-32a Pr-c
D2-32a Bu-n
D2-32a Bu-i
D2-32a Bu-c
D2-32a Bu-s
D2-32a Bu-t
D2-32a Pen-n
D2-32a Pen-c
D2-32a Hex-n
D2-32a Hex-c
D2-32a CH₂Pr-c
D2-32a CH₂Bu-c
D2-32a CH₂Pen-c
D2-32a CH₂Hex-c
D2-32a CH₂CH=CH₂
D2-32a CH₂CH=C(Cl)₂
D2-32a CH₂C≡CH
D2-32a CH₂CN
D2-32a CH₂CF₃
D2-32a CH₂OMe
D2-32a CH₂OCF₃
D2-32a CH₂SMe
D2-32a CH₂S(O)Me
D2-32a CH₂S(O)₂Me
D2-32a CH₂SCF₃
D2-32a CH₂S(O)CF₃
D2-32a CH₂S(O)₂CF₃
D2-32a CH₂CH(OMe)₂
D2-32a CH₂CH(SMe)₂
D2-32a CH₂C(O)Me
D2-32a CH₂C(O)CF₃
D2-32a CH₂C(O)OMe
D2-32a CH₂(D2-32a)
D2-32a CH₂(D2-33a)
D2-32a CH₂(D2-34a)
D2-32a CH₂(D2-37a)
D2-32a CH₂(D2-81a)
D2-32a CH₂(D2-82a)
D2-32a CH₂(D2-84a)
D2-32a CH₂(D2-85a)
D2-32a CH₂(D2-87a)
D2-32a CH₂(D2-92a)
D2-32a CH₂(D2-93a)
D2-32a CH₂(D2-95a)
D2-32a CH₂(D2-96a)
D2-32a CH₂(D2-98a)
D2-32a CH₂(D2-108a)
D2-32a CH₂(D2-108b,Z²=2-Cl)
D2-32a CH₂(D2-108b,Z²=3-Me)
D2-32a CH₂(D2-108b,Z²=4-OMe)
D2-32a CH₂(D2-108b,Z²=2-SMe)
D2-32a CH₂(D2-108b,Z²=3-CF₃)
D2-32a CH₂(D2-108b,Z²=4-OCF₃)
D2-32a CH₂(D2-108b,Z²=2-SCF₃)
D2-32a CH₂CH₂CN
D2-32a CH₂CH₂CF₃
D2-32a CH₂CH₂OMe
D2-32a CH₂CH₂SMe
D2-32a CH₂CH₂S(O)Me
D2-32a CH₂CH₂S(O)₂Me
D2-32a D2-32a
D2-32a D2-33a
D2-32a D2-34a
D2-32a D2-37a
D2-32a D2-81a
D2-32a D2-82a
D2-32a D2-84a
D2-32a D2-85a
D2-32a D2-87a
D2-32a D2-92a
D2-32a D2-93a
D2-32a D2-95a
D2-32a D2-96a
D2-32a D2-98a
D2-32a D2-108a
D2-32a D2-108b(Z²=2-Cl)
D2-32a D2-108b(Z²=3-Me)
D2-32a D2-108b(Z²=4-OMe)
D2-32a D2-108b(Z²=2-SMe)
D2-32a D2-108b(Z²=3-CF₃)
D2-32a D2-108b(Z²=4-OCF₃)
D2-32a D2-108b(Z²=2-SCF₃)
D2-32a C(O)Me
D2-32a C(O)CF₃
D2-32a C(O)OMe
D2-33a Me
D2-33a Et
D2-33a Pr-n
D2-33a Pr-i
D2-33a Pr-c
D2-33a Bu-n
D2-33a Bu-i
D2-33a Bu-c
D2-33a Bu-s
D2-33a Bu-t
D2-33a Pen-n
D2-33a Pen-c
D2-33a Hex-n
D2-33a Hex-c
D2-33a CH₂Pr-c
D2-33a CH₂Bu-c
D2-33a CH₂Pen-c
D2-33a CH₂Hex-c
D2-33a CH₂CH=CH₂
D2-33a CH₂CH=C(Cl)₂
D2-33a CH₂C≡CH
D2-33a CH₂CN
D2-33a CH₂CF₃
D2-33a CH₂OMe
D2-33a CH₂OCF₃
D2-33a CH₂SMe
D2-33a CH₂S(O)Me
D2-33a CH₂S(O)₂Me
D2-33a CH₂SCF₃
D2-33a CH₂S(O)CF₃
D2-33a CH₂S(O)₂CF₃
D2-33a CH₂CH(OMe)₂
D2-33a CH₂CH(SMe)₂
D2-33a CH₂C(O)Me
D2-33a CH₂C(O)CF₃
D2-33a CH₂C(O)OMe
D2-33a CH₂(D2-32a)
D2-33a CH₂(D2-33a)
D2-33a CH₂(D2-34a)
D2-33a CH₂(D2-37a)
D2-33a CH₂(D2-81a)
D2-33a CH₂(D2-82a)
D2-33a CH₂(D2-84a)
D2-33a CH₂(D2-85a)
D2-33a CH₂(D2-87a)
D2-33a CH₂(D2-92a)
D2-33a CH₂(D2-93a)
D2-33a CH₂(D2-95a)
D2-33a CH₂(D2-96a)
D2-33a CH₂(D2-98a)
D2-33a CH₂(D2-108a)
D2-33a CH₂(D2-108b,Z²=2-Cl)
D2-33a CH₂(D2-108b,Z²=3-Me)
D2-33a CH₂(D2-108b,Z²=4-OMe)
D2-33a CH₂(D2-108b,Z²=2-SMe)
D2-33a CH₂(D2-108b,Z²=3-CF₃)
D2-33a CH₂(D2-108b,Z²=4-OCF₃)
D2-33a CH₂(D2-108b,Z²=2-SCF₃)
D2-33a CH₂CH₂CN
D2-33a CH₂CH₂CF₃
D2-33a CH₂CH₂OMe
D2-33a CH₂CH₂SMe
D2-33a CH₂CH₂S(O)Me
D2-33a CH₂CH₂S(O)₂Me
D2-33a D2-32a
D2-33a D2-33a
D2-33a D2-34a
D2-33a D2-37a
D2-33a D2-81a
D2-33a D2-82a
D2-33a D2-84a
D2-33a D2-85a
D2-33a D2-87a
D2-33a D2-92a
D2-33a D2-93a
D2-33a D2-95a
D2-33a D2-96a
D2-33a D2-98a
D2-33a D2-108a
D2-33a D2-108b(Z²=2-Cl)
D2-33a D2-108b(Z²=3-Me)
D2-33a D2-108b(Z²=4-OMe)
D2-33a D2-108b(Z²=2-SMe)
D2-33a D2-108b(Z²=3-CF₃)
D2-33a D2-108b(Z²=4-OCF₃)
D2-33a D2-108b(Z²=2-SCF₃)
D2-33a C(O)Me
D2-33a C(O)CF₃
D2-33a C(O)OMe
D2-34a Me
D2-34a Et
D2-34a Pr-n
D2-34a Pr-i
D2-34a Pr-c
D2-34a Bu-n
D2-34a Bu-i
D2-34a Bu-c
D2-34a Bu-s
D2-34a Bu-t
D2-34a Pen-n
D2-34a Pen-c
D2-34a Hex-n
D2-34a Hex-c
D2-34a CH₂Pr-c
D2-34a CH₂Bu-c
D2-34a CH₂Pen-c
D2-34a CH₂Hex-c
D2-34a CH₂CH=CH₂
D2-34a CH₂CH=C(Cl)₂
D2-34a CH₂C≡CH
D2-34a CH₂CN
D2-34a CH₂CF₃
D2-34a CH₂OMe
D2-34a CH₂OCF₃
D2-34a CH₂SMe
D2-34a CH₂S(O)Me
D2-34a CH₂S(O)₂Me
D2-34a CH₂SCF₃
D2-34a CH₂S(O)CF₃
D2-34a CH₂S(O)₂CF₃
D2-34a CH₂CH(OMe)₂
D2-34a CH₂CH(SMe)₂
D2-34a CH₂C(O)Me
D2-34a CH₂C(O)CF₃
D2-34a CH₂C(O)OMe
D2-34a CH₂(D2-32a)
D2-34a CH₂(D2-33a)
D2-34a CH₂(D2-34a)
D2-34a CH₂(D2-37a)
D2-34a CH₂(D2-81a)
D2-34a CH₂(D2-82a)
D2-34a CH₂(D2-84a)
D2-34a CH₂(D2-85a)
D2-34a CH₂(D2-87a)
D2-34a CH₂(D2-92a)
D2-34a CH₂(D2-93a)
D2-34a CH₂(D2-95a)
D2-34a CH₂(D2-96a)
D2-34a CH₂(D2-98a)
D2-34a CH₂(D2-108a)
D2-34a CH₂(D2-108b,Z²=2-Cl)
D2-34a CH₂(D2-108b,Z²=3-Me)
D2-34a CH₂(D2-108b,Z²=4-OMe)
D2-34a CH₂(D2-108b,Z²=2-SMe)
D2-34a CH₂(D2-108b,Z²=3-CF₃)
D2-34a CH₂(D2-108b,Z²=4-OCF₃)
D2-34a CH₂(D2-108b,Z²=2-SCF₃)
D2-34a CH₂CH₂CN
D2-34a CH₂CH₂CF₃
D2-34a CH₂CH₂OMe
D2-34a CH₂CH₂SMe
D2-34a CH₂CH₂S(O)Me
D2-34a CH₂CH₂S(O)₂Me
D2-34a D2-32a
D2-34a D2-33a
D2-34a D2-34a
D2-34a D2-37a
D2-34a D2-81a
D2-34a D2-82a
D2-34a D2-84a
D2-34a D2-85a
D2-34a D2-87a
D2-34a D2-92a
D2-34a D2-93a
D2-34a D2-95a
D2-34a D2-96a
D2-34a D2-98a
D2-34a D2-108a
D2-34a D2-108b(Z²=2-Cl)
D2-34a D2-108b(Z²=3-Me)
D2-34a D2-108b(Z²=4-OMe)
D2-34a D2-108b(Z²=2-SMe)
D2-34a D2-108b(Z²=3-CF₃)
D2-34a D2-108b(Z²=4-OCF₃)
D2-34a D2-108b(Z²=2-SCF₃)
D2-34a C(O)Me
D2-34a C(O)CF₃
D2-34a C(O)OMe
D2-37a Me
D2-37a Et
D2-37a Pr-n
D2-37a Pr-i
D2-37a Pr-c
D2-37a Bu-n
D2-37a Bu-i
D2-37a Bu-c
D2-37a Bu-s
D2-37a Bu-t
D2-37a Pen-n
D2-37a Pen-c
D2-37a Hex-n
D2-37a Hex-c
D2-37a CH₂Pr-c
D2-37a CH₂Bu-c
D2-37a CH₂Pen-c
D2-37a CH₂Hex-c
D2-37a CH₂CH=CH₂
D2-37a CH₂CH=C(Cl)₂
D2-37a CH₂C≡CH
D2-37a CH₂CN
D2-37a CH₂CF₃
D2-37a CH₂OMe
D2-37a CH₂OCF₃
D2-37a CH₂SMe
D2-37a CH₂S(O)Me
D2-37a CH₂S(O)₂Me
D2-37a CH₂SCF₃
D2-37a CH₂S(O)CF₃
D2-37a CH₂S(O)₂CF₃
D2-37a CH₂CH(OMe)₂
D2-37a CH₂CH(SMe)₂
D2-37a CH₂C(O)Me
D2-37a CH₂C(O)CF₃
D2-37a CH₂C(O)OMe
D2-37a CH₂(D2-32a)
D2-37a CH₂(D2-33a)
D2-37a CH₂(D2-34a)
D2-37a CH₂(D2-37a)
D2-37a CH₂(D2-81a)
D2-37a CH₂(D2-82a)
D2-37a CH₂(D2-84a)
D2-37a CH₂(D2-85a)
D2-37a CH₂(D2-87a)
D2-37a CH₂(D2-92a)
D2-37a CH₂(D2-93a)
D2-37a CH₂(D2-95a)
D2-37a CH₂(D2-96a)
D2-37a CH₂(D2-98a)
D2-37a CH₂(D2-108a)
D2-37a CH₂(D2-108b,Z²=2-Cl)
D2-37a CH₂(D2-108b,Z²=3-Me)
D2-37a CH₂(D2-108b,Z²=4-OMe)
D2-37a CH₂(D2-108b,Z²=2-SMe)
D2-37a CH₂(D2-108b,Z²=3-CF₃)
D2-37a CH₂(D2-108b,Z²=4-OCF₃)
D2-37a CH₂(D2-108b,Z²=2-SCF₃)
D2-37a CH₂CH₂CN
D2-37a CH₂CH₂CF₃
D2-37a CH₂CH₂OMe
D2-37a CH₂CH₂SMe
D2-37a CH₂CH₂S(O)Me
D2-37a CH₂CH₂S(O)₂Me
D2-37a D2-32a
D2-37a D2-33a
D2-37a D2-34a
D2-37a D2-37a
D2-37a D2-81a
D2-37a D2-82a
D2-37a D2-84a
D2-37a D2-85a
D2-37a D2-87a
D2-37a D2-92a
D2-37a D2-93a
D2-37a D2-95a
D2-37a D2-96a
D2-37a D2-98a
D2-37a D2-108a
D2-37a D2-108b(Z²=2-Cl)
D2-37a D2-108b(Z²=3-Me)
D2-37a D2-108b(Z²=4-OMe)
D2-37a D2-108b(Z²=2-SMe)
D2-37a D2-108b(Z²=3-CF₃)
D2-37a D2-108b(Z²=4-OCF₃)
D2-37a D2-108b(Z²=2-SCF₃)
D2-37a C(O)Me
D2-37a C(O)CF₃
D2-37a C(O)OMe
D2-81a Me
D2-81a Et
D2-81a Pr-n
D2-81a Pr-i
D2-81a Pr-c
D2-81a Bu-n
D2-81a Bu-i
D2-81a Bu-c
D2-81a Bu-s
D2-81a Bu-t
D2-81a Pen-n
D2-81a Pen-c
D2-81a Hex-n
D2-81a Hex-c
D2-81a CH₂Pr-c
D2-81a CH₂Bu-c
D2-81a CH₂Pen-c
D2-81a CH₂Hex-c
D2-81a CH₂CH=CH₂
D2-81a CH₂CH=C(Cl)₂
D2-81a CH₂C≡CH
D2-81a CH₂CN
D2-81a CH₂CF₃
D2-81a CH₂OMe
D2-81a CH₂OCF₃
D2-81a CH₂SMe
D2-81a CH₂S(O)Me
D2-81a CH₂S(O)₂Me
D2-81a CH₂SCF₃
D2-81a CH₂S(O)CF₃
D2-81a CH₂S(O)₂CF₃
D2-81a CH₂CH(OMe)₂
D2-81a CH₂CH(SMe)₂
D2-81a CH₂C(O)Me
D2-81a CH₂C(O)CF₃
D2-81a CH₂C(O)OMe
D2-81a CH₂(D2-32a)
D2-81a CH₂(D2-33a)
D2-81a CH₂(D2-34a)
D2-81a CH₂(D2-37a)
D2-81a CH₂(D2-81a)
D2-81a CH₂(D2-82a)
D2-81a CH₂(D2-84a)
D2-81a CH₂(D2-85a)
D2-81a CH₂(D2-87a)
D2-81a CH₂(D2-92a)
D2-81a CH₂(D2-93a)
D2-81a CH₂(D2-95a)
D2-81a CH₂(D2-96a)
D2-81a CH₂(D2-98a)
D2-81a CH₂(D2-108a)
D2-81a CH₂(D2-108b,Z²=2-Cl)
D2-81a CH₂(D2-108b,Z²=3-Me)
D2-81a CH₂(D2-108b,Z²=4-OMe)
D2-81a CH₂(D2-108b,Z²=2-SMe)
D2-81a CH₂(D2-108b,Z²=3-CF₃)
D2-81a CH₂(D2-108b,Z²=4-OCF₃)
D2-81a CH₂(D2-108b,Z²=2-SCF₃)
D2-81a CH₂CH₂CN
D2-81a CH₂CH₂CF₃
D2-81a CH₂CH₂OMe
D2-81a CH₂CH₂SMe
D2-81a CH₂CH₂S(O)Me
D2-81a CH₂CH₂S(O)₂Me
D2-81a D2-32a
D2-81a D2-33a
D2-81a D2-34a
D2-81a D2-37a
D2-81a D2-81a
D2-81a D2-82a
D2-81a D2-84a
D2-81a D2-85a
D2-81a D2-87a
D2-81a D2-92a
D2-81a D2-93a
D2-81a D2-95a
D2-81a D2-96a
D2-81a D2-98a
D2-81a D2-108a
D2-81a D2-108b(Z²=2-Cl)
D2-81a D2-108b(Z²=3-Me)
D2-81a D2-108b(Z²=4-OMe)
D2-81a D2-108b(Z²=2-SMe)
D2-81a D2-108b(Z²=3-CF₃)
D2-81a D2-108b(Z²=4-OCF₃)
D2-81a D2-108b(Z²=2-SCF₃)
D2-81a C(O)Me
D2-81a C(O)CF₃
D2-81a C(O)OMe
D2-82a Me
D2-82a Et
D2-82a Pr-n
D2-82a Pr-i
D2-82a Pr-c
D2-82a Bu-n
D2-82a Bu-i
D2-82a Bu-c
D2-82a Bu-s
D2-82a Bu-t
D2-82a Pen-n
D2-82a Pen-c
D2-82a Hex-n
D2-82a Hex-c
D2-82a CH₂Pr-c
D2-82a CH₂Bu-c
D2-82a CH₂Pen-c
D2-82a CH₂Hex-c
D2-82a CH₂CH=CH₂
D2-82a CH₂CH=C(Cl)₂
D2-82a CH₂C≡CH
D2-82a CH₂CN
D2-82a CH₂CF₃
D2-82a CH₂OMe
D2-82a CH₂OCF₃
D2-82a CH₂SMe
D2-82a CH₂S(O)Me
D2-82a CH₂S(O)₂Me
D2-82a CH₂SCF₃
D2-82a CH₂S(O)CF₃
D2-82a CH₂S(O)₂CF₃
D2-82a CH₂CH(OMe)₂
D2-82a CH₂CH(SMe)₂
D2-82a CH₂C(O)Me
D2-82a CH₂C(O)CF₃
D2-82a CH₂C(O)OMe
D2-82a CH₂(D2-32a)
D2-82a CH₂(D2-33a)
D2-82a CH₂(D2-34a)
D2-82a CH₂(D2-37a)
D2-82a CH₂(D2-81a)
D2-82a CH₂(D2-82a)
D2-82a CH₂(D2-84a)
D2-82a CH₂(D2-85a)
D2-82a CH₂(D2-87a)
D2-82a CH₂(D2-92a)
D2-82a CH₂(D2-93a)
D2-82a CH₂(D2-95a)
D2-82a CH₂(D2-96a)
D2-82a CH₂(D2-98a)
D2-82a CH₂(D2-108a)
D2-82a CH₂(D2-108b,Z²=2-Cl)
D2-82a CH₂(D2-108b,Z²=3-Me)
D2-82a CH₂(D2-108b,Z²=4-OMe)
D2-82a CH₂(D2-108b,Z²=2-SMe)
D2-82a CH₂(D2-108b,Z²=3-CF₃)
D2-82a CH₂(D2-108b,Z²=4-OCF₃)
D2-82a CH₂(D2-108b,Z²=2-SCF₃)
D2-82a CH₂CH₂CN
D2-82a CH₂CH₂CF₃
D2-82a CH₂CH₂OMe
D2-82a CH₂CH₂SMe
D2-82a CH₂CH₂S(O)Me
D2-82a CH₂CH₂S(O)₂Me
D2-82a D2-32a
D2-82a D2-33a
D2-82a D2-34a
D2-82a D2-37a
D2-82a D2-81a
D2-82a D2-82a
D2-82a D2-84a
D2-82a D2-85a
D2-82a D2-87a
D2-82a D2-92a
D2-82a D2-93a
D2-82a D2-95a
D2-82a D2-96a
D2-82a D2-98a
D2-82a D2-108a
D2-82a D2-108b(Z²=2-Cl)
D2-82a D2-108b(Z²=3-Me)
D2-82a D2-108b(Z²=4-OMe)
D2-82a D2-108b(Z²=2-SMe)
D2-82a D2-108b(Z²=3-CF₃)
D2-82a D2-108b(Z²=4-OCF₃)
D2-82a D2-108b(Z²=2-SCF₃)
D2-82a C(O)Me
D2-82a C(O)CF₃
D2-82a C(O)OMe
D2-84a Me
D2-84a Et
D2-84a Pr-n
D2-84a Pr-i
D2-84a Pr-c
D2-84a Bu-n
D2-84a Bu-i
D2-84a Bu-c
D2-84a Bu-s
D2-84a Bu-t
D2-84a Pen-n
D2-84a Pen-c
D2-84a Hex-n
D2-84a Hex-c
D2-84a CH₂Pr-c
D2-84a CH₂Bu-c
D2-84a CH₂Pen-c
D2-84a CH₂Hex-c
D2-84a CH₂CH=CH₂
D2-84a CH₂CH=C(Cl)₂
D2-84a CH₂C≡CH
D2-84a CH₂CN
D2-84a CH₂CF₃
D2-84a CH₂OMe
D2-84a CH₂OCF₃
D2-84a CH₂SMe
D2-84a CH₂S(O)Me
D2-84a CH₂S(O)₂Me
D2-84a CH₂SCF₃
D2-84a CH₂S(O)CF₃
D2-84a CH₂S(O)₂CF₃
D2-84a CH₂CH(OMe)₂
D2-84a CH₂CH(SMe)₂
D2-84a CH₂C(O)Me
D2-84a CH₂C(O)CF₃
D2-84a CH₂C(O)OMe
D2-84a CH₂(D2-32a)
D2-84a CH₂(D2-33a)
D2-84a CH₂(D2-34a)
D2-84a CH₂(D2-37a)
D2-84a CH₂(D2-81a)
D2-84a CH₂(D2-82a)
D2-84a CH₂(D2-84a)
D2-84a CH₂(D2-85a)
D2-84a CH₂(D2-87a)
D2-84a CH₂(D2-92a)
D2-84a CH₂(D2-93a)
D2-84a CH₂(D2-95a)
D2-84a CH₂(D2-96a)
D2-84a CH₂(D2-98a)
D2-84a CH₂(D2-108a)
D2-84a CH₂(D2-108b,Z²=2-Cl)
D2-84a CH₂(D2-108b,Z²=3-Me)
D2-84a CH₂(D2-108b,Z²=4-OMe)
D2-84a CH₂(D2-108b,Z=²2-SMe)
D2-84a CH₂(D2-108b,Z²=3-CF₃)
D2-84a CH₂(D2-108b,Z²=4-OCF₃)
D2-84a CH₂(D2-108b,Z²=2-SCF₃)
D2-84a CH₂CH₂CN
D2-84a CH₂CH₂CF₃
D2-84a CH₂CH₂OMe
D2-84a CH₂CH₂SMe
D2-84a CH₂CH₂S(O)Me
D2-84a CH₂CH₂S(O)₂Me
D2-84a D2-32a
D2-84a D2-33a
D2-84a D2-34a
D2-84a D2-37a
D2-84a D2-81a
D2-84a D2-82a
D2-84a D2-84a
D2-84a D2-85a
D2-84a D2-87a
D2-84a D2-92a
D2-84a D2-93a
D2-84a D2-95a
D2-84a D2-96a
D2-84a D2-98a
D2-84a D2-108a
D2-84a D2-108b(Z²=2-Cl)
D2-84a D2-108b(Z²=3-Me)
D2-84a D2-108b(Z²=4-OMe)
D2-84a D2-108b(Z²=2-SMe)
D2-84a D2-108b(Z²=3-CF₃)
D2-84a D2-108b(Z²=4-OCF₃)
D2-84a D2-108b(Z²=2-SCF₃)
D2-84a C(O)Me
D2-84a C(O)CF₃
D2-84a C(O)OMe
D2-85a Me
D2-85a Et
D2-85a Pr-n
D2-85a Pr-i
D2-85a Pr-c
D2-85a Bu-n
D2-85a Bu-i
D2-85a Bu-c
D2-85a Bu-s
D2-85a Bu-t
D2-85a Pen-n
D2-85a Pen-c
D2-85a Hex-n
D2-85a Hex-c
D2-85a CH₂Pr-c
D2-85a CH₂Bu-c
D2-85a CH₂Pen-c
D2-85a CH₂Hex-c
D2-85a CH₂CH=CH₂
D2-85a CH₂CH=C(Cl)₂
D2-85a CH₂C≡CH
D2-85a CH₂CN
D2-85a CH₂CF₃
D2-85a CH₂OMe
D2-85a CH₂OCF₃
D2-85a CH₂SMe
D2-85a CH₂S(O)Me
D2-85a CH₂S(O)₂Me
D2-85a CH₂SCF₃
D2-85a CH₂S(O)CF₃
D2-85a CH₂S(O)₂CF₃
D2-85a CH₂CH(OMe)₂
D2-85a CH₂CH(SMe)₂
D2-85a CH₂C(O)Me
D2-85a CH₂C(O)CF₃
D2-85a CH₂C(O)OMe
D2-85a CH₂(D2-32a)
D2-85a CH₂(D2-33a)
D2-85a CH₂(D2-34a)
D2-85a CH₂(D2-37a)
D2-85a CH₂(D2-81a)
D2-85a CH₂(D2-82a)
D2-85a CH₂(D2-84a)
D2-85a CH₂(D2-85a)
D2-85a CH₂(D2-87a)
D2-85a CH₂(D2-92a)
D2-85a CH₂(D2-93a)
D2-85a CH₂(D2-95a)
D2-85a CH₂(D2-96a)
D2-85a CH₂(D2-98a)
D2-85a CH₂(D2-108a)
D2-85a CH₂(D2-108b,Z²=2-Cl)
D2-85a CH₂(D2-108b,Z²=3-Me)
D2-85a CH₂(D2-108b,Z²=4-OMe)
D2-85a CH₂(D2-108b,Z²=2-SMe)
D2-85a CH₂(D2-108b,Z²=3-CF₃)
D2-85a CH₂(D2-108b,Z²=4-OCF₃)
D2-85a CH₂(D2-108b,Z²=2-SCF₃)
D2-85a CH₂CH₂CN
D2-85a CH₂CH₂CF₃
D2-85a CH₂CH₂OMe
D2-85a CH₂CH₂SMe
D2-85a CH₂CH₂S(O)Me
D2-85a CH₂CH₂S(O)₂Me
D2-85a D2-32a
D2-85a D2-33a
D2-85a D2-34a
D2-85a D2-37a
D2-85a D2-81a
D2-85a D2-82a
D2-85a D2-84a
D2-85a D2-85a
D2-85a D2-87a
D2-85a D2-92a
D2-85a D2-93a
D2-85a D2-95a
D2-85a D2-96a
D2-85a D2-98a
D2-85a D2-108a
D2-85a D2-108b(Z²=2-Cl)
D2-85a D2-108b(Z²=3-Me)
D2-85a D2-108b(Z²=4-OMe)
D2-85a D2-108b(Z²=2-SMe)
D2-85a D2-108b(Z²=3-CF₃)
D2-85a D2-108b(Z²=4-OCF₃)
D2-85a D2-108b(Z²=2-SCF₃)
D2-85a C(O)Me
D2-85a C(O)CF₃
D2-85a C(O)OMe
D2-87a Me
D2-87a Et
D2-87a Pr-n
D2-87a Pr-i
D2-87a Pr-c
D2-87a Bu-n
D2-87a Bu-i
D2-87a Bu-c
D2-87a Bu-s
D2-87a Bu-t
D2-87a Pen-n
D2-87a Pen-c
D2-87a Hex-n
D2-87a Hex-c
D2-87a CH₂Pr-c
D2-87a CH₂Bu-c
D2-87a CH₂Pen-c
D2-87a CH₂Hex-c
D2-87a CH₂CH=CH₂
D2-87a CH₂CH=C(Cl)₂
D2-87a CH₂C≡CH
D2-87a CH₂CN
D2-87a CH₂CF₃
D2-87a CH₂OMe
D2-87a CH₂OCF₃
D2-87a CH₂SMe
D2-87a CH₂S(O)Me
D2-87a CH₂S(O)₂Me
D2-87a CH₂SCF₃
D2-87a CH₂S(O)CF₃
D2-87a CH₂S(O)₂CF₃
D2-87a CH₂CH(OMe)₂
D2-87a CH₂CH(SMe)₂
D2-87a CH₂C(O)Me
D2-87a CH₂C(O)CF₃
D2-87a CH₂C(O)OMe
D2-87a CH₂(D2-32a)
D2-87a CH₂(D2-33a)
D2-87a CH₂(D2-34a)
D2-87a CH₂(D2-37a)
D2-87a CH₂(D2-81a)
D2-87a CH₂(D2-82a)
D2-87a CH₂(D2-84a)
D2-87a CH₂(D2-85a)
D2-87a CH₂(D2-87a)
D2-87a CH₂(D2-92a)
D2-87a CH₂(D2-93a)
D2-87a CH₂(D2-95a)
D2-87a CH₂(D2-96a)
D2-87a CH₂(D2-98a)
D2-87a CH₂(D2-108a)
D2-87a CH₂(D2-108b,Z²=2-Cl)
D2-87a CH₂(D2-108b,Z²=3-Me)
D2-87a CH₂(D2-108b,Z²=4-OMe)
D2-87a CH₂(D2-108b,Z²=2-SMe)
D2-87a CH₂(D2-108b,Z²=3-CF₃)
D2-87a CH₂(D2-108b,Z²=4-OCF₃)
D2-87a CH₂(D2-108b,Z²=2-SCF₃)
D2-87a CH₂CH₂CN
D2-87a CH₂CH₂CF₃
D2-87a CH₂CH₂OMe
D2-87a CH₂CH₂SMe
D2-87a CH₂CH₂S(O)Me
D2-87a CH₂CH₂S(O)₂Me
D2-87a D2-32a
D2-87a D2-33a
D2-87a D2-34a
D2-87a D2-37a
D2-87a D2-81a
D2-87a D2-82a
D2-87a D2-84a
D2-87a D2-85a
D2-87a D2-87a
D2-87a D2-92a
D2-87a D2-93a
D2-87a D2-95a
D2-87a D2-96a
D2-87a D2-98a
D2-87a D2-108a
D2-87a D2-108b(Z²=2-Cl)
D2-87a D2-108b(Z²=3-Me)
D2-87a D2-108b(Z²=4-OMe)
D2-87a D2-108b(Z²=2-SMe)
D2-87a D2-108b(Z²=3-CF₃)
D2-87a D2-108b(Z²=4-OCF₃)
D2-87a D2-108b(Z²=2-SCF₃)
D2-87a C(O)Me
D2-87a C(O)CF₃
D2-87a C(O)OMe
D2-92a Me
D2-92a Et
D2-92a Pr-n
D2-92a Pr-i
D2-92a Pr-c
D2-92a Bu-n
D2-92a Bu-i
D2-92a Bu-c
D2-92a Bu-s
D2-92a Bu-t
D2-92a Pen-n
D2-92a Pen-c
D2-92a Hex-n
D2-92a Hex-c
D2-92a CH₂Pr-c
D2-92a CH₂Bu-c
D2-92a CH₂Pen-c
D2-92a CH₂Hex-c
D2-92a CH₂CH=CH₂
D2-92a CH₂CH=C(Cl)₂
D2-92a CH₂C≡CH
D2-92a CH₂CN
D2-92a CH₂CF₃
D2-92a CH₂OMe
D2-92a CH₂OCF₃
D2-92a CH₂SMe
D2-92a CH₂S(O)Me
D2-92a CH₂S(O)₂Me
D2-92a CH₂SCF₃
D2-92a CH₂S(O)CF₃
D2-92a CH₂S(O)₂CF₃
D2-92a CH₂CH(OMe)₂
D2-92a CH₂CH(SMe)₂
D2-92a CH₂C(O)Me
D2-92a CH₂C(O)CF₃
D2-92a CH₂C(O)OMe
D2-92a CH₂(D2-32a)
D2-92a CH₂(D2-33a)
D2-92a CH₂(D2-34a)
D2-92a CH₂(D2-37a)
D2-92a CH₂(D2-81a)
D2-92a CH₂(D2-82a)
D2-92a CH₂(D2-84a)
D2-92a CH₂(D2-85a)
D2-92a CH₂(D2-87a)
D2-92a CH₂(D2-92a)
D2-92a CH₂(D2-93a)
D2-92a CH₂(D2-95a)
D2-92a CH₂(D2-96a)
D2-92a CH₂(D2-98a)
D2-92a CH₂(D2-108a)
D2-92a CH₂(D2-108b,Z²=2-Cl)
D2-92a CH₂(D2-108b,Z²=3-Me)
D2-92a CH₂(D2-108b,Z²=4-OMe)
D2-92a CH₂(D2-108b,Z²=2-SMe)
D2-92a CH₂(D2-108b,Z²=3-CF₃)
D2-92a CH₂(D2-108b,Z²=4-OCF₃)
D2-92a CH₂(D2-108b,Z²=2-SCF₃)
D2-92a CH₂CH₂CN
D2-92a CH₂CH₂CF₃
D2-92a CH₂CH₂OMe
D2-92a CH₂CH₂SMe
D2-92a CH₂CH₂S(O)Me
D2-92a CH₂CH₂S(O)₂Me
D2-92a D2-32a
D2-92a D2-33a
D2-92a D2-34a
D2-92a D2-37a
D2-92a D2-81a
D2-92a D2-82a
D2-92a D2-84a
D2-92a D2-85a
D2-92a D2-87a
D2-92a D2-92a
D2-92a D2-93a
D2-92a D2-95a
D2-92a D2-96a
D2-92a D2-98a
D2-92a D2-108a
D2-92a D2-108b(Z²=2-Cl)
D2-92a D2-108b(Z²=3-Me)
D2-92a D2-108b(Z²=4-OMe)
D2-92a D2-108b(Z²=2-SMe)
D2-92a D2-108b(Z²=3-CF₃)
D2-92a D2-108b(Z²=4-OCF₃)
D2-92a D2-108b(Z²=2-SCF₃)
D2-92a C(O)Me
D2-92a C(O)CF₃
D2-92a C(O)OMe
D2-93a Me
D2-93a Et
D2-93a Pr-n
D2-93a Pr-i
D2-93a Pr-c
D2-93a Bu-n
D2-93a Bu-i
D2-93a Bu-c
D2-93a Bu-s
D2-93a Bu-t
D2-93a Pen-n
D2-93a Pen-c
D2-93a Hex-n
D2-93a Hex-c
D2-93a CH₂Pr-c
D2-93a CH₂Bu-c
D2-93a CH₂Pen-c
D2-93a CH₂Hex-c
D2-93a CH₂CH=CH₂
D2-93a CH₂CH=C(Cl)₂
D2-93a CH₂C≡CH
D2-93a CH₂CN
D2-93a CH₂CF₃
D2-93a CH₂OMe
D2-93a CH₂OCF₃
D2-93a CH₂SMe
D2-93a CH₂S(O)Me
D2-93a CH₂S(O)₂Me
D2-93a CH₂SCF₃
D2-93a CH₂S(O)CF₃
D2-93a CH₂S(O)₂CF₃
D2-93a CH₂CH(OMe)₂
D2-93a CH₂CH(SMe)₂
D2-93a CH₂C(O)Me
D2-93a CH₂C(O)CF₃
D2-93a CH₂C(O)OMe
D2-93a CH₂(D2-32a)
D2-93a CH₂(D2-33a)
D2-93a CH₂(D2-34a)
D2-93a CH₂(D2-37a)
D2-93a CH₂(D2-81a)
D2-93a CH₂(D2-82a)
D2-93a CH₂(D2-84a)
D2-93a CH₂(D2-85a)
D2-93a CH₂(D2-87a)
D2-93a CH₂(D2-92a)
D2-93a CH₂(D2-93a)
D2-93a CH₂(D2-95a)
D2-93a CH₂(D2-96a)
D2-93a CH₂(D2-98a)
D2-93a CH₂(D2-108a)
D2-93a CH₂(D2-108b,Z²=2-Cl)
D2-93a CH₂(D2-108b,Z²=3-Me)
D2-93a CH₂(D2-108b,Z²=4-OMe)
D2-93a CH₂(D2-108b,Z²=2-SMe)
D2-93a CH₂(D2-108b,Z²=3-CF₃)
D2-93a CH₂(D2-108b,Z²=4-OCF₃)
D2-93a CH₂(D2-108b,Z²=2-SCF₃)
D2-93a CH₂CH₂CN
D2-93a CH₂CH₂CF₃
D2-93a CH₂CH₂OMe
D2-93a CH₂CH₂SMe
D2-93a CH₂CH₂S(O)Me
D2-93a CH₂CH₂S(O)₂Me
D2-93a D2-32a
D2-93a D2-33a
D2-93a D2-34a
D2-93a D2-37a
D2-93a D2-81a
D2-93a D2-82a
D2-93a D2-84a
D2-93a D2-85a
D2-93a D2-87a
D2-93a D2-92a
D2-93a D2-93a
D2-93a D2-95a
D2-93a D2-96a
D2-93a D2-98a
D2-93a D2-108a
D2-93a D2-108b(Z²=2-Cl)
D2-93a D2-108b(Z²=3-Me)
D2-93a D2-108b(Z²=4-OMe)
D2-93a D2-108b(Z²=2-SMe)
D2-93a D2-108b(Z²=3-CF₃)
D2-93a D2-108b(Z²=4-OCF₃)
D2-93a D2-108b(Z²=2-SCF₃)
D2-93a C(O)Me
D2-93a C(O)CF₃
D2-93a C(O)OMe
D2-95a Me
D2-95a Et
D2-95a Pr-n
D2-95a Pr-i
D2-95a Pr-c
D2-95a Bu-n
D2-95a Bu-i
D2-95a Bu-c
D2-95a Bu-s
D2-95a Bu-t
D2-95a Pen-n
D2-95a Pen-c
D2-95a Hex-n
D2-95a Hex-c
D2-95a CH₂Pr-c
D2-95a CH₂Bu-c
D2-95a CH₂Pen-c
D2-95a CH₂Hex-c
D2-95a CH₂CH=CH₂
D2-95a CH₂CH=C(Cl)₂
D2-95a CH₂C≡CH
D2-95a CH₂CN
D2-95a CH₂CF₃
D2-95a CH₂OMe
D2-95a CH₂OCF₃
D2-95a CH₂SMe
D2-95a CH₂S(O)Me
D2-95a CH₂S(O)₂Me
D2-95a CH₂SCF₃
D2-95a CH₂S(O)CF₃
D2-95a CH₂S(O)₂CF₃
D2-95a CH₂CH(OMe)₂
D2-95a CH₂CH(SMe)₂
D2-95a CH₂C(O)Me
D2-95a CH₂C(O)CF₃
D2-95a CH₂C(O)OMe
D2-95a CH₂(D2-32a)
D2-95a CH₂(D2-33a)
D2-95a CH₂(D2-34a)
D2-95a CH₂(D2-37a)
D2-95a CH₂(D2-81a)
D2-95a CH₂(D2-82a)
D2-95a CH₂(D2-84a)
D2-95a CH₂(D2-85a)
D2-95a CH₂(D2-87a)
D2-95a CH₂(D2-92a)
D2-95a CH₂(D2-93a)
D2-95a CH₂(D2-95a)
D2-95a CH₂(D2-96a)
D2-95a CH₂(D2-98a)
D2-95a CH₂(D2-108a)
D2-95a CH₂(D2-108b,Z²=2-Cl)
D2-95a CH₂(D2-108b,Z²=3-Me)
D2-95a CH₂(D2-108b,Z²=4-OMe)
D2-95a CH₂(D2-108b,Z²=2-SMe)
D2-95a CH₂(D2-108b,Z²=3-CF₃)
D2-95a CH₂(D2-108b,Z²=4-OCF₃)
D2-95a CH₂(D2-108b,Z²=2-SCF₃)
D2-95a CH₂CH₂CN
D2-95a CH₂CH₂CF₃
D2-95a CH₂CH₂OMe
D2-95a CH₂CH₂SMe
D2-95a CH₂CH₂S(O)Me
D2-95a CH₂CH₂S(O)₂Me
D2-95a D2-32a
D2-95a D2-33a
D2-95a D2-34a
D2-95a D2-37a
D2-95a D2-81a
D2-95a D2-82a
D2-95a D2-84a
D2-95a D2-85a
D2-95a D2-87a
D2-95a D2-92a
D2-95a D2-93a
D2-95a D2-95a
D2-95a D2-96a
D2-95a D2-98a
D2-95a D2-108a
D2-95a D2-108b(Z²=2-Cl)
D2-95a D2-108b(Z²=3-Me)
D2-95a D2-108b(Z²=4-OMe)
D2-95a D2-108b(Z²=2-SMe)
D2-95a D2-108b(Z²=3-CF₃)
D2-95a D2-108b(Z²=4-OCF₃)
D2-95a D2-108b(Z²=2-SCF₃)
D2-95a C(O)Me
D2-95a C(O)CF₃
D2-95a C(O)OMe
D2-96a Me
D2-96a Et
D2-96a Pr-n
D2-96a Pr-i
D2-96a Pr-c
D2-96a Bu-n
D2-96a Bu-i
D2-96a Bu-c
D2-96a Bu-s
D2-96a Bu-t
D2-96a Pen-n
D2-96a Pen-c
D2-96a Hex-n
D2-96a Hex-c
D2-96a CH₂Pr-c
D2-96a CH₂Bu-c
D2-96a CH₂Pen-c
D2-96a CH₂Hex-c
D2-96a CH₂CH=CH₂
D2-96a CH₂CH=C(Cl)₂
D2-96a CH₂C≡CH
D2-96a CH₂CN
D2-96a CH₂CF₃
D2-96a CH₂OMe
D2-96a CH₂OCF₃
D2-96a CH₂SMe
D2-96a CH₂S(O)Me
D2-96a CH₂S(O)₂Me
D2-96a CH₂SCF₃
D2-96a CH₂S(O)CF₃
D2-96a CH₂S(O)₂CF₃
D2-96a CH₂CH(OMe)₂
D2-96a CH₂CH(SMe)₂
D2-96a CH₂C(O)Me
D2-96a CH₂C(O)CF₃
D2-96a CH₂C(O)OMe
D2-96a CH₂(D2-32a)
D2-96a CH₂(D2-33a)
D2-96a CH₂(D2-34a)
D2-96a CH₂(D2-37a)
D2-96a CH₂(D2-81a)
D2-96a CH₂(D2-82a)
D2-96a CH₂(D2-84a)
D2-96a CH₂(D2-85a)
D2-96a CH₂(D2-87a)
D2-96a CH₂(D2-92a)
D2-96a CH₂(D2-93a)
D2-96a CH₂(D2-95a)
D2-96a CH₂(D2-96a)
D2-96a CH₂(D2-98a)
D2-96a CH₂(D2-108a)
D2-96a CH₂(D2-108b,Z²=2-Cl)
D2-96a CH₂(D2-108b,Z²=3-Me)
D2-96a CH₂(D2-108b,Z²=4-OMe)
D2-96a CH₂(D2-108b,Z²=2-SMe)
D2-96a CH₂(D2-108b,Z²=3-CF₃)
D2-96a CH₂(D2-108b,Z²=4-OCF₃)
D2-96a CH₂(D2-108b,Z²=2-SCF₃)
D2-96a CH₂CH₂CN
D2-96a CH₂CH₂CF₃
D2-96a CH₂CH₂OMe
D2-96a CH₂CH₂SMe
D2-96a CH₂CH₂S(O)Me
D2-96a CH₂CH₂S(O)₂Me
D2-96a D2-32a
D2-96a D2-33a
D2-96a D2-34a
D2-96a D2-37a
D2-96a D2-81a
D2-96a D2-82a
D2-96a D2-84a
D2-96a D2-85a
D2-96a D2-87a
D2-96a D2-92a
D2-96a D2-93a
D2-96a D2-95a
D2-96a D2-96a
D2-96a D2-98a
D2-96a D2-108a
D2-96a D2-108b(Z²=2-Cl)
D2-96a D2-108b(Z²=3-Me)
D2-96a D2-108b(Z²=4-OMe)
D2-96a D2-108b(Z²=2-SMe)
D2-96a D2-108b(Z²=3-CF₃)
D2-96a D2-108b(Z²=4-OCF₃)
D2-96a D2-108b(Z²=2-SCF₃)
D2-96a C(O)Me
D2-96a C(O)CF₃
D2-96a C(O)OMe
D2-98a Me
D2-98a Et
D2-98a Pr-n
D2-98a Pr-i
D2-98a Pr-c
D2-98a Bu-n
D2-98a Bu-i
D2-98a Bu-c
D2-98a Bu-s
D2-98a Bu-t
D2-98a Pen-n
D2-98a Pen-c
D2-98a Hex-n
D2-98a Hex-c
D2-98a CH₂Pr-c
D2-98a CH₂Bu-c
D2-98a CH₂Pen-c
D2-98a CH₂Hex-c
D2-98a CH₂CH=CH₂
D2-98a CH₂CH=C(Cl)₂
D2-98a CH₂C≡CH
D2-98a CH₂CN
D2-98a CH₂CF₃
D2-98a CH₂OMe
D2-98a CH₂OCF₃
D2-98a CH₂SMe
D2-98a CH₂S(O)Me
D2-98a CH₂S(O)₂Me
D2-98a CH₂SCF₃
D2-98a CH₂S(O)CF₃
D2-98a CH₂S(O)₂CF₃
D2-98a CH₂CH(OMe)₂
D2-98a CH₂CH(SMe)₂
D2-98a CH₂C(O)Me
D2-98a CH₂C(O)CF₃
D2-98a CH₂C(O)OMe
D2-98a CH₂(D2-32a)
D2-98a CH₂(D2-33a)
D2-98a CH₂(D2-34a)
D2-98a CH₂(D2-37a)
D2-98a CH₂(D2-81a)
D2-98a CH₂(D2-82a)
D2-98a CH₂(D2-84a)
D2-98a CH₂(D2-85a)
D2-98a CH₂(D2-87a)
D2-98a CH₂(D2-92a)
D2-98a CH₂(D2-93a)
D2-98a CH₂(D2-95a)
D2-98a CH₂(D2-96a)
D2-98a CH₂(D2-98a)
D2-98a CH₂(D2-108a)
D2-98a CH₂(D2-108b,Z²=2-Cl)
D2-98a CH₂(D2-108b,Z²=3-Me)
D2-98a CH₂(D2-108b,Z²=4-OMe)
D2-98a CH₂(D2-108b,Z²=2-SMe)
D2-98a CH₂(D2-108b,Z²=3-CF₃)
D2-98a CH₂(D2-108b,Z²=4-OCF₃)
D2-98a CH₂(D2-108b,Z²=2-SCF₃)
D2-98a CH₂CH₂CN
D2-98a CH₂CH₂CF₃
D2-98a CH₂CH₂OMe
D2-98a CH₂CH₂SMe
D2-98a CH₂CH₂S(O)Me
D2-98a CH₂CH₂S(O)₂Me
D2-98a D2-32a
D2-98a D2-33a
D2-98a D2-34a
D2-98a D2-37a
D2-98a D2-81a
D2-98a D2-82a
D2-98a D2-84a
D2-98a D2-85a
D2-98a D2-87a
D2-98a D2-92a
D2-98a D2-93a
D2-98a D2-95a
D2-98a D2-96a
D2-98a D2-98a
D2-98a D2-108a
D2-98a D2-108b(Z²=2-Cl)
D2-98a D2-108b(Z²=3-Me)
D2-98a D2-108b(Z²=4-OMe)
D2-98a D2-108b(Z²=2-SMe)
D2-98a D2-108b(Z²=3-CF₃)
D2-98a D2-108b(Z²=4-OCF₃)
D2-98a D2-108b(Z²=2-SCF₃)
D2-98a C(O)Me
D2-98a C(O)CF₃
D2-98a C(O)OMe
D2-108a Me
D2-108a Et
D2-108a Pr-n
D2-108a Pr-i
D2-108a Pr-c
D2-108a Bu-n
D2-108a Bu-i
D2-108a Bu-c
D2-108a Bu-s
D2-108a Bu-t
D2-108a Pen-n
D2-108a Pen-c
D2-108a Hex-n
D2-108a Hex-c
D2-108a CH₂Pr-c
D2-108a CH₂Bu-c
D2-108a CH₂Pen-c
D2-108a CH₂Hex-c
D2-108a CH₂CH=CH₂
D2-108a CH₂CH=C(Cl)₂
D2-108a CH₂C≡CH
D2-108a CH₂CN
D2-108a CH₂CF₃
D2-108a CH₂OMe
D2-108a CH₂OCF₃
D2-108a CH₂SMe
D2-108a CH₂S(O)Me
D2-108a CH₂S(O)₂Me
D2-108a CH₂SCF₃
D2-108a CH₂S(O)CF₃
D2-108a CH₂S(O)₂CF₃
D2-108a CH₂CH(OMe)₂
D2-108a CH₂CH(SMe)₂
D2-108a CH₂C(O)Me
D2-108a CH₂C(O)CF₃
D2-108a CH₂C(O)OMe
D2-108a CH₂(D2-32a)
D2-108a CH₂(D2-33a)
D2-108a CH₂(D2-34a)
D2-108a CH₂(D2-37a)
D2-108a CH₂(D2-81a)
D2-108a CH₂(D2-82a)
D2-108a CH₂(D2-84a)
D2-108a CH₂(D2-85a)
D2-108a CH₂(D2-87a)
D2-108a CH₂(D2-92a)
D2-108a CH₂(D2-93a)
D2-108a CH₂(D2-95a)
D2-108a CH₂(D2-96a)
D2-108a CH₂(D2-98a)
D2-108a CH₂(D2-108a)
D2-108a CH₂(D2-108b,Z²=2-Cl)
D2-108a CH₂(D2-108b,Z²=3-Me)
D2-108a CH₂(D2-108b,Z²=4-OMe)
D2-108a CH₂(D2-108b,Z²=2-SMe)
D2-108a CH₂(D2-108b,Z²=3-CF₃)
D2-108a CH₂(D2-108b,Z²=4-OCF₃)
D2-108a CH₂(D2-108b,Z²=2-SCF₃)
D2-108a CH₂CH₂CN
D2-108a CH₂CH₂CF₃
D2-108a CH₂CH₂OMe
D2-108a CH₂CH₂SMe
D2-108a CH₂CH₂S(O)Me
D2-108a CH₂CH₂S(O)₂Me
D2-108a D2-32a
D2-108a D2-33a
D2-108a D2-34a
D2-108a D2-37a
D2-108a D2-81a
D2-108a D2-82a
D2-108a D2-84a
D2-108a D2-85a
D2-108a D2-87a
D2-108a D2-92a
D2-108a D2-93a
D2-108a D2-95a
D2-108a D2-96a
D2-108a D2-98a
D2-108a D2-108a
D2-108a D2-108b(Z²=2-Cl)
D2-108a D2-108b(Z²=3-Me)
D2-108a D2-108b(Z²=4-OMe)
D2-108a D2-108b(Z²=2-SMe)
D2-108a D2-108b(Z²=3-CF₃)
D2-108a D2-108b(Z²=4-OCF₃)
D2-108a D2-108b(Z²=2-SCF₃)
D2-108a C(O)Me
D2-108a C(O)CF₃
D2-108a C(O)OMe
C(O)NHCH₂CF₃ Me
C(O)NHCH₂CF₃ Et
C(O)NHCH₂CF₃ Pr-n
C(O)NHCH₂CF₃ Pr-i
C(O)NHCH₂CF₃ Pr-c
C(O)NHCH₂CF₃ Bu-n
C(O)NHCH₂CF₃ Bu-i
C(O)NHCH₂CF₃ Bu-c
C(O)NHCH₂CF₃ Bu-s
C(O)NHCH₂CF₃ Bu-t
C(O)NHCH₂CF₃ Pen-n
C(O)NHCH₂CF₃ Pen-c
C(O)NHCH₂CF₃ Hex-n
C(O)NHCH₂CF₃ Hex-c
C(O)NHCH₂CF₃ CH₂Pr-c
C(O)NHCH₂CF₃ CH₂Bu-c
C(O)NHCH₂CF₃ CH₂Pen-c
C(O)NHCH₂CF₃ CH₂Hex-c
C(O)NHCH₂CF₃ CH₂CH=CH₂
C(O)NHCH₂CF₃ CH₂CH=C(Cl)₂
C(O)NHCH₂CF₃ CH₂C≡CH
C(O)NHCH₂CF₃ CH₂CN
C(O)NHCH₂CF₃ CH₂CF₃
C(O)NHCH₂CF₃ CH₂OMe
C(O)NHCH₂CF₃ CH₂OCF₃
C(O)NHCH₂CF₃ CH₂SMe
C(O)NHCH₂CF₃ CH₂S(O)Me
C(O)NHCH₂CF₃ CH₂S(O)₂Me
C(O)NHCH₂CF₃ CH₂SCF₃
C(O)NHCH₂CF₃ CH₂S(O)CF₃
C(O)NHCH₂CF₃ CH₂S(O)₂CF₃
C(O)NHCH₂CF₃ CH₂CH(OMe)₂
C(O)NHCH₂CF₃ CH₂CH(SMe)₂
C(O)NHCH₂CF₃ CH₂C(O)Me
C(O)NHCH₂CF₃ CH₂C(O)CF₃
C(O)NHCH₂CF₃ CH₂C(O)OMe
C(O)NHCH₂CF₃ CH₂(D2-32a)
C(O)NHCH₂CF₃ CH₂(D2-33a)
C(O)NHCH₂CF₃ CH₂(D2-34a)
C(O)NHCH₂CF₃ CH₂(D2-37a)
C(O)NHCH₂CF₃ CH₂(D2-81a)
C(O)NHCH₂CF₃ CH₂(D2-82a)
C(O)NHCH₂CF₃ CH₂(D2-84a)
C(O)NHCH₂CF₃ CH₂(D2-85a)
C(O)NHCH₂CF₃ CH₂(D2-87a)
C(O)NHCH₂CF₃ CH₂(D2-92a)
C(O)NHCH₂CF₃ CH₂(D2-93a)
C(O)NHCH₂CF₃ CH₂(D2-95a)
C(O)NHCH₂CF₃ CH₂(D2-96a)
C(O)NHCH₂CF₃ CH₂(D2-98a)
C(O)NHCH₂CF₃ CH₂(D2-108a)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=2-Cl)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=3-Me)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=4-OMe)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=2-SMe)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=3-CF₃)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=4-OCF₃)
C(O)NHCH₂CF₃ CH₂(D2-108b,Z²=2-SCF₃)
C(O)NHCH₂CF₃ CH₂CH₂CN
C(O)NHCH₂CF₃ CH₂CH₂CF₃
C(O)NHCH₂CF₃ CH₂CH₂OMe
C(O)NHCH₂CF₃ CH₂CH₂SMe
C(O)NHCH₂CF₃ CH₂CH₂S(O)Me
C(O)NHCH₂CF₃ CH₂CH₂S(O)₂Me
C(O)NHCH₂CF₃ D2-32a
C(O)NHCH₂CF₃ D2-33a
C(O)NHCH₂CF₃ D2-34a
C(O)NHCH₂CF₃ D2-37a
C(O)NHCH₂CF₃ D2-81a
C(O)NHCH₂CF₃ D2-82a
C(O)NHCH₂CF₃ D2-84a
C(O)NHCH₂CF₃ D2-85a
C(O)NHCH₂CF₃ D2-87a
C(O)NHCH₂CF₃ D2-92a
C(O)NHCH₂CF₃ D2-93a
C(O)NHCH₂CF₃ D2-95a
C(O)NHCH₂CF₃ D2-96a
C(O)NHCH₂CF₃ D2-98a
C(O)NHCH₂CF₃ D2-108a
C(O)NHCH₂CF₃ D2-108b(Z²=2-Cl)
C(O)NHCH₂CF₃ D2-108b(Z²=3-Me)
C(O)NHCH₂CF₃ D2-108b(Z²=4-OMe)
C(O)NHCH₂CF₃ D2-108b(Z²=2-SMe)
C(O)NHCH₂CF₃ D2-108b(Z²=3-CF₃)
C(O)NHCH₂CF₃ D2-108b(Z²=4-OCF₃)
C(O)NHCH₂CF₃ D2-108b(Z²=2-SCF₃)
C(O)NHCH₂CF₃ C(O)Me
C(O)NHCH₂CF₃ C(O)CF₃
C(O)NHCH₂CF₃ C(O)OMe
C(O)OMe Me
C(O)OMe Et
C(O)OMe Pr-n
C(O)OMe Pr-i
C(O)OMe Pr-c
C(O)OMe Bu-n
C(O)OMe Bu-i
C(O)OMe Bu-c
C(O)OMe Bu-s
C(O)OMe Bu-t
C(O)OMe Pen-n
C(O)OMe Pen-c
C(O)OMe Hex-n
C(O)OMe Hex-c
C(O)OMe CH₂Pr-c
C(O)OMe CH₂Bu-c
C(O)OMe CH₂Pen-c
C(O)OMe CH₂Hex-c
C(O)OMe CH₂CH=CH₂
C(O)OMe CH₂CH=C(Cl)₂
C(O)OMe CH₂C≡CH
C(O)OMe CH₂CN
C(O)OMe CH₂CF₃
C(O)OMe CH₂OMe
C(O)OMe CH₂OCF₃
C(O)OMe CH₂SMe
C(O)OMe CH₂S(O)Me
C(O)OMe CH₂S(O)₂Me
C(O)OMe CH₂SCF₃
C(O)OMe CH₂S(O)CF₃
C(O)OMe CH₂S(O)₂CF₃
C(O)OMe CH₂CH(OMe)₂
C(O)OMe CH₂CH(SMe)₂
C(O)OMe CH₂C(O)Me
C(O)OMe CH₂C(O)CF₃
C(O)OMe CH₂C(O)OMe
C(O)OMe CH₂(D2-32a)
C(O)OMe CH₂(D2-33a)
C(O)OMe CH₂(D2-34a)
C(O)OMe CH₂(D2-37a)
C(O)OMe CH₂(D2-81a)
C(O)OMe CH₂(D2-82a)
C(O)OMe CH₂(D2-84a)
C(O)OMe CH₂(D2-85a)
C(O)OMe CH₂(D2-87a)
C(O)OMe CH₂(D2-92a)
C(O)OMe CH₂(D2-93a)
C(O)OMe CH₂(D2-95a)
C(O)OMe CH₂(D2-96a)
C(O)OMe CH₂(D2-98a)
C(O)OMe CH₂(D2-108a)
C(O)OMe CH₂(D2-108b,Z²=2-Cl)
C(O)OMe CH₂(D2-108b,Z²=3-Me)
C(O)OMe CH₂(D2-108b,Z²=4-OMe)
C(O)OMe CH₂(D2-108b,Z²=2-SMe)
C(O)OMe CH₂(D2-108b,Z²=3-CF₃)
C(O)OMe CH₂(D2-108b,Z²=4-OCF₃)
C(O)OMe CH₂(D2-108b,Z²=2-SCF₃)
C(O)OMe CH₂CH₂CN
C(O)OMe CH₂CH₂CF₃
C(O)OMe CH₂CH₂OMe
C(O)OMe CH₂CH₂SMe
C(O)OMe CH₂CH₂S(O)Me
C(O)OMe CH₂CH₂S(O)₂Me
C(O)OMe D2-32a
C(O)OMe D2-33a
C(O)OMe D2-34a
C(O)OMe D2-37a
C(O)OMe D2-81a
C(O)OMe D2-82a
C(O)OMe D2-84a
C(O)OMe D2-85a
C(O)OMe D2-87a
C(O)OMe D2-92a
C(O)OMe D2-93a
C(O)OMe D2-95a
C(O)OMe D2-96a
C(O)OMe D2-98a
C(O)OMe D2-108a
C(O)OMe D2-108b(Z²=2-Cl)
C(O)OMe D2-108b(Z²=3-Me)
C(O)OMe D2-108b(Z²=4-OMe)
C(O)OMe D2-108b(Z²=2-SMe)
C(O)OMe D2-108b(Z²=3-CF₃)
C(O)OMe D2-108b(Z²=4-OCF₃)
C(O)OMe D2-108b(Z²=2-SCF₃)
C(O)OMe C(O)Me
C(O)OMe C(O)CF₃
C(O)OMe C(O)OMe
C(O)OEt Me
C(O)OEt Et
C(O)OEt Pr-n
C(O)OEt Pr-i
C(O)OEt Pr-c
C(O)OEt Bu-n
C(O)OEt Bu-i
C(O)OEt Bu-c
C(O)OEt Bu-s
C(O)OEt Bu-t
C(O)OEt Pen-n
C(O)OEt Pen-c
C(O)OEt Hex-n
C(O)OEt Hex-c
C(O)OEt CH₂Pr-c
C(O)OEt CH₂Bu-c
C(O)OEt CH₂Pen-c
C(O)OEt CH₂Hex-c
C(O)OEt CH₂CH=CH₂
C(O)OEt CH₂CH=C(Cl)₂
C(O)OEt CH₂C≡CH
C(O)OEt CH₂CN
C(O)OEt CH₂CF₃
C(O)OEt CH₂OMe
C(O)OEt CH₂OCF₃
C(O)OEt CH₂SMe
C(O)OEt CH₂S(O)Me
C(O)OEt CH₂S(O)₂Me
C(O)OEt CH₂SCF₃
C(O)OEt CH₂S(O)CF₃
C(O)OEt CH₂S(O)₂CF₃
C(O)OEt CH₂CH(OMe)₂
C(O)OEt CH₂CH(SMe)₂
C(O)OEt CH₂C(O)Me
C(O)OEt CH₂C(O)CF₃
C(O)OEt CH₂C(O)OMe
C(O)OEt CH₂(D2-32a)
C(O)OEt CH₂(D2-33a)
C(O)OEt CH₂(D2-34a)
C(O)OEt CH₂(D2-37a)
C(O)OEt CH₂(D2-81a)
C(O)OEt CH₂(D2-82a)
C(O)OEt CH₂(D2-84a)
C(O)OEt CH₂(D2-85a)
C(O)OEt CH₂(D2-87a)
C(O)OEt CH₂(D2-92a)
C(O)OEt CH₂(D2-93a)
C(O)OEt CH₂(D2-95a)
C(O)OEt CH₂(D2-96a)
C(O)OEt CH₂(D2-98a)
C(O)OEt CH₂(D2-108a)
C(O)OEt CH₂(D2-108b,Z²=2-Cl)
C(O)OEt CH₂(D2-108b,Z²=3-Me)
C(O)OEt CH₂(D2-108b,Z²=4-OMe)
C(O)OEt CH₂(D2-108b,Z²=2-SMe)
C(O)OEt CH₂(D2-108b,Z²=3-CF₃)
C(O)OEt CH₂(D2-108b,Z²=4-OCF₃)
C(O)OEt CH₂(D2-108b,Z²=2-SCF₃)
C(O)OEt CH₂CH₂CN
C(O)OEt CH₂CH₂CF₃
C(O)OEt CH₂CH₂OMe
C(O)OEt CH₂CH₂SMe
C(O)OEt CH₂CH₂S(O)Me
C(O)OEt CH₂CH₂S(O)₂Me
C(O)OEt D2-32a
C(O)OEt D2-34a
C(O)OEt D2-37a
C(O)OEt D2-81a
C(O)OEt D2-82a
C(O)OEt D2-84a
C(O)OEt D2-85a
C(O)OEt D2-87a
C(O)OEt D2-92a
C(O)OEt D2-93a
C(O)OEt D2-95a
C(O)OEt D2-96a
C(O)OEt D2-98a
C(O)OEt D2-108a
C(O)OEt D2-108b(Z²=2-Cl)
C(O)OEt D2-108b(Z²=3-Me)
C(O)OEt D2-108b(Z²=4-OMe)
C(O)OEt D2-108b(Z²=2-SMe)
C(O)OEt D2-108b(Z²=3-CF₃)
C(O)OEt D2-108b(Z²=4-OCF₃)
C(O)OEt D2-108b(Z²=2-SCF₃)
C(O)OEt C(O)Me
C(O)OEt C(O)CF₃
C(O)OEt C(O)OMe
NHCH₂CF₃ Me
NHCH₂CF₃ Et
NHCH₂CF₃ Pr-n
NHCH₂CF₃ Pr-i
NHCH₂CF₃ Pr-c
NHCH₂CF₃ Bu-n
NHCH₂CF₃ Bu-i
NHCH₂CF₃ Bu-c
NHCH₂CF₃ Bu-s
NHCH₂CF₃ Bu-t
NHCH₂CF₃ Pen-n
NHCH₂CF₃ Pen-c
NHCH₂CF₃ Hex-n
NHCH₂CF₃ Hex-c
NHCH₂CF₃ CH₂Pr-c
NHCH₂CF₃ CH₂Bu-c
NHCH₂CF₃ CH₂Pen-c
NHCH₂CF₃ CH₂Hex-c
NHCH₂CF₃ CH₂CH=CH₂
NHCH₂CF₃ CH₂CH=C(Cl)₂
NHCH₂CF₃ CH₂C≡CH
NHCH₂CF₃ CH₂CN
NHCH₂CF₃ CH₂CF₃
NHCH₂CF₃ CH₂OMe
NHCH₂CF₃ CH₂OCF₃
NHCH₂CF₃ CH₂SMe
NHCH₂CF₃ CH₂S(O)Me
NHCH₂CF₃ CH₂S(O)₂Me
NHCH₂CF₃ CH₂SCF₃
NHCH₂CF₃ CH₂S(O)CF₃
NHCH₂CF₃ CH₂S(O)₂CF₃
NHCH₂CF₃ CH₂CH(OMe)₂
NHCH₂CF₃ CH₂CH(SMe)₂
NHCH₂CF₃ CH₂C(O)Me
NHCH₂CF₃ CH₂C(O)CF₃
NHCH₂CF₃ CH₂C(O)OMe
NHCH₂CF₃ CH₂(D2-32a)
NHCH₂CF₃ CH₂(D2-33a)
NHCH₂CF₃ CH₂(D2-34a)
NHCH₂CF₃ CH₂(D2-37a)
NHCH₂CF₃ CH₂(D2-81a)
NHCH₂CF₃ CH₂(D2-82a)
NHCH₂CF₃ CH₂(D2-84a)
NHCH₂CF₃ CH₂(D2-85a)
NHCH₂CF₃ CH₂(D2-87a)
NHCH₂CF₃ CH₂(D2-92a)
NHCH₂CF₃ CH₂(D2-93a)
NHCH₂CF₃ CH₂(D2-95a)
NHCH₂CF₃ CH₂(D2-96a)
NHCH₂CF₃ CH₂(D2-98a)
NHCH₂CF₃ CH₂(D2-108a)
NHCH₂CF₃ CH₂(D2-108b,Z²=2-Cl)
NHCH₂CF₃ CH₂(D2-108b,Z²=3-Me)
NHCH₂CF₃ CH₂(D2-108b,Z²=4-OMe)
NHCH₂CF₃ CH₂(D2-108b,Z²=2-SMe)
NHCH₂CF₃ CH₂(D2-108b,Z²=3-CF₃)
NHCH₂CF₃ CH₂(D2-108b,Z²=4-OCF₃)
NHCH₂CF₃ CH₂(D2-108b,Z²=2-SCF₃)
NHCH₂CF₃ CH₂CH₂CN
NHCH₂CF₃ CH₂CH₂CF₃
NHCH₂CF₃ CH₂CH₂OMe
NHCH₂CF₃ CH₂CH₂SMe
NHCH₂CF₃ CH₂CH₂S(O)Me
NHCH₂CF₃ CH₂CH₂S(O)₂Me
NHCH₂CF₃ D2-32a
NHCH₂CF₃ D2-34a
NHCH₂CF₃ D2-37a
NHCH₂CF₃ D2-81a
NHCH₂CF₃ D2-82a
NHCH₂CF₃ D2-84a
NHCH₂CF₃ D2-85a
NHCH₂CF₃ D2-87a
NHCH₂CF₃ D2-92a
NHCH₂CF₃ D2-93a
NHCH₂CF₃ D2-95a
NHCH₂CF₃ D2-98a
NHCH₂CF₃ D2-108a
NHCH₂CF₃ D2-108b(Z²=2-Cl)
NHCH₂CF₃ D2-108b(Z²=3-Me)
NHCH₂CF₃ D2-108b(Z²=4-OMe)
NHCH₂CF₃ D2-108b(Z²=2-SMe)
NHCH₂CF₃ D2-108b(Z²=4-OCF₃)
NHCH₂CF₃ D2-108b(Z²=2-SCF₃)
NHCH₂CF₃ C(O)Me
NHCH₂CF₃ C(O)CF₃
NHCH₂CF₃ C(O)OMe
D2-7b(X²=3-CF₂CF₃) Me
--------------------------------------
〔第２表〕 Table 1
--------------------------------------
R^a           R^b
--------------------------------------
H H
H Me
H Et
H Pr-n
H Pr-i
H Pr-c
H Bu-n
H Bu-i
H Bu-c
H Bu-s
H Bu-t
H Pen-n
H Pen-c
H Hex-n
H Hex-c
H CH₂Pr-c
H CH₂Bu-c
H CH₂Pen-c
H CH₂Hex-c
H CH₂CH = CH₂
H CH₂CH = C (Cl)₂
H CH₂C≡CH
H CH₂CN
H CH₂CF_Three
H CH₂OMe
H CH₂OCF_Three
H CH₂SMe
H CH₂S (O) Me
H CH₂S (O)₂Me
H CH₂SCF_Three
H CH₂S (O) CF_Three
H CH₂S (O)₂CF_Three
H CH₂CH (OMe)₂
H CH₂CH (SMe)₂
H CH₂C (O) Me
H CH₂C (O) CF_Three
H CH₂C (O) OMe
H CH₂(D2-32a)
H CH₂(D2-33a)
H CH₂(D2-34a)
H CH₂(D2-37a)
H CH₂(D2-81a)
H CH₂(D2-82a)
H CH₂(D2-84a)
H CH₂(D2-85a)
H CH₂(D2-87a)
H CH₂(D2-92a)
H CH₂(D2-93a)
H CH₂(D2-95a)
H CH₂(D2-96a)
H CH₂(D2-98a)
H CH₂(D2-108a)
H CH₂(D2-108b, Z²= 2-Cl)
H CH₂(D2-108b, Z²= 3-Me)
H CH₂(D2-108b, Z²= 4-OMe)
H CH₂(D2-108b, Z²= 2-SMe)
H CH₂(D2-108b, Z²= 3-CF_Three)
H CH₂(D2-108b, Z²= 4-OCF_Three)
H CH₂(D2-108b, Z²= 2-SCF_Three)
H CH₂CH₂CN
H CH₂CH₂CF_Three
H CH₂CH₂OMe
H CH₂CH₂SMe
H CH₂CH₂S (O) Me
H CH₂CH₂S (O)₂Me
H D2-32a
H D2-33a
H D2-34a
H D2-37a
H D2-81a
H D2-82a
H D2-84a
H D2-85a
H D2-87a
H D2-92a
H D2-93a
H D2-95a
H D2-96a
H D2-98a
H D2-108a
H D2-108b (Z²= 2-Cl)
H D2-108b (Z²= 3-Me)
H D2-108b (Z²= 4-OMe)
H D2-108b (Z²= 2-SMe)
H D2-108b (Z²= 3-CF_Three)
H D2-108b (Z²= 4-OCF_Three)
H D2-108b (Z²= 2-SCF_Three)
H C (O) Me
H C (O) CF_Three
H C (O) OMe
CF_Three           Me
CF_Three           Et
CF_Three           Pr-n
CF_Three           Pr-i
CF_Three           Pr-c
CF_Three           Bu-n
CF_Three           Bu-i
CF_Three           Bu-c
CF_Three           Bu-s
CF_Three           Bu-t
CF_Three           Pen-n
CF_Three           Pen-c
CF_Three           Hex-n
CF_Three           Hex-c
CF_Three           CH₂Pr-c
CF_Three           CH₂Bu-c
CF_Three           CH₂Pen-c
CF_Three           CH₂Hex-c
CF_Three           CH₂CH = CH₂
CF_Three           CH₂CH = C (Cl)₂
CF_Three           CH₂C≡CH
CF_Three           CH₂CN
CF_Three           CH₂CF_Three
CF_Three           CH₂OMe
CF_Three           CH₂OCF_Three
CF_Three           CH₂SMe
CF_Three           CH₂S (O) Me
CF_Three           CH₂S (O)₂Me
CF_Three           CH₂SCF_Three
CF_Three           CH₂S (O) CF_Three
CF_Three           CH₂S (O)₂CF_Three
CF_Three           CH₂CH (OMe)₂
CF_Three           CH₂CH (SMe)₂
CF_Three           CH₂C (O) Me
CF_Three           CH₂C (O) CF_Three
CF_Three           CH₂C (O) OMe
CF_Three           CH₂(D2-32a)
CF_Three           CH₂(D2-33a)
CF_Three           CH₂(D2-34a)
CF_Three           CH₂(D2-37a)
CF_Three           CH₂(D2-81a)
CF_Three           CH₂(D2-82a)
CF_Three           CH₂(D2-84a)
CF_Three           CH₂(D2-85a)
CF_Three           CH₂(D2-87a)
CF_Three           CH₂(D2-92a)
CF_Three           CH₂(D2-93a)
CF_Three           CH₂(D2-95a)
CF_Three           CH₂(D2-96a)
CF_Three           CH₂(D2-98a)
CF_Three           CH₂(D2-108a)
CF_Three           CH₂(D2-108b, Z²= 2-Cl)
CF_Three           CH₂(D2-108b, Z²= 3-Me)
CF_Three           CH₂(D2-108b, Z²= 4-OMe)
CF_Three           CH₂(D2-108b, Z²= 2-SMe)
CF_Three           CH₂(D2-108b, Z²= 3-CF_Three)
CF_Three           CH₂(D2-108b, Z²= 4-OCF_Three)
CF_Three           CH₂(D2-108b, Z²= 2-SCF_Three)
CF_Three           CH₂CH₂CN
CF_Three           CH₂CH₂CF_Three
CF_Three           CH₂CH₂OMe
CF_Three           CH₂CH₂SMe
CF_Three           CH₂CH₂S (O) Me
CF_Three           CH₂CH₂S (O)₂Me
CF_Three           D2-32a
CF_Three           D2-33a
CF_Three           D2-34a
CF_Three           D2-37a
CF_Three           D2-81a
CF_Three           D2-82a
CF_Three          D2-84a
CF_Three           D2-85a
CF_Three           D2-87a
CF_Three           D2-92a
CF_Three           D2-93a
CF_Three           D2-95a
CF_Three           D2-96a
CF_Three           D2-98a
CF_Three           D2-108a
CF_Three           D2-108b (Z²= 2-Cl)
CF_Three           D2-108b (Z²= 3-Me)
CF_Three           D2-108b (Z²= 4-OMe)
CF_Three           D2-108b (Z²= 2-SMe)
CF_Three           D2-108b (Z²= 3-CF_Three)
CF_Three           D2-108b (Z²= 4-OCF_Three)
CF_Three           D2-108b (Z²= 2-SCF_Three)
CF_Three           C (O) Me
CF_Three           C (O) CF_Three
CF_Three           C (O) OMe
Me Me
Me Et
Me Pr-n
Me Pr-i
Me Pr-c
Me Bu-n
Me Bu-i
Me Bu-c
Me Bu-s
Me Bu-t
Me Pen-n
Me Pen-c
Me Hex-n
Me Hex-c
Me CH₂Pr-c
Me CH₂Bu-c
Me CH₂Pen-c
Me CH₂Hex-c
Me CH₂CH = CH₂
Me CH₂CH = C (Cl)₂
Me CH₂C≡CH
Me CH₂CN
Me CH₂CF_Three
Me CH₂OMe
Me CH₂OCF_Three
Me CH₂SMe
Me CH₂S (O) Me
Me CH₂S (O)₂Me
Me CH₂SCF_Three
Me CH₂S (O) CF_Three
Me CH₂S (O)₂CF_Three
Me CH₂CH (OMe)₂
Me CH₂CH (SMe)₂
Me CH₂C (O) Me
Me CH₂C (O) CF_Three
Me CH₂C (O) OMe
Me CH₂(D2-32a)
Me CH₂(D2-33a)
Me CH₂(D2-34a)
Me CH₂(D2-37a)
Me CH₂(D2-81a)
Me CH₂(D2-82a)
Me CH₂(D2-84a)
Me CH₂(D2-85a)
Me CH₂(D2-87a)
Me CH₂(D2-92a)
Me CH₂(D2-93a)
Me CH₂(D2-95a)
Me CH₂(D2-96a)
Me CH₂(D2-98a)
Me CH₂(D2-108a)
Me CH₂(D2-108b, Z²= 2-Cl)
Me CH₂(D2-108b, Z²= 3-Me)
Me CH₂(D2-108b, Z²= 4-OMe)
Me CH₂(D2-108b, Z²= 2-SMe)
Me CH₂(D2-108b, Z²= 3-CF_Three)
Me CH₂(D2-108b, Z²= 4-OCF_Three)
Me CH₂(D2-108b, Z²= 2-SCF_Three)
Me CH₂CH₂CN
Me CH₂CH₂CF_Three
Me CH₂CH₂OMe
Me CH₂CH₂SMe
Me CH₂CH₂S (O) Me
Me CH₂CH₂S (O)₂Me
Me D2-32a
Me D2-33a
Me D2-34a
Me D2-37a
Me D2-81a
Me D2-82a
Me D2-84a
Me D2-85a
Me D2-87a
Me D2-92a
Me D2-93a
Me D2-95a
Me D2-96a
Me D2-98a
Me D2-108a
Me D2-108b (Z²= 2-Cl)
Me D2-108b (Z²= 3-Me)
Me D2-108b (Z²= 4-OMe)
Me D2-108b (Z²= 2-SMe)
Me D2-108b (Z²= 3-CF_Three)
Me D2-108b (Z²= 4-OCF_Three)
Me D2-108b (Z²= 2-SCF_Three)
Me C (O) Me
Me C (O) CF_Three
Me C (O) OMe
OMe Me
OMe Et
OMe Pr-n
OMe Pr-i
OMe Pr-c
OMe Bu-n
OMe Bu-i
OMe Bu-c
OMe Bu-s
OMe Bu-t
OMe Pen-n
OMe Pen-c
OMe Hex-n
OMe Hex-c
OMe CH₂Pr-c
OMe CH₂Bu-c
OMe CH₂Pen-c
OMe CH₂Hex-c
OMe CH₂CH = CH₂
OMe CH₂CH = C (Cl)₂
OMe CH₂C≡CH
OMe CH₂CN
OMe CH₂CF_Three
OMe CH₂OMe
OMe CH₂OCF_Three
OMe CH₂SMe
OMe CH₂S (O) Me
OMe CH₂S (O)₂Me
OMe CH₂SCF_Three
OMe CH₂S (O) CF_Three
OMe CH₂S (O)₂CF_Three
OMe CH₂CH (OMe)₂
OMe CH₂CH (SMe)₂
OMe CH₂C (O) Me
OMe CH₂C (O) CF_Three
OMe CH₂C (O) OMe
OMe CH₂(D2-32a)
OMe CH₂(D2-33a)
OMe CH₂(D2-34a)
OMe CH₂(D2-37a)
OMe CH₂(D2-81a)
OMe CH₂(D2-82a)
OMe CH₂(D2-84a)
OMe CH₂(D2-85a)
OMe CH₂(D2-87a)
OMe CH₂(D2-92a)
OMe CH₂(D2-93a)
OMe CH₂(D2-95a)
OMe CH₂(D2-96a)
OMe CH₂(D2-98a)
OMe CH₂(D2-108a)
OMe CH₂(D2-108b, Z²= 2-Cl)
OMe CH₂(D2-108b, Z²= 3-Me)
OMe CH₂(D2-108b, Z²= 4-OMe)
OMe CH₂(D2-108b, Z²= 2-SMe)
OMe CH₂(D2-108b, Z²= 3-CF_Three)
OMe CH₂(D2-108b, Z²= 4-OCF_Three)
OMe CH₂(D2-108b, Z²= 2-SCF_Three)
OMe CH₂CH₂CN
OMe CH₂CH₂CF_Three
OMe CH₂CH₂OMe
OMe CH₂CH₂SMe
OMe CH₂CH₂S (O) Me
OMe CH₂CH₂S (O)₂Me
OMe D2-32a
OMe D2-33a
OMe D2-34a
OMe D2-37a
OMe D2-81a
OMe D2-82a
OMe D2-84a
OMe D2-85a
OMe D2-87a
OMe D2-92a
OMe D2-93a
OMe D2-95a
OMe D2-96a
OMe D2-98a
OMe D2-108a
OMe D2-108b (Z²= 2-Cl)
OMe D2-108b (Z²= 3-Me)
OMe D2-108b (Z²= 4-OMe)
OMe D2-108b (Z²= 2-SMe)
OMe D2-108b (Z²= 3-CF_Three)
OMe D2-108b (Z²= 4-OCF_Three)
OMe D2-108b (Z²= 2-SCF_Three)
OMe C (O) Me
OMe C (O) CF_Three
OMe C (O) OMe
SMe Me
SMe Et
SMe Pr-n
SMe Pr-i
SMe Pr-c
SMe Bu-n
SMe Bu-i
SMe Bu-c
SMe Bu-s
SMe Bu-t
SMe Pen-n
SMe Pen-c
SMe Hex-n
SMe Hex-c
SMe CH₂Pr-c
SMe CH₂Bu-c
SMe CH₂Pen-c
SMe CH₂Hex-c
SMe CH₂CH = CH₂
SMe CH₂CH = C (Cl)₂
SMe CH₂C≡CH
SMe CH₂CN
SMe CH₂CF_Three
SMe CH₂OMe
SMe CH₂OCF_Three
SMe CH₂SMe
SMe CH₂S (O) Me
SMe CH₂S (O)₂Me
SMe CH₂SCF_Three
SMe CH₂S (O) CF_Three
SMe CH₂S (O)₂CF_Three
SMe CH₂CH (OMe)₂
SMe CH₂CH (SMe)₂
SMe CH₂C (O) Me
SMe CH₂C (O) CF_Three
SMe CH₂C (O) OMe
SMe CH₂(D2-32a)
SMe CH₂(D2-33a)
SMe CH₂(D2-34a)
SMe CH₂(D2-37a)
SMe CH₂(D2-81a)
SMe CH₂(D2-82a)
SMe CH₂(D2-84a)
SMe CH₂(D2-85a)
SMe CH₂(D2-87a)
SMe CH₂(D2-92a)
SMe CH₂(D2-93a)
SMe CH₂(D2-95a)
SMe CH₂(D2-96a)
SMe CH₂(D2-98a)
SMe CH₂(D2-108a)
SMe CH₂(D2-108b, Z²= 2-Cl)
SMe CH₂(D2-108b, Z²= 3-Me)
SMe CH₂(D2-108b, Z²= 4-OMe)
SMe CH₂(D2-108b, Z²= 2-SMe)
SMe CH₂(D2-108b, Z²= 3-CF_Three)
SMe CH₂(D2-108b, Z²= 4-OCF_Three)
SMe CH₂(D2-108b, Z²= 2-SCF_Three)
SMe CH₂CH₂CN
SMe CH₂CH₂CF_Three
SMe CH₂CH₂OMe
SMe CH₂CH₂SMe
SMe CH₂CH₂S (O) Me
SMe CH₂CH₂S (O)₂Me
SMe D2-32a
SMe D2-33a
SMe D2-34a
SMe D2-37a
SMe D2-81a
SMe D2-82a
SMe D2-84a
SMe D2-85a
SMe D2-87a
SMe D2-92a
SMe D2-93a
SMe D2-95a
SMe D2-96a
SMe D2-98a
SMe D2-108a
SMe D2-108b (Z²= 2-Cl)
SMe D2-108b (Z²= 3-Me)
SMe D2-108b (Z²= 4-OMe)
SMe D2-108b (Z²= 2-SMe)
SMe D2-108b (Z²= 3-CF_Three)
SMe D2-108b (Z²= 4-OCF_Three)
SMe D2-108b (Z²= 2-SCF_Three)
SMe C (O) Me
SMe C (O) CF_Three
SMe C (O) OMe
CH₂OMe Me
CH₂OMe Et
CH₂OMe Pr-n
CH₂OMe Pr-i
CH₂OMe Pr-c
CH₂OMe Bu-n
CH₂OMe Bu-i
CH₂OMe Bu-c
CH₂OMe Bu-s
CH₂OMe Bu-t
CH₂OMe Pen-n
CH₂OMe Pen-c
CH₂OMe Hex-n
CH₂OMe Hex-c
CH₂OMe CH₂Pr-c
CH₂OMe CH₂Bu-c
CH₂OMe CH₂Pen-c
CH₂OMe CH₂Hex-c
CH₂OMe CH₂CH = CH₂
CH₂OMe CH₂CH = C (Cl)₂
CH₂OMe CH₂C≡CH
CH₂OMe CH₂CN
CH₂OMe CH₂CF_Three
CH₂OMe CH₂OMe
CH₂OMe CH₂OCF_Three
CH₂OMe CH₂SMe
CH₂OMe CH₂S (O) Me
CH₂OMe CH₂S (O)₂Me
CH₂OMe CH₂SCF_Three
CH₂OMe CH₂S (O) CF_Three
CH₂OMe CH₂S (O)₂CF_Three
CH₂OMe CH₂CH (OMe)₂
CH₂OMe CH₂CH (SMe)₂
CH₂OMe CH₂C (O) Me
CH₂OMe CH₂C (O) CF_Three
CH₂OMe CH₂C (O) OMe
CH₂OMe CH₂(D2-32a)
CH₂OMe CH₂(D2-33a)
CH₂OMe CH₂(D2-34a)
CH₂OMe CH₂(D2-37a)
CH₂OMe CH₂(D2-81a)
CH₂OMe CH₂(D2-82a)
CH₂OMe CH₂(D2-84a)
CH₂OMe CH₂(D2-85a)
CH₂OMe CH₂(D2-87a)
CH₂OMe CH₂(D2-92a)
CH₂OMe CH₂(D2-93a)
CH₂OMe CH₂(D2-95a)
CH₂OMe CH₂(D2-96a)
CH₂OMe CH₂(D2-98a)
CH₂OMe CH₂(D2-108a)
CH₂OMe CH₂(D2-108b, Z²= 2-Cl)
CH₂OMe CH₂(D2-108b, Z²= 3-Me)
CH₂OMe CH₂(D2-108b, Z²= 4-OMe)
CH₂OMe CH₂(D2-108b, Z²= 2-SMe)
CH₂OMe CH₂(D2-108b, Z²= 3-CF_Three)
CH₂OMe CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂OMe CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂OMe CH₂CH₂CN
CH₂OMe CH₂CH₂CF_Three
CH₂OMe CH₂CH₂OMe
CH₂OMe CH₂CH₂SMe
CH₂OMe CH₂CH₂S (O) Me
CH₂OMe CH₂CH₂S (O)₂Me
CH₂OMe D2-32a
CH₂OMe D2-33a
CH₂OMe D2-34a
CH₂OMe D2-37a
CH₂OMe D2-81a
CH₂OMe D2-82a
CH₂OMe D2-84a
CH₂OMe D2-85a
CH₂OMe D2-87a
CH₂OMe D2-92a
CH₂OMe D2-93a
CH₂OMe D2-95a
CH₂OMe D2-96a
CH₂OMe D2-98a
CH₂OMe D2-108a
CH₂OMe D2-108b (Z²= 2-Cl)
CH₂OMe D2-108b (Z²= 3-Me)
CH₂OMe D2-108b (Z²= 4-OMe)
CH₂OMe D2-108b (Z²= 2-SMe)
CH₂OMe D2-108b (Z²= 3-CF_Three)
CH₂OMe D2-108b (Z²= 4-OCF_Three)
CH₂OMe D2-108b (Z²= 2-SCF_Three)
CH₂OMe C (O) Me
CH₂OMe C (O) CF_Three
CH₂OMe C (O) OMe
CH₂SMe Me
CH₂SMe Et
CH₂SMe Pr-n
CH₂SMe Pr-i
CH₂SMe Pr-c
CH₂SMe Bu-n
CH₂SMe Bu-i
CH₂SMe Bu-c
CH₂SMe Bu-s
CH₂SMe Bu-t
CH₂SMe Pen-n
CH₂SMe Pen-c
CH₂SMe Hex-n
CH₂SMe Hex-c
CH₂SMe CH₂Pr-c
CH₂SMe CH₂Bu-c
CH₂SMe CH₂Pen-c
CH₂SMe CH₂Hex-c
CH₂SMe CH₂CH = CH₂
CH₂SMe CH₂CH = C (Cl)₂
CH₂SMe CH₂C≡CH
CH₂SMe CH₂CN
CH₂SMe CH₂CF_Three
CH₂SMe CH₂OMe
CH₂SMe CH₂OCF_Three
CH₂SMe CH₂SMe
CH₂SMe CH₂S (O) Me
CH₂SMe CH₂S (O)₂Me
CH₂SMe CH₂SCF_Three
CH₂SMe CH₂S (O) CF_Three
CH₂SMe CH₂S (O)₂CF_Three
CH₂SMe CH₂CH (OMe)₂
CH₂SMe CH₂CH (SMe)₂
CH₂SMe CH₂C (O) Me
CH₂SMe CH₂C (O) CF_Three
CH₂SMe CH₂C (O) OMe
CH₂SMe CH₂(D2-32a)
CH₂SMe CH₂(D2-33a)
CH₂SMe CH₂(D2-34a)
CH₂SMe CH₂(D2-37a)
CH₂SMe CH₂(D2-81a)
CH₂SMe CH₂(D2-82a)
CH₂SMe CH₂(D2-84a)
CH₂SMe CH₂(D2-85a)
CH₂SMe CH₂(D2-87a)
CH₂SMe CH₂(D2-92a)
CH₂SMe CH₂(D2-93a)
CH₂SMe CH₂(D2-95a)
CH₂SMe CH₂(D2-96a)
CH₂SMe CH₂(D2-98a)
CH₂SMe CH₂(D2-108a)
CH₂SMe CH₂(D2-108b, Z²= 2-Cl)
CH₂SMe CH₂(D2-108b, Z²= 3-Me)
CH₂SMe CH₂(D2-108b, Z²= 4-OMe)
CH₂SMe CH₂(D2-108b, Z²= 2-SMe)
CH₂SMe CH₂(D2-108b, Z²= 3-CF_Three)
CH₂SMe CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂SMe CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂SMe CH₂CH₂CN
CH₂SMe CH₂CH₂CF_Three
CH₂SMe CH₂CH₂OMe
CH₂SMe CH₂CH₂SMe
CH₂SMe CH₂CH₂S (O) Me
CH₂SMe CH₂CH₂S (O)₂Me
CH₂SMe D2-32a
CH₂SMe D2-33a
CH₂SMe D2-34a
CH₂SMe D2-37a
CH₂SMe D2-81a
CH₂SMe D2-82a
CH₂SMe D2-84a
CH₂SMe D2-85a
CH₂SMe D2-87a
CH₂SMe D2-92a
CH₂SMe D2-93a
CH₂SMe D2-95a
CH₂SMe D2-96a
CH₂SMe D2-98a
CH₂SMe D2-108a
CH₂SMe D2-108b (Z²= 2-Cl)
CH₂SMe D2-108b (Z²= 3-Me)
CH₂SMe D2-108b (Z²= 4-OMe)
CH₂SMe D2-108b (Z²= 2-SMe)
CH₂SMe D2-108b (Z²= 3-CF_Three)
CH₂SMe D2-108b (Z²= 4-OCF_Three)
CH₂SMe D2-108b (Z²= 2-SCF_Three)
CH₂SMe C (O) Me
CH₂SMe C (O) CF_Three
CH₂SMe C (O) OMe
CH₂S (O) Me Me
CH₂S (O) Me Et
CH₂S (O) Me Pr-n
CH₂S (O) Me Pr-i
CH₂S (O) Me Pr-c
CH₂S (O) Me Bu-n
CH₂S (O) Me Bu-i
CH₂S (O) Me Bu-c
CH₂S (O) Me Bu-s
CH₂S (O) Me Bu-t
CH₂S (O) Me Pen-n
CH₂S (O) Me Pen-c
CH₂S (O) Me Hex-n
CH₂S (O) Me Hex-c
CH₂S (O) Me CH₂Pr-c
CH₂S (O) Me CH₂Bu-c
CH₂S (O) Me CH₂Pen-c
CH₂S (O) Me CH₂Hex-c
CH₂S (O) Me CH₂CH = CH₂
CH₂S (O) Me CH₂CH = C (Cl)₂
CH₂S (O) Me CH₂C≡CH
CH₂S (O) Me CH₂CN
CH₂S (O) Me CH₂CF_Three
CH₂S (O) Me CH₂OMe
CH₂S (O) Me CH₂OCF_Three
CH₂S (O) Me CH₂SMe
CH₂S (O) Me CH₂S (O) Me
CH₂S (O) Me CH₂S (O)₂Me
CH₂S (O) Me CH₂SCF_Three
CH₂S (O) Me CH₂S (O) CF_Three
CH₂S (O) Me CH₂S (O)₂CF_Three
CH₂S (O) Me CH₂CH (OMe)₂
CH₂S (O) Me CH₂CH (SMe)₂
CH₂S (O) Me CH₂C (O) Me
CH₂S (O) Me CH₂C (O) CF_Three
CH₂S (O) Me CH₂C (O) OMe
CH₂S (O) Me CH₂(D2-32a)
CH₂S (O) Me CH₂(D2-33a)
CH₂S (O) Me CH₂(D2-34a)
CH₂S (O) Me CH₂(D2-37a)
CH₂S (O) Me CH₂(D2-81a)
CH₂S (O) Me CH₂(D2-82a)
CH₂S (O) Me CH₂(D2-84a)
CH₂S (O) Me CH₂(D2-85a)
CH₂S (O) Me CH₂(D2-87a)
CH₂S (O) Me CH₂(D2-92a)
CH₂S (O) Me CH₂(D2-93a)
CH₂S (O) Me CH₂(D2-95a)
CH₂S (O) Me CH₂(D2-96a)
CH₂S (O) Me CH₂(D2-98a)
CH₂S (O) Me CH₂(D2-108a)
CH₂S (O) Me CH₂(D2-108b, Z²= 2-Cl)
CH₂S (O) Me CH₂(D2-108b, Z²= 3-Me)
CH₂S (O) Me CH₂(D2-108b, Z²= 4-OMe)
CH₂S (O) Me CH₂(D2-108b, Z²= 2-SMe)
CH₂S (O) Me CH₂(D2-108b, Z²= 3-CF_Three)
CH₂S (O) Me CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂S (O) Me CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂S (O) Me CH₂CH₂CN
CH₂S (O) Me CH₂CH₂CF_Three
CH₂S (O) Me CH₂CH₂OMe
CH₂S (O) Me CH₂CH₂SMe
CH₂S (O) Me CH₂CH₂S (O) Me
CH₂S (O) Me CH₂CH₂S (O)₂Me
CH₂S (O) Me D2-32a
CH₂S (O) Me D2-33a
CH₂S (O) Me D2-34a
CH₂S (O) Me D2-37a
CH₂S (O) Me D2-81a
CH₂S (O) Me D2-82a
CH₂S (O) Me D2-84a
CH₂S (O) Me D2-85a
CH₂S (O) Me D2-87a
CH₂S (O) Me D2-92a
CH₂S (O) Me D2-93a
CH₂S (O) Me D2-95a
CH₂S (O) Me D2-96a
CH₂S (O) Me D2-98a
CH₂S (O) Me D2-108a
CH₂S (O) Me D2-108b (Z²= 2-Cl)
CH₂S (O) Me D2-108b (Z²= 3-Me)
CH₂S (O) Me D2-108b (Z²= 4-OMe)
CH₂S (O) Me D2-108b (Z²= 2-SMe)
CH₂S (O) Me D2-108b (Z²= 3-CF_Three)
CH₂S (O) Me D2-108b (Z²= 4-OCF_Three)
CH₂S (O) Me D2-108b (Z²= 2-SCF_Three)
CH₂S (O) Me C (O) Me
CH₂S (O) Me C (O) CF_Three
CH₂S (O) Me C (O) OMe
CH₂S (O)₂Me Me
CH₂S (O)₂Me Et
CH₂S (O)₂Me Pr-n
CH₂S (O)₂Me Pr-i
CH₂S (O)₂Me Pr-c
CH₂S (O)₂Me Bu-n
CH₂S (O)₂Me Bu-i
CH₂S (O)₂Me Bu-c
CH₂S (O)₂Me Bu-s
CH₂S (O)₂Me Bu-t
CH₂S (O)₂Me Pen-n
CH₂S (O)₂Me Pen-c
CH₂S (O)₂Me Hex-n
CH₂S (O)₂Me Hex-c
CH₂S (O)₂Me CH₂Pr-c
CH₂S (O)₂Me CH₂Bu-c
CH₂S (O)₂Me CH₂Pen-c
CH₂S (O)₂Me CH₂Hex-c
CH₂S (O)₂Me CH₂CH = CH₂
CH₂S (O)₂Me CH₂CH = C (Cl)₂
CH₂S (O)₂Me CH₂C≡CH
CH₂S (O)₂Me CH₂CN
CH₂S (O)₂Me CH₂CF_Three
CH₂S (O)₂Me CH₂OMe
CH₂S (O)₂Me CH₂OCF_Three
CH₂S (O)₂Me CH₂SMe
CH₂S (O)₂Me CH₂S (O) Me
CH₂S (O)₂Me CH₂S (O)₂Me
CH₂S (O)₂Me CH₂SCF_Three
CH₂S (O)₂Me CH₂S (O) CF_Three
CH₂S (O)₂Me CH₂S (O)₂CF_Three
CH₂S (O)₂Me CH₂CH (OMe)₂
CH₂S (O)₂Me CH₂CH (SMe)₂
CH₂S (O)₂Me CH₂C (O) Me
CH₂S (O)₂Me CH₂C (O) CF_Three
CH₂S (O)₂Me CH₂C (O) OMe
CH₂S (O)₂Me CH₂(D2-32a)
CH₂S (O)₂Me CH₂(D2-33a)
CH₂S (O)₂Me CH₂(D2-34a)
CH₂S (O)₂Me CH₂(D2-37a)
CH₂S (O)₂Me CH₂(D2-81a)
CH₂S (O)₂Me CH₂(D2-82a)
CH₂S (O)₂Me CH₂(D2-84a)
CH₂S (O)₂Me CH₂(D2-85a)
CH₂S (O)₂Me CH₂(D2-87a)
CH₂S (O)₂Me CH₂(D2-92a)
CH₂S (O)₂Me CH₂(D2-93a)
CH₂S (O)₂Me CH₂(D2-95a)
CH₂S (O)₂Me CH₂(D2-96a)
CH₂S (O)₂Me CH₂(D2-98a)
CH₂S (O)₂Me CH₂(D2-108a)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 2-Cl)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 3-Me)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 4-OMe)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 2-SMe)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 3-CF_Three)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂S (O)₂Me CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂S (O)₂Me CH₂CH₂CN
CH₂S (O)₂Me CH₂CH₂CF_Three
CH₂S (O)₂Me CH₂CH₂OMe
CH₂S (O)₂Me CH₂CH₂SMe
CH₂S (O)₂Me CH₂CH₂S (O) Me
CH₂S (O)₂Me CH₂CH₂S (O)₂Me
CH₂S (O)₂Me D2-32a
CH₂S (O)₂Me D2-33a
CH₂S (O)₂Me D2-34a
CH₂S (O)₂Me D2-37a
CH₂S (O)₂Me D2-81a
CH₂S (O)₂Me D2-82a
CH₂S (O)₂Me D2-84a
CH₂S (O)₂Me D2-85a
CH₂S (O)₂Me D2-87a
CH₂S (O)₂Me D2-92a
CH₂S (O)₂Me D2-93a
CH₂S (O)₂Me D2-95a
CH₂S (O)₂Me D2-96a
CH₂S (O)₂Me D2-98a
CH₂S (O)₂Me D2-108a
CH₂S (O)₂Me D2-108b (Z²= 2-Cl)
CH₂S (O)₂Me D2-108b (Z²= 3-Me)
CH₂S (O)₂Me D2-108b (Z²= 4-OMe)
CH₂S (O)₂Me D2-108b (Z²= 2-SMe)
CH₂S (O)₂Me D2-108b (Z²= 3-CF_Three)
CH₂S (O)₂Me D2-108b (Z²= 4-OCF_Three)
CH₂S (O)₂Me D2-108b (Z²= 2-SCF_Three)
CH₂S (O)₂Me C (O) Me
CH₂S (O)₂Me C (O) CF_Three
CH₂S (O)₂Me C (O) OMe
CH₂SCF_Three       Me
CH₂SCF_Three       Et
CH₂SCF_Three       Pr-n
CH₂SCF_Three       Pr-i
CH₂SCF_Three       Pr-c
CH₂SCF_Three       Bu-n
CH₂SCF_Three       Bu-i
CH₂SCF_Three       Bu-c
CH₂SCF_Three       Bu-s
CH₂SCF_Three       Bu-t
CH₂SCF_Three       Pen-n
CH₂SCF_Three       Pen-c
CH₂SCF_Three       Hex-n
CH₂SCF_Three       Hex-c
CH₂SCF_Three       CH₂Pr-c
CH₂SCF_Three       CH₂Bu-c
CH₂SCF_Three       CH₂Pen-c
CH₂SCF_Three       CH₂Hex-c
CH₂SCF_Three       CH₂CH = CH₂
CH₂SCF_Three       CH₂CH = C (Cl)₂
CH₂SCF_Three       CH₂C≡CH
CH₂SCF_Three       CH₂CN
CH₂SCF_Three       CH₂CF_Three
CH₂SCF_Three       CH₂OMe
CH₂SCF_Three       CH₂OCF_Three
CH₂SCF_Three       CH₂SMe
CH₂SCF_Three       CH₂S (O) Me
CH₂SCF_Three       CH₂S (O)₂Me
CH₂SCF_Three       CH₂SCF_Three
CH₂SCF_Three       CH₂S (O) CF_Three
CH₂SCF_Three       CH₂S (O)₂CF_Three
CH₂SCF_Three       CH₂CH (OMe)₂
CH₂SCF_Three       CH₂CH (SMe)₂
CH₂SCF_Three       CH₂C (O) Me
CH₂SCF_Three       CH₂C (O) CF_Three
CH₂SCF_Three       CH₂C (O) OMe
CH₂SCF_Three       CH₂(D2-32a)
CH₂SCF_Three       CH₂(D2-33a)
CH₂SCF_Three       CH₂(D2-34a)
CH₂SCF_Three       CH₂(D2-37a)
CH₂SCF_Three       CH₂(D2-81a)
CH₂SCF_Three       CH₂(D2-82a)
CH₂SCF_Three       CH₂(D2-84a)
CH₂SCF_Three       CH₂(D2-85a)
CH₂SCF_Three       CH₂(D2-87a)
CH₂SCF_Three       CH₂(D2-92a)
CH₂SCF_Three       CH₂(D2-93a)
CH₂SCF_Three       CH₂(D2-95a)
CH₂SCF_Three       CH₂(D2-96a)
CH₂SCF_Three       CH₂(D2-98a)
CH₂SCF_Three       CH₂(D2-108a)
CH₂SCF_Three       CH₂(D2-108b, Z²= 2-Cl)
CH₂SCF_Three       CH₂(D2-108b, Z²= 3-Me)
CH₂SCF_Three       CH₂(D2-108b, Z²= 4-OMe)
CH₂SCF_Three       CH₂(D2-108b, Z²= 2-SMe)
CH₂SCF_Three       CH₂(D2-108b, Z²= 3-CF_Three)
CH₂SCF_Three       CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂SCF_Three       CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂SCF_Three       CH₂CH₂CN
CH₂SCF_Three       CH₂CH₂CF_Three
CH₂SCF_Three       CH₂CH₂OMe
CH₂SCF_Three       CH₂CH₂SMe
CH₂SCF_Three       CH₂CH₂S (O) Me
CH₂SCF_Three       CH₂CH₂S (O)₂Me
CH₂SCF_Three       D2-32a
CH₂SCF_Three       D2-33a
CH₂SCF_Three       D2-34a
CH₂SCF_Three       D2-37a
CH₂SCF_Three       D2-81a
CH₂SCF_Three       D2-82a
CH₂SCF_Three       D2-84a
CH₂SCF_Three       D2-85a
CH₂SCF_Three       D2-87a
CH₂SCF_Three       D2-92a
CH₂SCF_Three       D2-93a
CH₂SCF_Three       D2-95a
CH₂SCF_Three       D2-96a
CH₂SCF_Three       D2-98a
CH₂SCF_Three      D2-108a
CH₂SCF_Three       D2-108b (Z²= 2-Cl)
CH₂SCF_Three       D2-108b (Z²= 3-Me)
CH₂SCF_Three       D2-108b (Z²= 4-OMe)
CH₂SCF_Three       D2-108b (Z²= 2-SMe)
CH₂SCF_Three       D2-108b (Z²= 3-CF_Three)
CH₂SCF_Three       D2-108b (Z²= 4-OCF_Three)
CH₂SCF_Three       D2-108b (Z²= 2-SCF_Three)
CH₂SCF_Three       C (O) Me
CH₂SCF_Three       C (O) CF_Three
CH₂SCF_Three       C (O) OMe
CH₂S (O) CF_Three    Me
CH₂S (O) CF_Three    Et
CH₂S (O) CF_Three    Pr-n
CH₂S (O) CF_Three    Pr-i
CH₂S (O) CF_Three    Pr-c
CH₂S (O) CF_Three    Bu-n
CH₂S (O) CF_Three    Bu-i
CH₂S (O) CF_Three    Bu-c
CH₂S (O) CF_Three    Bu-s
CH₂S (O) CF_Three    Bu-t
CH₂S (O) CF_Three    Pen-n
CH₂S (O) CF_Three    Pen-c
CH₂S (O) CF_Three    Hex-n
CH₂S (O) CF_Three    Hex-c
CH₂S (O) CF_Three    CH₂Pr-c
CH₂S (O) CF_Three    CH₂Bu-c
CH₂S (O) CF_Three    CH₂Pen-c
CH₂S (O) CF_Three    CH₂Hex-c
CH₂S (O) CF_Three    CH₂CH = CH₂
CH₂S (O) CF_Three    CH₂CH = C (Cl)₂
CH₂S (O) CF_Three    CH₂C≡CH
CH₂S (O) CF_Three    CH₂CN
CH₂S (O) CF_Three    CH₂CF_Three
CH₂S (O) CF_Three    CH₂OMe
CH₂S (O) CF_Three    CH₂OCF_Three
CH₂S (O) CF_Three    CH₂SMe
CH₂S (O) CF_Three    CH₂S (O) Me
CH₂S (O) CF_Three    CH₂S (O)₂Me
CH₂S (O) CF_Three    CH₂SCF_Three
CH₂S (O) CF_Three    CH₂S (O) CF_Three
CH₂S (O) CF_Three    CH₂S (O)₂CF_Three
CH₂S (O) CF_Three    CH₂CH (OMe)₂
CH₂S (O) CF_Three    CH₂CH (SMe)₂
CH₂S (O) CF_Three    CH₂C (O) Me
CH₂S (O) CF_Three    CH₂C (O) CF_Three
CH₂S (O) CF_Three    CH₂C (O) OMe
CH₂S (O) CF_Three    CH₂(D2-32a)
CH₂S (O) CF_Three    CH₂(D2-33a)
CH₂S (O) CF_Three    CH₂(D2-34a)
CH₂S (O) CF_Three    CH₂(D2-37a)
CH₂S (O) CF_Three    CH₂(D2-81a)
CH₂S (O) CF_Three    CH₂(D2-82a)
CH₂S (O) CF_Three    CH₂(D2-84a)
CH₂S (O) CF_Three    CH₂(D2-85a)
CH₂S (O) CF_Three    CH₂(D2-87a)
CH₂S (O) CF_Three    CH₂(D2-92a)
CH₂S (O) CF_Three    CH₂(D2-93a)
CH₂S (O) CF_Three    CH₂(D2-95a)
CH₂S (O) CF_Three    CH₂(D2-96a)
CH₂S (O) CF_Three    CH₂(D2-98a)
CH₂S (O) CF_Three    CH₂(D2-108a)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 2-Cl)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 3-Me)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 4-OMe)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 2-SMe)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 3-CF_Three)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂S (O) CF_Three    CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂S (O) CF_Three    CH₂CH₂CN
CH₂S (O) CF_Three    CH₂CH₂CF_Three
CH₂S (O) CF_Three    CH₂CH₂OMe
CH₂S (O) CF_Three    CH₂CH₂SMe
CH₂S (O) CF_Three    CH₂CH₂S (O) Me
CH₂S (O) CF_Three    CH₂CH₂S (O)₂Me
CH₂S (O) CF_Three    D2-32a
CH₂S (O) CF_Three    D2-33a
CH₂S (O) CF_Three    D2-34a
CH₂S (O) CF_Three    D2-37a
CH₂S (O) CF_Three    D2-81a
CH₂S (O) CF_Three    D2-82a
CH₂S (O) CF_Three    D2-84a
CH₂S (O) CF_Three    D2-85a
CH₂S (O) CF_Three    D2-87a
CH₂S (O) CF_Three    D2-92a
CH₂S (O) CF_Three    D2-93a
CH₂S (O) CF_Three    D2-95a
CH₂S (O) CF_Three    D2-96a
CH₂S (O) CF_Three    D2-98a
CH₂S (O) CF_Three    D2-108a
CH₂S (O) CF_Three    D2-108b (Z²= 2-Cl)
CH₂S (O) CF_Three    D2-108b (Z²= 3-Me)
CH₂S (O) CF_Three    D2-108b (Z²= 4-OMe)
CH₂S (O) CF_Three    D2-108b (Z²= 2-SMe)
CH₂S (O) CF_Three    D2-108b (Z²= 3-CF_Three)
CH₂S (O) CF_Three    D2-108b (Z²= 4-OCF_Three)
CH₂S (O) CF_Three    D2-108b (Z²= 2-SCF_Three)
CH₂S (O) CF_Three    C (O) Me
CH₂S (O) CF_Three    C (O) CF_Three
CH₂S (O) CF_Three    C (O) OMe
CH₂S (O)₂CF_Three    Me
CH₂S (O)₂CF_Three    Et
CH₂S (O)₂CF_Three    Pr-n
CH₂S (O)₂CF_Three    Pr-i
CH₂S (O)₂CF_Three    Pr-c
CH₂S (O)₂CF_Three    Bu-n
CH₂S (O)₂CF_Three    Bu-i
CH₂S (O)₂CF_Three    Bu-c
CH₂S (O)₂CF_Three    Bu-s
CH₂S (O)₂CF_Three    Bu-t
CH₂S (O)₂CF_Three    Pen-n
CH₂S (O)₂CF_Three    Pen-c
CH₂S (O)₂CF_Three    Hex-n
CH₂S (O)₂CF_Three    Hex-c
CH₂S (O)₂CF_Three    CH₂Pr-c
CH₂S (O)₂CF_Three    CH₂Bu-c
CH₂S (O)₂CF_Three    CH₂Pen-c
CH₂S (O)₂CF_Three    CH₂Hex-c
CH₂S (O)₂CF_Three    CH₂CH = CH₂
CH₂S (O)₂CF_Three    CH₂CH = C (Cl)₂
CH₂S (O)₂CF_Three    CH₂C≡CH
CH₂S (O)₂CF_Three    CH₂CN
CH₂S (O)₂CF_Three    CH₂CF_Three
CH₂S (O)₂CF_Three    CH₂OMe
CH₂S (O)₂CF_Three    CH₂OCF_Three
CH₂S (O)₂CF_Three    CH₂SMe
CH₂S (O)₂CF_Three    CH₂S (O) Me
CH₂S (O)₂CF_Three    CH₂S (O)₂Me
CH₂S (O)₂CF_Three    CH₂SCF_Three
CH₂S (O)₂CF_Three    CH₂S (O) CF_Three
CH₂S (O)₂CF_Three    CH₂S (O)₂CF_Three
CH₂S (O)₂CF_Three    CH₂CH (OMe)₂
CH₂S (O)₂CF_Three    CH₂CH (SMe)₂
CH₂S (O)₂CF_Three    CH₂C (O) Me
CH₂S (O)₂CF_Three    CH₂C (O) CF_Three
CH₂S (O)₂CF_Three    CH₂C (O) OMe
CH₂S (O)₂CF_Three    CH₂(D2-32a)
CH₂S (O)₂CF_Three    CH₂(D2-33a)
CH₂S (O)₂CF_Three    CH₂(D2-34a)
CH₂S (O)₂CF_Three    CH₂(D2-37a)
CH₂S (O)₂CF_Three    CH₂(D2-81a)
CH₂S (O)₂CF_Three    CH₂(D2-82a)
CH₂S (O)₂CF_Three    CH₂(D2-84a)
CH₂S (O)₂CF_Three    CH₂(D2-85a)
CH₂S (O)₂CF_Three    CH₂(D2-87a)
CH₂S (O)₂CF_Three    CH₂(D2-92a)
CH₂S (O)₂CF_Three    CH₂(D2-93a)
CH₂S (O)₂CF_Three    CH₂(D2-95a)
CH₂S (O)₂CF_Three    CH₂(D2-96a)
CH₂S (O)₂CF_Three    CH₂(D2-98a)
CH₂S (O)₂CF_Three    CH₂(D2-108a)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 2-Cl)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 3-Me)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 4-OMe)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 2-SMe)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 3-CF_Three)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 4-OCF_Three)
CH₂S (O)₂CF_Three    CH₂(D2-108b, Z²= 2-SCF_Three)
CH₂S (O)₂CF_Three    CH₂CH₂CN
CH₂S (O)₂CF_Three    CH₂CH₂CF_Three
CH₂S (O)₂CF_Three    CH₂CH₂OMe
CH₂S (O)₂CF_Three    CH₂CH₂SMe
CH₂S (O)₂CF_Three    CH₂CH₂S (O) Me
CH₂S (O)₂CF_Three    CH₂CH₂S (O)₂Me
CH₂S (O)₂CF_Three    D2-32a
CH₂S (O)₂CF_Three    D2-33a
CH₂S (O)₂CF_Three    D2-34a
CH₂S (O)₂CF_Three    D2-37a
CH₂S (O)₂CF_Three    D2-81a
CH₂S (O)₂CF_Three    D2-82a
CH₂S (O)₂CF_Three    D2-84a
CH₂S (O)₂CF_Three    D2-85a
CH₂S (O)₂CF_Three    D2-87a
CH₂S (O)₂CF_Three    D2-92a
CH₂S (O)₂CF_Three    D2-93a
CH₂S (O)₂CF_Three    D2-95a
CH₂S (O)₂CF_Three    D2-96a
CH₂S (O)₂CF_Three    D2-98a
CH₂S (O)₂CF_Three    D2-108a
CH₂S (O)₂CF_Three    D2-108b (Z²= 2-Cl)
CH₂S (O)₂CF_Three    D2-108b (Z²= 3-Me)
CH₂S (O)₂CF_Three    D2-108b (Z²= 4-OMe)
CH₂S (O)₂CF_Three    D2-108b (Z²= 2-SMe)
CH₂S (O)₂CF_Three    D2-108b (Z²= 3-CF_Three)
CH₂S (O)₂CF_Three    D2-108b (Z²= 4-OCF_Three)
CH₂S (O)₂CF_Three    D2-108b (Z²= 2-SCF_Three)
CH₂S (O)₂CF_Three    C (O) Me
CH₂S (O)₂CF_Three    C (O) CF_Three
CH₂S (O)₂CF_Three    C (O) OMe
D2-32a Me
D2-32a Et
D2-32a Pr-n
D2-32a Pr-i
D2-32a Pr-c
D2-32a Bu-n
D2-32a Bu-i
D2-32a Bu-c
D2-32a Bu-s
D2-32a Bu-t
D2-32a Pen-n
D2-32a Pen-c
D2-32a Hex-n
D2-32a Hex-c
D2-32a CH₂Pr-c
D2-32a CH₂Bu-c
D2-32a CH₂Pen-c
D2-32a CH₂Hex-c
D2-32a CH₂CH = CH₂
D2-32a CH₂CH = C (Cl)₂
D2-32a CH₂C≡CH
D2-32a CH₂CN
D2-32a CH₂CF_Three
D2-32a CH₂OMe
D2-32a CH₂OCF_Three
D2-32a CH₂SMe
D2-32a CH₂S (O) Me
D2-32a CH₂S (O)₂Me
D2-32a CH₂SCF_Three
D2-32a CH₂S (O) CF_Three
D2-32a CH₂S (O)₂CF_Three
D2-32a CH₂CH (OMe)₂
D2-32a CH₂CH (SMe)₂
D2-32a CH₂C (O) Me
D2-32a CH₂C (O) CF_Three
D2-32a CH₂C (O) OMe
D2-32a CH₂(D2-32a)
D2-32a CH₂(D2-33a)
D2-32a CH₂(D2-34a)
D2-32a CH₂(D2-37a)
D2-32a CH₂(D2-81a)
D2-32a CH₂(D2-82a)
D2-32a CH₂(D2-84a)
D2-32a CH₂(D2-85a)
D2-32a CH₂(D2-87a)
D2-32a CH₂(D2-92a)
D2-32a CH₂(D2-93a)
D2-32a CH₂(D2-95a)
D2-32a CH₂(D2-96a)
D2-32a CH₂(D2-98a)
D2-32a CH₂(D2-108a)
D2-32a CH₂(D2-108b, Z²= 2-Cl)
D2-32a CH₂(D2-108b, Z²= 3-Me)
D2-32a CH₂(D2-108b, Z²= 4-OMe)
D2-32a CH₂(D2-108b, Z²= 2-SMe)
D2-32a CH₂(D2-108b, Z²= 3-CF_Three)
D2-32a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-32a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-32a CH₂CH₂CN
D2-32a CH₂CH₂CF_Three
D2-32a CH₂CH₂OMe
D2-32a CH₂CH₂SMe
D2-32a CH₂CH₂S (O) Me
D2-32a CH₂CH₂S (O)₂Me
D2-32a D2-32a
D2-32a D2-33a
D2-32a D2-34a
D2-32a D2-37a
D2-32a D2-81a
D2-32a D2-82a
D2-32a D2-84a
D2-32a D2-85a
D2-32a D2-87a
D2-32a D2-92a
D2-32a D2-93a
D2-32a D2-95a
D2-32a D2-96a
D2-32a D2-98a
D2-32a D2-108a
D2-32a D2-108b (Z²= 2-Cl)
D2-32a D2-108b (Z²= 3-Me)
D2-32a D2-108b (Z²= 4-OMe)
D2-32a D2-108b (Z²= 2-SMe)
D2-32a D2-108b (Z²= 3-CF_Three)
D2-32a D2-108b (Z²= 4-OCF_Three)
D2-32a D2-108b (Z²= 2-SCF_Three)
D2-32a C (O) Me
D2-32a C (O) CF_Three
D2-32a C (O) OMe
D2-33a Me
D2-33a Et
D2-33a Pr-n
D2-33a Pr-i
D2-33a Pr-c
D2-33a Bu-n
D2-33a Bu-i
D2-33a Bu-c
D2-33a Bu-s
D2-33a Bu-t
D2-33a Pen-n
D2-33a Pen-c
D2-33a Hex-n
D2-33a Hex-c
D2-33a CH₂Pr-c
D2-33a CH₂Bu-c
D2-33a CH₂Pen-c
D2-33a CH₂Hex-c
D2-33a CH₂CH = CH₂
D2-33a CH₂CH = C (Cl)₂
D2-33a CH₂C≡CH
D2-33a CH₂CN
D2-33a CH₂CF_Three
D2-33a CH₂OMe
D2-33a CH₂OCF_Three
D2-33a CH₂SMe
D2-33a CH₂S (O) Me
D2-33a CH₂S (O)₂Me
D2-33a CH₂SCF_Three
D2-33a CH₂S (O) CF_Three
D2-33a CH₂S (O)₂CF_Three
D2-33a CH₂CH (OMe)₂
D2-33a CH₂CH (SMe)₂
D2-33a CH₂C (O) Me
D2-33a CH₂C (O) CF_Three
D2-33a CH₂C (O) OMe
D2-33a CH₂(D2-32a)
D2-33a CH₂(D2-33a)
D2-33a CH₂(D2-34a)
D2-33a CH₂(D2-37a)
D2-33a CH₂(D2-81a)
D2-33a CH₂(D2-82a)
D2-33a CH₂(D2-84a)
D2-33a CH₂(D2-85a)
D2-33a CH₂(D2-87a)
D2-33a CH₂(D2-92a)
D2-33a CH₂(D2-93a)
D2-33a CH₂(D2-95a)
D2-33a CH₂(D2-96a)
D2-33a CH₂(D2-98a)
D2-33a CH₂(D2-108a)
D2-33a CH₂(D2-108b, Z²= 2-Cl)
D2-33a CH₂(D2-108b, Z²= 3-Me)
D2-33a CH₂(D2-108b, Z²= 4-OMe)
D2-33a CH₂(D2-108b, Z²= 2-SMe)
D2-33a CH₂(D2-108b, Z²= 3-CF_Three)
D2-33a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-33a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-33a CH₂CH₂CN
D2-33a CH₂CH₂CF_Three
D2-33a CH₂CH₂OMe
D2-33a CH₂CH₂SMe
D2-33a CH₂CH₂S (O) Me
D2-33a CH₂CH₂S (O)₂Me
D2-33a D2-32a
D2-33a D2-33a
D2-33a D2-34a
D2-33a D2-37a
D2-33a D2-81a
D2-33a D2-82a
D2-33a D2-84a
D2-33a D2-85a
D2-33a D2-87a
D2-33a D2-92a
D2-33a D2-93a
D2-33a D2-95a
D2-33a D2-96a
D2-33a D2-98a
D2-33a D2-108a
D2-33a D2-108b (Z²= 2-Cl)
D2-33a D2-108b (Z²= 3-Me)
D2-33a D2-108b (Z²= 4-OMe)
D2-33a D2-108b (Z²= 2-SMe)
D2-33a D2-108b (Z²= 3-CF_Three)
D2-33a D2-108b (Z²= 4-OCF_Three)
D2-33a D2-108b (Z²= 2-SCF_Three)
D2-33a C (O) Me
D2-33a C (O) CF_Three
D2-33a C (O) OMe
D2-34a Me
D2-34a Et
D2-34a Pr-n
D2-34a Pr-i
D2-34a Pr-c
D2-34a Bu-n
D2-34a Bu-i
D2-34a Bu-c
D2-34a Bu-s
D2-34a Bu-t
D2-34a Pen-n
D2-34a Pen-c
D2-34a Hex-n
D2-34a Hex-c
D2-34a CH₂Pr-c
D2-34a CH₂Bu-c
D2-34a CH₂Pen-c
D2-34a CH₂Hex-c
D2-34a CH₂CH = CH₂
D2-34a CH₂CH = C (Cl)₂
D2-34a CH₂C≡CH
D2-34a CH₂CN
D2-34a CH₂CF_Three
D2-34a CH₂OMe
D2-34a CH₂OCF_Three
D2-34a CH₂SMe
D2-34a CH₂S (O) Me
D2-34a CH₂S (O)₂Me
D2-34a CH₂SCF_Three
D2-34a CH₂S (O) CF_Three
D2-34a CH₂S (O)₂CF_Three
D2-34a CH₂CH (OMe)₂
D2-34a CH₂CH (SMe)₂
D2-34a CH₂C (O) Me
D2-34a CH₂C (O) CF_Three
D2-34a CH₂C (O) OMe
D2-34a CH₂(D2-32a)
D2-34a CH₂(D2-33a)
D2-34a CH₂(D2-34a)
D2-34a CH₂(D2-37a)
D2-34a CH₂(D2-81a)
D2-34a CH₂(D2-82a)
D2-34a CH₂(D2-84a)
D2-34a CH₂(D2-85a)
D2-34a CH₂(D2-87a)
D2-34a CH₂(D2-92a)
D2-34a CH₂(D2-93a)
D2-34a CH₂(D2-95a)
D2-34a CH₂(D2-96a)
D2-34a CH₂(D2-98a)
D2-34a CH₂(D2-108a)
D2-34a CH₂(D2-108b, Z²= 2-Cl)
D2-34a CH₂(D2-108b, Z²= 3-Me)
D2-34a CH₂(D2-108b, Z²= 4-OMe)
D2-34a CH₂(D2-108b, Z²= 2-SMe)
D2-34a CH₂(D2-108b, Z²= 3-CF_Three)
D2-34a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-34a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-34a CH₂CH₂CN
D2-34a CH₂CH₂CF_Three
D2-34a CH₂CH₂OMe
D2-34a CH₂CH₂SMe
D2-34a CH₂CH₂S (O) Me
D2-34a CH₂CH₂S (O)₂Me
D2-34a D2-32a
D2-34a D2-33a
D2-34a D2-34a
D2-34a D2-37a
D2-34a D2-81a
D2-34a D2-82a
D2-34a D2-84a
D2-34a D2-85a
D2-34a D2-87a
D2-34a D2-92a
D2-34a D2-93a
D2-34a D2-95a
D2-34a D2-96a
D2-34a D2-98a
D2-34a D2-108a
D2-34a D2-108b (Z²= 2-Cl)
D2-34a D2-108b (Z²= 3-Me)
D2-34a D2-108b (Z²= 4-OMe)
D2-34a D2-108b (Z²= 2-SMe)
D2-34a D2-108b (Z²= 3-CF_Three)
D2-34a D2-108b (Z²= 4-OCF_Three)
D2-34a D2-108b (Z²= 2-SCF_Three)
D2-34a C (O) Me
D2-34a C (O) CF_Three
D2-34a C (O) OMe
D2-37a Me
D2-37a Et
D2-37a Pr-n
D2-37a Pr-i
D2-37a Pr-c
D2-37a Bu-n
D2-37a Bu-i
D2-37a Bu-c
D2-37a Bu-s
D2-37a Bu-t
D2-37a Pen-n
D2-37a Pen-c
D2-37a Hex-n
D2-37a Hex-c
D2-37a CH₂Pr-c
D2-37a CH₂Bu-c
D2-37a CH₂Pen-c
D2-37a CH₂Hex-c
D2-37a CH₂CH = CH₂
D2-37a CH₂CH = C (Cl)₂
D2-37a CH₂C≡CH
D2-37a CH₂CN
D2-37a CH₂CF_Three
D2-37a CH₂OMe
D2-37a CH₂OCF_Three
D2-37a CH₂SMe
D2-37a CH₂S (O) Me
D2-37a CH₂S (O)₂Me
D2-37a CH₂SCF_Three
D2-37a CH₂S (O) CF_Three
D2-37a CH₂S (O)₂CF_Three
D2-37a CH₂CH (OMe)₂
D2-37a CH₂CH (SMe)₂
D2-37a CH₂C (O) Me
D2-37a CH₂C (O) CF_Three
D2-37a CH₂C (O) OMe
D2-37a CH₂(D2-32a)
D2-37a CH₂(D2-33a)
D2-37a CH₂(D2-34a)
D2-37a CH₂(D2-37a)
D2-37a CH₂(D2-81a)
D2-37a CH₂(D2-82a)
D2-37a CH₂(D2-84a)
D2-37a CH₂(D2-85a)
D2-37a CH₂(D2-87a)
D2-37a CH₂(D2-92a)
D2-37a CH₂(D2-93a)
D2-37a CH₂(D2-95a)
D2-37a CH₂(D2-96a)
D2-37a CH₂(D2-98a)
D2-37a CH₂(D2-108a)
D2-37a CH₂(D2-108b, Z²= 2-Cl)
D2-37a CH₂(D2-108b, Z²= 3-Me)
D2-37a CH₂(D2-108b, Z²= 4-OMe)
D2-37a CH₂(D2-108b, Z²= 2-SMe)
D2-37a CH₂(D2-108b, Z²= 3-CF_Three)
D2-37a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-37a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-37a CH₂CH₂CN
D2-37a CH₂CH₂CF_Three
D2-37a CH₂CH₂OMe
D2-37a CH₂CH₂SMe
D2-37a CH₂CH₂S (O) Me
D2-37a CH₂CH₂S (O)₂Me
D2-37a D2-32a
D2-37a D2-33a
D2-37a D2-34a
D2-37a D2-37a
D2-37a D2-81a
D2-37a D2-82a
D2-37a D2-84a
D2-37a D2-85a
D2-37a D2-87a
D2-37a D2-92a
D2-37a D2-93a
D2-37a D2-95a
D2-37a D2-96a
D2-37a D2-98a
D2-37a D2-108a
D2-37a D2-108b (Z²= 2-Cl)
D2-37a D2-108b (Z²= 3-Me)
D2-37a D2-108b (Z²= 4-OMe)
D2-37a D2-108b (Z²= 2-SMe)
D2-37a D2-108b (Z²= 3-CF_Three)
D2-37a D2-108b (Z²= 4-OCF_Three)
D2-37a D2-108b (Z²= 2-SCF_Three)
D2-37a C (O) Me
D2-37a C (O) CF_Three
D2-37a C (O) OMe
D2-81a Me
D2-81a Et
D2-81a Pr-n
D2-81a Pr-i
D2-81a Pr-c
D2-81a Bu-n
D2-81a Bu-i
D2-81a Bu-c
D2-81a Bu-s
D2-81a Bu-t
D2-81a Pen-n
D2-81a Pen-c
D2-81a Hex-n
D2-81a Hex-c
D2-81a CH₂Pr-c
D2-81a CH₂Bu-c
D2-81a CH₂Pen-c
D2-81a CH₂Hex-c
D2-81a CH₂CH = CH₂
D2-81a CH₂CH = C (Cl)₂
D2-81a CH₂C≡CH
D2-81a CH₂CN
D2-81a CH₂CF_Three
D2-81a CH₂OMe
D2-81a CH₂OCF_Three
D2-81a CH₂SMe
D2-81a CH₂S (O) Me
D2-81a CH₂S (O)₂Me
D2-81a CH₂SCF_Three
D2-81a CH₂S (O) CF_Three
D2-81a CH₂S (O)₂CF_Three
D2-81a CH₂CH (OMe)₂
D2-81a CH₂CH (SMe)₂
D2-81a CH₂C (O) Me
D2-81a CH₂C (O) CF_Three
D2-81a CH₂C (O) OMe
D2-81a CH₂(D2-32a)
D2-81a CH₂(D2-33a)
D2-81a CH₂(D2-34a)
D2-81a CH₂(D2-37a)
D2-81a CH₂(D2-81a)
D2-81a CH₂(D2-82a)
D2-81a CH₂(D2-84a)
D2-81a CH₂(D2-85a)
D2-81a CH₂(D2-87a)
D2-81a CH₂(D2-92a)
D2-81a CH₂(D2-93a)
D2-81a CH₂(D2-95a)
D2-81a CH₂(D2-96a)
D2-81a CH₂(D2-98a)
D2-81a CH₂(D2-108a)
D2-81a CH₂(D2-108b, Z²= 2-Cl)
D2-81a CH₂(D2-108b, Z²= 3-Me)
D2-81a CH₂(D2-108b, Z²= 4-OMe)
D2-81a CH₂(D2-108b, Z²= 2-SMe)
D2-81a CH₂(D2-108b, Z²= 3-CF_Three)
D2-81a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-81a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-81a CH₂CH₂CN
D2-81a CH₂CH₂CF_Three
D2-81a CH₂CH₂OMe
D2-81a CH₂CH₂SMe
D2-81a CH₂CH₂S (O) Me
D2-81a CH₂CH₂S (O)₂Me
D2-81a D2-32a
D2-81a D2-33a
D2-81a D2-34a
D2-81a D2-37a
D2-81a D2-81a
D2-81a D2-82a
D2-81a D2-84a
D2-81a D2-85a
D2-81a D2-87a
D2-81a D2-92a
D2-81a D2-93a
D2-81a D2-95a
D2-81a D2-96a
D2-81a D2-98a
D2-81a D2-108a
D2-81a D2-108b (Z²= 2-Cl)
D2-81a D2-108b (Z²= 3-Me)
D2-81a D2-108b (Z²= 4-OMe)
D2-81a D2-108b (Z²= 2-SMe)
D2-81a D2-108b (Z²= 3-CF_Three)
D2-81a D2-108b (Z²= 4-OCF_Three)
D2-81a D2-108b (Z²= 2-SCF_Three)
D2-81a C (O) Me
D2-81a C (O) CF_Three
D2-81a C (O) OMe
D2-82a Me
D2-82a Et
D2-82a Pr-n
D2-82a Pr-i
D2-82a Pr-c
D2-82a Bu-n
D2-82a Bu-i
D2-82a Bu-c
D2-82a Bu-s
D2-82a Bu-t
D2-82a Pen-n
D2-82a Pen-c
D2-82a Hex-n
D2-82a Hex-c
D2-82a CH₂Pr-c
D2-82a CH₂Bu-c
D2-82a CH₂Pen-c
D2-82a CH₂Hex-c
D2-82a CH₂CH = CH₂
D2-82a CH₂CH = C (Cl)₂
D2-82a CH₂C≡CH
D2-82a CH₂CN
D2-82a CH₂CF_Three
D2-82a CH₂OMe
D2-82a CH₂OCF_Three
D2-82a CH₂SMe
D2-82a CH₂S (O) Me
D2-82a CH₂S (O)₂Me
D2-82a CH₂SCF_Three
D2-82a CH₂S (O) CF_Three
D2-82a CH₂S (O)₂CF_Three
D2-82a CH₂CH (OMe)₂
D2-82a CH₂CH (SMe)₂
D2-82a CH₂C (O) Me
D2-82a CH₂C (O) CF_Three
D2-82a CH₂C (O) OMe
D2-82a CH₂(D2-32a)
D2-82a CH₂(D2-33a)
D2-82a CH₂(D2-34a)
D2-82a CH₂(D2-37a)
D2-82a CH₂(D2-81a)
D2-82a CH₂(D2-82a)
D2-82a CH₂(D2-84a)
D2-82a CH₂(D2-85a)
D2-82a CH₂(D2-87a)
D2-82a CH₂(D2-92a)
D2-82a CH₂(D2-93a)
D2-82a CH₂(D2-95a)
D2-82a CH₂(D2-96a)
D2-82a CH₂(D2-98a)
D2-82a CH₂(D2-108a)
D2-82a CH₂(D2-108b, Z²= 2-Cl)
D2-82a CH₂(D2-108b, Z²= 3-Me)
D2-82a CH₂(D2-108b, Z²= 4-OMe)
D2-82a CH₂(D2-108b, Z²= 2-SMe)
D2-82a CH₂(D2-108b, Z²= 3-CF_Three)
D2-82a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-82a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-82a CH₂CH₂CN
D2-82a CH₂CH₂CF_Three
D2-82a CH₂CH₂OMe
D2-82a CH₂CH₂SMe
D2-82a CH₂CH₂S (O) Me
D2-82a CH₂CH₂S (O)₂Me
D2-82a D2-32a
D2-82a D2-33a
D2-82a D2-34a
D2-82a D2-37a
D2-82a D2-81a
D2-82a D2-82a
D2-82a D2-84a
D2-82a D2-85a
D2-82a D2-87a
D2-82a D2-92a
D2-82a D2-93a
D2-82a D2-95a
D2-82a D2-96a
D2-82a D2-98a
D2-82a D2-108a
D2-82a D2-108b (Z²= 2-Cl)
D2-82a D2-108b (Z²= 3-Me)
D2-82a D2-108b (Z²= 4-OMe)
D2-82a D2-108b (Z²= 2-SMe)
D2-82a D2-108b (Z²= 3-CF_Three)
D2-82a D2-108b (Z²= 4-OCF_Three)
D2-82a D2-108b (Z²= 2-SCF_Three)
D2-82a C (O) Me
D2-82a C (O) CF_Three
D2-82a C (O) OMe
D2-84a Me
D2-84a Et
D2-84a Pr-n
D2-84a Pr-i
D2-84a Pr-c
D2-84a Bu-n
D2-84a Bu-i
D2-84a Bu-c
D2-84a Bu-s
D2-84a Bu-t
D2-84a Pen-n
D2-84a Pen-c
D2-84a Hex-n
D2-84a Hex-c
D2-84a CH₂Pr-c
D2-84a CH₂Bu-c
D2-84a CH₂Pen-c
D2-84a CH₂Hex-c
D2-84a CH₂CH = CH₂
D2-84a CH₂CH = C (Cl)₂
D2-84a CH₂C≡CH
D2-84a CH₂CN
D2-84a CH₂CF_Three
D2-84a CH₂OMe
D2-84a CH₂OCF_Three
D2-84a CH₂SMe
D2-84a CH₂S (O) Me
D2-84a CH₂S (O)₂Me
D2-84a CH₂SCF_Three
D2-84a CH₂S (O) CF_Three
D2-84a CH₂S (O)₂CF_Three
D2-84a CH₂CH (OMe)₂
D2-84a CH₂CH (SMe)₂
D2-84a CH₂C (O) Me
D2-84a CH₂C (O) CF_Three
D2-84a CH₂C (O) OMe
D2-84a CH₂(D2-32a)
D2-84a CH₂(D2-33a)
D2-84a CH₂(D2-34a)
D2-84a CH₂(D2-37a)
D2-84a CH₂(D2-81a)
D2-84a CH₂(D2-82a)
D2-84a CH₂(D2-84a)
D2-84a CH₂(D2-85a)
D2-84a CH₂(D2-87a)
D2-84a CH₂(D2-92a)
D2-84a CH₂(D2-93a)
D2-84a CH₂(D2-95a)
D2-84a CH₂(D2-96a)
D2-84a CH₂(D2-98a)
D2-84a CH₂(D2-108a)
D2-84a CH₂(D2-108b, Z²= 2-Cl)
D2-84a CH₂(D2-108b, Z²= 3-Me)
D2-84a CH₂(D2-108b, Z²= 4-OMe)
D2-84a CH₂(D2-108b, Z =²2-SMe)
D2-84a CH₂(D2-108b, Z²= 3-CF_Three)
D2-84a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-84a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-84a CH₂CH₂CN
D2-84a CH₂CH₂CF_Three
D2-84a CH₂CH₂OMe
D2-84a CH₂CH₂SMe
D2-84a CH₂CH₂S (O) Me
D2-84a CH₂CH₂S (O)₂Me
D2-84a D2-32a
D2-84a D2-33a
D2-84a D2-34a
D2-84a D2-37a
D2-84a D2-81a
D2-84a D2-82a
D2-84a D2-84a
D2-84a D2-85a
D2-84a D2-87a
D2-84a D2-92a
D2-84a D2-93a
D2-84a D2-95a
D2-84a D2-96a
D2-84a D2-98a
D2-84a D2-108a
D2-84a D2-108b (Z²= 2-Cl)
D2-84a D2-108b (Z²= 3-Me)
D2-84a D2-108b (Z²= 4-OMe)
D2-84a D2-108b (Z²= 2-SMe)
D2-84a D2-108b (Z²= 3-CF_Three)
D2-84a D2-108b (Z²= 4-OCF_Three)
D2-84a D2-108b (Z²= 2-SCF_Three)
D2-84a C (O) Me
D2-84a C (O) CF_Three
D2-84a C (O) OMe
D2-85a Me
D2-85a Et
D2-85a Pr-n
D2-85a Pr-i
D2-85a Pr-c
D2-85a Bu-n
D2-85a Bu-i
D2-85a Bu-c
D2-85a Bu-s
D2-85a Bu-t
D2-85a Pen-n
D2-85a Pen-c
D2-85a Hex-n
D2-85a Hex-c
D2-85a CH₂Pr-c
D2-85a CH₂Bu-c
D2-85a CH₂Pen-c
D2-85a CH₂Hex-c
D2-85a CH₂CH = CH₂
D2-85a CH₂CH = C (Cl)₂
D2-85a CH₂C≡CH
D2-85a CH₂CN
D2-85a CH₂CF_Three
D2-85a CH₂OMe
D2-85a CH₂OCF_Three
D2-85a CH₂SMe
D2-85a CH₂S (O) Me
D2-85a CH₂S (O)₂Me
D2-85a CH₂SCF_Three
D2-85a CH₂S (O) CF_Three
D2-85a CH₂S (O)₂CF_Three
D2-85a CH₂CH (OMe)₂
D2-85a CH₂CH (SMe)₂
D2-85a CH₂C (O) Me
D2-85a CH₂C (O) CF_Three
D2-85a CH₂C (O) OMe
D2-85a CH₂(D2-32a)
D2-85a CH₂(D2-33a)
D2-85a CH₂(D2-34a)
D2-85a CH₂(D2-37a)
D2-85a CH₂(D2-81a)
D2-85a CH₂(D2-82a)
D2-85a CH₂(D2-84a)
D2-85a CH₂(D2-85a)
D2-85a CH₂(D2-87a)
D2-85a CH₂(D2-92a)
D2-85a CH₂(D2-93a)
D2-85a CH₂(D2-95a)
D2-85a CH₂(D2-96a)
D2-85a CH₂(D2-98a)
D2-85a CH₂(D2-108a)
D2-85a CH₂(D2-108b, Z²= 2-Cl)
D2-85a CH₂(D2-108b, Z²= 3-Me)
D2-85a CH₂(D2-108b, Z²= 4-OMe)
D2-85a CH₂(D2-108b, Z²= 2-SMe)
D2-85a CH₂(D2-108b, Z²= 3-CF_Three)
D2-85a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-85a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-85a CH₂CH₂CN
D2-85a CH₂CH₂CF_Three
D2-85a CH₂CH₂OMe
D2-85a CH₂CH₂SMe
D2-85a CH₂CH₂S (O) Me
D2-85a CH₂CH₂S (O)₂Me
D2-85a D2-32a
D2-85a D2-33a
D2-85a D2-34a
D2-85a D2-37a
D2-85a D2-81a
D2-85a D2-82a
D2-85a D2-84a
D2-85a D2-85a
D2-85a D2-87a
D2-85a D2-92a
D2-85a D2-93a
D2-85a D2-95a
D2-85a D2-96a
D2-85a D2-98a
D2-85a D2-108a
D2-85a D2-108b (Z²= 2-Cl)
D2-85a D2-108b (Z²= 3-Me)
D2-85a D2-108b (Z²= 4-OMe)
D2-85a D2-108b (Z²= 2-SMe)
D2-85a D2-108b (Z²= 3-CF_Three)
D2-85a D2-108b (Z²= 4-OCF_Three)
D2-85a D2-108b (Z²= 2-SCF_Three)
D2-85a C (O) Me
D2-85a C (O) CF_Three
D2-85a C (O) OMe
D2-87a Me
D2-87a Et
D2-87a Pr-n
D2-87a Pr-i
D2-87a Pr-c
D2-87a Bu-n
D2-87a Bu-i
D2-87a Bu-c
D2-87a Bu-s
D2-87a Bu-t
D2-87a Pen-n
D2-87a Pen-c
D2-87a Hex-n
D2-87a Hex-c
D2-87a CH₂Pr-c
D2-87a CH₂Bu-c
D2-87a CH₂Pen-c
D2-87a CH₂Hex-c
D2-87a CH₂CH = CH₂
D2-87a CH₂CH = C (Cl)₂
D2-87a CH₂C≡CH
D2-87a CH₂CN
D2-87a CH₂CF_Three
D2-87a CH₂OMe
D2-87a CH₂OCF_Three
D2-87a CH₂SMe
D2-87a CH₂S (O) Me
D2-87a CH₂S (O)₂Me
D2-87a CH₂SCF_Three
D2-87a CH₂S (O) CF_Three
D2-87a CH₂S (O)₂CF_Three
D2-87a CH₂CH (OMe)₂
D2-87a CH₂CH (SMe)₂
D2-87a CH₂C (O) Me
D2-87a CH₂C (O) CF_Three
D2-87a CH₂C (O) OMe
D2-87a CH₂(D2-32a)
D2-87a CH₂(D2-33a)
D2-87a CH₂(D2-34a)
D2-87a CH₂(D2-37a)
D2-87a CH₂(D2-81a)
D2-87a CH₂(D2-82a)
D2-87a CH₂(D2-84a)
D2-87a CH₂(D2-85a)
D2-87a CH₂(D2-87a)
D2-87a CH₂(D2-92a)
D2-87a CH₂(D2-93a)
D2-87a CH₂(D2-95a)
D2-87a CH₂(D2-96a)
D2-87a CH₂(D2-98a)
D2-87a CH₂(D2-108a)
D2-87a CH₂(D2-108b, Z²= 2-Cl)
D2-87a CH₂(D2-108b, Z²= 3-Me)
D2-87a CH₂(D2-108b, Z²= 4-OMe)
D2-87a CH₂(D2-108b, Z²= 2-SMe)
D2-87a CH₂(D2-108b, Z²= 3-CF_Three)
D2-87a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-87a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-87a CH₂CH₂CN
D2-87a CH₂CH₂CF_Three
D2-87a CH₂CH₂OMe
D2-87a CH₂CH₂SMe
D2-87a CH₂CH₂S (O) Me
D2-87a CH₂CH₂S (O)₂Me
D2-87a D2-32a
D2-87a D2-33a
D2-87a D2-34a
D2-87a D2-37a
D2-87a D2-81a
D2-87a D2-82a
D2-87a D2-84a
D2-87a D2-85a
D2-87a D2-87a
D2-87a D2-92a
D2-87a D2-93a
D2-87a D2-95a
D2-87a D2-96a
D2-87a D2-98a
D2-87a D2-108a
D2-87a D2-108b (Z²= 2-Cl)
D2-87a D2-108b (Z²= 3-Me)
D2-87a D2-108b (Z²= 4-OMe)
D2-87a D2-108b (Z²= 2-SMe)
D2-87a D2-108b (Z²= 3-CF_Three)
D2-87a D2-108b (Z²= 4-OCF_Three)
D2-87a D2-108b (Z²= 2-SCF_Three)
D2-87a C (O) Me
D2-87a C (O) CF_Three
D2-87a C (O) OMe
D2-92a Me
D2-92a Et
D2-92a Pr-n
D2-92a Pr-i
D2-92a Pr-c
D2-92a Bu-n
D2-92a Bu-i
D2-92a Bu-c
D2-92a Bu-s
D2-92a Bu-t
D2-92a Pen-n
D2-92a Pen-c
D2-92a Hex-n
D2-92a Hex-c
D2-92a CH₂Pr-c
D2-92a CH₂Bu-c
D2-92a CH₂Pen-c
D2-92a CH₂Hex-c
D2-92a CH₂CH = CH₂
D2-92a CH₂CH = C (Cl)₂
D2-92a CH₂C≡CH
D2-92a CH₂CN
D2-92a CH₂CF_Three
D2-92a CH₂OMe
D2-92a CH₂OCF_Three
D2-92a CH₂SMe
D2-92a CH₂S (O) Me
D2-92a CH₂S (O)₂Me
D2-92a CH₂SCF_Three
D2-92a CH₂S (O) CF_Three
D2-92a CH₂S (O)₂CF_Three
D2-92a CH₂CH (OMe)₂
D2-92a CH₂CH (SMe)₂
D2-92a CH₂C (O) Me
D2-92a CH₂C (O) CF_Three
D2-92a CH₂C (O) OMe
D2-92a CH₂(D2-32a)
D2-92a CH₂(D2-33a)
D2-92a CH₂(D2-34a)
D2-92a CH₂(D2-37a)
D2-92a CH₂(D2-81a)
D2-92a CH₂(D2-82a)
D2-92a CH₂(D2-84a)
D2-92a CH₂(D2-85a)
D2-92a CH₂(D2-87a)
D2-92a CH₂(D2-92a)
D2-92a CH₂(D2-93a)
D2-92a CH₂(D2-95a)
D2-92a CH₂(D2-96a)
D2-92a CH₂(D2-98a)
D2-92a CH₂(D2-108a)
D2-92a CH₂(D2-108b, Z²= 2-Cl)
D2-92a CH₂(D2-108b, Z²= 3-Me)
D2-92a CH₂(D2-108b, Z²= 4-OMe)
D2-92a CH₂(D2-108b, Z²= 2-SMe)
D2-92a CH₂(D2-108b, Z²= 3-CF_Three)
D2-92a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-92a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-92a CH₂CH₂CN
D2-92a CH₂CH₂CF_Three
D2-92a CH₂CH₂OMe
D2-92a CH₂CH₂SMe
D2-92a CH₂CH₂S (O) Me
D2-92a CH₂CH₂S (O)₂Me
D2-92a D2-32a
D2-92a D2-33a
D2-92a D2-34a
D2-92a D2-37a
D2-92a D2-81a
D2-92a D2-82a
D2-92a D2-84a
D2-92a D2-85a
D2-92a D2-87a
D2-92a D2-92a
D2-92a D2-93a
D2-92a D2-95a
D2-92a D2-96a
D2-92a D2-98a
D2-92a D2-108a
D2-92a D2-108b (Z²= 2-Cl)
D2-92a D2-108b (Z²= 3-Me)
D2-92a D2-108b (Z²= 4-OMe)
D2-92a D2-108b (Z²= 2-SMe)
D2-92a D2-108b (Z²= 3-CF_Three)
D2-92a D2-108b (Z²= 4-OCF_Three)
D2-92a D2-108b (Z²= 2-SCF_Three)
D2-92a C (O) Me
D2-92a C (O) CF_Three
D2-92a C (O) OMe
D2-93a Me
D2-93a Et
D2-93a Pr-n
D2-93a Pr-i
D2-93a Pr-c
D2-93a Bu-n
D2-93a Bu-i
D2-93a Bu-c
D2-93a Bu-s
D2-93a Bu-t
D2-93a Pen-n
D2-93a Pen-c
D2-93a Hex-n
D2-93a Hex-c
D2-93a CH₂Pr-c
D2-93a CH₂Bu-c
D2-93a CH₂Pen-c
D2-93a CH₂Hex-c
D2-93a CH₂CH = CH₂
D2-93a CH₂CH = C (Cl)₂
D2-93a CH₂C≡CH
D2-93a CH₂CN
D2-93a CH₂CF_Three
D2-93a CH₂OMe
D2-93a CH₂OCF_Three
D2-93a CH₂SMe
D2-93a CH₂S (O) Me
D2-93a CH₂S (O)₂Me
D2-93a CH₂SCF_Three
D2-93a CH₂S (O) CF_Three
D2-93a CH₂S (O)₂CF_Three
D2-93a CH₂CH (OMe)₂
D2-93a CH₂CH (SMe)₂
D2-93a CH₂C (O) Me
D2-93a CH₂C (O) CF_Three
D2-93a CH₂C (O) OMe
D2-93a CH₂(D2-32a)
D2-93a CH₂(D2-33a)
D2-93a CH₂(D2-34a)
D2-93a CH₂(D2-37a)
D2-93a CH₂(D2-81a)
D2-93a CH₂(D2-82a)
D2-93a CH₂(D2-84a)
D2-93a CH₂(D2-85a)
D2-93a CH₂(D2-87a)
D2-93a CH₂(D2-92a)
D2-93a CH₂(D2-93a)
D2-93a CH₂(D2-95a)
D2-93a CH₂(D2-96a)
D2-93a CH₂(D2-98a)
D2-93a CH₂(D2-108a)
D2-93a CH₂(D2-108b, Z²= 2-Cl)
D2-93a CH₂(D2-108b, Z²= 3-Me)
D2-93a CH₂(D2-108b, Z²= 4-OMe)
D2-93a CH₂(D2-108b, Z²= 2-SMe)
D2-93a CH₂(D2-108b, Z²= 3-CF_Three)
D2-93a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-93a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-93a CH₂CH₂CN
D2-93a CH₂CH₂CF_Three
D2-93a CH₂CH₂OMe
D2-93a CH₂CH₂SMe
D2-93a CH₂CH₂S (O) Me
D2-93a CH₂CH₂S (O)₂Me
D2-93a D2-32a
D2-93a D2-33a
D2-93a D2-34a
D2-93a D2-37a
D2-93a D2-81a
D2-93a D2-82a
D2-93a D2-84a
D2-93a D2-85a
D2-93a D2-87a
D2-93a D2-92a
D2-93a D2-93a
D2-93a D2-95a
D2-93a D2-96a
D2-93a D2-98a
D2-93a D2-108a
D2-93a D2-108b (Z²= 2-Cl)
D2-93a D2-108b (Z²= 3-Me)
D2-93a D2-108b (Z²= 4-OMe)
D2-93a D2-108b (Z²= 2-SMe)
D2-93a D2-108b (Z²= 3-CF_Three)
D2-93a D2-108b (Z²= 4-OCF_Three)
D2-93a D2-108b (Z²= 2-SCF_Three)
D2-93a C (O) Me
D2-93a C (O) CF_Three
D2-93a C (O) OMe
D2-95a Me
D2-95a Et
D2-95a Pr-n
D2-95a Pr-i
D2-95a Pr-c
D2-95a Bu-n
D2-95a Bu-i
D2-95a Bu-c
D2-95a Bu-s
D2-95a Bu-t
D2-95a Pen-n
D2-95a Pen-c
D2-95a Hex-n
D2-95a Hex-c
D2-95a CH₂Pr-c
D2-95a CH₂Bu-c
D2-95a CH₂Pen-c
D2-95a CH₂Hex-c
D2-95a CH₂CH = CH₂
D2-95a CH₂CH = C (Cl)₂
D2-95a CH₂C≡CH
D2-95a CH₂CN
D2-95a CH₂CF_Three
D2-95a CH₂OMe
D2-95a CH₂OCF_Three
D2-95a CH₂SMe
D2-95a CH₂S (O) Me
D2-95a CH₂S (O)₂Me
D2-95a CH₂SCF_Three
D2-95a CH₂S (O) CF_Three
D2-95a CH₂S (O)₂CF_Three
D2-95a CH₂CH (OMe)₂
D2-95a CH₂CH (SMe)₂
D2-95a CH₂C (O) Me
D2-95a CH₂C (O) CF_Three
D2-95a CH₂C (O) OMe
D2-95a CH₂(D2-32a)
D2-95a CH₂(D2-33a)
D2-95a CH₂(D2-34a)
D2-95a CH₂(D2-37a)
D2-95a CH₂(D2-81a)
D2-95a CH₂(D2-82a)
D2-95a CH₂(D2-84a)
D2-95a CH₂(D2-85a)
D2-95a CH₂(D2-87a)
D2-95a CH₂(D2-92a)
D2-95a CH₂(D2-93a)
D2-95a CH₂(D2-95a)
D2-95a CH₂(D2-96a)
D2-95a CH₂(D2-98a)
D2-95a CH₂(D2-108a)
D2-95a CH₂(D2-108b, Z²= 2-Cl)
D2-95a CH₂(D2-108b, Z²= 3-Me)
D2-95a CH₂(D2-108b, Z²= 4-OMe)
D2-95a CH₂(D2-108b, Z²= 2-SMe)
D2-95a CH₂(D2-108b, Z²= 3-CF_Three)
D2-95a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-95a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-95a CH₂CH₂CN
D2-95a CH₂CH₂CF_Three
D2-95a CH₂CH₂OMe
D2-95a CH₂CH₂SMe
D2-95a CH₂CH₂S (O) Me
D2-95a CH₂CH₂S (O)₂Me
D2-95a D2-32a
D2-95a D2-33a
D2-95a D2-34a
D2-95a D2-37a
D2-95a D2-81a
D2-95a D2-82a
D2-95a D2-84a
D2-95a D2-85a
D2-95a D2-87a
D2-95a D2-92a
D2-95a D2-93a
D2-95a D2-95a
D2-95a D2-96a
D2-95a D2-98a
D2-95a D2-108a
D2-95a D2-108b (Z²= 2-Cl)
D2-95a D2-108b (Z²= 3-Me)
D2-95a D2-108b (Z²= 4-OMe)
D2-95a D2-108b (Z²= 2-SMe)
D2-95a D2-108b (Z²= 3-CF_Three)
D2-95a D2-108b (Z²= 4-OCF_Three)
D2-95a D2-108b (Z²= 2-SCF_Three)
D2-95a C (O) Me
D2-95a C (O) CF_Three
D2-95a C (O) OMe
D2-96a Me
D2-96a Et
D2-96a Pr-n
D2-96a Pr-i
D2-96a Pr-c
D2-96a Bu-n
D2-96a Bu-i
D2-96a Bu-c
D2-96a Bu-s
D2-96a Bu-t
D2-96a Pen-n
D2-96a Pen-c
D2-96a Hex-n
D2-96a Hex-c
D2-96a CH₂Pr-c
D2-96a CH₂Bu-c
D2-96a CH₂Pen-c
D2-96a CH₂Hex-c
D2-96a CH₂CH = CH₂
D2-96a CH₂CH = C (Cl)₂
D2-96a CH₂C≡CH
D2-96a CH₂CN
D2-96a CH₂CF_Three
D2-96a CH₂OMe
D2-96a CH₂OCF_Three
D2-96a CH₂SMe
D2-96a CH₂S (O) Me
D2-96a CH₂S (O)₂Me
D2-96a CH₂SCF_Three
D2-96a CH₂S (O) CF_Three
D2-96a CH₂S (O)₂CF_Three
D2-96a CH₂CH (OMe)₂
D2-96a CH₂CH (SMe)₂
D2-96a CH₂C (O) Me
D2-96a CH₂C (O) CF_Three
D2-96a CH₂C (O) OMe
D2-96a CH₂(D2-32a)
D2-96a CH₂(D2-33a)
D2-96a CH₂(D2-34a)
D2-96a CH₂(D2-37a)
D2-96a CH₂(D2-81a)
D2-96a CH₂(D2-82a)
D2-96a CH₂(D2-84a)
D2-96a CH₂(D2-85a)
D2-96a CH₂(D2-87a)
D2-96a CH₂(D2-92a)
D2-96a CH₂(D2-93a)
D2-96a CH₂(D2-95a)
D2-96a CH₂(D2-96a)
D2-96a CH₂(D2-98a)
D2-96a CH₂(D2-108a)
D2-96a CH₂(D2-108b, Z²= 2-Cl)
D2-96a CH₂(D2-108b, Z²= 3-Me)
D2-96a CH₂(D2-108b, Z²= 4-OMe)
D2-96a CH₂(D2-108b, Z²= 2-SMe)
D2-96a CH₂(D2-108b, Z²= 3-CF_Three)
D2-96a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-96a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-96a CH₂CH₂CN
D2-96a CH₂CH₂CF_Three
D2-96a CH₂CH₂OMe
D2-96a CH₂CH₂SMe
D2-96a CH₂CH₂S (O) Me
D2-96a CH₂CH₂S (O)₂Me
D2-96a D2-32a
D2-96a D2-33a
D2-96a D2-34a
D2-96a D2-37a
D2-96a D2-81a
D2-96a D2-82a
D2-96a D2-84a
D2-96a D2-85a
D2-96a D2-87a
D2-96a D2-92a
D2-96a D2-93a
D2-96a D2-95a
D2-96a D2-96a
D2-96a D2-98a
D2-96a D2-108a
D2-96a D2-108b (Z²= 2-Cl)
D2-96a D2-108b (Z²= 3-Me)
D2-96a D2-108b (Z²= 4-OMe)
D2-96a D2-108b (Z²= 2-SMe)
D2-96a D2-108b (Z²= 3-CF_Three)
D2-96a D2-108b (Z²= 4-OCF_Three)
D2-96a D2-108b (Z²= 2-SCF_Three)
D2-96a C (O) Me
D2-96a C (O) CF_Three
D2-96a C (O) OMe
D2-98a Me
D2-98a Et
D2-98a Pr-n
D2-98a Pr-i
D2-98a Pr-c
D2-98a Bu-n
D2-98a Bu-i
D2-98a Bu-c
D2-98a Bu-s
D2-98a Bu-t
D2-98a Pen-n
D2-98a Pen-c
D2-98a Hex-n
D2-98a Hex-c
D2-98a CH₂Pr-c
D2-98a CH₂Bu-c
D2-98a CH₂Pen-c
D2-98a CH₂Hex-c
D2-98a CH₂CH = CH₂
D2-98a CH₂CH = C (Cl)₂
D2-98a CH₂C≡CH
D2-98a CH₂CN
D2-98a CH₂CF_Three
D2-98a CH₂OMe
D2-98a CH₂OCF_Three
D2-98a CH₂SMe
D2-98a CH₂S (O) Me
D2-98a CH₂S (O)₂Me
D2-98a CH₂SCF_Three
D2-98a CH₂S (O) CF_Three
D2-98a CH₂S (O)₂CF_Three
D2-98a CH₂CH (OMe)₂
D2-98a CH₂CH (SMe)₂
D2-98a CH₂C (O) Me
D2-98a CH₂C (O) CF_Three
D2-98a CH₂C (O) OMe
D2-98a CH₂(D2-32a)
D2-98a CH₂(D2-33a)
D2-98a CH₂(D2-34a)
D2-98a CH₂(D2-37a)
D2-98a CH₂(D2-81a)
D2-98a CH₂(D2-82a)
D2-98a CH₂(D2-84a)
D2-98a CH₂(D2-85a)
D2-98a CH₂(D2-87a)
D2-98a CH₂(D2-92a)
D2-98a CH₂(D2-93a)
D2-98a CH₂(D2-95a)
D2-98a CH₂(D2-96a)
D2-98a CH₂(D2-98a)
D2-98a CH₂(D2-108a)
D2-98a CH₂(D2-108b, Z²= 2-Cl)
D2-98a CH₂(D2-108b, Z²= 3-Me)
D2-98a CH₂(D2-108b, Z²= 4-OMe)
D2-98a CH₂(D2-108b, Z²= 2-SMe)
D2-98a CH₂(D2-108b, Z²= 3-CF_Three)
D2-98a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-98a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-98a CH₂CH₂CN
D2-98a CH₂CH₂CF_Three
D2-98a CH₂CH₂OMe
D2-98a CH₂CH₂SMe
D2-98a CH₂CH₂S (O) Me
D2-98a CH₂CH₂S (O)₂Me
D2-98a D2-32a
D2-98a D2-33a
D2-98a D2-34a
D2-98a D2-37a
D2-98a D2-81a
D2-98a D2-82a
D2-98a D2-84a
D2-98a D2-85a
D2-98a D2-87a
D2-98a D2-92a
D2-98a D2-93a
D2-98a D2-95a
D2-98a D2-96a
D2-98a D2-98a
D2-98a D2-108a
D2-98a D2-108b (Z²= 2-Cl)
D2-98a D2-108b (Z²= 3-Me)
D2-98a D2-108b (Z²= 4-OMe)
D2-98a D2-108b (Z²= 2-SMe)
D2-98a D2-108b (Z²= 3-CF_Three)
D2-98a D2-108b (Z²= 4-OCF_Three)
D2-98a D2-108b (Z²= 2-SCF_Three)
D2-98a C (O) Me
D2-98a C (O) CF_Three
D2-98a C (O) OMe
D2-108a Me
D2-108a Et
D2-108a Pr-n
D2-108a Pr-i
D2-108a Pr-c
D2-108a Bu-n
D2-108a Bu-i
D2-108a Bu-c
D2-108a Bu-s
D2-108a Bu-t
D2-108a Pen-n
D2-108a Pen-c
D2-108a Hex-n
D2-108a Hex-c
D2-108a CH₂Pr-c
D2-108a CH₂Bu-c
D2-108a CH₂Pen-c
D2-108a CH₂Hex-c
D2-108a CH₂CH = CH₂
D2-108a CH₂CH = C (Cl)₂
D2-108a CH₂C≡CH
D2-108a CH₂CN
D2-108a CH₂CF_Three
D2-108a CH₂OMe
D2-108a CH₂OCF_Three
D2-108a CH₂SMe
D2-108a CH₂S (O) Me
D2-108a CH₂S (O)₂Me
D2-108a CH₂SCF_Three
D2-108a CH₂S (O) CF_Three
D2-108a CH₂S (O)₂CF_Three
D2-108a CH₂CH (OMe)₂
D2-108a CH₂CH (SMe)₂
D2-108a CH₂C (O) Me
D2-108a CH₂C (O) CF_Three
D2-108a CH₂C (O) OMe
D2-108a CH₂(D2-32a)
D2-108a CH₂(D2-33a)
D2-108a CH₂(D2-34a)
D2-108a CH₂(D2-37a)
D2-108a CH₂(D2-81a)
D2-108a CH₂(D2-82a)
D2-108a CH₂(D2-84a)
D2-108a CH₂(D2-85a)
D2-108a CH₂(D2-87a)
D2-108a CH₂(D2-92a)
D2-108a CH₂(D2-93a)
D2-108a CH₂(D2-95a)
D2-108a CH₂(D2-96a)
D2-108a CH₂(D2-98a)
D2-108a CH₂(D2-108a)
D2-108a CH₂(D2-108b, Z²= 2-Cl)
D2-108a CH₂(D2-108b, Z²= 3-Me)
D2-108a CH₂(D2-108b, Z²= 4-OMe)
D2-108a CH₂(D2-108b, Z²= 2-SMe)
D2-108a CH₂(D2-108b, Z²= 3-CF_Three)
D2-108a CH₂(D2-108b, Z²= 4-OCF_Three)
D2-108a CH₂(D2-108b, Z²= 2-SCF_Three)
D2-108a CH₂CH₂CN
D2-108a CH₂CH₂CF_Three
D2-108a CH₂CH₂OMe
D2-108a CH₂CH₂SMe
D2-108a CH₂CH₂S (O) Me
D2-108a CH₂CH₂S (O)₂Me
D2-108a D2-32a
D2-108a D2-33a
D2-108a D2-34a
D2-108a D2-37a
D2-108a D2-81a
D2-108a D2-82a
D2-108a D2-84a
D2-108a D2-85a
D2-108a D2-87a
D2-108a D2-92a
D2-108a D2-93a
D2-108a D2-95a
D2-108a D2-96a
D2-108a D2-98a
D2-108a D2-108a
D2-108a D2-108b (Z²= 2-Cl)
D2-108a D2-108b (Z²= 3-Me)
D2-108a D2-108b (Z²= 4-OMe)
D2-108a D2-108b (Z²= 2-SMe)
D2-108a D2-108b (Z²= 3-CF_Three)
D2-108a D2-108b (Z²= 4-OCF_Three)
D2-108a D2-108b (Z²= 2-SCF_Three)
D2-108a C (O) Me
D2-108a C (O) CF_Three
D2-108a C (O) OMe
C (O) NHCH₂CF_Three    Me
C (O) NHCH₂CF_Three    Et
C (O) NHCH₂CF_Three    Pr-n
C (O) NHCH₂CF_Three    Pr-i
C (O) NHCH₂CF_Three    Pr-c
C (O) NHCH₂CF_Three    Bu-n
C (O) NHCH₂CF_Three    Bu-i
C (O) NHCH₂CF_Three    Bu-c
C (O) NHCH₂CF_Three    Bu-s
C (O) NHCH₂CF_Three    Bu-t
C (O) NHCH₂CF_Three    Pen-n
C (O) NHCH₂CF_Three    Pen-c
C (O) NHCH₂CF_Three    Hex-n
C (O) NHCH₂CF_Three    Hex-c
C (O) NHCH₂CF_Three    CH₂Pr-c
C (O) NHCH₂CF_Three    CH₂Bu-c
C (O) NHCH₂CF_Three    CH₂Pen-c
C (O) NHCH₂CF_Three    CH₂Hex-c
C (O) NHCH₂CF_Three    CH₂CH = CH₂
C (O) NHCH₂CF_Three    CH₂CH = C (Cl)₂
C (O) NHCH₂CF_Three    CH₂C≡CH
C (O) NHCH₂CF_Three    CH₂CN
C (O) NHCH₂CF_Three    CH₂CF_Three
C (O) NHCH₂CF_Three    CH₂OMe
C (O) NHCH₂CF_Three    CH₂OCF_Three
C (O) NHCH₂CF_Three    CH₂SMe
C (O) NHCH₂CF_Three    CH₂S (O) Me
C (O) NHCH₂CF_Three    CH₂S (O)₂Me
C (O) NHCH₂CF_Three    CH₂SCF_Three
C (O) NHCH₂CF_Three    CH₂S (O) CF_Three
C (O) NHCH₂CF_Three    CH₂S (O)₂CF_Three
C (O) NHCH₂CF_Three    CH₂CH (OMe)₂
C (O) NHCH₂CF_Three    CH₂CH (SMe)₂
C (O) NHCH₂CF_Three    CH₂C (O) Me
C (O) NHCH₂CF_Three    CH₂C (O) CF_Three
C (O) NHCH₂CF_Three    CH₂C (O) OMe
C (O) NHCH₂CF_Three    CH₂(D2-32a)
C (O) NHCH₂CF_Three    CH₂(D2-33a)
C (O) NHCH₂CF_Three    CH₂(D2-34a)
C (O) NHCH₂CF_Three    CH₂(D2-37a)
C (O) NHCH₂CF_Three    CH₂(D2-81a)
C (O) NHCH₂CF_Three    CH₂(D2-82a)
C (O) NHCH₂CF_Three    CH₂(D2-84a)
C (O) NHCH₂CF_Three    CH₂(D2-85a)
C (O) NHCH₂CF_Three    CH₂(D2-87a)
C (O) NHCH₂CF_Three    CH₂(D2-92a)
C (O) NHCH₂CF_Three    CH₂(D2-93a)
C (O) NHCH₂CF_Three    CH₂(D2-95a)
C (O) NHCH₂CF_Three    CH₂(D2-96a)
C (O) NHCH₂CF_Three    CH₂(D2-98a)
C (O) NHCH₂CF_Three    CH₂(D2-108a)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 2-Cl)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 3-Me)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 4-OMe)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 2-SMe)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 3-CF_Three)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 4-OCF_Three)
C (O) NHCH₂CF_Three    CH₂(D2-108b, Z²= 2-SCF_Three)
C (O) NHCH₂CF_Three    CH₂CH₂CN
C (O) NHCH₂CF_Three    CH₂CH₂CF_Three
C (O) NHCH₂CF_Three    CH₂CH₂OMe
C (O) NHCH₂CF_Three    CH₂CH₂SMe
C (O) NHCH₂CF_Three    CH₂CH₂S (O) Me
C (O) NHCH₂CF_Three    CH₂CH₂S (O)₂Me
C (O) NHCH₂CF_Three    D2-32a
C (O) NHCH₂CF_Three    D2-33a
C (O) NHCH₂CF_Three    D2-34a
C (O) NHCH₂CF_Three    D2-37a
C (O) NHCH₂CF_Three    D2-81a
C (O) NHCH₂CF_Three    D2-82a
C (O) NHCH₂CF_Three    D2-84a
C (O) NHCH₂CF_Three    D2-85a
C (O) NHCH₂CF_Three    D2-87a
C (O) NHCH₂CF_Three    D2-92a
C (O) NHCH₂CF_Three    D2-93a
C (O) NHCH₂CF_Three    D2-95a
C (O) NHCH₂CF_Three    D2-96a
C (O) NHCH₂CF_Three    D2-98a
C (O) NHCH₂CF_Three    D2-108a
C (O) NHCH₂CF_Three    D2-108b (Z²= 2-Cl)
C (O) NHCH₂CF_Three    D2-108b (Z²= 3-Me)
C (O) NHCH₂CF_Three    D2-108b (Z²= 4-OMe)
C (O) NHCH₂CF_Three    D2-108b (Z²= 2-SMe)
C (O) NHCH₂CF_Three    D2-108b (Z²= 3-CF_Three)
C (O) NHCH₂CF_Three    D2-108b (Z²= 4-OCF_Three)
C (O) NHCH₂CF_Three    D2-108b (Z²= 2-SCF_Three)
C (O) NHCH₂CF_Three    C (O) Me
C (O) NHCH₂CF_Three    C (O) CF_Three
C (O) NHCH₂CF_Three    C (O) OMe
C (O) OMe Me
C (O) OMe Et
C (O) OMe Pr-n
C (O) OMe Pr-i
C (O) OMe Pr-c
C (O) OMe Bu-n
C (O) OMe Bu-i
C (O) OMe Bu-c
C (O) OMe Bu-s
C (O) OMe Bu-t
C (O) OMe Pen-n
C (O) OMe Pen-c
C (O) OMe Hex-n
C (O) OMe Hex-c
C (O) OMe CH₂Pr-c
C (O) OMe CH₂Bu-c
C (O) OMe CH₂Pen-c
C (O) OMe CH₂Hex-c
C (O) OMe CH₂CH = CH₂
C (O) OMe CH₂CH = C (Cl)₂
C (O) OMe CH₂C≡CH
C (O) OMe CH₂CN
C (O) OMe CH₂CF_Three
C (O) OMe CH₂OMe
C (O) OMe CH₂OCF_Three
C (O) OMe CH₂SMe
C (O) OMe CH₂S (O) Me
C (O) OMe CH₂S (O)₂Me
C (O) OMe CH₂SCF_Three
C (O) OMe CH₂S (O) CF_Three
C (O) OMe CH₂S (O)₂CF_Three
C (O) OMe CH₂CH (OMe)₂
C (O) OMe CH₂CH (SMe)₂
C (O) OMe CH₂C (O) Me
C (O) OMe CH₂C (O) CF_Three
C (O) OMe CH₂C (O) OMe
C (O) OMe CH₂(D2-32a)
C (O) OMe CH₂(D2-33a)
C (O) OMe CH₂(D2-34a)
C (O) OMe CH₂(D2-37a)
C (O) OMe CH₂(D2-81a)
C (O) OMe CH₂(D2-82a)
C (O) OMe CH₂(D2-84a)
C (O) OMe CH₂(D2-85a)
C (O) OMe CH₂(D2-87a)
C (O) OMe CH₂(D2-92a)
C (O) OMe CH₂(D2-93a)
C (O) OMe CH₂(D2-95a)
C (O) OMe CH₂(D2-96a)
C (O) OMe CH₂(D2-98a)
C (O) OMe CH₂(D2-108a)
C (O) OMe CH₂(D2-108b, Z²= 2-Cl)
C (O) OMe CH₂(D2-108b, Z²= 3-Me)
C (O) OMe CH₂(D2-108b, Z²= 4-OMe)
C (O) OMe CH₂(D2-108b, Z²= 2-SMe)
C (O) OMe CH₂(D2-108b, Z²= 3-CF_Three)
C (O) OMe CH₂(D2-108b, Z²= 4-OCF_Three)
C (O) OMe CH₂(D2-108b, Z²= 2-SCF_Three)
C (O) OMe CH₂CH₂CN
C (O) OMe CH₂CH₂CF_Three
C (O) OMe CH₂CH₂OMe
C (O) OMe CH₂CH₂SMe
C (O) OMe CH₂CH₂S (O) Me
C (O) OMe CH₂CH₂S (O)₂Me
C (O) OMe D2-32a
C (O) OMe D2-33a
C (O) OMe D2-34a
C (O) OMe D2-37a
C (O) OMe D2-81a
C (O) OMe D2-82a
C (O) OMe D2-84a
C (O) OMe D2-85a
C (O) OMe D2-87a
C (O) OMe D2-92a
C (O) OMe D2-93a
C (O) OMe D2-95a
C (O) OMe D2-96a
C (O) OMe D2-98a
C (O) OMe D2-108a
C (O) OMe D2-108b (Z²= 2-Cl)
C (O) OMe D2-108b (Z²= 3-Me)
C (O) OMe D2-108b (Z²= 4-OMe)
C (O) OMe D2-108b (Z²= 2-SMe)
C (O) OMe D2-108b (Z²= 3-CF_Three)
C (O) OMe D2-108b (Z²= 4-OCF_Three)
C (O) OMe D2-108b (Z²= 2-SCF_Three)
C (O) OMe C (O) Me
C (O) OMe C (O) CF_Three
C (O) OMe C (O) OMe
C (O) OEt Me
C (O) OEt Et
C (O) OEt Pr-n
C (O) OEt Pr-i
C (O) OEt Pr-c
C (O) OEt Bu-n
C (O) OEt Bu-i
C (O) OEt Bu-c
C (O) OEt Bu-s
C (O) OEt Bu-t
C (O) OEt Pen-n
C (O) OEt Pen-c
C (O) OEt Hex-n
C (O) OEt Hex-c
C (O) OEt CH₂Pr-c
C (O) OEt CH₂Bu-c
C (O) OEt CH₂Pen-c
C (O) OEt CH₂Hex-c
C (O) OEt CH₂CH = CH₂
C (O) OEt CH₂CH = C (Cl)₂
C (O) OEt CH₂C≡CH
C (O) OEt CH₂CN
C (O) OEt CH₂CF_Three
C (O) OEt CH₂OMe
C (O) OEt CH₂OCF_Three
C (O) OEt CH₂SMe
C (O) OEt CH₂S (O) Me
C (O) OEt CH₂S (O)₂Me
C (O) OEt CH₂SCF_Three
C (O) OEt CH₂S (O) CF_Three
C (O) OEt CH₂S (O)₂CF_Three
C (O) OEt CH₂CH (OMe)₂
C (O) OEt CH₂CH (SMe)₂
C (O) OEt CH₂C (O) Me
C (O) OEt CH₂C (O) CF_Three
C (O) OEt CH₂C (O) OMe
C (O) OEt CH₂(D2-32a)
C (O) OEt CH₂(D2-33a)
C (O) OEt CH₂(D2-34a)
C (O) OEt CH₂(D2-37a)
C (O) OEt CH₂(D2-81a)
C (O) OEt CH₂(D2-82a)
C (O) OEt CH₂(D2-84a)
C (O) OEt CH₂(D2-85a)
C (O) OEt CH₂(D2-87a)
C (O) OEt CH₂(D2-92a)
C (O) OEt CH₂(D2-93a)
C (O) OEt CH₂(D2-95a)
C (O) OEt CH₂(D2-96a)
C (O) OEt CH₂(D2-98a)
C (O) OEt CH₂(D2-108a)
C (O) OEt CH₂(D2-108b, Z²= 2-Cl)
C (O) OEt CH₂(D2-108b, Z²= 3-Me)
C (O) OEt CH₂(D2-108b, Z²= 4-OMe)
C (O) OEt CH₂(D2-108b, Z²= 2-SMe)
C (O) OEt CH₂(D2-108b, Z²= 3-CF_Three)
C (O) OEt CH₂(D2-108b, Z²= 4-OCF_Three)
C (O) OEt CH₂(D2-108b, Z²= 2-SCF_Three)
C (O) OEt CH₂CH₂CN
C (O) OEt CH₂CH₂CF_Three
C (O) OEt CH₂CH₂OMe
C (O) OEt CH₂CH₂SMe
C (O) OEt CH₂CH₂S (O) Me
C (O) OEt CH₂CH₂S (O)₂Me
C (O) OEt D2-32a
C (O) OEt D2-34a
C (O) OEt D2-37a
C (O) OEt D2-81a
C (O) OEt D2-82a
C (O) OEt D2-84a
C (O) OEt D2-85a
C (O) OEt D2-87a
C (O) OEt D2-92a
C (O) OEt D2-93a
C (O) OEt D2-95a
C (O) OEt D2-96a
C (O) OEt D2-98a
C (O) OEt D2-108a
C (O) OEt D2-108b (Z²= 2-Cl)
C (O) OEt D2-108b (Z²= 3-Me)
C (O) OEt D2-108b (Z²= 4-OMe)
C (O) OEt D2-108b (Z²= 2-SMe)
C (O) OEt D2-108b (Z²= 3-CF_Three)
C (O) OEt D2-108b (Z²= 4-OCF_Three)
C (O) OEt D2-108b (Z²= 2-SCF_Three)
C (O) OEt C (O) Me
C (O) OEt C (O) CF_Three
C (O) OEt C (O) OMe
NHCH₂CF_Three        Me
NHCH₂CF_Three        Et
NHCH₂CF_Three        Pr-n
NHCH₂CF_Three        Pr-i
NHCH₂CF_Three        Pr-c
NHCH₂CF_Three        Bu-n
NHCH₂CF_Three        Bu-i
NHCH₂CF_Three        Bu-c
NHCH₂CF_Three        Bu-s
NHCH₂CF_Three        Bu-t
NHCH₂CF_Three        Pen-n
NHCH₂CF_Three        Pen-c
NHCH₂CF_Three        Hex-n
NHCH₂CF_Three        Hex-c
NHCH₂CF_Three        CH₂Pr-c
NHCH₂CF_Three        CH₂Bu-c
NHCH₂CF_Three        CH₂Pen-c
NHCH₂CF_Three        CH₂Hex-c
NHCH₂CF_Three        CH₂CH = CH₂
NHCH₂CF_Three        CH₂CH = C (Cl)₂
NHCH₂CF_Three        CH₂C≡CH
NHCH₂CF_Three        CH₂CN
NHCH₂CF_Three        CH₂CF_Three
NHCH₂CF_Three        CH₂OMe
NHCH₂CF_Three        CH₂OCF_Three
NHCH₂CF_Three        CH₂SMe
NHCH₂CF_Three        CH₂S (O) Me
NHCH₂CF_Three        CH₂S (O)₂Me
NHCH₂CF_Three        CH₂SCF_Three
NHCH₂CF_Three        CH₂S (O) CF_Three
NHCH₂CF_Three        CH₂S (O)₂CF_Three
NHCH₂CF_Three        CH₂CH (OMe)₂
NHCH₂CF_Three        CH₂CH (SMe)₂
NHCH₂CF_Three        CH₂C (O) Me
NHCH₂CF_Three        CH₂C (O) CF_Three
NHCH₂CF_Three        CH₂C (O) OMe
NHCH₂CF_Three        CH₂(D2-32a)
NHCH₂CF_Three        CH₂(D2-33a)
NHCH₂CF_Three        CH₂(D2-34a)
NHCH₂CF_Three        CH₂(D2-37a)
NHCH₂CF_Three        CH₂(D2-81a)
NHCH₂CF_Three        CH₂(D2-82a)
NHCH₂CF_Three        CH₂(D2-84a)
NHCH₂CF_Three        CH₂(D2-85a)
NHCH₂CF_Three        CH₂(D2-87a)
NHCH₂CF_Three        CH₂(D2-92a)
NHCH₂CF_Three        CH₂(D2-93a)
NHCH₂CF_Three        CH₂(D2-95a)
NHCH₂CF_Three        CH₂(D2-96a)
NHCH₂CF_Three        CH₂(D2-98a)
NHCH₂CF_Three        CH₂(D2-108a)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 2-Cl)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 3-Me)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 4-OMe)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 2-SMe)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 3-CF_Three)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 4-OCF_Three)
NHCH₂CF_Three        CH₂(D2-108b, Z²= 2-SCF_Three)
NHCH₂CF_Three        CH₂CH₂CN
NHCH₂CF_Three        CH₂CH₂CF_Three
NHCH₂CF_Three        CH₂CH₂OMe
NHCH₂CF_Three        CH₂CH₂SMe
NHCH₂CF_Three        CH₂CH₂S (O) Me
NHCH₂CF_Three        CH₂CH₂S (O)₂Me
NHCH₂CF_Three        D2-32a
NHCH₂CF_Three        D2-34a
NHCH₂CF_Three        D2-37a
NHCH₂CF_Three        D2-81a
NHCH₂CF_Three        D2-82a
NHCH₂CF_Three        D2-84a
NHCH₂CF_Three        D2-85a
NHCH₂CF_Three        D2-87a
NHCH₂CF_Three        D2-92a
NHCH₂CF_Three        D2-93a
NHCH₂CF_Three        D2-95a
NHCH₂CF_Three        D2-98a
NHCH₂CF_Three        D2-108a
NHCH₂CF_Three        D2-108b (Z²= 2-Cl)
NHCH₂CF_Three        D2-108b (Z²= 3-Me)
NHCH₂CF_Three        D2-108b (Z²= 4-OMe)
NHCH₂CF_Three        D2-108b (Z²= 2-SMe)
NHCH₂CF_Three        D2-108b (Z²= 4-OCF_Three)
NHCH₂CF_Three        D2-108b (Z²= 2-SCF_Three)
NHCH₂CF_Three        C (O) Me
NHCH₂CF_Three        C (O) CF_Three
NHCH₂CF_Three        C (O) OMe
D2-7b (X²= 3-CF₂CF_Three) Me
--------------------------------------
[Table 2]

第２表
-------------------------
R^b1
-------------------------
H
Me
Et
Pr-n
Pr-i
Pr-c
Bu-n
Bu-i
Bu-c
Bu-s
Bu-t
Pen-n
Pen-c
Hex-n
Hex-c
CH₂Pr-c
CH₂Bu-c
CH₂Pen-c
CH₂Hex-c
CH₂CH=CH₂
CH₂CH=C(Cl)₂
CH₂C≡CH
CH₂CN
CH₂CF₃
CH₂OMe
CH₂OCF₃
CH₂OH
CH₂Cl
CF₂CF₃
SMe
S(O)Me
S(O)₂Me
SEt
S(O)Et
S(O)₂Et
C(O)NHEt
C(O)NHCH₂CF₃
C(O)OEt
CH₂SMe
CH₂S(O)Me
CH₂S(O)₂Me
CH₂SCF₃
CH₂S(O)CF₃
CH₂S(O)₂CF₃
CH₂CH₂CH(Me)SMe
CH₂CH₂CH(Me)S(O)Me
CH₂CH₂CH(Me)S(O)₂Me
CH₂CH₂CH₂SEt
CH₂CH₂CH₂S(O)Et
CH₂CH₂CH₂S(O)₂Et
CH(Me)CH₂CH₂SEt
CH(Me)CH₂CH₂S(O)Et
CH(Me)CH₂CH₂S(O)₂Et
CH₂CH(Me)CH₂SEt
CH₂CH(Me)CH₂S(O)Et
CH₂CH(Me)CH₂S(O)₂Et
CH₂CH₂CH(Me)SEt
CH₂CH₂CH(Me)S(O)Et
CH₂CH₂CH(Me)S(O)₂Et
CH₂CH₂CH₂SPr-n
CH₂CH₂CH₂S(O)Pr-n
CH₂CH₂CH₂S(O)₂Pr-n
CH(Me)CH₂CH₂SPr-n
CH₂CH₂CH₂SMe
CH₂CH₂CH₂S(O)Me
CH₂CH₂CH₂S(O)₂Me
CH(Me)CH₂CH₂SMe
CH(Me)CH₂CH₂S(O)Me
CH(Me)CH₂CH₂S(O)₂Me
CH₂CH(Me)CH₂SMe
CH₂CH(Me)CH₂S(O)Me
CH₂CH(Me)CH₂S(O)₂Me
CH(Me)CH₂CH₂S(O)Pr-n
CH(Me)CH₂CH₂S(O)₂Pr-n
CH₂CH(Me)CH₂SPr-n
CH₂CH(Me)CH₂S(O)Pr-n
CH₂CH(Me)CH₂S(O)₂Pr-n
CH₂CH₂CH(Me)SMe
CH₂CH₂CH(Me)S(O)Me
CH₂CH₂CH(Me)S(O)₂Me
CH₂CH₂CH₂CH₂SMe
CH₂CH₂CH₂CH₂S(O)Me
CH₂CH₂CH₂CH₂S(O)₂Me
CH₂CH₂CH₂CH₂SEt
CH₂CH₂CH₂CH₂S(O)Et
CH₂CH₂CH₂CH₂S(O)₂Et
CH₂CH₂CH₂CH₂SPr-n
CH₂CH₂CH₂CH₂S(O)Pr-n
CH₂CH₂CH₂CH₂S(O)₂Pr-n
CH₂CH(OMe)₂
CH₂CH(SMe)₂
CH₂C(O)Me
CH₂C(O)CF₃
CH₂C(O)OMe
CH₂(D2-32a)
CH₂(D2-33a)
CH₂(D2-34a)
CH₂(D2-37a)
CH₂(D2-81a)
CH₂(D2-82a)
CH₂(D2-84a)
CH₂(D2-85a)
CH₂(D2-87a)
CH₂(D2-92a)
CH₂(D2-93a)
CH₂(D2-95a)
CH₂(D2-96a)
CH₂(D2-98a)
CH₂(D2-108a)
CH₂(D2-108b,Z²=2-Cl)
CH₂(D2-108b,Z²=3-Me)
CH₂(D2-108b,Z²=4-OMe)
CH₂(D2-108b,Z²=2-SMe)
CH₂(D2-108b,Z²=3-CF₃)
CH₂(D2-108b,Z²=4-OCF₃)
CH₂(D2-108b,Z²=2-SCF₃)
CH₂CH₂CN
CH₂CH₂CF₃
CH₂CH₂OMe
CH₂CH₂SMe
CH₂CH₂S(O)Me
CH₂CH₂S(O)₂Me
D2-32a
D2-33a
D2-34a
D2-37a
D2-81a
D2-82a
D2-84a
D2-85a
D2-87a
D2-92a
D2-93a
D2-95a
D2-96a
D2-98a
D2-108a
D2-108b(Z²=2-Cl)
D2-108b(Z²=3-Me)
D2-108b(Z²=4-OMe)
D2-108b(Z²=2-SMe)
D2-108b(Z²=3-CF₃)
D2-108b(Z²=4-OCF₃)
D2-108b(Z²=2-SCF₃)
C(O)Me
C(O)CF₃
C(O)OMe
-------------------------
〔第３表〕 Table 2
-------------------------
R ^b1
-------------------------
H
Me
Et
Pr-n
Pr-i
Pr-c
Bu-n
Bu-i
Bu-c
Bu-s
Bu-t
Pen-n
Pen-c
Hex-n
Hex-c
CH ₂ Pr-c
CH ₂ Bu-c
CH ₂ Pen-c
CH ₂ Hex-c
CH ₂ CH = CH ₂
CH ₂ CH = C (Cl) ₂
CH ₂ C≡CH
CH ₂ CN
CH ₂ CF ₃
CH ₂ OMe
CH ₂ OCF ₃
CH ₂ OH
CH ₂ Cl
CF ₂ CF ₃
SMe
S (O) Me
S (O) ₂ Me
SEt
S (O) Et
S (O) ₂ Et
C (O) NHEt
C (O) NHCH ₂ CF ₃
C (O) OEt
CH ₂ SMe
CH ₂ S (O) Me
CH ₂ S (O) ₂ Me
CH ₂ SCF ₃
CH ₂ S (O) CF ₃
CH ₂ S (O) ₂ CF ₃
CH ₂ CH ₂ CH (Me) SMe
CH ₂ CH ₂ CH (Me) S (O) Me
CH ₂ CH ₂ CH (Me) S (O) ₂ Me
CH ₂ CH ₂ CH ₂ SEt
CH ₂ CH ₂ CH ₂ S (O) Et
CH ₂ CH ₂ CH ₂ S (O) ₂ Et
CH (Me) CH ₂ CH ₂ SEt
CH (Me) CH ₂ CH ₂ S (O) Et
CH (Me) CH ₂ CH ₂ S (O) ₂ Et
CH ₂ CH (Me) CH ₂ SEt
CH ₂ CH (Me) CH ₂ S (O) Et
CH ₂ CH (Me) CH ₂ S (O) ₂ Et
CH ₂ CH ₂ CH (Me) SEt
CH ₂ CH ₂ CH (Me) S (O) Et
CH ₂ CH ₂ CH (Me) S (O) ₂ Et
CH ₂ CH ₂ CH ₂ SPr-n
CH ₂ CH ₂ CH ₂ S (O) Pr-n
CH ₂ CH ₂ CH ₂ S (O) ₂ Pr-n
CH (Me) CH ₂ CH ₂ SPr-n
CH ₂ CH ₂ CH ₂ SMe
CH ₂ CH ₂ CH ₂ S (O) Me
CH ₂ CH ₂ CH ₂ S (O) ₂ Me
CH (Me) CH ₂ CH ₂ SMe
CH (Me) CH ₂ CH ₂ S (O) Me
CH (Me) CH ₂ CH ₂ S (O) ₂ Me
CH ₂ CH (Me) CH ₂ SMe
CH ₂ CH (Me) CH ₂ S (O) Me
CH ₂ CH (Me) CH ₂ S (O) ₂ Me
CH (Me) CH ₂ CH ₂ S (O) Pr-n
CH (Me) CH ₂ CH ₂ S (O) ₂ Pr-n
CH ₂ CH (Me) CH ₂ SPr-n
CH ₂ CH (Me) CH ₂ S (O) Pr-n
CH ₂ CH (Me) CH ₂ S (O) ₂ Pr-n
CH ₂ CH ₂ CH (Me) SMe
CH ₂ CH ₂ CH (Me) S (O) Me
CH ₂ CH ₂ CH (Me) S (O) ₂ Me
CH ₂ CH ₂ CH ₂ CH ₂ SMe
CH ₂ CH ₂ CH ₂ CH ₂ S (O) Me
CH ₂ CH ₂ CH ₂ CH ₂ S (O) ₂ Me
CH ₂ CH ₂ CH ₂ CH ₂ SEt
CH ₂ CH ₂ CH ₂ CH ₂ S (O) Et
CH ₂ CH ₂ CH ₂ CH ₂ S (O) ₂ Et
CH ₂ CH ₂ CH ₂ CH ₂ SPr-n
CH ₂ CH ₂ CH ₂ CH ₂ S (O) Pr-n
CH ₂ CH ₂ CH ₂ CH ₂ S (O) ₂ Pr-n
CH ₂ CH (OMe) ₂
CH ₂ CH (SMe) ₂
CH ₂ C (O) Me
CH ₂ C (O) CF ₃
CH ₂ C (O) OMe
CH ₂ (D2-32a)
CH ₂ (D2-33a)
CH ₂ (D2-34a)
CH ₂ (D2-37a)
CH ₂ (D2-81a)
CH ₂ (D2-82a)
CH ₂ (D2-84a)
CH ₂ (D2-85a)
CH ₂ (D2-87a)
CH ₂ (D2-92a)
CH ₂ (D2-93a)
CH ₂ (D2-95a)
CH ₂ (D2-96a)
CH ₂ (D2-98a)
CH ₂ (D2-108a)
CH ₂ (D2-108b, Z ² = 2-Cl)
CH ₂ (D2-108b, Z ² = 3-Me)
CH ₂ (D2-108b, Z ² = 4-OMe)
CH ₂ (D2-108b, Z ² = 2-SMe)
CH ₂ (D2-108b, Z ² = 3-CF ₃ )
CH ₂ (D2-108b, Z ² = 4-OCF ₃ )
CH ₂ (D2-108b, Z ² = 2-SCF ₃ )
CH ₂ CH ₂ CN
CH ₂ CH ₂ CF ₃
CH ₂ CH ₂ OMe
CH ₂ CH ₂ SMe
CH ₂ CH ₂ S (O) Me
CH ₂ CH ₂ S (O) ₂ Me
D2-32a
D2-33a
D2-34a
D2-37a
D2-81a
D2-82a
D2-84a
D2-85a
D2-87a
D2-92a
D2-93a
D2-95a
D2-96a
D2-98a
D2-108a
D2-108b (Z ² = 2-Cl)
D2-108b (Z ² = 3-Me)
D2-108b (Z ² = 4-OMe)
D2-108b (Z ² = 2-SMe)
D2-108b (Z ² = 3-CF ₃ )
D2-108b (Z ² = 4-OCF ₃ )
D2-108b (Z ² = 2-SCF ₃ )
C (O) Me
C (O) CF ₃
C (O) OMe
-------------------------
[Table 3]

第３表
―――――――――――――――――――
R^ｃ
―――――――――――――――――――
H
Si(Me)₃
CH₂SMe
SMe
S(O)Me
S(O)₂Me
C(O)SMe
C(O)NHEt
D2-32b(X²=5-CF₃)
H
Me
Et
n-Pr
i-Pr
c-Pr
n-Bu
i-Bu
s-Bu
t-Bu
c-Bu
n-Pen
c-Pen
n-Hex
c-Hex
Hep
Oct
CH₂Pr-c
CH₂Bu-i
CH₂Bu-s
CH₂Bu-t
CH₂Bu-c
CH₂Pen-c
CH₂Hex-c
CH(CH₃)Pr-n
CH(CH₃)Pr-i
CH(CH₃)Pr-n
CH(CH₃)Bu-i
CH(Et)₂
C(CH₃)₂Et
C(CH₃)₂Pr-n
CH₂CH₂F
CH₂CH₂Cl
CH₂CH₂Br
CH₂CHF₂
CH₂CHFCl
CH₂CHCl₂
CH₂CHFBr
CH₂CF₂Cl
CH₂CFCl₂
CH₂CCl₃
CH₂CF₂Br
CH₂CFClBr
CH₂CCl₂Br
CH(CH₃)CH₂F
CH(CH₃)CH₂Cl
CH(CH₃)CH₂Br
CH₂CHFCH₃
CH₂CHClCH₃
CH₂CHBrCH₃
CH₂CFClCH₃
CH₂CHClCH₂Cl
CH₂CHBrCH₂F
CH₂CHClCH₂Br
CH₂CHBrCH₂Cl
CH₂CHBrCHCl₂
CH₂CClBrCH₃
CH₂CHBrCH₂Br
CH₂CH₂CF₃
CH₂CH₂CF₂Br
CH₂CClBrCH₂Cl
CH₂CF₂CF₂H
CH₂CHClCF₃
CH₂CF₂CF₃
CH₂CF(CH₃)₂
CH₂CHFCH₂CH₃
CH₂CHClCH₂CH₃
CH₂CF₂CHFCF₃
CH₂CF₂CF₂CHF₂
CH₂CF₂CF₂CF₃
C(CH₃)₂CH₂Cl
C(CH₃)₂CH₂Br
C(CH₃)₂CHBrCH₂Br
CH₂CF₃
CH(CF₃)Me
CH(CF₃)Et
CH(CF₃)OH
CH(CF₃)OMe
CH₂CH(OMe)₂
CH₂CH(OEt)₂
CH₂CN
CH(Me)CN
C(Me)₂CN
CH(OMe)CN
CH₂CH₂CN
CH₂C(O)Me
CH₂C(O)OMe
CH₂C(O)OEt
CH₂C(O)OCH₂CF₃
CH(Me)C(O)OMe
CH(Me)C(O)OEt
CH(Me)C(O)OCH₂CF₃
CH(OMe)C(O)OMe
CH(OMe)C(O)OEt
CH(OMe)C(O)OCH₂CF₃
CH(Ph)C(O)OMe
CH(Ph)C(O)OEt
CH(Ph)C(O)OCH₂CF₃
CH(CF₃)C(O)OMe
CH(CF₃)C(O)OEt
CH(CF₃)C(O)OCH₂CF₃
CH₂CH₂C(O)OMe
CH₂CH₂C(O)OEt
CH₂CH₂C(O)OCH₂CF₃
CH₂CH(Me)C(O)OMe
CH₂CH(Me)C(O)OEt
CH(Me)CH₂C(O)OMe
CH(Me)CH₂C(O)OEt
CH₂C(O)NH₂
CH₂C(O)NHMe
CH₂C(O)NHEt
CH₂C(O)NHPr-n
CH₂C(O)NHPr-i
CH₂C(O)NHPr-c
CH₂C(O)NHBu-n
CH₂C(O)NHBu-i
CH₂C(O)NHBu-s
CH₂C(O)NHBu-t
CH₂C(O)NHBu-c
CH₂C(O)NHHex-n
CH₂C(O)NHHex-c
CH₂C(O)N(Me)₂
CH₂C(O)N(Et)₂
CH₂C(O)N(n-Pr)₂
CH₂C(O)N(Me)Et
CH₂C(O)N(Me)Pr-n
CH₂C(O)N(Me)Pr-i
CH₂C(O)NHCH₂CH₂F
CH₂C(O)NHCH₂CH₂Cl
CH₂C(O)NHCH₂CH₂Br
CH₂C(O)N(Me)CH₂CH₂F
CH₂C(O)N(Me)CH₂CH₂Cl
CH₂C(O)N(Me)CH₂CH₂Br
CH₂C(O)NHCH₂CF₃
CH₂C(O)N(Me)CH₂CF₃
CH₂C(O)NHCH₂CF₂Cl
CH₂C(O)NHCH₂CN
CH₂C(O)NHCH₂CH=CH₂
CH₂C(O)NHCH₂CH≡CH
CH₂C(O)NHCH₂CH₂CH₂Cl
CH₂C(O)NHCH₂CH₂OCH₃
CH₂C(O)NHCH₂CH₂SCH₃
CH₂C(O)NHCH₂CH₂SO₂CH₃
CH(Me)C(O)NH₂
CH(Me)C(O)NHMe
CH(Me)C(O)NHEt
CH(Me)C(O)NHPr-n
CH(Me)C(O)NHPr-i
CH(Me)C(O)NHPr-c
CH(Me)C(O)NHBu-n
CH(Me)C(O)NHBu-i
CH(Me)C(O)NHBu-s
CH(Me)C(O)NHBu-t
CH(Me)C(O)NHBu-c
CH(Me)C(O)NHHex-n
CH(Me)C(O)NHHex-c
CH(Me)C(O)N(Me)₂
CH(Me)C(O)N(Et)₂
CH(Me)C(O)N(n-Pr)₂
CH(Me)C(O)N(Me)Et
CH(Me)C(O)N(Me)Pr-n
CH(Me)C(O)N(Me)Pr-i
CH(Me)C(O)NHCH₂CH₂F
CH(Me)C(O)NHCH₂CH₂Cl
CH(Me)C(O)NHCH₂CH₂Br
CH(Me)C(O)NHCH₂CF₃
CH(Et)C(O)NHCH₂CF₃
CH(i-Pr)C(O)NHCH₂CF₃
CH(CH₂OCH₃)C(O)NHCH₂CF₃
CH(CH₂SCH₃)C(O)NHCH₂CF₃
CH(Ph)C(O)NHCH₂CF₃
CH(CH₂Ph)C(O)NHCH₂CF₃
CH(CF₃)C(O)NHMe
CH(CF₃)C(O)NHEt
CH(CF₃)C(O)NHPr-n
CH(CF₃)C(O)NHPr-i
CH(CF₃)C(O)NHPr-c
CH(CF₃)C(O)NHBu-n
CH(CF₃)C(O)NHBu-i
CH(CF₃)C(O)NHBu-s
CH(CF₃)C(O)NHBu-t
CH(CF₃)C(O)NHBu-c
CH(CF₃)C(O)NHHex-n
CH(CF₃)C(O)NHHex-c
CH(CF₃)C(O)N(Me)₂
CH(CF₃)C(O)N(Et)₂
CH(CF₃)C(O)N(n-Pr)₂
CH(CF₃)C(O)N(Me)Et
CH(CF₃)C(O)N(Me)Pr-n
CH(CF₃)C(O)N(Me)Pr-i
CH(CF₃)C(O)NHCH₂CH₂F
CH(CF₃)C(O)NHCH₂CH₂Cl
CH(CF₃)C(O)NHCH₂CH₂Br
CH(CF₃)C(O)NHCH₂CF₃
CH₂CH₂C(O)NHCH₂CF₃
CH₂C(O)N(Me)₂
CH₂C(O)N(Et)₂
CH₂C(O)N(n-Pr)₂
CH₂CH=CH₂
CH₂C(Me)=CH₂
CH₂C(Et)=CH₂
CH(Me)CH=CH₂
CH₂CH=C(Me)₂
CH₂C(Me)=CHCH₃
CH(Me)CH=CHCH₃
CH₂C(F)=CH₂
CH₂CH=CHCl
CH₂C(Cl)=CH₂
CH₂CH=CCl₂
CH₂CH=CHBr
CH₂C(Br)=CH₂
CH₂C(Br)=CHBr
CH₂C(Me)=CHBr
CH₂CH=C(Cl)CH₃
CH₂CH=C(Br)CH₃
CH₂C(OMe)=CH₂
CH₂C(Br)=CHOMe
CH₂C(Br)=CHOEt
CH₂C(Br)=CHPh
CH₂C≡CH
CH₂C≡CCl
CH₂C≡CBr
CH₂C≡CI
CH₂C≡CPh
CH₂OMe
CH₂CH₂OH
CH₂CH₂OMe
CH₂CH₂OEt
CH₂CH₂OPr-n
CH₂CH₂OPr-i
CH₂CH₂OBu-i
CH₂CH₂OCH₂CH₂Cl
CH₂CH₂OCH₂CF₃
CH₂CH₂OCH₂CH₂OCH₃
CH₂CH₂OCH₂CH₂SCH₃
CH₂CH₂OC(O)CH₃
CH₂CH(Me)OH
CH₂CH(Me)OMe
CH₂CH(Me)OCH₂CF₃
CH(Me)CH₂OH
CH(Me)CH₂OMe
CH(Me)CH₂OCH₂CF₃
CH(Ph)CH₂OH
CH(Ph)CH₂OMe
CH(Ph)CH₂OCH₂CF₃
C(Me)₂CH₂OH
C(Me)₂CH₂OMe
C(Me)₂CH₂OCH₂CF₃
CH₂CH₂CH₂OH
CH₂CH₂CH₂OMe
CH₂CH₂CH₂OCH₂CF₃
CH₂CH₂CH₂CH₂OH
CH₂CH₂CH₂CH₂OMe
CH₂CH₂CH₂CH₂OCH₂CF₃
CH₂SMe
CH(CF₃)SMe
CH(CF₃)SEt
CH₂CH₂SMe
CH₂CH₂S(O)Me
CH₂CH₂S(O)₂Me
CH₂CH₂SEt
CH₂CH₂S(O)Et
CH₂CH₂S(O)₂Et
CH₂CH₂SPr-n
CH₂CH₂S(O)Pr-n
CH₂CH₂S(O)₂Pr-n
CH₂CH₂SPr-i
CH₂CH₂S(O)Pr-i
CH₂CH₂S(O)₂Pr-i
CH₂CH₂SCH₂CF₃
CH₂CH₂S(O)CH₂CF₃
CH₂CH₂S(O)₂CH₂CF₃
CH₂CH₂SCH₂CH₂OH
CH₂CH₂S(O)CH₂CH₂OH
CH₂CH₂S(O)₂CH₂CH₂OH
CH₂CH₂SCH₂CH₂OMe
CH₂CH₂S(O)CH₂CH₂OMe
CH₂CH₂S(O)₂CH₂CH₂OMe
CH₂CH₂SCH₂C(O)OMe
CH₂CH₂S(O)CH₂C(O)OMe
CH₂CH₂S(O)₂CH₂C(O)OMe
CH₂CH₂SCH₂C(O)NHMe
CH₂CH₂S(O)CH₂C(O)NHMe
CH₂CH₂S(O)₂CH₂C(O)NHMe
CH₂CH₂SCH₂C(O)NMe
CH₂CH₂S(O)CH₂C(O)NMe
CH₂CH₂S(O)₂CH₂C(O)N(Me)₂
CH₂CH₂SCH₂CH=CH₂
CH₂CH₂SCH₂CH≡CH
CH₂CH₂S(O)₂NHMe
CH₂CH₂S(O)₂N(Me)₂
CH₂CH₂S(O)₂NHEt
CH₂CH₂S(O)₂N(Et)₂
CH₂CH₂S(O)₂NHPr-n
CH₂CH₂S(O)₂N(Pr-n)₂
CH₂CH₂S(O)₂NHPr-i
CH₂CH₂S(O)₂N(Pr-i)₂
CH₂CH₂S(O)₂NHPr-c
CH₂CH₂S(O)₂NHBu-t
CH₂CH₂S(O)₂NHCH₂CF₃
CH₂CH₂S(O)₂NHCH₂CH₂OMe
CH₂CH₂S(O)₂NHCH₂CH₂SMe
CH₂CH₂S(O)₂NHCH₂CH=CH₂
CH₂CH₂S(O)₂NHCH₂CH≡CH
CH₂CH₂S(O)(=NCN)Me
CH₂CH(Me)SMe
CH₂CH(Me)S(O)Me
CH₂CH(Me)S(O)₂Me
CH₂CH(Me)SEt
CH₂CH(Me)S(O)Et
CH₂CH(Me)S(O)₂Et
CH₂CH(Et)SMe
CH₂CH(Et)S(O)Me
CH₂CH(Et)S(O)₂Me
CH₂CH(n-Pr)SMe
CH₂CH(n-Pr)S(O)Me
CH₂CH(n-Pr)S(O)₂Me
CH₂CH(i-Pr)SMe
CH₂CH(i-Pr)S(O)Me
CH₂CH(i-Pr)S(O)₂Me
CH₂CH(Ph)SMe
CH₂CH(Ph)S(O)Me
CH₂CH(Ph)S(O)₂Me
CH(Me)CH₂SMe
CH(Me)CH₂S(O)Me
CH(Me)CH₂S(O)₂Me
CH(Me)CH₂SEt
CH(Me)CH₂S(O)Et
CH(Me)CH₂S(O)₂Et
CH(Me)CH₂SPr-n
CH(Me)CH₂S(O)Pr-n
CH(Me)CH₂S(O)₂Pr-n
CH(Me)CH₂SPr-i
CH(Me)CH₂S(O)Pr-i
CH(Me)CH₂S(O)₂Pr-i
CH(Me)CH₂SPh
CH(Me)CH₂S(O)Ph
CH(Me)CH₂S(O)₂Ph
CH(Ph)CH₂SMe
CH(Ph)CH₂S(O)Me
CH(Ph)CH₂S(O)₂Me
CH(Me)CH(Me)SMe
CH(Me)CH(Me)S(O)Me
CH(Me)CH(Me)S(O)₂Me
C(Me)₂CH₂SMe
C(Me)₂CH₂S(O)Me
C(Me)₂CH₂S(O)₂Me
CH₂CH₂CH₂SMe
CH₂CH₂CH₂S(O)Me
CH₂CH₂CH₂S(O)₂Me
CH₂CH₂CH(Me)SMe
CH₂CH₂CH(Me)S(O)Me
CH₂CH₂CH(Me)S(O)₂Me
CH₂CH(Me)CH₂SMe
CH₂CH(Me)CH₂S(O)Me
CH₂CH(Me)CH₂S(O)₂Me
CH(Me)CH₂CH₂SMe
CH(Me)CH₂CH₂S(O)Me
CH(Me)CH₂CH₂S(O)₂Me
C(Me)₂CH₂CH₂SMe
C(Me)₂CH₂CH₂S(O)Me
C(Me)₂CH₂CH₂S(O)₂Me
CH(Me)(CH₂)₃SMe
CH(Me)(CH₂)₃S(O)Me
CH(Me)(CH₂)₃S(O)₂Me
CH(Me)(CH₂)₄SMe
CH(Me)(CH₂)₄S(O)Me
CH(Me)(CH₂)₄S(O)₂Me
CH₂NHC(O)Me
CH₂NHC(O)Et
CH₂NHC(O)Pr-n
CH₂CH₂NHC(O)Me
CH₂CH₂NHC(O)Et
CH₂CH₂NHC(O)Pr-n
CH₂CH₂NHC(O)Pr-i
CH₂CH₂NHC(O)Pr-c
CH₂CH₂NHC(O)Bu-n
CH₂CH₂NHC(O)Bu-i
CH₂CH₂NHC(O)Bu-s
CH₂CH₂NHC(O)Bu-t
CH₂CH₂NHC(O)CF₃
CH₂CH₂NHC(O)CF₂Cl
CH₂CH₂NHC(O)Ph
CH₂CH₂NHC(O)CH₂CF₃
CH₂CH₂NHC(O)CH₂SMe
CH₂CH₂NHC(O)CH₂S(O)Me
CH₂CH₂NHC(O)CH₂S(O)₂Me
CH₂CH₂N(Me)C(O)Me
CH₂CH₂N(Me)C(O)Et
CH₂CH₂N(Me)C(O)CF₃
CH₂CH₂N(Me)C(O)CH₂CF₃
CH₂CH₂N(Me)C(O)CH₂SMe
CH ₂CH₂N(Me)C(O)CH₂S(O)Me
CH ₂CH₂N(Me)C(O)CH₂S(O)₂Me
CH₂CH₂NHC(O)OMe
CH₂CH₂NHC(O)OEt
CH₂CH₂NHC(O)OPr-n
CH₂CH₂NHC(O)OBu-t
CH₂CH₂NHC(O)NHEt
CH₂CH₂NHC(O)NHPr-n
CH₂CH₂NHC(O)NHPr-i
CH₂CH₂NHC(O)NHBu-t
CH₂CH₂NHC(O)N(Me)₂
CH₂CH₂NHSO₂Me
CH₂CH₂NHSO₂Et
CH₂CH₂NHSO₂CF₃
CH₂CH₂NHSO₂Ph
CH₂CH₂NHSO₂N(Me)₂
CH₂CH₂NHP(S)(OMe)₂
CH₂CH₂NHP(S)(OEt)₂
CH₂CH₂N(Me)SO₂Me
CH₂CH₂N(Me)SO₂CF₃
CH₂CH₂N(Me)OMe
CH₂CH(Me)NHC(O)Me
CH₂CH(Me)NHC(O)CF₃
CH₂CH(Me)NHC(O)CH₂CF₃
CH₂CH(Me)NHC(O)CH₂SMe
CH(Me)NHC(O)CH₂S(O)Me
CH(Me)NHC(O)CH₂S(O)₂Me
CH₂CH(Me)NHC(O)OMe
CH(Me)CH₂NHC(O)Me
CH(Me)CH₂NHC(O)CF₃
CH(Me)CH₂NHC(O)CH₂CF₃
CH(Me)CH₂NHC(O)CH₂SMe
CH(Me)CH₂NHC(O)CH₂S(O)Me
CH(Me)CH₂NHC(O)CH₂S(O)₂Me
CH(Me)CH₂NHC(O)OMe
CH₂CH₂CH₂NHC(O)Me
CH₂CH₂CH₂NHC(O)OMe
D2-1a
D2-1b
D2-2a
D2-2b
D2-5a
D2-5b
D2-5c
D2-6a
D2-6b
D2-6c
D2-7a
D2-8a
D2-8b
D2-8c
D2-9a
D2-9b
D2-9c
D2-10a
D2-10b
D2-10c
D2-11a
D2-12a
D2-12b
D2-12c
D2-13a
D2-13b
D2-14a
D2-14b
D2-15a
D2-15b
D2-16a
D2-17a
D2-18a
D2-19a
D2-21a
D2-21b
D2-22a
D2-23a
D2-23b
D2-24a
D2-25a
D2-27a
D2-30a
D2-31a
D2-32a
D2-34a
D2-36a
D2-37a
D2-41a
D2-43a
D2-45a
D2-46a
D2-49a
D2-51a
D2-53a
D2-59a
D2-61a
D2-63a
D2-68a
D2-75a
D2-76a
D2-76b
D2-77a
D2-77b
D2-78a
D2-78b
D2-79a
D2-81a
D2-82a
D2-84a
D2-85a
D2-87a
D2-90a
D2-100a
D2-100b
D2-100c
D2-100d
D2-100e
D2-101a
D2-101b
D2-101c
D2-101d
D2-102a
D2-102b
D2-102c
D2-102d
D2-102e
D2-102f
D2-103a
D2-108a
CH₂(D2-1a)
CH₂(D2-1b)
CH₂(D2-2a)
CH₂(D2-2b)
CH₂(D2-4a)
CH₂(D2-4b)
CH₂(D2-5a)
CH₂(D2-5b)
CH₂(D2-5c)
CH₂(D2-6a)
CH₂(D2-6b)
CH₂(D2-6c)
CH₂(D2-7a)
CH₂(D2-8a)
CH₂(D2-8b)
CH₂(D2-8c)
CH₂(D2-9a)
CH₂(D2-9b)
CH₂(D2-9c)
CH₂(D2-10a)
CH₂(D2-10b)
CH₂(D2-10c)
CH₂(D2-12a)
CH₂(D2-12b)
CH₂(D2-12c)
CH₂(D2-13a)
CH₂(D2-13b)
CH₂(D2-14a)
CH₂(D2-14b)
CH₂(D2-15a)
CH₂(D2-15b)
CH₂(D2-16a)
CH₂(D2-17a)
CH₂(D2-18a)
CH₂(D2-19a)
CH₂(D2-20a)
CH₂(D2-21a)
CH₂(D2-21b)
CH₂(D2-23a)
CH₂(D2-23b)
CH₂(D2-25a)
CH₂(D2-27a)
CH₂(D2-30a)
CH₂(D2-31a)
CH₂(D2-32a)
CH₂(D2-33a)
CH₂(D2-34a)
CH₂(D2-35a)
CH₂(D2-35b)
CH₂(D2-36a)
CH₂(D2-37a)
CH₂(D2-38a)
CH₂(D2-39a)
CH₂(D2-40a)
CH₂(D2-41a)
CH₂(D2-42a)
CH₂(D2-43a)
CH₂(D2-45a)
CH₂(D2-46a)
CH₂(D2-49a)
CH₂(D2-51a)
CH₂(D2-53a)
CH₂(D2-59a)
CH₂(D2-61a)
CH₂(D2-63a)
CH₂(D2-68a)
CH₂(D2-75a)
CH₂(D2-76a)
CH₂(D2-76b)
CH₂(D2-77a)
CH₂(D2-77b)
CH₂(D2-78a)
CH₂(D2-78b)
CH₂(D2-79a)
CH₂(D2-81a)
CH₂(D2-82a)
CH₂(D2-84a)
CH₂(D2-85a)
CH₂(D2-87a)
CH₂(D2-90a)
CH₂(D2-100a)
CH₂(D2-100b)
CH₂(D2-100c)
CH₂(D2-100d)
CH₂(D2-100e)
CH₂(D2-101a)
CH₂(D2-101b)
CH₂(D2-101c)
CH₂(D2-101d)
CH₂(D2-102a)
CH₂(D2-102b)
CH₂(D2-102c)
CH₂(D2-102d)
CH₂(D2-102e)
CH₂(D2-102f)
CH₂(D2-103a)
CH₂(D2-108a)
CH(Me)(D2-1a)
CH(Me)(D2-2a)
CH(Me)(D2-5a)
CH(Me)(D2-5c)
CH(Me)(D2-6c)
CH(Me)(D2-8c)
CH(Me)(D2-9b)
CH(Me)(D2-9c)
CH(Me)(D2-10b)
CH(Me)(D2-10c)
CH(Me)(D2-12b)
CH(Me)(D2-12c)
CH(Me)(D2-13b)
CH(Me)(D2-14a)
CH(Me)(D2-14b)
CH(Me)(D2-15a)
CH(Me)(D2-15b)
CH(Me)(D2-16a)
CH(Me)(D2-17a)
CH(Me)(D2-18a)
CH(Me)(D2-23b)
CH(Me)(D2-27a)
CH(Me)(D2-31a)
CH(Me)(D2-32a)
CH(Me)(D2-35a)
CH(Me)(D2-36a)
CH(Me)(D2-37a)
CH(Me)(D2-39a)
CH(Me)(D2-41a)
CH₂C(O)NH(D2-1a)
CH₂C(O)NH(D2-2a)
CH₂C(O)NH(D2-5a)
CH₂C(O)NH(D2-5c)
CH₂C(O)NH(D2-6c)
CH₂C(O)NH(D2-8c)
CH₂C(O)NH(D2-9b)
CH₂C(O)NH(D2-9c)
CH₂C(O)NH(D2-10b)
CH₂C(O)NH(D2-10c)
CH₂C(O)NH(D2-12b)
CH₂C(O)NH(D2-12c)
CH₂C(O)NH(D2-13b)
CH₂C(O)NH(D2-14a)
CH₂C(O)NH(D2-14b)
CH₂C(O)NH(D2-15a)
CH₂C(O)NH(D2-15b)
CH₂C(O)NH(D2-16a)
CH₂C(O)NH(D2-17a)
CH₂C(O)NH(D2-18a)
CH₂C(O)NH(D2-23b)
CH₂C(O)NH(D2-27a)
CH₂C(O)NH(D2-31a)
CH₂C(O)NH(D2-32a)
CH₂C(O)NH(D2-35a)
CH₂C(O)NH(D2-36a)
CH₂C(O)NH(D2-37a)
CH₂C(O)NH(D2-39a)
CH₂C(O)NH(D2-41a)
CH₂C(O)NH(D2-45a)
CH₂C(O)NH(D2-46a)
CH₂C(O)NH(D2-49a)
CH₂C(O)NH(D2-51a)
CH₂C(O)NH(D2-53a)
CH₂C(O)NH(D2-59a)
CH₂C(O)NH(D2-61a)
CH₂C(O)NH(D2-63a)
CH₂C(O)NH(D2-68a)
CH₂C(O)NH(D2-75a)
CH₂C(O)NH(D2-76a)
CH₂C(O)NH(D2-76b)
CH₂C(O)NH(D2-77a)
CH₂C(O)NH(D2-77b)
CH₂C(O)NH(D2-78a)
CH₂C(O)NH(D2-78b)
CH₂C(O)NH(D2-79a)
CH₂C(O)NH(D2-82a)
CH₂C(O)NH(D2-84a)
CH₂C(O)NH(D2-85a)
CH₂C(O)NH(D2-87a)
CH₂C(O)NH(D2-90a)
CH₂C(O)NH(D2-100a)
CH₂C(O)NH(D2-100b)
CH₂C(O)NH(D2-100c)
CH₂C(O)NH(D2-100d)
CH₂C(O)NH(D2-100e)
CH₂C(O)NH(D2-101a)
CH₂C(O)NH(D2-101b)
CH₂C(O)NH(D2-101c)
CH₂C(O)NH(D2-101d)
CH₂C(O)NH(D2-108a)
CH₂C(O)NHCH₂(D2-1a)
CH₂C(O)NHCH₂(D2-2a)
CH₂C(O)NHCH₂(D2-5a)
CH₂C(O)NHCH₂(D2-5c)
CH₂C(O)NHCH₂(D2-6c)
CH₂C(O)NHCH₂(D2-8c)
CH₂C(O)NHCH₂(D2-9b)
CH₂C(O)NHCH₂(D2-9c)
CH₂C(O)NHCH₂(D2-10b)
CH₂C(O)NHCH₂(D2-10c)
CH₂C(O)NHCH₂(D2-12b)
CH₂C(O)NHCH₂(D2-12c)
CH₂C(O)NHCH₂(D2-13b)
CH₂C(O)NHCH₂(D2-14a)
CH₂C(O)NHCH₂(D2-14b)
CH₂C(O)NHCH₂(D2-15a)
CH₂C(O)NHCH₂(D2-15b)
CH₂C(O)NHCH₂(D2-16a)
CH₂C(O)NHCH₂(D2-17a)
CH₂C(O)NHCH₂(D2-18a)
CH₂C(O)NHCH₂(D2-23b)
CH₂C(O)NHCH₂(D2-27a)
CH₂C(O)NHCH₂(D2-31a)
CH₂C(O)NHCH₂(D2-32a)
CH₂C(O)NHCH₂(D2-35a)
CH₂C(O)NHCH₂(D2-36a)
CH₂C(O)NHCH₂(D2-37a)
CH₂C(O)NHCH₂(D2-39a)
CH₂C(O)NHCH₂(D2-41a)
CH₂C(O)NHCH₂(D2-45a)
CH₂C(O)NHCH₂(D2-46a)
CH₂C(O)NHCH₂(D2-49a)
CH₂C(O)NHCH₂(D2-51a)
CH₂C(O)NHCH₂(D2-53a)
CH₂C(O)NHCH₂(D2-59a)
CH₂C(O)NHCH₂(D2-61a)
CH₂C(O)NHCH₂(D2-63a)
CH₂C(O)NHCH₂(D2-68a)
CH₂C(O)NHCH₂(D2-75a)
CH₂C(O)NHCH₂(D2-76a)
CH₂C(O)NHCH₂(D2-76b)
CH₂C(O)NHCH₂(D2-77a)
CH₂C(O)NHCH₂(D2-77b)
CH₂C(O)NHCH₂(D2-78a)
CH₂C(O)NHCH₂(D2-78b)
CH₂C(O)NHCH₂(D2-79a)
CH₂C(O)NHCH₂(D2-82a)
CH₂C(O)NHCH₂(D2-84a)
CH₂C(O)NHCH₂(D2-85a)
CH₂C(O)NHCH₂(D2-87a)
CH₂C(O)NHCH₂(D2-90a)
CH₂C(O)NHCH₂(D2-102a)
CH₂C(O)NHCH₂(D2-102b)
CH₂C(O)NHCH₂(D2-102c)
CH₂C(O)NHCH₂(D2-102d)
CH₂C(O)NHCH₂(D2-102e)
CH₂C(O)NHCH₂(D2-102f)
CH₂C(O)NHCH₂(D2-103a)
CH₂C(O)NHCH₂(D2-108a)
NH(D2-7a)
NH(D2-10c)
NH(D2-22a)
NH(D2-24a)
NH(D2-32a)
NC(O)Me(D2-32a)
NC(O)OMe(D2-32a)
NC(O)Et(D2-32a)
NC(O)OEt(D2-32a)
NC(O)CH₂CF₃(D2-32a)
NSO₂Me(D2-32a)
NSO₂CF₃(D2-32a)
NSO₂Ph(D2-32a)
NH(D2-35a)
NH(D2-36a)
NH(D2-37a)
NH(D2-39a)
NH(D2-43a)
NH(D2-45a)
NH(D2-49a)
NH(D2-51a)
NH(D2-53a)
NH(D2-59a)
NH(D2-61a)
NH(D2-63a)
NH(D2-108a)
NH{D2-32b(3-Cl)}
NH{D2-32b(4-Cl)}
NH{D2-32b(5-Cl)}
NH{D2-32b(6-Cl)}
NH{D2-32b(4-CF₃)}
NH{D2-108b(2-Cl)}
NH{D2-108b(3-Cl)}
NH{D2-108b(4-Cl)}
NH{D2-108b(2-Me)}
NH{D2-108b(3-Me)}
NH{D2-108b(4-Me)}
CH₂CH₂(D2-1a)
CH₂CH₂(D2-1b)
CH₂CH₂(D2-2a)
CH₂CH₂(D2-2b)
CH₂CH₂(D2-5c)
CH₂CH₂(D2-6c)
CH₂CH₂(D2-7a)
CH₂CH₂(D2-8c)
CH₂CH₂(D2-9b)
CH₂CH₂(D2-10b)
CH₂CH₂(D2-10c)
CH₂CH₂(D2-11a)
CH₂CH₂(D2-20a)
CH₂CH₂(D2-22a)
CH₂CH₂(D2-24a)
CH₂CH₂(D2-26a)
CH₂CH₂(D2-28a)
CH₂CH₂(D2-29a)
CH₂CH₂(D2-32a)
CH₂CH₂(D2-36a)
CH₂CH₂(D2-37a)
CH₂CH₂OCH₂(D2-1a)
CH₂CH₂OCH₂(D2-1b)
CH₂CH₂OCH₂(D2-2a)
CH₂CH₂OCH₂(D2-2b)
CH₂CH₂OCH₂(D2-4a)
CH₂CH₂OCH₂(D2-4b)
CH₂CH₂OCH₂(D2-5a)
CH₂CH₂OCH₂(D2-5b)
CH₂CH₂OCH₂(D2-5c)
CH₂CH₂OCH₂(D2-6a)
CH₂CH₂OCH₂(D2-6b)
CH₂CH₂OCH₂(D2-6c)
CH₂CH₂OCH₂(D2-7a)
CH₂CH₂OCH₂(D2-8a)
CH₂CH₂OCH₂(D2-8b)
CH₂CH₂OCH₂(D2-8c)
CH₂CH₂OCH₂(D2-9a)
CH₂CH₂OCH₂(D2-9b)
CH₂CH₂OCH₂(D2-9c)
CH₂CH₂OCH₂(D2-10a)
CH₂CH₂OCH₂(D2-10b)
CH₂CH₂OCH₂(D2-10c)
CH₂CH₂OCH₂(D2-12a)
CH₂CH₂OCH₂(D2-12b)
CH₂CH₂OCH₂(D2-12c)
CH₂CH₂OCH₂(D2-13a)
CH₂CH₂OCH₂(D2-13b)
CH₂CH₂OCH₂(D2-14a)
CH₂CH₂OCH₂(D2-14b)
CH₂CH₂OCH₂(D2-15a)
CH₂CH₂OCH₂(D2-15b)
CH₂CH₂OCH₂(D2-16a)
CH₂CH₂OCH₂(D2-17a)
CH₂CH₂OCH₂(D2-18a)
CH₂CH₂OCH₂(D2-19a)
CH₂CH₂OCH₂(D2-20a)
CH₂CH₂OCH₂(D2-21a)
CH₂CH₂OCH₂(D2-21b)
CH₂CH₂OCH₂(D2-23a)
CH₂CH₂OCH₂(D2-23b)
CH₂CH₂OCH₂(D2-25a)
CH₂CH₂OCH₂(D2-27a)
CH₂CH₂OCH₂(D2-30a)
CH₂CH₂OCH₂(D2-31a)
CH₂CH₂OCH₂(D2-32a)
CH₂CH₂OCH₂(D2-33a)
CH₂CH₂OCH₂(D2-34a)
CH₂CH₂OCH₂(D2-35a)
CH₂CH₂OCH₂(D2-35b)
CH₂CH₂OCH₂(D2-36a)
CH₂CH₂OCH₂(D2-37a)
CH₂CH₂OCH₂(D2-38a)
CH₂CH₂OCH₂(D2-39a)
CH₂CH₂OCH₂(D2-40a)
CH₂CH₂OCH₂(D2-41a)
CH₂CH₂OCH₂(D2-42a)
CH₂CH₂OCH₂(D2-43a)
CH₂CH₂OCH₂(D2-45a)
CH₂CH₂OCH₂(D2-46a)
CH₂CH₂OCH₂(D2-49a)
CH₂CH₂OCH₂(D2-51a)
CH₂CH₂OCH₂(D2-53a)
CH₂CH₂OCH₂(D2-59a)
CH₂CH₂OCH₂(D2-61a)
CH₂CH₂OCH₂(D2-63a)
CH₂CH₂OCH₂(D2-68a)
CH₂CH₂OCH₂(D2-75a)
CH₂CH₂OCH₂(D2-76a)
CH₂CH₂OCH₂(D2-76b)
CH₂CH₂OCH₂(D2-77a)
CH₂CH₂OCH₂(D2-77b)
CH₂CH₂OCH₂(D2-78a)
CH₂CH₂OCH₂(D2-78b)
CH₂CH₂OCH₂(D2-79a)
CH₂CH₂OCH₂(D2-81a)
CH₂CH₂OCH₂(D2-82a)
CH₂CH₂OCH₂(D2-84a)
CH₂CH₂OCH₂(D2-85a)
CH₂CH₂OCH₂(D2-87a)
CH₂CH₂OCH₂(D2-90a)
CH₂CH₂OCH₂(D2-100a)
CH₂CH₂OCH₂(D2-100b)
CH₂CH₂OCH₂(D2-100c)
CH₂CH₂OCH₂(D2-100d)
CH₂CH₂OCH₂(D2-100e)
CH₂CH₂OCH₂(D2-101a)
CH₂CH₂OCH₂(D2-101b)
CH₂CH₂OCH₂(D2-101c)
CH₂CH₂OCH₂(D2-101d)
CH₂CH₂OCH₂(D2-102a)
CH₂CH₂OCH₂(D2-102b)
CH₂CH₂OCH₂(D2-102c)
CH₂CH₂OCH₂(D2-102d)
CH₂CH₂OCH₂(D2-102e)
CH₂CH₂OCH₂(D2-102f)
CH₂CH₂OCH₂(D2-103a)
CH₂CH₂OCH₂(D2-108a)
CH₂CH₂SCH₂(D2-1a)
CH₂CH₂SCH₂(D2-1b)
CH₂CH₂SCH₂(D2-2a)
CH₂CH₂SCH₂(D2-2b)
CH₂CH₂SCH₂(D2-4a)
CH₂CH₂SCH₂(D2-4b)
CH₂CH₂SCH₂(D2-5a)
CH₂CH₂SCH₂(D2-5b)
CH₂CH₂SCH₂(D2-5c)
CH₂CH₂SCH₂(D2-6a)
CH₂CH₂SCH₂(D2-6b)
CH₂CH₂SCH₂(D2-6c)
CH₂CH₂SCH₂(D2-7a)
CH₂CH₂SCH₂(D2-8a)
CH₂CH₂SCH₂(D2-8b)
CH₂CH₂SCH₂(D2-8c)
CH₂CH₂SCH₂(D2-9a)
CH₂CH₂SCH₂(D2-9b)
CH₂CH₂SCH₂(D2-9c)
CH₂CH₂SCH₂(D2-10a)
CH₂CH₂SCH₂(D2-10b)
CH₂CH₂SCH₂(D2-10c)
CH₂CH₂SCH₂(D2-12a)
CH₂CH₂SCH₂(D2-12b)
CH₂CH₂SCH₂(D2-12c)
CH₂CH₂SCH₂(D2-13a)
CH₂CH₂SCH₂(D2-13b)
CH₂CH₂OCH₂(D2-14a)
CH₂CH₂SCH₂(D2-14b)
CH₂CH₂SCH₂(D2-15a)
CH₂CH₂SCH₂(D2-15b)
CH₂CH₂SCH₂(D2-16a)
CH₂CH₂SCH₂(D2-17a)
CH₂CH₂SCH₂(D2-18a)
CH₂CH₂SCH₂(D2-19a)
CH₂CH₂SCH₂(D2-20a)
CH₂CH₂SCH₂(D2-21a)
CH₂CH₂SCH₂(D2-21b)
CH₂CH₂SCH₂(D2-23a)
CH₂CH₂SCH₂(D2-23b)
CH₂CH₂SCH₂(D2-25a)
CH₂CH₂SCH₂(D2-27a)
CH₂CH₂SCH₂(D2-30a)
CH₂CH₂SCH₂(D2-31a)
CH₂CH₂SCH₂(D2-32a)
CH₂CH₂SCH₂(D2-33a)
CH₂CH₂SCH₂(D2-34a)
CH₂CH₂SCH₂(D2-35a)
CH₂CH₂SCH₂(D2-35b)
CH₂CH₂SCH₂(D2-36a)
CH₂CH₂SCH₂(D2-37a)
CH₂CH₂SCH₂(D2-38a)
CH₂CH₂SCH₂(D2-39a)
CH₂CH₂SCH₂(D2-40a)
CH₂CH₂SCH₂(D2-41a)
CH₂CH₂SCH₂(D2-42a)
CH₂CH₂SCH₂(D2-43a)
CH₂CH₂SCH₂(D2-45a)
CH₂CH₂SCH₂(D2-46a)
CH₂CH₂SCH₂(D2-49a)
CH₂CH₂SCH₂(D2-51a)
CH₂CH₂SCH₂(D2-53a)
CH₂CH₂SCH₂(D2-59a)
CH₂CH₂SCH₂(D2-61a)
CH₂CH₂SCH₂(D2-63a)
CH₂CH₂SCH₂(D2-68a)
CH₂CH₂SCH₂(D2-75a)
CH₂CH₂SCH₂(D2-76a)
CH₂CH₂SCH₂(D2-76b)
CH₂CH₂SCH₂(D2-77a)
CH₂CH₂SCH₂(D2-77b)
CH₂CH₂SCH₂(D2-78a)
CH₂CH₂SCH₂(D2-78b)
CH₂CH₂SCH₂(D2-79a)
CH₂CH₂SCH₂(D2-81a)
CH₂CH₂SCH₂(D2-82a)
CH₂CH₂SCH₂(D2-84a)
CH₂CH₂SCH₂(D2-85a)
CH₂CH₂SCH₂(D2-87a)
CH₂CH₂SCH₂(D2-90a)
CH₂CH₂SCH₂(D2-100a)
CH₂CH₂SCH₂(D2-100b)
CH₂CH₂SCH₂(D2-100c)
CH₂CH₂SCH₂(D2-100d)
CH₂CH₂SCH₂(D2-100e)
CH₂CH₂SCH₂(D2-101a)
CH₂CH₂SCH₂(D2-101b)
CH₂CH₂SCH₂(D2-101c)
CH₂CH₂SCH₂(D2-101d)
CH₂CH₂SCH₂(D2-102a)
CH₂CH₂SCH₂(D2-102b)
CH₂CH₂SCH₂(D2-102c)
CH₂CH₂SCH₂(D2-102d)
CH₂CH₂SCH₂(D2-102e)
CH₂CH₂SCH₂(D2-102f)
CH₂CH₂SCH₂(D2-103a)
CH₂CH₂SCH₂(D2-108a)
CH₂{D2-1c(3-Me)}
CH₂{D2-1d(5-Cl)}
CH₂{D2-2c(5-Br)}
CH₂{D2-2d(5-Cl)}
CH₂{D2-4c(5-Cl)}
CH₂{D2-4d(5-Cl)}
CH₂{D2-5d(3-Me)}
CH₂{D2-5e(3-Me)}
CH₂{D2-5f(5-Me)}
CH₂{D2-6d(3-Cl)}
CH₂{D2-6e(3-Me)}
CH₂{D2-6f(5-Me)}
CH₂{D2-7a(3-Me)}
CH₂{D2-8d(3-Cl)}
CH₂{D2-8e(3-CF₃)}
CH₂{D2-8f(5-Me)}
CH₂{D2-9d(2-Me)}
CH₂{D2-9e(2-Me)}
CH₂{D2-9f(4-Me)}
CH₂{D2-10e(2-Me)}
CH₂{D2-10f(2-Cl)}
CH₂{D2-10e(2-Br)}
CH₂{D2-12d(4-Me)}
CH₂{D2-12e(5-Me)}
CH₂{D2-12f(5-Cl)}
CH₂{D2-13c(Me)}
CH₂{D2-13d(Cl)}
CH₂{D2-14c(Me)}
CH₂{D2-14d(Me)}
CH₂{D2-15c(Cl)}
CH₂{D2-15d(Me)}
CH₂{D2-16b(Ph)}
CH₂{D2-17b(Ph)}
CH₂{D2-18b(Me)}
CH₂{D2-19b(Cl)}
CH₂{D2-20b(Me)}
CH₂{D2-21c(Me)}
CH₂{D2-21d(Me)}
CH₂{D2-23c(t-Bu)}
CH₂{D2-23d(Ph)}
CH₂{D2-25b(Me)}
CH₂{D2-27a(Me)}
CH₂{D2-32b(3-Cl)}
CH₂{D2-32b(4-Cl)}
CH₂{D2-32b(5-Cl)}
CH₂{D2-32b(6-Cl)}
CH₂{D2-32b(3-Me)}
CH₂{D2-32b(4-Me)}
CH₂{D2-32b(5-Me)}
CH₂{D2-32b(6-Me)}
CH₂{D2-32b(5-CF₃)}
CH₂{D2-33b(4-CF₃)}
CH₂{D2-34b(3-Cl)}
CH₂{D2-35c(3-Cl)}
CH₂{D2-35d(3-Cl)}
CH₂{D2-36b(2-Me)}
CH₂{D2-37b(4-Me)}
CH₂{D2-38b(2-Me)}
CH₂{D2-39b(5-Me)}
CH₂{D2-108b(2-Cl)}
CH₂{D2-108b(3-Cl)}
CH₂{D2-108b(4-Cl)}
CH₂{D2-108b(2-Me)}
CH₂{D2-108b(3-Me)}
CH₂{D2-108b(4-Me)}
CH₂{D2-108b(2-CF₃)}
CH₂{D2-108b(3-CF₃)}
CH₂{D2-108b(4-CF₃)}
CH₂{D2-108b(2-OMe)}
CH₂{D2-108b(3-OMe)}
CH₂{D2-108b(4-OMe)}
CH₂CH₂{D2-7b(4-Cl)}
CH₂CH₂{D2-10e(2-Cl)}
CH₂CH₂{D2-11b(2-Me)}
CH₂CH₂{D2-20b(4-Me)}
CH₂CH₂{D2-22b(3-SMe)}
CH₂CH₂{D2-24b(3-Me)}
CH₂CH₂{D2-26b(4-CO₂Me)}
CH₂CH₂{D2-28b(Me)}
CH₂CH₂{D2-29a(Ph)}
CH₂CH₂{D2-32b(3-Cl)}
CH₂CH₂{D2-36b(2-Me)}
CH₂CH₂{D2-37b(4-Me)
―――――――――――――――――――
〔第４表〕 Table 3 ―――――――――――――――――――
R ^c
―――――――――――――――――――
H
Si (Me) ₃
CH ₂ SMe
SMe
S (O) Me
S (O) ₂ Me
C (O) SMe
C (O) NHEt
D2-32b (X ² = 5-CF ₃ )
H
Me
Et
NPR
i-Pr
c-Pr
n-Bu
i-Bu
s-Bu
t-Bu
c-Bu
n-Pen
c-Pen
n-Hex
c-Hex
Hep
Oct
CH ₂ Pr-c
CH ₂ Bu-i
CH ₂ Bu-s
CH ₂ Bu-t
CH ₂ Bu-c
CH ₂ Pen-c
CH ₂ Hex-c
CH (CH ₃ ) Pr-n
CH (CH ₃ ) Pr-i
CH (CH ₃ ) Pr-n
CH (CH ₃ ) Bu-i
CH (Et) ₂
C (CH ₃ ) ₂ Et
C (CH ₃ ) ₂ Pr-n
CH ₂ CH ₂ F
CH ₂ CH ₂ Cl
CH ₂ CH ₂ Br
CH ₂ CHF ₂
CH ₂ CHFCl
CH ₂ CHCl ₂
CH ₂ CHFBr
CH ₂ CF ₂ Cl
CH ₂ CFCl ₂
CH ₂ CCl ₃
CH ₂ CF ₂ Br
CH ₂ CFClBr
CH ₂ CCl ₂ Br
CH (CH ₃ ) CH ₂ F
CH (CH ₃ ) CH ₂ Cl
CH (CH ₃ ) CH ₂ Br
CH ₂ CHFCH ₃
CH ₂ CHClCH ₃
CH ₂ CHBrCH ₃
CH ₂ CFClCH ₃
CH ₂ CHClCH ₂ Cl
CH ₂ CHBrCH ₂ F
CH ₂ CHClCH ₂ Br
CH ₂ CHBrCH ₂ Cl
CH ₂ CHBrCHCl ₂
CH ₂ CClBrCH ₃
CH ₂ CHBrCH ₂ Br
CH ₂ CH ₂ CF ₃
CH ₂ CH ₂ CF ₂ Br
CH ₂ CClBrCH ₂ Cl
CH ₂ CF ₂ CF ₂ H
CH ₂ CHClCF ₃
CH ₂ CF ₂ CF ₃
CH ₂ CF (CH ₃ ) ₂
CH ₂ CHFCH ₂ CH ₃
CH ₂ CHClCH ₂ CH ₃
CH ₂ CF ₂ CHFCF ₃
CH ₂ CF ₂ CF ₂ CHF ₂
CH ₂ CF ₂ CF ₂ CF ₃
C (CH ₃ ) ₂ CH ₂ Cl
C (CH ₃ ) ₂ CH ₂ Br
C (CH ₃ ) ₂ CHBrCH ₂ Br
CH ₂ CF ₃
CH (CF ₃ ) Me
CH (CF ₃ ) Et
CH (CF ₃ ) OH
CH (CF ₃ ) OMe
CH ₂ CH (OMe) ₂
CH ₂ CH (OEt) ₂
CH ₂ CN
CH (Me) CN
C (Me) ₂ CN
CH (OMe) CN
CH ₂ CH ₂ CN
CH ₂ C (O) Me
CH ₂ C (O) OMe
CH ₂ C (O) OEt
CH ₂ C (O) OCH ₂ CF ₃
CH (Me) C (O) OMe
CH (Me) C (O) OEt
CH (Me) C (O) OCH ₂ CF ₃
CH (OMe) C (O) OMe
CH (OMe) C (O) OEt
CH (OMe) C (O) OCH ₂ CF ₃
CH (Ph) C (O) OMe
CH (Ph) C (O) OEt
CH (Ph) C (O) OCH ₂ CF ₃
CH (CF ₃ ) C (O) OMe
CH (CF ₃ ) C (O) OEt
CH (CF ₃ ) C (O) OCH ₂ CF ₃
CH ₂ CH ₂ C (O) OMe
CH ₂ CH ₂ C (O) OEt
CH ₂ CH ₂ C (O) OCH ₂ CF ₃
CH ₂ CH (Me) C (O) OMe
CH ₂ CH (Me) C (O) OEt
CH (Me) CH ₂ C (O) OMe
CH (Me) CH ₂ C (O) OEt
CH ₂ C (O) NH ₂
CH ₂ C (O) NHMe
CH ₂ C (O) NHEt
CH ₂ C (O) NHPr-n
CH ₂ C (O) NHPr-i
CH ₂ C (O) NHPr-c
CH ₂ C (O) NHBu-n
CH ₂ C (O) NHBu-i
CH ₂ C (O) NHBu-s
CH ₂ C (O) NHBu-t
CH ₂ C (O) NHBu-c
CH ₂ C (O) NHHex-n
CH ₂ C (O) NHHex-c
CH ₂ C (O) N (Me) ₂
CH ₂ C (O) N (Et) ₂
CH ₂ C (O) N (n-Pr) ₂
CH ₂ C (O) N (Me) Et
CH ₂ C (O) N (Me) Pr-n
CH ₂ C (O) N (Me) Pr-i
CH ₂ C (O) NHCH ₂ CH ₂ F
CH ₂ C (O) NHCH ₂ CH ₂ Cl
CH ₂ C (O) NHCH ₂ CH ₂ Br
CH ₂ C (O) N (Me) CH ₂ CH ₂ F
CH ₂ C (O) N (Me) CH ₂ CH ₂ Cl
CH ₂ C (O) N (Me) CH ₂ CH ₂ Br
CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ C (O) N (Me) CH ₂ CF ₃
CH ₂ C (O) NHCH ₂ CF ₂ Cl
CH ₂ C (O) NHCH ₂ CN
CH ₂ C (O) NHCH ₂ CH = CH ₂
CH ₂ C (O) NHCH ₂ CH≡CH
CH ₂ C (O) NHCH ₂ CH ₂ CH ₂ Cl
CH ₂ C (O) NHCH ₂ CH ₂ OCH ₃
CH ₂ C (O) NHCH ₂ CH ₂ SCH ₃
CH ₂ C (O) NHCH ₂ CH ₂ SO ₂ CH ₃
CH (Me) C (O) NH ₂
CH (Me) C (O) NHMe
CH (Me) C (O) NHEt
CH (Me) C (O) NHPr-n
CH (Me) C (O) NHPr-i
CH (Me) C (O) NHPr-c
CH (Me) C (O) NHBu-n
CH (Me) C (O) NHBu-i
CH (Me) C (O) NHBu-s
CH (Me) C (O) NHBu-t
CH (Me) C (O) NHBu-c
CH (Me) C (O) NHHex-n
CH (Me) C (O) NHHex-c
CH (Me) C (O) N (Me) ₂
CH (Me) C (O) N (Et) ₂
CH (Me) C (O) N (n-Pr) ₂
CH (Me) C (O) N (Me) Et
CH (Me) C (O) N (Me) Pr-n
CH (Me) C (O) N (Me) Pr-i
CH (Me) C (O) NHCH ₂ CH ₂ F
CH (Me) C (O) NHCH ₂ CH ₂ Cl
CH (Me) C (O) NHCH ₂ CH ₂ Br
CH (Me) C (O) NHCH ₂ CF ₃
CH (Et) C (O) NHCH ₂ CF ₃
CH (i-Pr) C (O) NHCH ₂ CF ₃
CH (CH ₂ OCH ₃ ) C (O) NHCH ₂ CF ₃
CH (CH ₂ SCH ₃ ) C (O) NHCH ₂ CF ₃
CH (Ph) C (O) NHCH ₂ CF ₃
CH (CH ₂ Ph) C (O) NHCH ₂ CF ₃
CH (CF ₃ ) C (O) NHMe
CH (CF ₃ ) C (O) NHEt
CH (CF ₃ ) C (O) NHPr-n
CH (CF ₃ ) C (O) NHPr-i
CH (CF ₃ ) C (O) NHPr-c
CH (CF ₃ ) C (O) NHBu-n
CH (CF ₃ ) C (O) NHBu-i
CH (CF ₃ ) C (O) NHBu-s
CH (CF ₃ ) C (O) NHBu-t
CH (CF ₃ ) C (O) NHBu-c
CH (CF ₃ ) C (O) NHHex-n
CH (CF ₃ ) C (O) NHHex-c
CH (CF ₃ ) C (O) N (Me) ₂
CH (CF ₃ ) C (O) N (Et) ₂
CH (CF ₃ ) C (O) N (n-Pr) ₂
CH (CF ₃ ) C (O) N (Me) Et
CH (CF ₃ ) C (O) N (Me) Pr-n
CH (CF ₃ ) C (O) N (Me) Pr-i
CH (CF ₃ ) C (O) NHCH ₂ CH ₂ F
CH (CF ₃ ) C (O) NHCH ₂ CH ₂ Cl
CH (CF ₃ ) C (O) NHCH ₂ CH ₂ Br
CH (CF ₃ ) C (O) NHCH ₂ CF ₃
CH ₂ CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ C (O) N (Me) ₂
CH ₂ C (O) N (Et) ₂
CH ₂ C (O) N (n-Pr) ₂
CH ₂ CH = CH ₂
CH ₂ C (Me) = CH ₂
CH ₂ C (Et) = CH ₂
CH (Me) CH = CH ₂
CH ₂ CH = C (Me) ₂
CH ₂ C (Me) = CHCH ₃
CH (Me) CH = CHCH ₃
CH ₂ C (F) = CH ₂
CH ₂ CH = CHCl
CH ₂ C (Cl) = CH ₂
CH ₂ CH = CCl ₂
CH ₂ CH = CHBr
CH ₂ C (Br) = CH ₂
CH ₂ C (Br) = CHBr
CH ₂ C (Me) = CHBr
CH ₂ CH = C (Cl) CH ₃
CH ₂ CH = C (Br) CH ₃
CH ₂ C (OMe) = CH ₂
CH ₂ C (Br) = CHOMe
CH ₂ C (Br) = CHOEt
CH ₂ C (Br) = CHPh
CH ₂ C≡CH
CH ₂ C≡CCl
CH ₂ C≡CBr
CH ₂ C≡CI
CH ₂ C≡CPh
CH ₂ OMe
CH ₂ CH ₂ OH
CH ₂ CH ₂ OMe
CH ₂ CH ₂ OEt
CH ₂ CH ₂ OPr-n
CH ₂ CH ₂ OPr-i
CH ₂ CH ₂ OBu-i
CH ₂ CH ₂ OCH ₂ CH ₂ Cl
CH ₂ CH ₂ OCH ₂ CF ₃
CH ₂ CH ₂ OCH ₂ CH ₂ OCH ₃
CH ₂ CH ₂ OCH ₂ CH ₂ SCH ₃
CH ₂ CH ₂ OC (O) CH ₃
CH ₂ CH (Me) OH
CH ₂ CH (Me) OMe
CH ₂ CH (Me) OCH ₂ CF ₃
CH (Me) CH ₂ OH
CH (Me) CH ₂ OMe
CH (Me) CH ₂ OCH ₂ CF ₃
CH (Ph) CH ₂ OH
CH (Ph) CH ₂ OMe
CH (Ph) CH ₂ OCH ₂ CF ₃
C (Me) ₂ CH ₂ OH
C (Me) ₂ CH ₂ OMe
C (Me) ₂ CH ₂ OCH ₂ CF ₃
CH ₂ CH ₂ CH ₂ OH
CH ₂ CH ₂ CH ₂ OMe
CH ₂ CH ₂ CH ₂ OCH ₂ CF ₃
CH ₂ CH ₂ CH ₂ CH ₂ OH
CH ₂ CH ₂ CH ₂ CH ₂ OMe
CH ₂ CH ₂ CH ₂ CH ₂ OCH ₂ CF ₃
CH ₂ SMe
CH (CF ₃ ) SMe
CH (CF ₃ ) SEt
CH ₂ CH ₂ SMe
CH ₂ CH ₂ S (O) Me
CH ₂ CH ₂ S (O) ₂ Me
CH ₂ CH ₂ SEt
CH ₂ CH ₂ S (O) Et
CH ₂ CH ₂ S (O) ₂ Et
CH ₂ CH ₂ SPr-n
CH ₂ CH ₂ S (O) Pr-n
CH ₂ CH ₂ S (O) ₂ Pr-n
CH ₂ CH ₂ SPr-i
CH ₂ CH ₂ S (O) Pr-i
CH ₂ CH ₂ S (O) ₂ Pr-i
CH ₂ CH ₂ SCH ₂ CF ₃
CH ₂ CH ₂ S (O) CH ₂ CF ₃
CH ₂ CH ₂ S (O) ₂ CH ₂ CF ₃
CH ₂ CH ₂ SCH ₂ CH ₂ OH
CH ₂ CH ₂ S (O) CH ₂ CH ₂ OH
CH ₂ CH ₂ S (O) ₂ CH ₂ CH ₂ OH
CH ₂ CH ₂ SCH ₂ CH ₂ OMe
CH ₂ CH ₂ S (O) CH ₂ CH ₂ OMe
CH ₂ CH ₂ S (O) ₂ CH ₂ CH ₂ OMe
CH ₂ CH ₂ SCH ₂ C (O) OMe
CH ₂ CH ₂ S (O) CH ₂ C (O) OMe
CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) OMe
CH ₂ CH ₂ SCH ₂ C (O) NHMe
CH ₂ CH ₂ S (O) CH ₂ C (O) NHMe
CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) NHMe
CH ₂ CH ₂ SCH ₂ C (O) NMe
CH ₂ CH ₂ S (O) CH ₂ C (O) NMe
CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) N (Me) ₂
CH ₂ CH ₂ SCH ₂ CH = CH ₂
CH ₂ CH ₂ SCH ₂ CH≡CH
CH ₂ CH ₂ S (O) ₂ NHMe
CH ₂ CH ₂ S (O) ₂ N (Me) ₂
CH ₂ CH ₂ S (O) ₂ NHEt
CH ₂ CH ₂ S (O) ₂ N (Et) ₂
CH ₂ CH ₂ S (O) ₂ NHPr-n
CH ₂ CH ₂ S (O) ₂ N (Pr-n) ₂
CH ₂ CH ₂ S (O) ₂ NHPr-i
CH ₂ CH ₂ S (O) ₂ N (Pr-i) ₂
CH ₂ CH ₂ S (O) ₂ NHPr-c
CH ₂ CH ₂ S (O) ₂ NHBu-t
CH ₂ CH ₂ S (O) ₂ NHCH ₂ CF ₃
CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH ₂ OMe
CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH ₂ SMe
CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH = CH ₂
CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH≡CH
CH ₂ CH ₂ S (O) (= NCN) Me
CH ₂ CH (Me) SMe
CH ₂ CH (Me) S (O) Me
CH ₂ CH (Me) S (O) ₂ Me
CH ₂ CH (Me) SEt
CH ₂ CH (Me) S (O) Et
CH ₂ CH (Me) S (O) ₂ Et
CH ₂ CH (Et) SMe
CH ₂ CH (Et) S (O) Me
CH ₂ CH (Et) S (O) ₂ Me
CH ₂ CH (n-Pr) SMe
CH ₂ CH (n-Pr) S (O) Me
CH ₂ CH (n-Pr) S (O) ₂ Me
CH ₂ CH (i-Pr) SMe
CH ₂ CH (i-Pr) S (O) Me
CH ₂ CH (i-Pr) S (O) ₂ Me
CH ₂ CH (Ph) SMe
CH ₂ CH (Ph) S (O) Me
CH ₂ CH (Ph) S (O) ₂ Me
CH (Me) CH ₂ SMe
CH (Me) CH ₂ S (O) Me
CH (Me) CH ₂ S (O) ₂ Me
CH (Me) CH ₂ SEt
CH (Me) CH ₂ S (O) Et
CH (Me) CH ₂ S (O) ₂ Et
CH (Me) CH ₂ SPr-n
CH (Me) CH ₂ S (O) Pr-n
CH (Me) CH ₂ S (O) ₂ Pr-n
CH (Me) CH ₂ SPr-i
CH (Me) CH ₂ S (O) Pr-i
CH (Me) CH ₂ S (O) ₂ Pr-i
CH (Me) CH ₂ SPh
CH (Me) CH ₂ S (O) Ph
CH (Me) CH ₂ S (O) ₂ Ph
CH (Ph) CH ₂ SMe
CH (Ph) CH ₂ S (O) Me
CH (Ph) CH ₂ S (O) ₂ Me
CH (Me) CH (Me) SMe
CH (Me) CH (Me) S (O) Me
CH (Me) CH (Me) S (O) ₂ Me
C (Me) ₂ CH ₂ SMe
C (Me) ₂ CH ₂ S (O) Me
C (Me) ₂ CH ₂ S (O) ₂ Me
CH ₂ CH ₂ CH ₂ SMe
CH ₂ CH ₂ CH ₂ S (O) Me
CH ₂ CH ₂ CH ₂ S (O) ₂ Me
CH ₂ CH ₂ CH (Me) SMe
CH ₂ CH ₂ CH (Me) S (O) Me
CH ₂ CH ₂ CH (Me) S (O) ₂ Me
CH ₂ CH (Me) CH ₂ SMe
CH ₂ CH (Me) CH ₂ S (O) Me
CH ₂ CH (Me) CH ₂ S (O) ₂ Me
CH (Me) CH ₂ CH ₂ SMe
CH (Me) CH ₂ CH ₂ S (O) Me
CH (Me) CH ₂ CH ₂ S (O) ₂ Me
C (Me) ₂ CH ₂ CH ₂ SMe
C (Me) ₂ CH ₂ CH ₂ S (O) Me
C (Me) ₂ CH ₂ CH ₂ S (O) ₂ Me
CH (Me) (CH ₂ ) ₃ SMe
CH (Me) (CH ₂ ) ₃ S (O) Me
CH (Me) (CH ₂ ) ₃ S (O) ₂ Me
CH (Me) (CH ₂ ) ₄ SMe
CH (Me) (CH ₂ ) ₄ S (O) Me
CH (Me) (CH ₂ ) ₄ S (O) ₂ Me
CH ₂ NHC (O) Me
CH ₂ NHC (O) Et
CH ₂ NHC (O) Pr-n
CH ₂ CH ₂ NHC (O) Me
CH ₂ CH ₂ NHC (O) Et
CH ₂ CH ₂ NHC (O) Pr-n
CH ₂ CH ₂ NHC (O) Pr-i
CH ₂ CH ₂ NHC (O) Pr-c
CH ₂ CH ₂ NHC (O) Bu-n
CH ₂ CH ₂ NHC (O) Bu-i
CH ₂ CH ₂ NHC (O) Bu-s
CH ₂ CH ₂ NHC (O) Bu-t
CH ₂ CH ₂ NHC (O) CF ₃
CH ₂ CH ₂ NHC (O) CF ₂ Cl
CH ₂ CH ₂ NHC (O) Ph
CH ₂ CH ₂ NHC (O) CH ₂ CF ₃
CH ₂ CH ₂ NHC (O) CH ₂ SMe
CH ₂ CH ₂ NHC (O) CH ₂ S (O) Me
CH ₂ CH ₂ NHC (O) CH ₂ S (O) ₂ Me
CH ₂ CH ₂ N (Me) C (O) Me
CH ₂ CH ₂ N (Me) C (O) Et
CH ₂ CH ₂ N (Me) C (O) CF ₃
CH ₂ CH ₂ N (Me) C (O) CH ₂ CF ₃
CH ₂ CH ₂ N (Me) C (O) CH ₂ SMe
CH ₂ CH ₂ N (Me) C (O) CH ₂ S (O) Me
CH ₂ CH ₂ N (Me) C (O) CH ₂ S (O) ₂ Me
CH ₂ CH ₂ NHC (O) OMe
CH ₂ CH ₂ NHC (O) OEt
CH ₂ CH ₂ NHC (O) OPr-n
CH ₂ CH ₂ NHC (O) OBu-t
CH ₂ CH ₂ NHC (O) NHEt
CH ₂ CH ₂ NHC (O) NHPr-n
CH ₂ CH ₂ NHC (O) NHPr-i
CH ₂ CH ₂ NHC (O) NHBu-t
CH ₂ CH ₂ NHC (O) N (Me) ₂
CH ₂ CH ₂ NHSO ₂ Me
CH ₂ CH ₂ NHSO ₂ Et
CH ₂ CH ₂ NHSO ₂ CF ₃
CH ₂ CH ₂ NHSO ₂ Ph
CH ₂ CH ₂ NHSO ₂ N (Me) ₂
CH ₂ CH ₂ NHP (S) (OMe) ₂
CH ₂ CH ₂ NHP (S) (OEt) ₂
CH ₂ CH ₂ N (Me) SO ₂ Me
CH ₂ CH ₂ N (Me) SO ₂ CF ₃
CH ₂ CH ₂ N (Me) OMe
CH ₂ CH (Me) NHC (O) Me
CH ₂ CH (Me) NHC (O) CF ₃
CH ₂ CH (Me) NHC (O) CH ₂ CF ₃
CH ₂ CH (Me) NHC (O) CH ₂ SMe
CH (Me) NHC (O) CH ₂ S (O) Me
CH (Me) NHC (O) CH ₂ S (O) ₂ Me
CH ₂ CH (Me) NHC (O) OMe
CH (Me) CH ₂ NHC (O) Me
CH (Me) CH ₂ NHC (O) CF ₃
CH (Me) CH ₂ NHC (O) CH ₂ CF ₃
CH (Me) CH ₂ NHC (O) CH ₂ SMe
CH (Me) CH ₂ NHC (O) CH ₂ S (O) Me
CH (Me) CH ₂ NHC (O) CH ₂ S (O) ₂ Me
CH (Me) CH ₂ NHC (O) OMe
CH ₂ CH ₂ CH ₂ NHC (O) Me
CH ₂ CH ₂ CH ₂ NHC (O) OMe
D2-1a
D2-1b
D2-2a
D2-2b
D2-5a
D2-5b
D2-5c
D2-6a
D2-6b
D2-6c
D2-7a
D2-8a
D2-8b
D2-8c
D2-9a
D2-9b
D2-9c
D2-10a
D2-10b
D2-10c
D2-11a
D2-12a
D2-12b
D2-12c
D2-13a
D2-13b
D2-14a
D2-14b
D2-15a
D2-15b
D2-16a
D2-17a
D2-18a
D2-19a
D2-21a
D2-21b
D2-22a
D2-23a
D2-23b
D2-24a
D2-25a
D2-27a
D2-30a
D2-31a
D2-32a
D2-34a
D2-36a
D2-37a
D2-41a
D2-43a
D2-45a
D2-46a
D2-49a
D2-51a
D2-53a
D2-59a
D2-61a
D2-63a
D2-68a
D2-75a
D2-76a
D2-76b
D2-77a
D2-77b
D2-78a
D2-78b
D2-79a
D2-81a
D2-82a
D2-84a
D2-85a
D2-87a
D2-90a
D2-100a
D2-100b
D2-100c
D2-100d
D2-100e
D2-101a
D2-101b
D2-101c
D2-101d
D2-102a
D2-102b
D2-102c
D2-102d
D2-102e
D2-102f
D2-103a
D2-108a
CH ₂ (D2-1a)
CH ₂ (D2-1b)
CH ₂ (D2-2a)
CH ₂ (D2-2b)
CH ₂ (D2-4a)
CH ₂ (D2-4b)
CH ₂ (D2-5a)
CH ₂ (D2-5b)
CH ₂ (D2-5c)
CH ₂ (D2-6a)
CH ₂ (D2-6b)
CH ₂ (D2-6c)
CH ₂ (D2-7a)
CH ₂ (D2-8a)
CH ₂ (D2-8b)
CH ₂ (D2-8c)
CH ₂ (D2-9a)
CH ₂ (D2-9b)
CH ₂ (D2-9c)
CH ₂ (D2-10a)
CH ₂ (D2-10b)
CH ₂ (D2-10c)
CH ₂ (D2-12a)
CH ₂ (D2-12b)
CH ₂ (D2-12c)
CH ₂ (D2-13a)
CH ₂ (D2-13b)
CH ₂ (D2-14a)
CH ₂ (D2-14b)
CH ₂ (D2-15a)
CH ₂ (D2-15b)
CH ₂ (D2-16a)
CH ₂ (D2-17a)
CH ₂ (D2-18a)
CH ₂ (D2-19a)
CH ₂ (D2-20a)
CH ₂ (D2-21a)
CH ₂ (D2-21b)
CH ₂ (D2-23a)
CH ₂ (D2-23b)
CH ₂ (D2-25a)
CH ₂ (D2-27a)
CH ₂ (D2-30a)
CH ₂ (D2-31a)
CH ₂ (D2-32a)
CH ₂ (D2-33a)
CH ₂ (D2-34a)
CH ₂ (D2-35a)
CH ₂ (D2-35b)
CH ₂ (D2-36a)
CH ₂ (D2-37a)
CH ₂ (D2-38a)
CH ₂ (D2-39a)
CH ₂ (D2-40a)
CH ₂ (D2-41a)
CH ₂ (D2-42a)
CH ₂ (D2-43a)
CH ₂ (D2-45a)
CH ₂ (D2-46a)
CH ₂ (D2-49a)
CH ₂ (D2-51a)
CH ₂ (D2-53a)
CH ₂ (D2-59a)
CH ₂ (D2-61a)
CH ₂ (D2-63a)
CH ₂ (D2-68a)
CH ₂ (D2-75a)
CH ₂ (D2-76a)
CH ₂ (D2-76b)
CH ₂ (D2-77a)
CH ₂ (D2-77b)
CH ₂ (D2-78a)
CH ₂ (D2-78b)
CH ₂ (D2-79a)
CH ₂ (D2-81a)
CH ₂ (D2-82a)
CH ₂ (D2-84a)
CH ₂ (D2-85a)
CH ₂ (D2-87a)
CH ₂ (D2-90a)
CH ₂ (D2-100a)
CH ₂ (D2-100b)
CH ₂ (D2-100c)
CH ₂ (D2-100d)
CH ₂ (D2-100e)
CH ₂ (D2-101a)
CH ₂ (D2-101b)
CH ₂ (D2-101c)
CH ₂ (D2-101d)
CH ₂ (D2-102a)
CH ₂ (D2-102b)
CH ₂ (D2-102c)
CH ₂ (D2-102d)
CH ₂ (D2-102e)
CH ₂ (D2-102f)
CH ₂ (D2-103a)
CH ₂ (D2-108a)
CH (Me) (D2-1a)
CH (Me) (D2-2a)
CH (Me) (D2-5a)
CH (Me) (D2-5c)
CH (Me) (D2-6c)
CH (Me) (D2-8c)
CH (Me) (D2-9b)
CH (Me) (D2-9c)
CH (Me) (D2-10b)
CH (Me) (D2-10c)
CH (Me) (D2-12b)
CH (Me) (D2-12c)
CH (Me) (D2-13b)
CH (Me) (D2-14a)
CH (Me) (D2-14b)
CH (Me) (D2-15a)
CH (Me) (D2-15b)
CH (Me) (D2-16a)
CH (Me) (D2-17a)
CH (Me) (D2-18a)
CH (Me) (D2-23b)
CH (Me) (D2-27a)
CH (Me) (D2-31a)
CH (Me) (D2-32a)
CH (Me) (D2-35a)
CH (Me) (D2-36a)
CH (Me) (D2-37a)
CH (Me) (D2-39a)
CH (Me) (D2-41a)
CH ₂ C (O) NH (D2-1a)
CH ₂ C (O) NH (D2-2a)
CH ₂ C (O) NH (D2-5a)
CH ₂ C (O) NH (D2-5c)
CH ₂ C (O) NH (D2-6c)
CH ₂ C (O) NH (D2-8c)
CH ₂ C (O) NH (D2-9b)
CH ₂ C (O) NH (D2-9c)
CH ₂ C (O) NH (D2-10b)
CH ₂ C (O) NH (D2-10c)
CH ₂ C (O) NH (D2-12b)
CH ₂ C (O) NH (D2-12c)
CH ₂ C (O) NH (D2-13b)
CH ₂ C (O) NH (D2-14a)
CH ₂ C (O) NH (D2-14b)
CH ₂ C (O) NH (D2-15a)
CH ₂ C (O) NH (D2-15b)
CH ₂ C (O) NH (D2-16a)
CH ₂ C (O) NH (D2-17a)
CH ₂ C (O) NH (D2-18a)
CH ₂ C (O) NH (D2-23b)
CH ₂ C (O) NH (D2-27a)
CH ₂ C (O) NH (D2-31a)
CH ₂ C (O) NH (D2-32a)
CH ₂ C (O) NH (D2-35a)
CH ₂ C (O) NH (D2-36a)
CH ₂ C (O) NH (D2-37a)
CH ₂ C (O) NH (D2-39a)
CH ₂ C (O) NH (D2-41a)
CH ₂ C (O) NH (D2-45a)
CH ₂ C (O) NH (D2-46a)
CH ₂ C (O) NH (D2-49a)
CH ₂ C (O) NH (D2-51a)
CH ₂ C (O) NH (D2-53a)
CH ₂ C (O) NH (D2-59a)
CH ₂ C (O) NH (D2-61a)
CH ₂ C (O) NH (D2-63a)
CH ₂ C (O) NH (D2-68a)
CH ₂ C (O) NH (D2-75a)
CH ₂ C (O) NH (D2-76a)
CH ₂ C (O) NH (D2-76b)
CH ₂ C (O) NH (D2-77a)
CH ₂ C (O) NH (D2-77b)
CH ₂ C (O) NH (D2-78a)
CH ₂ C (O) NH (D2-78b)
CH ₂ C (O) NH (D2-79a)
CH ₂ C (O) NH (D2-82a)
CH ₂ C (O) NH (D2-84a)
CH ₂ C (O) NH (D2-85a)
CH ₂ C (O) NH (D2-87a)
CH ₂ C (O) NH (D2-90a)
CH ₂ C (O) NH (D2-100a)
CH ₂ C (O) NH (D2-100b)
CH ₂ C (O) NH (D2-100c)
CH ₂ C (O) NH (D2-100d)
CH ₂ C (O) NH (D2-100e)
CH ₂ C (O) NH (D2-101a)
CH ₂ C (O) NH (D2-101b)
CH ₂ C (O) NH (D2-101c)
CH ₂ C (O) NH (D2-101d)
CH ₂ C (O) NH (D2-108a)
CH ₂ C (O) NHCH ₂ (D2-1a)
CH ₂ C (O) NHCH ₂ (D2-2a)
CH ₂ C (O) NHCH ₂ (D2-5a)
CH ₂ C (O) NHCH ₂ (D2-5c)
CH ₂ C (O) NHCH ₂ (D2-6c)
CH ₂ C (O) NHCH ₂ (D2-8c)
CH ₂ C (O) NHCH ₂ (D2-9b)
CH ₂ C (O) NHCH ₂ (D2-9c)
CH ₂ C (O) NHCH ₂ (D2-10b)
CH ₂ C (O) NHCH ₂ (D2-10c)
CH ₂ C (O) NHCH ₂ (D2-12b)
CH ₂ C (O) NHCH ₂ (D2-12c)
CH ₂ C (O) NHCH ₂ (D2-13b)
CH ₂ C (O) NHCH ₂ (D2-14a)
CH ₂ C (O) NHCH ₂ (D2-14b)
CH ₂ C (O) NHCH ₂ (D2-15a)
CH ₂ C (O) NHCH ₂ (D2-15b)
CH ₂ C (O) NHCH ₂ (D2-16a)
CH ₂ C (O) NHCH ₂ (D2-17a)
CH ₂ C (O) NHCH ₂ (D2-18a)
CH ₂ C (O) NHCH ₂ (D2-23b)
CH ₂ C (O) NHCH ₂ (D2-27a)
CH ₂ C (O) NHCH ₂ (D2-31a)
CH ₂ C (O) NHCH ₂ (D2-32a)
CH ₂ C (O) NHCH ₂ (D2-35a)
CH ₂ C (O) NHCH ₂ (D2-36a)
CH ₂ C (O) NHCH ₂ (D2-37a)
CH ₂ C (O) NHCH ₂ (D2-39a)
CH ₂ C (O) NHCH ₂ (D2-41a)
CH ₂ C (O) NHCH ₂ (D2-45a)
CH ₂ C (O) NHCH ₂ (D2-46a)
CH ₂ C (O) NHCH ₂ (D2-49a)
CH ₂ C (O) NHCH ₂ (D2-51a)
CH ₂ C (O) NHCH ₂ (D2-53a)
CH ₂ C (O) NHCH ₂ (D2-59a)
CH ₂ C (O) NHCH ₂ (D2-61a)
CH ₂ C (O) NHCH ₂ (D2-63a)
CH ₂ C (O) NHCH ₂ (D2-68a)
CH ₂ C (O) NHCH ₂ (D2-75a)
CH ₂ C (O) NHCH ₂ (D2-76a)
CH ₂ C (O) NHCH ₂ (D2-76b)
CH ₂ C (O) NHCH ₂ (D2-77a)
CH ₂ C (O) NHCH ₂ (D2-77b)
CH ₂ C (O) NHCH ₂ (D2-78a)
CH ₂ C (O) NHCH ₂ (D2-78b)
CH ₂ C (O) NHCH ₂ (D2-79a)
CH ₂ C (O) NHCH ₂ (D2-82a)
CH ₂ C (O) NHCH ₂ (D2-84a)
CH ₂ C (O) NHCH ₂ (D2-85a)
CH ₂ C (O) NHCH ₂ (D2-87a)
CH ₂ C (O) NHCH ₂ (D2-90a)
CH ₂ C (O) NHCH ₂ (D2-102a)
CH ₂ C (O) NHCH ₂ (D2-102b)
CH ₂ C (O) NHCH ₂ (D2-102c)
CH ₂ C (O) NHCH ₂ (D2-102d)
CH ₂ C (O) NHCH ₂ (D2-102e)
CH ₂ C (O) NHCH ₂ (D2-102f)
CH ₂ C (O) NHCH ₂ (D2-103a)
CH ₂ C (O) NHCH ₂ (D2-108a)
NH (D2-7a)
NH (D2-10c)
NH (D2-22a)
NH (D2-24a)
NH (D2-32a)
NC (O) Me (D2-32a)
NC (O) OMe (D2-32a)
NC (O) Et (D2-32a)
NC (O) OEt (D2-32a)
NC (O) CH ₂ CF ₃ (D2-32a)
NSO ₂ Me (D2-32a)
NSO ₂ CF ₃ (D2-32a)
NSO ₂ Ph (D2-32a)
NH (D2-35a)
NH (D2-36a)
NH (D2-37a)
NH (D2-39a)
NH (D2-43a)
NH (D2-45a)
NH (D2-49a)
NH (D2-51a)
NH (D2-53a)
NH (D2-59a)
NH (D2-61a)
NH (D2-63a)
NH (D2-108a)
NH {D2-32b (3-Cl)}
NH {D2-32b (4-Cl)}
NH {D2-32b (5-Cl)}
NH {D2-32b (6-Cl)}
NH {D2-32b (4-CF ₃ )}
NH {D2-108b (2-Cl)}
NH {D2-108b (3-Cl)}
NH {D2-108b (4-Cl)}
NH {D2-108b (2-Me)}
NH {D2-108b (3-Me)}
NH {D2-108b (4-Me)}
CH ₂ CH ₂ (D2-1a)
CH ₂ CH ₂ (D2-1b)
CH ₂ CH ₂ (D2-2a)
CH ₂ CH ₂ (D2-2b)
CH ₂ CH ₂ (D2-5c)
CH ₂ CH ₂ (D2-6c)
CH ₂ CH ₂ (D2-7a)
CH ₂ CH ₂ (D2-8c)
CH ₂ CH ₂ (D2-9b)
CH ₂ CH ₂ (D2-10b)
CH ₂ CH ₂ (D2-10c)
CH ₂ CH ₂ (D2-11a)
CH ₂ CH ₂ (D2-20a)
CH ₂ CH ₂ (D2-22a)
CH ₂ CH ₂ (D2-24a)
CH ₂ CH ₂ (D2-26a)
CH ₂ CH ₂ (D2-28a)
CH ₂ CH ₂ (D2-29a)
CH ₂ CH ₂ (D2-32a)
CH ₂ CH ₂ (D2-36a)
CH ₂ CH ₂ (D2-37a)
CH ₂ CH ₂ OCH ₂ (D2-1a)
CH ₂ CH ₂ OCH ₂ (D2-1b)
CH ₂ CH ₂ OCH ₂ (D2-2a)
CH ₂ CH ₂ OCH ₂ (D2-2b)
CH ₂ CH ₂ OCH ₂ (D2-4a)
CH ₂ CH ₂ OCH ₂ (D2-4b)
CH ₂ CH ₂ OCH ₂ (D2-5a)
CH ₂ CH ₂ OCH ₂ (D2-5b)
CH ₂ CH ₂ OCH ₂ (D2-5c)
CH ₂ CH ₂ OCH ₂ (D2-6a)
CH ₂ CH ₂ OCH ₂ (D2-6b)
CH ₂ CH ₂ OCH ₂ (D2-6c)
CH ₂ CH ₂ OCH ₂ (D2-7a)
CH ₂ CH ₂ OCH ₂ (D2-8a)
CH ₂ CH ₂ OCH ₂ (D2-8b)
CH ₂ CH ₂ OCH ₂ (D2-8c)
CH ₂ CH ₂ OCH ₂ (D2-9a)
CH ₂ CH ₂ OCH ₂ (D2-9b)
CH ₂ CH ₂ OCH ₂ (D2-9c)
CH ₂ CH ₂ OCH ₂ (D2-10a)
CH ₂ CH ₂ OCH ₂ (D2-10b)
CH ₂ CH ₂ OCH ₂ (D2-10c)
CH ₂ CH ₂ OCH ₂ (D2-12a)
CH ₂ CH ₂ OCH ₂ (D2-12b)
CH ₂ CH ₂ OCH ₂ (D2-12c)
CH ₂ CH ₂ OCH ₂ (D2-13a)
CH ₂ CH ₂ OCH ₂ (D2-13b)
CH ₂ CH ₂ OCH ₂ (D2-14a)
CH ₂ CH ₂ OCH ₂ (D2-14b)
CH ₂ CH ₂ OCH ₂ (D2-15a)
CH ₂ CH ₂ OCH ₂ (D2-15b)
CH ₂ CH ₂ OCH ₂ (D2-16a)
CH ₂ CH ₂ OCH ₂ (D2-17a)
CH ₂ CH ₂ OCH ₂ (D2-18a)
CH ₂ CH ₂ OCH ₂ (D2-19a)
CH ₂ CH ₂ OCH ₂ (D2-20a)
CH ₂ CH ₂ OCH ₂ (D2-21a)
CH ₂ CH ₂ OCH ₂ (D2-21b)
CH ₂ CH ₂ OCH ₂ (D2-23a)
CH ₂ CH ₂ OCH ₂ (D2-23b)
CH ₂ CH ₂ OCH ₂ (D2-25a)
CH ₂ CH ₂ OCH ₂ (D2-27a)
CH ₂ CH ₂ OCH ₂ (D2-30a)
CH ₂ CH ₂ OCH ₂ (D2-31a)
CH ₂ CH ₂ OCH ₂ (D2-32a)
CH ₂ CH ₂ OCH ₂ (D2-33a)
CH ₂ CH ₂ OCH ₂ (D2-34a)
CH ₂ CH ₂ OCH ₂ (D2-35a)
CH ₂ CH ₂ OCH ₂ (D2-35b)
CH ₂ CH ₂ OCH ₂ (D2-36a)
CH ₂ CH ₂ OCH ₂ (D2-37a)
CH ₂ CH ₂ OCH ₂ (D2-38a)
CH ₂ CH ₂ OCH ₂ (D2-39a)
CH ₂ CH ₂ OCH ₂ (D2-40a)
CH ₂ CH ₂ OCH ₂ (D2-41a)
CH ₂ CH ₂ OCH ₂ (D2-42a)
CH ₂ CH ₂ OCH ₂ (D2-43a)
CH ₂ CH ₂ OCH ₂ (D2-45a)
CH ₂ CH ₂ OCH ₂ (D2-46a)
CH ₂ CH ₂ OCH ₂ (D2-49a)
CH ₂ CH ₂ OCH ₂ (D2-51a)
CH ₂ CH ₂ OCH ₂ (D2-53a)
CH ₂ CH ₂ OCH ₂ (D2-59a)
CH ₂ CH ₂ OCH ₂ (D2-61a)
CH ₂ CH ₂ OCH ₂ (D2-63a)
CH ₂ CH ₂ OCH ₂ (D2-68a)
CH ₂ CH ₂ OCH ₂ (D2-75a)
CH ₂ CH ₂ OCH ₂ (D2-76a)
CH ₂ CH ₂ OCH ₂ (D2-76b)
CH ₂ CH ₂ OCH ₂ (D2-77a)
CH ₂ CH ₂ OCH ₂ (D2-77b)
CH ₂ CH ₂ OCH ₂ (D2-78a)
CH ₂ CH ₂ OCH ₂ (D2-78b)
CH ₂ CH ₂ OCH ₂ (D2-79a)
CH ₂ CH ₂ OCH ₂ (D2-81a)
CH ₂ CH ₂ OCH ₂ (D2-82a)
CH ₂ CH ₂ OCH ₂ (D2-84a)
CH ₂ CH ₂ OCH ₂ (D2-85a)
CH ₂ CH ₂ OCH ₂ (D2-87a)
CH ₂ CH ₂ OCH ₂ (D2-90a)
CH ₂ CH ₂ OCH ₂ (D2-100a)
CH ₂ CH ₂ OCH ₂ (D2-100b)
CH ₂ CH ₂ OCH ₂ (D2-100c)
CH ₂ CH ₂ OCH ₂ (D2-100d)
CH ₂ CH ₂ OCH ₂ (D2-100e)
CH ₂ CH ₂ OCH ₂ (D2-101a)
CH ₂ CH ₂ OCH ₂ (D2-101b)
CH ₂ CH ₂ OCH ₂ (D2-101c)
CH ₂ CH ₂ OCH ₂ (D2-101d)
CH ₂ CH ₂ OCH ₂ (D2-102a)
CH ₂ CH ₂ OCH ₂ (D2-102b)
CH ₂ CH ₂ OCH ₂ (D2-102c)
CH ₂ CH ₂ OCH ₂ (D2-102d)
CH ₂ CH ₂ OCH ₂ (D2-102e)
CH ₂ CH ₂ OCH ₂ (D2-102f)
CH ₂ CH ₂ OCH ₂ (D2-103a)
CH ₂ CH ₂ OCH ₂ (D2-108a)
CH ₂ CH ₂ SCH ₂ (D2-1a)
CH ₂ CH ₂ SCH ₂ (D2-1b)
CH ₂ CH ₂ SCH ₂ (D2-2a)
CH ₂ CH ₂ SCH ₂ (D2-2b)
CH ₂ CH ₂ SCH ₂ (D2-4a)
CH ₂ CH ₂ SCH ₂ (D2-4b)
CH ₂ CH ₂ SCH ₂ (D2-5a)
CH ₂ CH ₂ SCH ₂ (D2-5b)
CH ₂ CH ₂ SCH ₂ (D2-5c)
CH ₂ CH ₂ SCH ₂ (D2-6a)
CH ₂ CH ₂ SCH ₂ (D2-6b)
CH ₂ CH ₂ SCH ₂ (D2-6c)
CH ₂ CH ₂ SCH ₂ (D2-7a)
CH ₂ CH ₂ SCH ₂ (D2-8a)
CH ₂ CH ₂ SCH ₂ (D2-8b)
CH ₂ CH ₂ SCH ₂ (D2-8c)
CH ₂ CH ₂ SCH ₂ (D2-9a)
CH ₂ CH ₂ SCH ₂ (D2-9b)
CH ₂ CH ₂ SCH ₂ (D2-9c)
CH ₂ CH ₂ SCH ₂ (D2-10a)
CH ₂ CH ₂ SCH ₂ (D2-10b)
CH ₂ CH ₂ SCH ₂ (D2-10c)
CH ₂ CH ₂ SCH ₂ (D2-12a)
CH ₂ CH ₂ SCH ₂ (D2-12b)
CH ₂ CH ₂ SCH ₂ (D2-12c)
CH ₂ CH ₂ SCH ₂ (D2-13a)
CH ₂ CH ₂ SCH ₂ (D2-13b)
CH ₂ CH ₂ OCH ₂ (D2-14a)
CH ₂ CH ₂ SCH ₂ (D2-14b)
CH ₂ CH ₂ SCH ₂ (D2-15a)
CH ₂ CH ₂ SCH ₂ (D2-15b)
CH ₂ CH ₂ SCH ₂ (D2-16a)
CH ₂ CH ₂ SCH ₂ (D2-17a)
CH ₂ CH ₂ SCH ₂ (D2-18a)
CH ₂ CH ₂ SCH ₂ (D2-19a)
CH ₂ CH ₂ SCH ₂ (D2-20a)
CH ₂ CH ₂ SCH ₂ (D2-21a)
CH ₂ CH ₂ SCH ₂ (D2-21b)
CH ₂ CH ₂ SCH ₂ (D2-23a)
CH ₂ CH ₂ SCH ₂ (D2-23b)
CH ₂ CH ₂ SCH ₂ (D2-25a)
CH ₂ CH ₂ SCH ₂ (D2-27a)
CH ₂ CH ₂ SCH ₂ (D2-30a)
CH ₂ CH ₂ SCH ₂ (D2-31a)
CH ₂ CH ₂ SCH ₂ (D2-32a)
CH ₂ CH ₂ SCH ₂ (D2-33a)
CH ₂ CH ₂ SCH ₂ (D2-34a)
CH ₂ CH ₂ SCH ₂ (D2-35a)
CH ₂ CH ₂ SCH ₂ (D2-35b)
CH ₂ CH ₂ SCH ₂ (D2-36a)
CH ₂ CH ₂ SCH ₂ (D2-37a)
CH ₂ CH ₂ SCH ₂ (D2-38a)
CH ₂ CH ₂ SCH ₂ (D2-39a)
CH ₂ CH ₂ SCH ₂ (D2-40a)
CH ₂ CH ₂ SCH ₂ (D2-41a)
CH ₂ CH ₂ SCH ₂ (D2-42a)
CH ₂ CH ₂ SCH ₂ (D2-43a)
CH ₂ CH ₂ SCH ₂ (D2-45a)
CH ₂ CH ₂ SCH ₂ (D2-46a)
CH ₂ CH ₂ SCH ₂ (D2-49a)
CH ₂ CH ₂ SCH ₂ (D2-51a)
CH ₂ CH ₂ SCH ₂ (D2-53a)
CH ₂ CH ₂ SCH ₂ (D2-59a)
CH ₂ CH ₂ SCH ₂ (D2-61a)
CH ₂ CH ₂ SCH ₂ (D2-63a)
CH ₂ CH ₂ SCH ₂ (D2-68a)
CH ₂ CH ₂ SCH ₂ (D2-75a)
CH ₂ CH ₂ SCH ₂ (D2-76a)
CH ₂ CH ₂ SCH ₂ (D2-76b)
CH ₂ CH ₂ SCH ₂ (D2-77a)
CH ₂ CH ₂ SCH ₂ (D2-77b)
CH ₂ CH ₂ SCH ₂ (D2-78a)
CH ₂ CH ₂ SCH ₂ (D2-78b)
CH ₂ CH ₂ SCH ₂ (D2-79a)
CH ₂ CH ₂ SCH ₂ (D2-81a)
CH ₂ CH ₂ SCH ₂ (D2-82a)
CH ₂ CH ₂ SCH ₂ (D2-84a)
CH ₂ CH ₂ SCH ₂ (D2-85a)
CH ₂ CH ₂ SCH ₂ (D2-87a)
CH ₂ CH ₂ SCH ₂ (D2-90a)
CH ₂ CH ₂ SCH ₂ (D2-100a)
CH ₂ CH ₂ SCH ₂ (D2-100b)
CH ₂ CH ₂ SCH ₂ (D2-100c)
CH ₂ CH ₂ SCH ₂ (D2-100d)
CH ₂ CH ₂ SCH ₂ (D2-100e)
CH ₂ CH ₂ SCH ₂ (D2-101a)
CH ₂ CH ₂ SCH ₂ (D2-101b)
CH ₂ CH ₂ SCH ₂ (D2-101c)
CH ₂ CH ₂ SCH ₂ (D2-101d)
CH ₂ CH ₂ SCH ₂ (D2-102a)
CH ₂ CH ₂ SCH ₂ (D2-102b)
CH ₂ CH ₂ SCH ₂ (D2-102c)
CH ₂ CH ₂ SCH ₂ (D2-102d)
CH ₂ CH ₂ SCH ₂ (D2-102e)
CH ₂ CH ₂ SCH ₂ (D2-102f)
CH ₂ CH ₂ SCH ₂ (D2-103a)
CH ₂ CH ₂ SCH ₂ (D2-108a)
CH ₂ {D2-1c (3-Me)}
CH ₂ {D2-1d (5-Cl)}
CH ₂ {D2-2c (5-Br)}
CH ₂ {D2-2d (5-Cl)}
CH ₂ {D2-4c (5-Cl)}
CH ₂ {D2-4d (5-Cl)}
CH ₂ {D2-5d (3-Me)}
CH ₂ {D2-5e (3-Me)}
CH ₂ {D2-5f (5-Me)}
CH ₂ {D2-6d (3-Cl)}
CH ₂ {D2-6e (3-Me)}
CH ₂ {D2-6f (5-Me)}
CH ₂ {D2-7a (3-Me)}
CH ₂ {D2-8d (3-Cl)}
CH ₂ {D2-8e (3-CF ₃ )}
CH ₂ {D2-8f (5-Me)}
CH ₂ {D2-9d (2-Me)}
CH ₂ {D2-9e (2-Me)}
CH ₂ {D2-9f (4-Me)}
CH ₂ {D2-10e (2-Me)}
CH ₂ {D2-10f (2-Cl)}
CH ₂ {D2-10e (2-Br)}
CH ₂ {D2-12d (4-Me)}
CH ₂ {D2-12e (5-Me)}
CH ₂ {D2-12f (5-Cl)}
CH ₂ {D2-13c (Me)}
CH ₂ {D2-13d (Cl)}
CH ₂ {D2-14c (Me)}
CH ₂ {D2-14d (Me)}
CH ₂ {D2-15c (Cl)}
CH ₂ {D2-15d (Me)}
CH ₂ {D2-16b (Ph)}
CH ₂ {D2-17b (Ph)}
CH ₂ {D2-18b (Me)}
CH ₂ {D2-19b (Cl)}
CH ₂ {D2-20b (Me)}
CH ₂ {D2-21c (Me)}
CH ₂ {D2-21d (Me)}
CH ₂ {D2-23c (t-Bu)}
CH ₂ {D2-23d (Ph)}
CH ₂ {D2-25b (Me)}
CH ₂ {D2-27a (Me)}
CH ₂ {D2-32b (3-Cl)}
CH ₂ {D2-32b (4-Cl)}
CH ₂ {D2-32b (5-Cl)}
CH ₂ {D2-32b (6-Cl)}
CH ₂ {D2-32b (3-Me)}
CH ₂ {D2-32b (4-Me)}
CH ₂ {D2-32b (5-Me)}
CH ₂ {D2-32b (6-Me)}
CH ₂ {D2-32b (5-CF ₃ )}
CH ₂ {D2-33b (4-CF ₃ )}
CH ₂ {D2-34b (3-Cl)}
CH ₂ {D2-35c (3-Cl)}
CH ₂ {D2-35d (3-Cl)}
CH ₂ {D2-36b (2-Me)}
CH ₂ {D2-37b (4-Me)}
CH ₂ {D2-38b (2-Me)}
CH ₂ {D2-39b (5-Me)}
CH ₂ {D2-108b (2-Cl)}
CH ₂ {D2-108b (3-Cl)}
CH ₂ {D2-108b (4-Cl)}
CH ₂ {D2-108b (2-Me)}
CH ₂ {D2-108b (3-Me)}
CH ₂ {D2-108b (4-Me)}
CH ₂ {D2-108b (2-CF ₃ )}
CH ₂ {D2-108b (3-CF ₃ )}
CH ₂ {D2-108b (4-CF ₃ )}
CH ₂ {D2-108b (2-OMe)}
CH ₂ {D2-108b (3-OMe)}
CH ₂ {D2-108b (4-OMe)}
CH ₂ CH ₂ {D2-7b (4-Cl)}
CH ₂ CH ₂ {D2-10e (2-Cl)}
CH ₂ CH ₂ {D2-11b (2-Me)}
CH ₂ CH ₂ {D2-20b (4-Me)}
CH ₂ CH ₂ {D2-22b (3-SMe)}
CH ₂ CH ₂ {D2-24b (3-Me)}
CH ₂ CH ₂ {D2-26b (4-CO ₂ Me)}
CH ₂ CH ₂ {D2-28b (Me)}
CH ₂ CH ₂ {D2-29a (Ph)}
CH ₂ CH ₂ {D2-32b (3-Cl)}
CH ₂ CH ₂ {D2-36b (2-Me)}
CH ₂ CH ₂ {D2-37b (4-Me)
―――――――――――――――――――
[Table 4]

―――――――――――――――――――――――――
R^ｄ R^e R^f
―――――――――――――――――――――――――
H H SMe
H H C(O)OEt
H H C(O)NHCH₂CF₃
H H C(O)N(Me)CH₂CF₃
H H D2-7b(X²=3-CF₂CF₃)
H H D2-108a
H H D2-108b(Z²=4-CF₃)
H -CH₂CH₂N(CH₂CF₃)C(O)-
H -CH₂CH₂NHC(O)-
H H Si(Me)₃
H H CH₂SMe
H H S(O)Me
H H S(O)₂Me
H H C(O)SMe
H H C(O)NHEt
H H D2-32b(X²=5-CF₃)
H H H
H H Me
H H Et
H H n-Pr
H H i-Pr
H H c-Pr
H H n-Bu
H H i-Bu
H H s-Bu
H H t-Bu
H H c-Bu
H H n-Pen
H H c-Pen
H H n-Hex
H H c-Hex
H H Hep
H H Oct
H H CH₂Pr-c
H H CH₂Bu-i
H H CH₂Bu-s
H H CH₂Bu-t
H H CH₂Bu-c
H H CH₂Pen-c
H H CH₂Hex-c
H H CH(CH₃)Pr-n
H H CH(CH₃)Pr-i
H H CH(CH₃)Pr-n
H H CH(CH₃)Bu-i
H H CH(Et)₂
H H C(CH₃)₂Et
H H C(CH₃)₂Pr-n
H H CH₂CH₂F
H H CH₂CH₂Cl
H H CH₂CH₂Br
H H CH₂CHF₂
H H CH₂CHFCl
H H CH₂CHCl₂
H H CH₂CHFBr
H H CH₂CF₂Cl
H H CH₂CFCl₂
H H CH₂CCl₃
H H CH₂CF₂Br
H H CH₂CFClBr
H H CH₂CCl₂Br
H H CH(CH₃)CH₂F
H H CH(CH₃)CH₂Cl
H H CH(CH₃)CH₂Br
H H CH₂CHFCH₃
H H CH₂CHClCH₃
H H CH₂CHBrCH₃
H H CH₂CFClCH₃
H H CH₂CHClCH₂Cl
H H CH₂CHBrCH₂F
H H CH₂CHClCH₂Br
H H CH₂CHBrCH₂Cl
H H CH₂CHBrCHCl₂
H H CH₂CClBrCH₃
H H CH₂CHBrCH₂Br
H H CH₂CH₂CF₃
H H CH₂CH₂CF₂Br
H H CH₂CClBrCH₂Cl
H H CH₂CF₂CF₂H
H H CH₂CHClCF₃
H H CH₂CF₂CF₃
H H CH₂CF(CH₃)₂
H H CH₂CHFCH₂CH₃
H H CH₂CHClCH₂CH₃
H H CH₂CF₂CHFCF₃
H H CH₂CF₂CF₂CHF₂
H H CH₂CF₂CF₂CF₃
H H C(CH₃)₂CH₂Cl
H H C(CH₃)₂CH₂Br
H H C(CH₃)₂CHBrCH₂Br
H H CH₂CF₃
H H CH(CF₃)Me
Me H CH(CF₃)Et
OMe H CH(CF₃)OH
H H CH(CF₃)OMe
H H CH₂CH(OMe)₂
H H CH₂CH(OEt)₂
SMe H CH₂CN
CN H CH(Me)CN
H H C(Me)₂CN
H H CH(OMe)CN
H H CH₂CH₂CN
H H CH₂C(O)Me
H C(O)OMe CH₂C(O)OMe
H H CH₂C(O)OEt
H H CH₂C(O)OCH₂CF₃
H H CH(Me)C(O)OMe
H H CH(Me)C(O)OEt
H H CH(Me)C(O)OCH₂CF₃
H Me CH(OMe)C(O)OMe
H Et CH(OMe)C(O)OEt
H n-Pr CH(OMe)C(O)OCH₂CF₃
H i-Pr CH(Ph)C(O)OMe
H CH₂OCH₃ CH(Ph)C(O)OEt
H CH₂CH₂OEt CH(Ph)C(O)OCH₂CF₃
H CH₂SCH₃ CH(CF₃)C(O)OMe
H CH₂CN CH(CF₃)C(O)OEt
H CH₂CO₂Me CH(CF₃)C(O)OCH₂CF₃
H CH₂CO₂Et CH₂CH₂C(O)OMe
H CH₂CH=CH₂ CH₂CH₂C(O)OEt
H CH₂CH≡CH CH₂CH₂C(O)OCH₂CF₃
H C(O)CH₃ CH₂CH(Me)C(O)OMe
H C(O)Et CH₂CH(Me)C(O)OEt
H C(O)Pr-n CH(Me)CH₂C(O)OMe
H C(O)Pr-c CH(Me)CH₂C(O)OEt
H C(O)Bu-t CH₂C(O)NH₂
H C(O)CH₂OCH CH₂C(O)NHMe
H C(O)CH₂SCH CH₂C(O)NHEt
H C(O)OMe CH₂C(O)NHPr-n
H C(O)OEt CH₂C(O)NHPr-i
H C(O)CH₂CH₂C CH₂C(O)NHPr-c
H C(O)CH₂CH₂O CH₂C(O)NHBu-n
H C(O)OCH₂CH CH₂C(O)NHBu-i
H C(O)SCH₃ CH₂C(O)NHBu-s
H C(S)OCH₃ CH₂C(O)NHBu-t
H C(S)SCH₃ CH₂C(O)NHBu-c
H SMe CH₂C(O)NHHex-n
H SPh CH₂C(O)NHHex-c
H SNEt₂ CH₂C(O)N(Me)₂
H SO₂Me CH₂C(O)N(Et)₂
H SO₂Et CH₂C(O)N(n-Pr)₂
H SO₂Ph CH₂C(O)N(Me)Et
H SO₂NMe₂ CH₂C(O)N(Me)Pr-n
H NH₂ CH₂C(O)N(Me)Pr-i
H NHMe CH₂C(O)NHCH₂CH₂F
H NHCHO CH₂C(O)NHCH₂CH₂Cl
H NHC(O)CH₃ CH₂C(O)NHCH₂CH₂Br
H NHC(O)OCH₃ CH₂C(O)N(Me)CH₂CH₂F
H N=C(CH₃)₂ CH₂C(O)N(Me)CH₂CH₂Cl
H N=CHPh CH₂C(O)N(Me)CH₂CH₂Br
Me H CH₂C(O)NHCH₂CF₃
Et H CH₂C(O)N(Me)CH₂CF₃
n-Pr H CH₂C(O)NHCH₂CF₂Cl
i-Pr H CH₂C(O)NHCH₂CN
CH₂OCH₃ H CH₂C(O)NHCH₂CH=CH₂
CH₂CH₂OEt H CH₂C(O)NHCH₂CH≡CH
CH₂SCH₃ H CH₂C(O)NHCH₂CH₂CH₂Cl
CH₂CN H CH₂C(O)NHCH₂CH₂OCH₃
CH₂CO₂Me H CH₂C(O)NHCH₂CH₂SCH₃
CH₂CO₂Et H CH₂C(O)NHCH₂CH₂SO₂CH₃
CH₂CH=CH₂ H CH(Me)C(O)NH₂
CH₂CH≡CH H CH(Me)C(O)NHMe
C(O)CH₃ H CH(Me)C(O)NHEt
C(O)Et H CH(Me)C(O)NHPr-n
C(O)Pr-n H CH(Me)C(O)NHPr-i
C(O)Pr-c H CH(Me)C(O)NHPr-c
C(O)Bu-t H CH(Me)C(O)NHBu-n
H H CH(Me)C(O)NHBu-i
H H CH(Me)C(O)NHBu-s
C(O)OMe H CH(Me)C(O)NHBu-t
C(O)OEt H CH(Me)C(O)NHBu-c
H H CH(Me)C(O)NHHex-n
H H CH(Me)C(O)NHHex-c
H H CH(Me)C(O)N(Me)₂
C(O)SCH₃ H CH(Me)C(O)N(Et)₂
C(S)OCH₃ H CH(Me)C(O)N(n-Pr)₂
C(S)SCH₃ H CH(Me)C(O)N(Me)Et
SMe H CH(Me)C(O)N(Me)Pr-n
SPh H CH(Me)C(O)N(Me)Pr-i
SNEt₂ H CH(Me))NHCH₂CH₂F
SO₂Me H CH(Me)C(O)NHCH₂CH₂Cl
SO₂Et H CH(Me)C(O)NHCH₂CH₂Br
SO₂Ph H CH(Me)C(O)NHCH₂CF₃
SO₂NMe₂ H CH(Et)C(O)NHCH₂CF₃
NH₂ H CH(i-Pr)C(O)NHCH₂CF₃
NHMe H CH(CH₂OCH₃)C(O)NHCH₂CF₃
NHCHO H CH(CH₂SCH₃)C(O)NHCH₂CF₃
NHC(O)CH₃ H CH(Ph)C(O)NHCH₂CF₃
H H CH(CH₂Ph)C(O)NHCH₂CF₃
N=C(CH₃)₂ H CH(CF₃)C(O)NHMe
N=CHPh H CH(CF₃)C(O)NHEt
H H CH(CF₃)C(O)NHPr-n
H H CH(CF₃)C(O)NHPr-i
H H CH(CF₃)C(O)NHPr-c
H H CH(CF₃)C(O)NHBu-n
H H CH(CF₃)C(O)NHBu-i
H H CH(CF₃)C(O)NHBu-s
H H CH(CF₃)C(O)NHBu-t
H H CH(CF₃)C(O)NHBu-c
H H CH(CF₃)C(O)NHHex-n
H H CH(CF₃)C(O)NHHex-c
H H CH(CF₃)C(O)N(Me)₂
H H CH(CF₃)C(O)N(Et)₂
H H CH(CF₃)C(O)N(n-Pr)₂
H H CH(CF₃)C(O)N(Me)Et
H H CH(CF₃)C(O)N(Me)Pr-n
H H CH(CF₃)C(O)N(Me)Pr-i
H H CH(CF₃)C(O)NHCH₂CH₂F
H H CH(CF₃)C(O)NHCH₂CH₂Cl
H H CH(CF₃)C(O)NHCH₂CH₂Br
H H CH(CF₃)C(O)NHCH₂CF₃
H H CH₂CH₂C(O)NHCH₂CF₃
H H CH₂C(O)N(Me)₂
H H CH₂C(O)N(Et)₂
H H CH₂C(O)N(n-Pr)₂
H H CH₂CH=CH₂
H H CH₂C(Me)=CH₂
H H CH₂C(Et)=CH₂
H H CH(Me)CH=CH₂
H H CH₂CH=C(Me)₂
H H CH₂C(Me)=CHCH₃
H H CH(Me)CH=CHCH₃
H H CH₂C(F)=CH₂
H H CH₂CH=CHCl
H H CH₂C(Cl)=CH₂
H H CH₂CH=CCl₂
H H CH₂CH=CHBr
H H CH₂C(Br)=CH₂
H H CH₂C(Br)=CHBr
H H CH₂C(Me)=CHBr
H H CH₂CH=C(Cl)CH₃
H H CH₂CH=C(Br)CH₃
H H CH₂C(OMe)=CH₂
H H CH₂C(Br)=CHOMe
H H CH₂C(Br)=CHOEt
H H CH₂C(Br)=CHPh
H H CH₂C≡CH
H H CH₂C≡CCl
H H CH₂C≡CBr
H H CH₂C≡CI
H H CH₂C≡CPh
H H CH₂OMe
H H CH₂CH₂OH
H H CH₂CH₂OMe
H H CH₂CH₂OEt
H H CH₂CH₂OPr-n
H H CH₂CH₂OPr-i
H H CH₂CH₂OBu-i
H H CH₂CH₂OCH₂CH₂Cl
H H CH₂CH₂OCH₂CF₃
H H CH₂CH₂OCH₂CH₂OCH₃
H H CH₂CH₂OCH₂CH₂SCH₃
H H CH₂CH₂OC(O)CH₃
H H CH₂CH(Me)OH
H H CH₂CH(Me)OMe
H H CH₂CH(Me)OCH₂CF₃
H H CH(Me)CH₂OH
H H CH(Me)CH₂OMe
H H CH(Me)CH₂OCH₂CF₃
H H CH(Ph)CH₂OH
H H CH(Ph)CH₂OMe
H H CH(Ph)CH₂OCH₂CF₃
H H C(Me)₂CH₂OH
H H C(Me)₂CH₂OMe
H H C(Me)₂CH₂OCH₂CF₃
H H CH₂CH₂CH₂OH
H H CH₂CH₂CH₂OMe
H H CH₂CH₂CH₂OCH₂CF₃
H H CH₂CH₂CH₂CH₂OH
H H CH₂CH₂CH₂CH₂OMe
H H CH₂CH₂CH₂CH₂OCH₂CF₃
H H CH₂SMe
H H CH(CF₃)SMe
H H CH(CF₃)SEt
H H CH₂CH₂SMe
H H CH₂CH₂S(O)Me
H H CH₂CH₂S(O)₂Me
H H CH₂CH₂SEt
H H CH₂CH₂S(O)Et
H H CH₂CH₂S(O)₂Et
H H CH₂CH₂SPr-n
H H CH₂CH₂S(O)Pr-n
H H CH₂CH₂S(O)₂Pr-n
H H CH₂CH₂SPr-i
H H CH₂CH₂S(O)Pr-i
H H CH₂CH₂S(O)₂Pr-i
H H CH₂CH₂SCH₂CF₃
H H CH₂CH₂S(O)CH₂CF₃
H H CH₂CH₂S(O)₂CH₂CF₃
H H CH₂CH₂SCH₂CH₂OH
H H CH₂CH₂S(O)CH₂CH₂OH
H H CH₂CH₂S(O)₂CH₂CH₂OH
H H CH₂CH₂SCH₂CH₂OMe
H H CH₂CH₂S(O)CH₂CH₂OMe
H H CH₂CH₂S(O)₂CH₂CH₂OMe
H H CH₂CH₂SCH₂C(O)OMe
H H CH₂CH₂S(O)CH₂C(O)OMe
H H CH₂CH₂S(O)₂CH₂C(O)OMe
H H CH₂CH₂SCH₂C(O)NHMe
H H CH₂CH₂S(O)CH₂C(O)NHMe
H H CH₂CH₂S(O)₂CH₂C(O)NHMe
H H CH₂CH₂SCH₂C(O)NMe
H H CH₂CH₂S(O)CH₂C(O)NMe
H H CH₂CH₂S(O)₂CH₂C(O)N(Me)₂
H H CH₂CH₂SCH₂CH=CH₂
H H CH₂CH₂SCH₂CH≡CH
H H CH₂CH₂S(O)₂NHMe
H H CH₂CH₂S(O)₂N(Me)₂
H H CH₂CH₂S(O)₂NHEt
H H CH₂CH₂S(O)₂N(Et)₂
H H CH₂CH₂S(O)₂NHPr-n
H H CH₂CH₂S(O)₂N(Pr-n)₂
H H CH₂CH₂S(O)₂NHPr-i
H H CH₂CH₂S(O)₂N(Pr-i)₂
H H CH₂CH₂S(O)₂NHPr-c
H H CH₂CH₂S(O)₂NHBu-t
H H CH₂CH₂S(O)₂NHCH₂CF₃
H H CH₂CH₂S(O)₂NHCH₂CH₂OMe
H H CH₂CH₂S(O)₂NHCH₂CH₂SMe
H H CH₂CH₂S(O)₂NHCH₂CH=CH₂
H H CH₂CH₂S(O)₂NHCH₂CH≡CH
H H CH₂CH₂S(O)(=NCN)Me
H H CH₂CH(Me)SMe
H H CH₂CH(Me)S(O)Me
H H CH₂CH(Me)S(O)₂Me
H H CH₂CH(Me)SEt
H H CH₂CH(Me)S(O)Et
H H CH₂CH(Me)S(O)₂Et
H H CH₂CH(Et)SMe
H H CH₂CH(Et)S(O)Me
H H CH₂CH(Et)S(O)₂Me
H H CH₂CH(n-Pr)SMe
H H CH₂CH(n-Pr)S(O)Me
H H CH₂CH(n-Pr)S(O)₂Me
H H CH₂CH(i-Pr)SMe
H H CH₂CH(i-Pr)S(O)Me
H H CH₂CH(i-Pr)S(O)₂Me
H H CH₂CH(Ph)SMe
H H CH₂CH(Ph)S(O)Me
H H CH₂CH(Ph)S(O)₂Me
H H CH(Me)CH₂SMe
H H CH(Me)CH₂S(O)Me
H H CH(Me)CH₂S(O)₂Me
H H CH(Me)CH₂SEt
H H CH(Me)CH₂S(O)Et
H H CH(Me)CH₂S(O)₂Et
H H CH(Me)CH₂SPr-n
H H CH(Me)CH₂S(O)Pr-n
H H CH(Me)CH₂S(O)₂Pr-n
H H CH(Me)CH₂SPr-i
H H CH(Me)CH₂S(O)Pr-i
H H CH(Me)CH₂S(O)₂Pr-i
H H CH(Me)CH₂SPh
H H CH(Me)CH₂S(O)Ph
H H CH(Me)CH₂S(O)₂Ph
H H CH(Ph)CH₂SMe
H H CH(Ph)CH₂S(O)Me
H H CH(Ph)CH₂S(O)₂Me
H H CH(Me)CH(Me)SMe
H H CH(Me)CH(Me)S(O)Me
H H CH(Me)CH(Me)S(O)₂Me
H H C(Me)₂CH₂SMe
H H C(Me)₂CH₂S(O)Me
H H C(Me)₂CH₂S(O)₂Me
H H CH₂CH₂CH₂SMe
H H CH₂CH₂CH₂S(O)Me
H H CH₂CH₂CH₂S(O)₂Me
H H CH₂CH₂CH(Me)SMe
H H CH₂CH₂CH(Me)S(O)Me
H H CH₂CH₂CH(Me)S(O)₂Me
H H CH₂CH(Me)CH₂SMe
H H CH₂CH(Me)CH₂S(O)Me
H H CH₂CH(Me)CH₂S(O)₂Me
H H CH(Me)CH₂CH₂SMe
H H CH(Me)CH₂CH₂S(O)Me
H H CH(Me)CH₂CH₂S(O)₂Me
H H C(Me)₂CH₂CH₂SMe
H H C(Me)₂CH₂CH₂S(O)Me
H H C(Me)₂CH₂CH₂S(O)₂Me
H H CH(Me)(CH₂)₃SMe
H H CH(Me)(CH₂)₃S(O)Me
H H CH(Me)(CH₂)₃S(O)₂Me
H H CH(Me)(CH₂)₄SMe
H H CH(Me)(CH₂)₄S(O)Me
H H CH(Me)(CH₂)₄S(O)₂Me
H H CH₂NHC(O)Me
H H CH₂NHC(O)Et
H H CH₂NHC(O)Pr-n
H H CH₂CH₂NHC(O)Me
H H CH₂CH₂NHC(O)Et
H H CH₂CH₂NHC(O)Pr-n
H H CH₂CH₂NHC(O)Pr-i
H H CH₂CH₂NHC(O)Pr-c
H H CH₂CH₂NHC(O)Bu-n
H H CH₂CH₂NHC(O)Bu-i
H H CH₂CH₂NHC(O)Bu-s
H H CH₂CH₂NHC(O)Bu-t
H H CH₂CH₂NHC(O)CF₃
H H CH₂CH₂NHC(O)CF₂Cl
H H CH₂CH₂NHC(O)Ph
H H CH₂CH₂NHC(O)CH₂CF₃
H H CH₂CH₂NHC(O)CH₂SMe
H H CH₂CH₂NHC(O)CH₂S(O)Me
H H CH₂CH₂NHC(O)CH₂S(O)₂Me
H H CH₂CH₂N(Me)C(O)Me
H H CH₂CH₂N(Me)C(O)Et
H H CH₂CH₂N(Me)C(O)CF₃
H H CH₂CH₂N(Me)C(O)CH₂CF₃
H H CH₂CH₂N(Me)C(O)CH₂SMe
H H CH ₂CH₂N(Me)C(O)CH₂S(O)Me
H H CH ₂CH₂N(Me)C(O)CH₂S(O)₂Me
H H CH₂CH₂NHC(O)OMe
H H CH₂CH₂NHC(O)OEt
H H CH₂CH₂NHC(O)OPr-n
H H CH₂CH₂NHC(O)OBu-t
H H CH₂CH₂NHC(O)NHEt
H H CH₂CH₂NHC(O)NHPr-n
H H CH₂CH₂NHC(O)NHPr-i
H H CH₂CH₂NHC(O)NHBu-t
H H CH₂CH₂NHC(O)N(Me)₂
H H CH₂CH₂NHSO₂Me
H H CH₂CH₂NHSO₂Et
H H CH₂CH₂NHSO₂CF₃
H H CH₂CH₂NHSO₂Ph
H H CH₂CH₂NHSO₂N(Me)₂
H H CH₂CH₂NHP(S)(OMe)₂
H H CH₂CH₂NHP(S)(OEt)₂
H H CH₂CH₂N(Me)SO₂Me
H H CH₂CH₂N(Me)SO₂CF₃
H H CH₂CH₂N(Me)OMe
H H CH₂CH(Me)NHC(O)Me
H H CH₂CH(Me)NHC(O)CF₃
H H CH₂CH(Me)NHC(O)CH₂CF₃
H H CH₂CH(Me)NHC(O)CH₂SMe
H H CH(Me)NHC(O)CH₂S(O)Me
H H CH(Me)NHC(O)CH₂S(O)₂Me
H H CH₂CH(Me)NHC(O)OMe
H H CH(Me)CH₂NHC(O)Me
H H CH(Me)CH₂NHC(O)CF₃
H H CH(Me)CH₂NHC(O)CH₂CF₃
H H CH(Me)CH₂NHC(O)CH₂SMe
H H CH(Me)CH₂NHC(O)CH₂S(O)Me
H H CH(Me)CH₂NHC(O)CH₂S(O)₂Me
H H CH(Me)CH₂NHC(O)OMe
H H CH₂CH₂CH₂NHC(O)Me
H H CH₂CH₂CH₂NHC(O)OMe
H H D2-1a
H H D2-1b
H H D2-2a
H H D2-2b
H H D2-5a
H H D2-5b
H H D2-5c
H H D2-6a
H H D2-6b
H H D2-6c
H H D2-7a
H H D2-8a
H H D2-8b
H H D2-8c
H H D2-9a
H H D2-9b
H H D2-9c
H H D2-10a
H H D2-10b
H H D2-10c
H H D2-11a
H H D2-12a
H H D2-12b
H H D2-12c
H H D2-13a
H H D2-13b
H H D2-14a
H H D2-14b
H H D2-15a
H H D2-15b
H H D2-16a
H H D2-17a
H H D2-18a
H H D2-19a
H H D2-21a
H H D2-21b
H H D2-22a
H H D2-23a
H H D2-23b
H H D2-24a
H H D2-25a
H H D2-27a
H H D2-30a
H H D2-31a
H H D2-32a
H H D2-34a
H H D2-36a
H H D2-37a
H H D2-41a
H H D2-43a
H H D2-45a
H H D2-46a
H H D2-49a
H H D2-51a
H H D2-53a
H H D2-59a
H H D2-61a
H H D2-63a
H H D2-68a
H H D2-75a
H H D2-76a
H H D2-76b
H H D2-77a
H H D2-77b
H H D2-78a
H H D2-78b
H H D2-79a
H H D2-81a
H H D2-82a
H H D2-84a
H H D2-85a
H H D2-87a
H H D2-90a
H H D2-100a
H H D2-100b
H H D2-100c
H H D2-100d
H H D2-100e
H H D2-101a
H H D2-101b
H H D2-101c
H H D2-101d
H H D2-102a
H H D2-102b
H H D2-102c
H H D2-102d
H H D2-102e
H H D2-102f
H H D2-103a
H H D2-108a
H H CH₂(D2-1a)
H H CH₂(D2-1b)
H H CH₂(D2-2a)
H H CH₂(D2-2b)
H H CH₂(D2-4a)
H H CH₂(D2-4b)
H H CH₂(D2-5a)
H H CH₂(D2-5b)
H H CH₂(D2-5c)
H H CH₂(D2-6a)
H H CH₂(D2-6b)
H H CH₂(D2-6c)
H H CH₂(D2-7a)
H H CH₂(D2-8a)
H H CH₂(D2-8b)
H H CH₂(D2-8c)
H H CH₂(D2-9a)
H H CH₂(D2-9b)
H H CH₂(D2-9c)
H H CH₂(D2-10a)
H H CH₂(D2-10b)
H H CH₂(D2-10c)
H H CH₂(D2-12a)
H H CH₂(D2-12b)
H H CH₂(D2-12c)
H H CH₂(D2-13a)
H H CH₂(D2-13b)
H H CH₂(D2-14a)
H H CH₂(D2-14b)
H H CH₂(D2-15a)
H H CH₂(D2-15b)
H H CH₂(D2-16a)
H H CH₂(D2-17a)
H H CH₂(D2-18a)
H H CH₂(D2-19a)
H H CH₂(D2-20a)
H H CH₂(D2-21a)
H H CH₂(D2-21b)
H H CH₂(D2-23a)
H H CH₂(D2-23b)
H H CH₂(D2-25a)
H H CH₂(D2-27a)
H H CH₂(D2-30a)
H H CH₂(D2-31a)
H H CH₂(D2-32a)
H H CH₂(D2-33a)
H H CH₂(D2-34a)
H H CH₂(D2-35a)
H H CH₂(D2-35b)
H H CH₂(D2-36a)
H H CH₂(D2-37a)
H H CH₂(D2-38a)
H H CH₂(D2-39a)
H H CH₂(D2-40a)
H H CH₂(D2-41a)
H H CH₂(D2-42a)
H H CH₂(D2-43a)
H H CH₂(D2-45a)
H H CH₂(D2-46a)
H H CH₂(D2-49a)
H H CH₂(D2-51a)
H H CH₂(D2-53a)
H H CH₂(D2-59a)
H H CH₂(D2-61a)
H H CH₂(D2-63a)
H H CH₂(D2-68a)
H H CH₂(D2-75a)
H H CH₂(D2-76a)
H H CH₂(D2-76b)
H H CH₂(D2-77a)
H H CH₂(D2-77b)
H H CH₂(D2-78a)
H H CH₂(D2-78b)
H H CH₂(D2-79a)
H H CH₂(D2-81a)
H H CH₂(D2-82a)
H H CH₂(D2-84a)
H H CH₂(D2-85a)
H H CH₂(D2-87a)
H H CH₂(D2-90a)
H H CH₂(D2-100a)
H H CH₂(D2-100b)
H H CH₂(D2-100c)
H H CH₂(D2-100d)
H H CH₂(D2-100e)
H H CH₂(D2-101a)
H H CH₂(D2-101b)
H H CH₂(D2-101c)
H H CH₂(D2-101d)
H H CH₂(D2-102a)
H H CH₂(D2-102b)
H H CH₂(D2-102c)
H H CH₂(D2-102d)
H H CH₂(D2-102e)
H H CH₂(D2-102f)
H H CH₂(D2-103a)
H H CH₂(D2-108a)
H H CH(Me)(D2-1a)
H H CH(Me)(D2-2a)
H H CH(Me)(D2-5a)
H H CH(Me)(D2-5c)
H H CH(Me)(D2-6c)
H H CH(Me)(D2-8c)
H H CH(Me)(D2-9b)
H H CH(Me)(D2-9c)
H H CH(Me)(D2-10b)
H H CH(Me)(D2-10c)
H H CH(Me)(D2-12b)
H H CH(Me)(D2-12c)
H H CH(Me)(D2-13b)
H H CH(Me)(D2-14a)
H H CH(Me)(D2-14b)
H H CH(Me)(D2-15a)
H H CH(Me)(D2-15b)
H H CH(Me)(D2-16a)
H H CH(Me)(D2-17a)
H H CH(Me)(D2-18a)
H H CH(Me)(D2-23b)
H H CH(Me)(D2-27a)
H H CH(Me)(D2-31a)
H H CH(Me)(D2-32a)
H H CH(Me)(D2-35a)
H H CH(Me)(D2-36a)
H H CH(Me)(D2-37a)
H H CH(Me)(D2-39a)
H H CH(Me)(D2-41a)
H H CH₂C(O)NH(D2-1a)
H H CH₂C(O)NH(D2-2a)
H H CH₂C(O)NH(D2-5a)
H H CH₂C(O)NH(D2-5c)
H H CH₂C(O)NH(D2-6c)
H H CH₂C(O)NH(D2-8c)
H H CH₂C(O)NH(D2-9b)
H H CH₂C(O)NH(D2-9c)
H H CH₂C(O)NH(D2-10b)
H H CH₂C(O)NH(D2-10c)
H H CH₂C(O)NH(D2-12b)
H H CH₂C(O)NH(D2-12c)
H H CH₂C(O)NH(D2-13b)
H H CH₂C(O)NH(D2-14a)
H H CH₂C(O)NH(D2-14b)
H H CH₂C(O)NH(D2-15a)
H H CH₂C(O)NH(D2-15b)
H H CH₂C(O)NH(D2-16a)
H H CH₂C(O)NH(D2-17a)
H H CH₂C(O)NH(D2-18a)
H H CH₂C(O)NH(D2-23b)
H H CH₂C(O)NH(D2-27a)
H H CH₂C(O)NH(D2-31a)
H H CH₂C(O)NH(D2-32a)
H H CH₂C(O)NH(D2-35a)
H H CH₂C(O)NH(D2-36a)
H H CH₂C(O)NH(D2-37a)
H H CH₂C(O)NH(D2-39a)
H H CH₂C(O)NH(D2-41a)
H H CH₂C(O)NH(D2-45a)
H H CH₂C(O)NH(D2-46a)
H H CH₂C(O)NH(D2-49a)
H H CH₂C(O)NH(D2-51a)
H H CH₂C(O)NH(D2-53a)
H H CH₂C(O)NH(D2-59a)
H H CH₂C(O)NH(D2-61a)
H H CH₂C(O)NH(D2-63a)
H H CH₂C(O)NH(D2-68a)
H H CH₂C(O)NH(D2-75a)
H H CH₂C(O)NH(D2-76a)
H H CH₂C(O)NH(D2-76b)
H H CH₂C(O)NH(D2-77a)
H H CH₂C(O)NH(D2-77b)
H H CH₂C(O)NH(D2-78a)
H H CH₂C(O)NH(D2-78b)
H H CH₂C(O)NH(D2-79a)
H H CH₂C(O)NH(D2-82a)
H H CH₂C(O)NH(D2-84a)
H H CH₂C(O)NH(D2-85a)
H H CH₂C(O)NH(D2-87a)
H H CH₂C(O)NH(D2-90a)
H H CH₂C(O)NH(D2-100a)
H H CH₂C(O)NH(D2-100b)
H H CH₂C(O)NH(D2-100c)
H H CH₂C(O)NH(D2-100d)
H H CH₂C(O)NH(D2-100e)
H H CH₂C(O)NH(D2-101a)
H H CH₂C(O)NH(D2-101b)
H H CH₂C(O)NH(D2-101c)
H H CH₂C(O)NH(D2-101d)
H H CH₂C(O)NH(D2-108a)
H H CH₂C(O)NHCH₂(D2-1a)
H H CH₂C(O)NHCH₂(D2-2a)
H H CH₂C(O)NHCH₂(D2-5a)
H H CH₂C(O)NHCH₂(D2-5c)
H H CH₂C(O)NHCH₂(D2-6c)
H H CH₂C(O)NHCH₂(D2-8c)
H H CH₂C(O)NHCH₂(D2-9b)
H H CH₂C(O)NHCH₂(D2-9c)
H H CH₂C(O)NHCH₂(D2-10b)
H H CH₂C(O)NHCH₂(D2-10c)
H H CH₂C(O)NHCH₂(D2-12b)
H H CH₂C(O)NHCH₂(D2-12c)
H H CH₂C(O)NHCH₂(D2-13b)
H H CH₂C(O)NHCH₂(D2−14a)
H H CH₂C(O)NHCH₂(D2-14b)
H H CH₂C(O)NHCH₂(D2-15a)
H H CH₂C(O)NHCH₂(D2-15b)
H H CH₂C(O)NHCH₂(D2-16a)
H H CH₂C(O)NHCH₂(D2-17a)
H H CH₂C(O)NHCH₂(D2-18a)
H H CH₂C(O)NHCH₂(D2-23b)
H H CH₂C(O)NHCH₂(D2-27a)
H H CH₂C(O)NHCH₂(D2-31a)
H H CH₂C(O)NHCH₂(D2-32a)
H H CH₂C(O)NHCH₂(D2-35a)
H H CH₂C(O)NHCH₂(D2-36a)
H H CH₂C(O)NHCH₂(D2-37a)
H H CH₂C(O)NHCH₂(D2-39a)
H H CH₂C(O)NHCH₂(D2-41a)
H H CH₂C(O)NHCH₂(D2-45a)
H H CH₂C(O)NHCH₂(D2-46a)
H H CH₂C(O)NHCH₂(D2-49a)
H H CH₂C(O)NHCH₂(D2-51a)
H H CH₂C(O)NHCH₂(D2-53a)
H H CH₂C(O)NHCH₂(D2-59a)
H H CH₂C(O)NHCH₂(D2-61a)
H H CH₂C(O)NHCH₂(D2-63a)
H H CH₂C(O)NHCH₂(D2-68a)
H H CH₂C(O)NHCH₂(D2-75a)
H H CH₂C(O)NHCH₂(D2-76a)
H H CH₂C(O)NHCH₂(D2-76b)
H H CH₂C(O)NHCH₂(D2-77a)
H H CH₂C(O)NHCH₂(D2-77b)
H H CH₂C(O)NHCH₂(D2-78a)
H H CH₂C(O)NHCH₂(D2-78b)
H H CH₂C(O)NHCH₂(D2-79a)
H H CH₂C(O)NHCH₂(D2-82a)
H H CH₂C(O)NHCH₂(D2-84a)
H H CH₂C(O)NHCH₂(D2-85a)
H H CH₂C(O)NHCH₂(D2-87a)
H H CH₂C(O)NHCH₂(D2-90a)
H H CH₂C(O)NHCH₂(D2-102a)
H H CH₂C(O)NHCH₂(D2-102b)
H H CH₂C(O)NHCH₂(D2-102c)
H H CH₂C(O)NHCH₂(D2-102d)
H H CH₂C(O)NHCH₂(D2-102e)
H H CH₂C(O)NHCH₂(D2-102f)
H H CH₂C(O)NHCH₂(D2-103a)
H H CH₂C(O)NHCH₂(D2-108a)
H H NH(D2-7a)
H H NH(D2-10c)
H H NH(D2-22a)
H H NH(D2-24a)
H H NH(D2-32a)
H H NC(O)Me(D2-32a)
H H NC(O)OMe(D2-32a)
H H NC(O)Et(D2-32a)
H H NC(O)OEt(D2-32a)
H H NC(O)CH₂CF₃(D2-32a)
H H NSO₂Me(D2-32a)
H H NSO₂CF₃(D2-32a)
H H NSO₂Ph(D2-32a)
H H NH(D2-35a)
H H NH(D2-36a)
H H NH(D2-37a)
H H NH(D2-39a)
H H NH(D2-43a)
H H NH(D2-45a)
H H NH(D2-49a)
H H NH(D2-51a)
H H NH(D2-53a)
H H NH(D2-59a)
H H NH(D2-61a)
H H NH(D2-63a)
H H NH(D2-108a)
H H NH{D2-32b(3-Cl)}
H H NH{D2-32b(4-Cl)}
H H NH{D2-32b(5-Cl)}
H H NH{D2-32b(6-Cl)}
H H NH{D2-32b(4-CF₃)}
H H NH{D2-108b(2-Cl)}
H H NH{D2-108b(3-Cl)}
H H NH{D2-108b(4-Cl)}
H H NH{D2-108b(2-Me)}
H H NH{D2-108b(3-Me)}
H H NH{D2-108b(4-Me)}
H H CH₂CH₂(D2-1a)
H H CH₂CH₂(D2-1b)
H H CH₂CH₂(D2-2a)
H H CH₂CH₂(D2-2b)
H H CH₂CH₂(D2-5c)
H H CH₂CH₂(D2-6c)
H H CH₂CH₂(D2-7a)
H H CH₂CH₂(D2-8c)
H H CH₂CH₂(D2-9b)
H H CH₂CH₂(D2-10b)
H H CH₂CH₂(D2-10c)
H H CH₂CH₂(D2-11a)
H H CH₂CH₂(D2-20a)
H H CH₂CH₂(D2-22a)
H H CH₂CH₂(D2-24a)
H H CH₂CH₂(D2-26a)
H H CH₂CH₂(D2-28a)
H H CH₂CH₂(D2-29a)
H H CH₂CH₂(D2-32a)
H H CH₂CH₂(D2-36a)
H H CH₂CH₂(D2-37a)
H H CH₂CH₂OCH₂(D2-1a)
H H CH₂CH₂OCH₂(D2-1b)
H H CH₂CH₂OCH₂(D2-2a)
H H CH₂CH₂OCH₂(D2-2b)
H H CH₂CH₂OCH₂(D2-4a)
H H CH₂CH₂OCH₂(D2-4b)
H H CH₂CH₂OCH₂(D2-5a)
H H CH₂CH₂OCH₂(D2-5b)
H H CH₂CH₂OCH₂(D2-5c)
H H CH₂CH₂OCH₂(D2-6a)
H H CH₂CH₂OCH₂(D2-6b)
H H CH₂CH₂OCH₂(D2-6c)
H H CH₂CH₂OCH₂(D2-7a)
H H CH₂CH₂OCH₂(D2-8a)
H H CH₂CH₂OCH₂(D2-8b)
H H CH₂CH₂OCH₂(D2-8c)
H H CH₂CH₂OCH₂(D2-9a)
H H CH₂CH₂OCH₂(D2-9b)
H H CH₂CH₂OCH₂(D2-9c)
H H CH₂CH₂OCH₂(D2-10a)
H H CH₂CH₂OCH₂(D2-10b)
H H CH₂CH₂OCH₂(D2-10c)
H H CH₂CH₂OCH₂(D2-12a)
H H CH₂CH₂OCH₂(D2-12b)
H H CH₂CH₂OCH₂(D2-12c)
H H CH₂CH₂OCH₂(D2-13a)
H H CH₂CH₂OCH₂(D2-13b)
H H CH₂CH₂OCH₂(D2-14a)
H H CH₂CH₂OCH₂(D2-14b)
H H CH₂CH₂OCH₂(D2-15a)
H H CH₂CH₂OCH₂(D2-15b)
H H CH₂CH₂OCH₂(D2-16a)
H H CH₂CH₂OCH₂(D2-17a)
H H CH₂CH₂OCH₂(D2-18a)
H H CH₂CH₂OCH₂(D2-19a)
H H CH₂CH₂OCH₂(D2-20a)
H H CH₂CH₂OCH₂(D2-21a)
H H CH₂CH₂OCH₂(D2-21b)
H H CH₂CH₂OCH₂(D2-23a)
H H CH₂CH₂OCH₂(D2-23b)
H H CH₂CH₂OCH₂(D2-25a)
H H CH₂CH₂OCH₂(D2-27a)
H H CH₂CH₂OCH₂(D2-30a)
H H CH₂CH₂OCH₂(D2-31a)
H H CH₂CH₂OCH₂(D2-32a)
H H CH₂CH₂OCH₂(D2-33a)
H H CH₂CH₂OCH₂(D2-34a)
H H CH₂CH₂OCH₂(D2-35a)
H H CH₂CH₂OCH₂(D2-35b)
H H CH₂CH₂OCH₂(D2-36a)
H H CH₂CH₂OCH₂(D2-37a)
H H CH₂CH₂OCH₂(D2-38a)
Me H CH₂CH₂OCH₂(D2-39a)
Me H CH₂CH₂OCH₂(D2-40a)
Me H CH₂CH₂OCH₂(D2-41a)
Me H CH₂CH₂OCH₂(D2-42a)
Me H CH₂CH₂OCH₂(D2-43a)
Me H CH₂CH₂OCH₂(D2-45a)
H H CH₂CH₂OCH₂(D2-46a)
H H CH₂CH₂OCH₂(D2-49a)
H H CH₂CH₂OCH₂(D2-51a)
H H CH₂CH₂OCH₂(D2-53a)
H H CH₂CH₂OCH₂(D2-59a)
H H CH₂CH₂OCH₂(D2-61a)
H H CH₂CH₂OCH₂(D2-63a)
H H CH₂CH₂OCH₂(D2-68a)
H H CH₂CH₂OCH₂(D2-75a)
H H CH₂CH₂OCH₂(D2-76a)
H H CH₂CH₂OCH₂(D2-76b)
H H CH₂CH₂OCH₂(D2-77a)
H H CH₂CH₂OCH₂(D2-77b)
H H CH₂CH₂OCH₂(D2-78a)
H H CH₂CH₂OCH₂(D2-78b)
H H CH₂CH₂OCH₂(D2-79a)
H H CH₂CH₂OCH₂(D2-81a)
H H CH₂CH₂OCH₂(D2-82a)
H H CH₂CH₂OCH₂(D2-84a)
H H CH₂CH₂OCH₂(D2-85a)
H H CH₂CH₂OCH₂(D2-87a)
H H CH₂CH₂OCH₂(D2-90a)
H H CH₂CH₂OCH₂(D2-100a)
H H CH₂CH₂OCH₂(D2-100b)
H H CH₂CH₂OCH₂(D2-100c)
H H CH₂CH₂OCH₂(D2-100d)
H H CH₂CH₂OCH₂(D2-100e)
H H CH₂CH₂OCH₂(D2-101a)
H H CH₂CH₂OCH₂(D2-101b)
H H CH₂CH₂OCH₂(D2-101c)
H H CH₂CH₂OCH₂(D2-101d)
H H CH₂CH₂OCH₂(D2-102a)
H H CH₂CH₂OCH₂(D2-102b)
H H CH₂CH₂OCH₂(D2-102c)
H H CH₂CH₂OCH₂(D2-102d)
H H CH₂CH₂OCH₂(D2-102e)
H H CH₂CH₂OCH₂(D2-102f)
H H CH₂CH₂OCH₂(D2-103a)
H H CH₂CH₂OCH₂(D2-108a)
H H CH₂CH₂SCH₂(D2-1a)
H H CH₂CH₂SCH₂(D2-1b)
H H CH₂CH₂SCH₂(D2-2a)
H H CH₂CH₂SCH₂(D2-2b)
H H CH₂CH₂SCH₂(D2-4a)
H H CH₂CH₂SCH₂(D2-4b)
H H CH₂CH₂SCH₂(D2-5a)
H H CH₂CH₂SCH₂(D2-5b)
H H CH₂CH₂SCH₂(D2-5c)
H H CH₂CH₂SCH₂(D2-6a)
H H CH₂CH₂SCH₂(D2-6b)
H H CH₂CH₂SCH₂(D2-6c)
H H CH₂CH₂SCH₂(D2-7a)
H H CH₂CH₂SCH₂(D2-8a)
H H CH₂CH₂SCH₂(D2-8b)
H H CH₂CH₂SCH₂(D2-8c)
H H CH₂CH₂SCH₂(D2-9a)
H H CH₂CH₂SCH₂(D2-9b)
H H CH₂CH₂SCH₂(D2-9c)
H H CH₂CH₂SCH₂(D2-10a)
H H CH₂CH₂SCH₂(D2-10b)
H H CH₂CH₂SCH₂(D2-10c)
H H CH₂CH₂SCH₂(D2-12a)
H H CH₂CH₂SCH₂(D2-12b)
H H CH₂CH₂SCH₂(D2-12c)
H H CH₂CH₂SCH₂(D2-13a)
H H CH₂CH₂SCH₂(D2-13b)
H H CH₂CH₂OCH₂(D2-14a)
H H CH₂CH₂SCH₂(D2-14b)
H H CH₂CH₂SCH₂(D2-15a)
H H CH₂CH₂SCH₂(D2-15b)
H H CH₂CH₂SCH₂(D2-16a)
H H CH₂CH₂SCH₂(D2-17a)
H H CH₂CH₂SCH₂(D2-18a)
H H CH₂CH₂SCH₂(D2-19a)
H H CH₂CH₂SCH₂(D2-20a)
H H CH₂CH₂SCH₂(D2-21a)
H H CH₂CH₂SCH₂(D2-21b)
H H CH₂CH₂SCH₂(D2-23a)
H H CH₂CH₂SCH₂(D2-23b)
H H CH₂CH₂SCH₂(D2-25a)
H H CH₂CH₂SCH₂(D2-27a)
H H CH₂CH₂SCH₂(D2-30a)
H H CH₂CH₂SCH₂(D2-31a)
H H CH₂CH₂SCH₂(D2-32a)
H H CH₂CH₂SCH₂(D2-33a)
H H CH₂CH₂SCH₂(D2-34a)
H H CH₂CH₂SCH₂(D2-35a)
H H CH₂CH₂SCH₂(D2-35b)
H H CH₂CH₂SCH₂(D2-36a)
H H CH₂CH₂SCH₂(D2-37a)
H H CH₂CH₂SCH₂(D2-38a)
H H CH₂CH₂SCH₂(D2-39a)
H H CH₂CH₂SCH₂(D2-40a)
H H CH₂CH₂SCH₂(D2-41a)
H H CH₂CH₂SCH₂(D2-42a)
H H CH₂CH₂SCH₂(D2-43a)
H H CH₂CH₂SCH₂(D2-45a)
H H CH₂CH₂SCH₂(D2-46a)
H H CH₂CH₂SCH₂(D2-49a)
H H CH₂CH₂SCH₂(D2-51a)
H H CH₂CH₂SCH₂(D2-53a)
H H CH₂CH₂SCH₂(D2-59a)
H H CH₂CH₂SCH₂(D2-61a)
H H CH₂CH₂SCH₂(D2-63a)
H H CH₂CH₂SCH₂(D2-68a)
H H CH₂CH₂SCH₂(D2-75a)
H H CH₂CH₂SCH₂(D2-76a)
H H CH₂CH₂SCH₂(D2-76b)
H H CH₂CH₂SCH₂(D2-77a)
H H CH₂CH₂SCH₂(D2-77b)
H H CH₂CH₂SCH₂(D2-78a)
H H CH₂CH₂SCH₂(D2-78b)
H H CH₂CH₂SCH₂(D2-79a)
H H CH₂CH₂SCH₂(D2-81a)
H H CH₂CH₂SCH₂(D2-82a)
H H CH₂CH₂SCH₂(D2-84a)
H H CH₂CH₂SCH₂(D2-85a)
H H CH₂CH₂SCH₂(D2-87a)
H H CH₂CH₂SCH₂(D2-90a)
H H CH₂CH₂SCH₂(D2-100a)
H H CH₂CH₂SCH₂(D2-100b)
H H CH₂CH₂SCH₂(D2-100c)
H H CH₂CH₂SCH₂(D2-100d)
H H CH₂CH₂SCH₂(D2-100e)
H H CH₂CH₂SCH₂(D2-101a)
H H CH₂CH₂SCH₂(D2-101b)
H H CH₂CH₂SCH₂(D2-101c)
H H CH₂CH₂SCH₂(D2-101d)
H H CH₂CH₂SCH₂(D2-102a)
H H CH₂CH₂SCH₂(D2-102b)
H H CH₂CH₂SCH₂(D2-102c)
H H CH₂CH₂SCH₂(D2-102d)
H H CH₂CH₂SCH₂(D2-102e)
H H CH₂CH₂SCH₂(D2-102f)
H H CH₂CH₂SCH₂(D2-103a)
H H CH₂CH₂SCH₂(D2-108a)
H H CH₂{D2-1c(3-Me)}
H H CH₂{D2-1d(5-Cl)}
H H CH₂{D2-2c(5-Br)}
H H CH₂{D2-2d(5-Cl)}
H H CH₂{D2-4c(5-Cl)}
H H CH₂{D2-4d(5-Cl)}
H H CH₂{D2-5d(3-Me)}
H H CH₂{D2-5e(3-Me)}
H H CH₂{D2-5f(5-Me)}
H H CH₂{D2-6d(3-Cl)}
H H CH₂{D2-6e(3-Me)}
H H CH₂{D2-6f(5-Me)}
H H CH₂{D2-7a(3-Me)}
H H CH₂{D2-8d(3-Cl)}
H H CH₂{D2-8e(3-CF₃)}
H H CH₂{D2-8f(5-Me)}
H H CH₂{D2-9d(2-Me)}
H H CH₂{D2-9e(2-Me)}
H H CH₂{D2-9f(4-Me)}
H H CH₂{D2-10e(2-Me)}
H H CH₂{D2-10f(2-Cl)}
H H CH₂{D2-10e(2-Br)}
H H CH₂{D2-12d(4-Me)}
H H CH₂{D2-12e(5-Me)}
H H CH₂{D2-12f(5-Cl)}
H H CH₂{D2-13c(Me)}
H H CH₂{D2-13d(Cl)}
H H CH₂{D2-14c(Me)}
H H CH₂{D2-14d(Me)}
H H CH₂{D2-15c(Cl)}
H H CH₂{D2-15d(Me)}
H H CH₂{D2-16b(Ph)}
H H CH₂{D2-17b(Ph)}
H H CH₂{D2-18b(Me)}
H H CH₂{D2-19b(Cl)}
H H CH₂{D2-20b(Me)}
H H CH₂{D2-21c(Me)}
H H CH₂{D2-21d(Me)}
H H CH₂{D2-23c(t-Bu)}
H H CH₂{D2-23d(Ph)}
H H CH₂{D2-25b(Me)}
H H CH₂{D2-27a(Me)}
H H CH₂{D2-32b(3-Cl)}
H H CH₂{D2-32b(4-Cl)}
H H CH₂{D2-32b(5-Cl)}
H H CH₂{D2-32b(6-Cl)}
H H CH₂{D2-32b(3-Me)}
H H CH₂{D2-32b(4-Me)}
H H CH₂{D2-32b(5-Me)}
H H CH₂{D2-32b(6-Me)}
H H CH₂{D2-32b(5-CF₃)}
H H CH₂{D2-33b(4-CF₃)}
H H CH₂{D2-34b(3-Cl)}
H H CH₂{D2-35c(3-Cl)}
H H CH₂{D2-35d(3-Cl)}
H H CH₂{D2-36b(2-Me)}
H H CH₂{D2-37b(4-Me)}
H H CH₂{D2-38b(2-Me)}
H H CH₂{D2-39b(5-Me)}
H H CH₂{D2-108b(2-Cl)}
H H CH₂{D2-108b(3-Cl)}
H H CH₂{D2-108b(4-Cl)}
H H CH₂{D2-108b(2-Me)}
H H CH₂{D2-108b(3-Me)}
H H CH₂{D2-108b(4-Me)}
H H CH₂{D2-108b(2-CF₃)}
H H CH₂{D2-108b(3-CF₃)}
H H CH₂{D2-108b(4-CF₃)}
H H CH₂{D2-108b(2-OMe)}
H H CH₂{D2-108b(3-OMe)}
H H CH₂{D2-108b(4-OMe)}
H H CH₂CH₂{D2-7b(4-Cl)}
H H CH₂CH₂{D2-10e(2-Cl)}
H H CH₂CH₂{D2-11b(2-Me)}
H H CH₂CH₂{D2-20b(4-Me)}
H H CH₂CH₂{D2-22b(3-SMe)}
H H CH₂CH₂{D2-24b(3-Me)}
H H CH₂CH₂{D2-26b(4-CO₂Me)}
H H CH₂CH₂{D2-28b(Me)}
H H CH₂CH₂{D2-29a(Ph)}
H H CH₂CH₂{D2-32b(3-Cl)}
H H CH₂CH₂{D2-36b(2-Me)}
H H CH₂CH₂{D2-37b(4-Me)
――――――――――――――――――――――――――
〔第５表〕 ―――――――――――――――――――――――――
R ^d R ^e R ^f
―――――――――――――――――――――――――
HH SMe
HHC (O) OEt
HHC (O) NHCH ₂ CF ₃
HHC (O) N (Me) CH ₂ CF ₃
HH D2-7b (X ² = 3-CF ₂ CF ₃ )
HH D2-108a
HH D2-108b (Z ² = 4-CF ₃ )
H -CH ₂ CH ₂ N (CH ₂ CF ₃ ) C (O)-
H -CH ₂ CH ₂ NHC (O)-
HH Si (Me) ₃
HH CH ₂ SMe
HHS (O) Me
HHS (O) ₂ Me
HHC (O) SMe
HHC (O) NHEt
HH D2-32b (X ² = 5-CF ₃ )
HHH
HH Me
HH Et
HH n-Pr
HH i-Pr
HH c-Pr
HH n-Bu
HH i-Bu
HH s-Bu
HH t-Bu
HH c-Bu
HH n-Pen
HH c-Pen
HH n-Hex
HH c-Hex
HH Hep
HH Oct
HH CH ₂ Pr-c
HH CH ₂ Bu-i
HH CH ₂ Bu-s
HH CH ₂ Bu-t
HH CH ₂ Bu-c
HH CH ₂ Pen-c
HH CH ₂ Hex-c
HH CH (CH ₃ ) Pr-n
HH CH (CH ₃ ) Pr-i
HH CH (CH ₃ ) Pr-n
HH CH (CH ₃ ) Bu-i
HH CH (Et) ₂
HHC (CH ₃ ) ₂ Et
HHC (CH ₃ ) ₂ Pr-n
HH CH ₂ CH ₂ F
HH CH ₂ CH ₂ Cl
HH CH ₂ CH ₂ Br
HH CH ₂ CHF ₂
HH CH ₂ CHFCl
HH CH ₂ CHCl ₂
HH CH ₂ CHFBr
HH CH ₂ CF ₂ Cl
HH CH ₂ CFCl ₂
HH CH ₂ CCl ₃
HH CH ₂ CF ₂ Br
HH CH ₂ CFClBr
HH CH ₂ CCl ₂ Br
HH CH (CH ₃ ) CH ₂ F
HH CH (CH ₃ ) CH ₂ Cl
HH CH (CH ₃ ) CH ₂ Br
HH CH ₂ CHFCH ₃
HH CH ₂ CHClCH ₃
HH CH ₂ CHBrCH ₃
HH CH ₂ CFClCH ₃
HH CH ₂ CHClCH ₂ Cl
HH CH ₂ CHBrCH ₂ F
HH CH ₂ CHClCH ₂ Br
HH CH ₂ CHBrCH ₂ Cl
HH CH ₂ CHBrCHCl ₂
HH CH ₂ CClBrCH ₃
HH CH ₂ CHBrCH ₂ Br
HH CH ₂ CH ₂ CF ₃
HH CH ₂ CH ₂ CF ₂ Br
HH CH ₂ CClBrCH ₂ Cl
HH CH ₂ CF ₂ CF ₂ H
HH CH ₂ CHClCF ₃
HH CH ₂ CF ₂ CF ₃
HH CH ₂ CF (CH ₃ ) ₂
HH CH ₂ CHFCH ₂ CH ₃
HH CH ₂ CHClCH ₂ CH ₃
HH CH ₂ CF ₂ CHFCF ₃
HH CH ₂ CF ₂ CF ₂ CHF ₂
HH CH ₂ CF ₂ CF ₂ CF ₃
HHC (CH ₃ ) ₂ CH ₂ Cl
HHC (CH ₃ ) ₂ CH ₂ Br
HHC (CH ₃ ) ₂ CHBrCH ₂ Br
HH CH ₂ CF ₃
HH CH (CF ₃ ) Me
Me H CH (CF ₃ ) Et
OMe H CH (CF ₃ ) OH
HH CH (CF ₃ ) OMe
HH CH ₂ CH (OMe) ₂
HH CH ₂ CH (OEt) ₂
SMe H CH ₂ CN
CN H CH (Me) CN
HHC (Me) ₂ CN
HH CH (OMe) CN
HH CH ₂ CH ₂ CN
HH CH ₂ C (O) Me
HC (O) OMe CH ₂ C (O) OMe
HH CH ₂ C (O) OEt
HH CH ₂ C (O) OCH ₂ CF ₃
HH CH (Me) C (O) OMe
HH CH (Me) C (O) OEt
HH CH (Me) C (O) OCH ₂ CF ₃
H Me CH (OMe) C (O) OMe
H Et CH (OMe) C (O) OEt
H n-Pr CH (OMe) C (O) OCH ₂ CF ₃
H i-Pr CH (Ph) C (O) OMe
H CH ₂ OCH ₃ CH (Ph) C (O) OEt
H CH ₂ CH ₂ OEt CH (Ph) C (O) OCH ₂ CF ₃
H CH ₂ SCH ₃ CH (CF ₃ ) C (O) OMe
H CH ₂ CN CH (CF ₃ ) C (O) OEt
H CH ₂ CO ₂ Me CH (CF ₃ ) C (O) OCH ₂ CF ₃
H CH ₂ CO ₂ Et CH ₂ CH ₂ C (O) OMe
H CH ₂ CH = CH ₂ CH ₂ CH ₂ C (O) OEt
H CH ₂ CH≡CH CH ₂ CH ₂ C (O) OCH ₂ CF ₃
HC (O) CH ₃ CH ₂ CH (Me) C (O) OMe
HC (O) Et CH ₂ CH (Me) C (O) OEt
HC (O) Pr-n CH (Me) CH ₂ C (O) OMe
HC (O) Pr-c CH (Me) CH ₂ C (O) OEt
HC (O) Bu-t CH ₂ C (O) NH ₂
HC (O) CH ₂ OCH CH ₂ C (O) NHMe
HC (O) CH ₂ SCH CH ₂ C (O) NHEt
HC (O) OMe CH ₂ C (O) NHPr-n
HC (O) OEt CH ₂ C (O) NHPr-i
HC (O) CH ₂ CH ₂ C CH ₂ C (O) NHPr-c
HC (O) CH ₂ CH ₂ O CH ₂ C (O) NHBu-n
HC (O) OCH ₂ CH CH ₂ C (O) NHBu-i
HC (O) SCH ₃ CH ₂ C (O) NHBu-s
HC (S) OCH ₃ CH ₂ C (O) NHBu-t
HC (S) SCH ₃ CH ₂ C (O) NHBu-c
H SMe CH ₂ C (O) NHHex-n
H SPh CH ₂ C (O) NHHex-c
H SNEt ₂ CH ₂ C (O) N (Me) ₂
H SO ₂ Me CH ₂ C (O) N (Et) ₂
H SO ₂ Et CH ₂ C (O) N (n-Pr) ₂
H SO ₂ Ph CH ₂ C (O) N (Me) Et
H SO ₂ NMe ₂ CH ₂ C (O) N (Me) Pr-n
H NH ₂ CH ₂ C (O) N (Me) Pr-i
H NHMe CH ₂ C (O) NHCH ₂ CH ₂ F
H NHCHO CH ₂ C (O) NHCH ₂ CH ₂ Cl
H NHC (O) CH ₃ CH ₂ C (O) NHCH ₂ CH ₂ Br
H NHC (O) OCH ₃ CH ₂ C (O) N (Me) CH ₂ CH ₂ F
HN = C (CH ₃ ) ₂ CH ₂ C (O) N (Me) CH ₂ CH ₂ Cl
HN = CHPh CH ₂ C (O) N (Me) CH ₂ CH ₂ Br
Me H CH ₂ C (O) NHCH ₂ CF ₃
Et H CH ₂ C (O) N (Me) CH ₂ CF ₃
n-Pr H CH ₂ C (O) NHCH ₂ CF ₂ Cl
i-Pr H CH ₂ C (O) NHCH ₂ CN
CH ₂ OCH ₃ H CH ₂ C (O) NHCH ₂ CH = CH ₂
CH ₂ CH ₂ OEt H CH ₂ C (O) NHCH ₂ CH≡CH
CH ₂ SCH ₃ H CH ₂ C (O) NHCH ₂ CH ₂ CH ₂ Cl
CH ₂ CN H CH ₂ C (O) NHCH ₂ CH ₂ OCH ₃
CH ₂ CO ₂ Me H CH ₂ C (O) NHCH ₂ CH ₂ SCH ₃
CH ₂ CO ₂ Et H CH ₂ C (O) NHCH ₂ CH ₂ SO ₂ CH ₃
CH ₂ CH = CH ₂ H CH (Me) C (O) NH ₂
CH ₂ CH≡CH H CH (Me) C (O) NHMe
C (O) CH ₃ H CH (Me) C (O) NHEt
C (O) Et H CH (Me) C (O) NHPr-n
C (O) Pr-n H CH (Me) C (O) NHPr-i
C (O) Pr-c H CH (Me) C (O) NHPr-c
C (O) Bu-t H CH (Me) C (O) NHBu-n
HH CH (Me) C (O) NHBu-i
HH CH (Me) C (O) NHBu-s
C (O) OMe H CH (Me) C (O) NHBu-t
C (O) OEt H CH (Me) C (O) NHBu-c
HH CH (Me) C (O) NHHex-n
HH CH (Me) C (O) NHHex-c
HH CH (Me) C (O) N (Me) ₂
C (O) SCH ₃ H CH (Me) C (O) N (Et) ₂
C (S) OCH ₃ H CH (Me) C (O) N (n-Pr) ₂
C (S) SCH ₃ H CH (Me) C (O) N (Me) Et
SMe H CH (Me) C (O) N (Me) Pr-n
SPh H CH (Me) C (O) N (Me) Pr-i
SNEt ₂ H CH (Me)) NHCH ₂ CH ₂ F
SO ₂ Me H CH (Me) C (O) NHCH ₂ CH ₂ Cl
SO ₂ Et H CH (Me) C (O) NHCH ₂ CH ₂ Br
SO ₂ Ph H CH (Me) C (O) NHCH ₂ CF ₃
SO ₂ NMe ₂ H CH (Et) C (O) NHCH ₂ CF ₃
NH ₂ H CH (i-Pr) C (O) NHCH ₂ CF ₃
NHMe H CH (CH ₂ OCH ₃ ) C (O) NHCH ₂ CF ₃
NHCHO H CH (CH ₂ SCH ₃ ) C (O) NHCH ₂ CF ₃
NHC (O) CH ₃ H CH (Ph) C (O) NHCH ₂ CF ₃
HH CH (CH ₂ Ph) C (O) NHCH ₂ CF ₃
N = C (CH ₃ ) ₂ H CH (CF ₃ ) C (O) NHMe
N = CHPh H CH (CF ₃ ) C (O) NHEt
HH CH (CF ₃ ) C (O) NHPr-n
HH CH (CF ₃ ) C (O) NHPr-i
HH CH (CF ₃ ) C (O) NHPr-c
HH CH (CF ₃ ) C (O) NHBu-n
HH CH (CF ₃ ) C (O) NHBu-i
HH CH (CF ₃ ) C (O) NHBu-s
HH CH (CF ₃ ) C (O) NHBu-t
HH CH (CF ₃ ) C (O) NHBu-c
HH CH (CF ₃ ) C (O) NHHex-n
HH CH (CF ₃ ) C (O) NHHex-c
HH CH (CF ₃ ) C (O) N (Me) ₂
HH CH (CF ₃ ) C (O) N (Et) ₂
HH CH (CF ₃ ) C (O) N (n-Pr) ₂
HH CH (CF ₃ ) C (O) N (Me) Et
HH CH (CF ₃ ) C (O) N (Me) Pr-n
HH CH (CF ₃ ) C (O) N (Me) Pr-i
HH CH (CF ₃ ) C (O) NHCH ₂ CH ₂ F
HH CH (CF ₃ ) C (O) NHCH ₂ CH ₂ Cl
HH CH (CF ₃ ) C (O) NHCH ₂ CH ₂ Br
HH CH (CF ₃ ) C (O) NHCH ₂ CF ₃
HH CH ₂ CH ₂ C (O) NHCH ₂ CF ₃
HH CH ₂ C (O) N (Me) ₂
HH CH ₂ C (O) N (Et) ₂
HH CH ₂ C (O) N (n-Pr) ₂
HH CH ₂ CH = CH ₂
HH CH ₂ C (Me) = CH ₂
HH CH ₂ C (Et) = CH ₂
HH CH (Me) CH = CH ₂
HH CH ₂ CH = C (Me) ₂
HH CH ₂ C (Me) = CHCH ₃
HH CH (Me) CH = CHCH ₃
HH CH ₂ C (F) = CH ₂
HH CH ₂ CH = CHCl
HH CH ₂ C (Cl) = CH ₂
HH CH ₂ CH = CCl ₂
HH CH ₂ CH = CHBr
HH CH ₂ C (Br) = CH ₂
HH CH ₂ C (Br) = CHBr
HH CH ₂ C (Me) = CHBr
HH CH ₂ CH = C (Cl) CH ₃
HH CH ₂ CH = C (Br) CH ₃
HH CH ₂ C (OMe) = CH ₂
HH CH ₂ C (Br) = CHOMe
HH CH ₂ C (Br) = CHOEt
HH CH ₂ C (Br) = CHPh
HH CH ₂ C≡CH
HH CH ₂ C≡CCl
HH CH ₂ C≡CBr
HH CH ₂ C≡CI
HH CH ₂ C≡CPh
HH CH ₂ OMe
HH CH ₂ CH ₂ OH
HH CH ₂ CH ₂ OMe
HH CH ₂ CH ₂ OEt
HH CH ₂ CH ₂ OPr-n
HH CH ₂ CH ₂ OPr-i
HH CH ₂ CH ₂ OBu-i
HH CH ₂ CH ₂ OCH ₂ CH ₂ Cl
HH CH ₂ CH ₂ OCH ₂ CF ₃
HH CH ₂ CH ₂ OCH ₂ CH ₂ OCH ₃
HH CH ₂ CH ₂ OCH ₂ CH ₂ SCH ₃
HH CH ₂ CH ₂ OC (O) CH ₃
HH CH ₂ CH (Me) OH
HH CH ₂ CH (Me) OMe
HH CH ₂ CH (Me) OCH ₂ CF ₃
HH CH (Me) CH ₂ OH
HH CH (Me) CH ₂ OMe
HH CH (Me) CH ₂ OCH ₂ CF ₃
HH CH (Ph) CH ₂ OH
HH CH (Ph) CH ₂ OMe
HH CH (Ph) CH ₂ OCH ₂ CF ₃
HHC (Me) ₂ CH ₂ OH
HHC (Me) ₂ CH ₂ OMe
HHC (Me) ₂ CH ₂ OCH ₂ CF ₃
HH CH ₂ CH ₂ CH ₂ OH
HH CH ₂ CH ₂ CH ₂ OMe
HH CH ₂ CH ₂ CH ₂ OCH ₂ CF ₃
HH CH ₂ CH ₂ CH ₂ CH ₂ OH
HH CH ₂ CH ₂ CH ₂ CH ₂ OMe
HH CH ₂ CH ₂ CH ₂ CH ₂ OCH ₂ CF ₃
HH CH ₂ SMe
HH CH (CF ₃ ) SMe
HH CH (CF ₃ ) SEt
HH CH ₂ CH ₂ SMe
HH CH ₂ CH ₂ S (O) Me
HH CH ₂ CH ₂ S (O) ₂ Me
HH CH ₂ CH ₂ SEt
HH CH ₂ CH ₂ S (O) Et
HH CH ₂ CH ₂ S (O) ₂ Et
HH CH ₂ CH ₂ SPr-n
HH CH ₂ CH ₂ S (O) Pr-n
HH CH ₂ CH ₂ S (O) ₂ Pr-n
HH CH ₂ CH ₂ SPr-i
HH CH ₂ CH ₂ S (O) Pr-i
HH CH ₂ CH ₂ S (O) ₂ Pr-i
HH CH ₂ CH ₂ SCH ₂ CF ₃
HH CH ₂ CH ₂ S (O) CH ₂ CF ₃
HH CH ₂ CH ₂ S (O) ₂ CH ₂ CF ₃
HH CH ₂ CH ₂ SCH ₂ CH ₂ OH
HH CH ₂ CH ₂ S (O) CH ₂ CH ₂ OH
HH CH ₂ CH ₂ S (O) ₂ CH ₂ CH ₂ OH
HH CH ₂ CH ₂ SCH ₂ CH ₂ OMe
HH CH ₂ CH ₂ S (O) CH ₂ CH ₂ OMe
HH CH ₂ CH ₂ S (O) ₂ CH ₂ CH ₂ OMe
HH CH ₂ CH ₂ SCH ₂ C (O) OMe
HH CH ₂ CH ₂ S (O) CH ₂ C (O) OMe
HH CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) OMe
HH CH ₂ CH ₂ SCH ₂ C (O) NHMe
HH CH ₂ CH ₂ S (O) CH ₂ C (O) NHMe
HH CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) NHMe
HH CH ₂ CH ₂ SCH ₂ C (O) NMe
HH CH ₂ CH ₂ S (O) CH ₂ C (O) NMe
HH CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) N (Me) ₂
HH CH ₂ CH ₂ SCH ₂ CH = CH ₂
HH CH ₂ CH ₂ SCH ₂ CH≡CH
HH CH ₂ CH ₂ S (O) ₂ NHMe
HH CH ₂ CH ₂ S (O) ₂ N (Me) ₂
HH CH ₂ CH ₂ S (O) ₂ NHEt
HH CH ₂ CH ₂ S (O) ₂ N (Et) ₂
HH CH ₂ CH ₂ S (O) ₂ NHPr-n
HH CH ₂ CH ₂ S (O) ₂ N (Pr-n) ₂
HH CH ₂ CH ₂ S (O) ₂ NHPr-i
HH CH ₂ CH ₂ S (O) ₂ N (Pr-i) ₂
HH CH ₂ CH ₂ S (O) ₂ NHPr-c
HH CH ₂ CH ₂ S (O) ₂ NHBu-t
HH CH ₂ CH ₂ S (O) ₂ NHCH ₂ CF ₃
HH CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH ₂ OMe
HH CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH ₂ SMe
HH CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH = CH ₂
HH CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH≡CH
HH CH ₂ CH ₂ S (O) (= NCN) Me
HH CH ₂ CH (Me) SMe
HH CH ₂ CH (Me) S (O) Me
HH CH ₂ CH (Me) S (O) ₂ Me
HH CH ₂ CH (Me) SEt
HH CH ₂ CH (Me) S (O) Et
HH CH ₂ CH (Me) S (O) ₂ Et
HH CH ₂ CH (Et) SMe
HH CH ₂ CH (Et) S (O) Me
HH CH ₂ CH (Et) S (O) ₂ Me
HH CH ₂ CH (n-Pr) SMe
HH CH ₂ CH (n-Pr) S (O) Me
HH CH ₂ CH (n-Pr) S (O) ₂ Me
HH CH ₂ CH (i-Pr) SMe
HH CH ₂ CH (i-Pr) S (O) Me
HH CH ₂ CH (i-Pr) S (O) ₂ Me
HH CH ₂ CH (Ph) SMe
HH CH ₂ CH (Ph) S (O) Me
HH CH ₂ CH (Ph) S (O) ₂ Me
HH CH (Me) CH ₂ SMe
HH CH (Me) CH ₂ S (O) Me
HH CH (Me) CH ₂ S (O) ₂ Me
HH CH (Me) CH ₂ SEt
HH CH (Me) CH ₂ S (O) Et
HH CH (Me) CH ₂ S (O) ₂ Et
HH CH (Me) CH ₂ SPr-n
HH CH (Me) CH ₂ S (O) Pr-n
HH CH (Me) CH ₂ S (O) ₂ Pr-n
HH CH (Me) CH ₂ SPr-i
HH CH (Me) CH ₂ S (O) Pr-i
HH CH (Me) CH ₂ S (O) ₂ Pr-i
HH CH (Me) CH ₂ SPh
HH CH (Me) CH ₂ S (O) Ph
HH CH (Me) CH ₂ S (O) ₂ Ph
HH CH (Ph) CH ₂ SMe
HH CH (Ph) CH ₂ S (O) Me
HH CH (Ph) CH ₂ S (O) ₂ Me
HH CH (Me) CH (Me) SMe
HH CH (Me) CH (Me) S (O) Me
HH CH (Me) CH (Me) S (O) ₂ Me
HHC (Me) ₂ CH ₂ SMe
HHC (Me) ₂ CH ₂ S (O) Me
HHC (Me) ₂ CH ₂ S (O) ₂ Me
HH CH ₂ CH ₂ CH ₂ SMe
HH CH ₂ CH ₂ CH ₂ S (O) Me
HH CH ₂ CH ₂ CH ₂ S (O) ₂ Me
HH CH ₂ CH ₂ CH (Me) SMe
HH CH ₂ CH ₂ CH (Me) S (O) Me
HH CH ₂ CH ₂ CH (Me) S (O) ₂ Me
HH CH ₂ CH (Me) CH ₂ SMe
HH CH ₂ CH (Me) CH ₂ S (O) Me
HH CH ₂ CH (Me) CH ₂ S (O) ₂ Me
HH CH (Me) CH ₂ CH ₂ SMe
HH CH (Me) CH ₂ CH ₂ S (O) Me
HH CH (Me) CH ₂ CH ₂ S (O) ₂ Me
HHC (Me) ₂ CH ₂ CH ₂ SMe
HHC (Me) ₂ CH ₂ CH ₂ S (O) Me
HHC (Me) ₂ CH ₂ CH ₂ S (O) ₂ Me
HH CH (Me) (CH ₂ ) ₃ SMe
HH CH (Me) (CH ₂ ) ₃ S (O) Me
HH CH (Me) (CH ₂ ) ₃ S (O) ₂ Me
HH CH (Me) (CH ₂ ) ₄ SMe
HH CH (Me) (CH ₂ ) ₄ S (O) Me
HH CH (Me) (CH ₂ ) ₄ S (O) ₂ Me
HH CH ₂ NHC (O) Me
HH CH ₂ NHC (O) Et
HH CH ₂ NHC (O) Pr-n
HH CH ₂ CH ₂ NHC (O) Me
HH CH ₂ CH ₂ NHC (O) Et
HH CH ₂ CH ₂ NHC (O) Pr-n
HH CH ₂ CH ₂ NHC (O) Pr-i
HH CH ₂ CH ₂ NHC (O) Pr-c
HH CH ₂ CH ₂ NHC (O) Bu-n
HH CH ₂ CH ₂ NHC (O) Bu-i
HH CH ₂ CH ₂ NHC (O) Bu-s
HH CH ₂ CH ₂ NHC (O) Bu-t
HH CH ₂ CH ₂ NHC (O) CF ₃
HH CH ₂ CH ₂ NHC (O) CF ₂ Cl
HH CH ₂ CH ₂ NHC (O) Ph
HH CH ₂ CH ₂ NHC (O) CH ₂ CF ₃
HH CH ₂ CH ₂ NHC (O) CH ₂ SMe
HH CH ₂ CH ₂ NHC (O) CH ₂ S (O) Me
HH CH ₂ CH ₂ NHC (O) CH ₂ S (O) ₂ Me
HH CH ₂ CH ₂ N (Me) C (O) Me
HH CH ₂ CH ₂ N (Me) C (O) Et
HH CH ₂ CH ₂ N (Me) C (O) CF ₃
HH CH ₂ CH ₂ N (Me) C (O) CH ₂ CF ₃
HH CH ₂ CH ₂ N (Me) C (O) CH ₂ SMe
HH CH ₂ CH ₂ N (Me) C (O) CH ₂ S (O) Me
HH CH ₂ CH ₂ N (Me) C (O) CH ₂ S (O) ₂ Me
HH CH ₂ CH ₂ NHC (O) OMe
HH CH ₂ CH ₂ NHC (O) OEt
HH CH ₂ CH ₂ NHC (O) OPr-n
HH CH ₂ CH ₂ NHC (O) OBu-t
HH CH ₂ CH ₂ NHC (O) NHEt
HH CH ₂ CH ₂ NHC (O) NHPr-n
HH CH ₂ CH ₂ NHC (O) NHPr-i
HH CH ₂ CH ₂ NHC (O) NHBu-t
HH CH ₂ CH ₂ NHC (O) N (Me) ₂
HH CH ₂ CH ₂ NHSO ₂ Me
HH CH ₂ CH ₂ NHSO ₂ Et
HH CH ₂ CH ₂ NHSO ₂ CF ₃
HH CH ₂ CH ₂ NHSO ₂ Ph
HH CH ₂ CH ₂ NHSO ₂ N (Me) ₂
HH CH ₂ CH ₂ NHP (S) (OMe) ₂
HH CH ₂ CH ₂ NHP (S) (OEt) ₂
HH CH ₂ CH ₂ N (Me) SO ₂ Me
HH CH ₂ CH ₂ N (Me) SO ₂ CF ₃
HH CH ₂ CH ₂ N (Me) OMe
HH CH ₂ CH (Me) NHC (O) Me
HH CH ₂ CH (Me) NHC (O) CF ₃
HH CH ₂ CH (Me) NHC (O) CH ₂ CF ₃
HH CH ₂ CH (Me) NHC (O) CH ₂ SMe
HH CH (Me) NHC (O) CH ₂ S (O) Me
HH CH (Me) NHC (O) CH ₂ S (O) ₂ Me
HH CH ₂ CH (Me) NHC (O) OMe
HH CH (Me) CH ₂ NHC (O) Me
HH CH (Me) CH ₂ NHC (O) CF ₃
HH CH (Me) CH ₂ NHC (O) CH ₂ CF ₃
HH CH (Me) CH ₂ NHC (O) CH ₂ SMe
HH CH (Me) CH ₂ NHC (O) CH ₂ S (O) Me
HH CH (Me) CH ₂ NHC (O) CH ₂ S (O) ₂ Me
HH CH (Me) CH ₂ NHC (O) OMe
HH CH ₂ CH ₂ CH ₂ NHC (O) Me
HH CH ₂ CH ₂ CH ₂ NHC (O) OMe
HH D2-1a
HH D2-1b
HH D2-2a
HH D2-2b
HH D2-5a
HH D2-5b
HH D2-5c
HH D2-6a
HH D2-6b
HH D2-6c
HH D2-7a
HH D2-8a
HH D2-8b
HH D2-8c
HH D2-9a
HH D2-9b
HH D2-9c
HH D2-10a
HH D2-10b
HH D2-10c
HH D2-11a
HH D2-12a
HH D2-12b
HH D2-12c
HH D2-13a
HH D2-13b
HH D2-14a
HH D2-14b
HH D2-15a
HH D2-15b
HH D2-16a
HH D2-17a
HH D2-18a
HH D2-19a
HH D2-21a
HH D2-21b
HH D2-22a
HH D2-23a
HH D2-23b
HH D2-24a
HH D2-25a
HH D2-27a
HH D2-30a
HH D2-31a
HH D2-32a
HH D2-34a
HH D2-36a
HH D2-37a
HH D2-41a
HH D2-43a
HH D2-45a
HH D2-46a
HH D2-49a
HH D2-51a
HH D2-53a
HH D2-59a
HH D2-61a
HH D2-63a
HH D2-68a
HH D2-75a
HH D2-76a
HH D2-76b
HH D2-77a
HH D2-77b
HH D2-78a
HH D2-78b
HH D2-79a
HH D2-81a
HH D2-82a
HH D2-84a
HH D2-85a
HH D2-87a
HH D2-90a
HH D2-100a
HH D2-100b
HH D2-100c
HH D2-100d
HH D2-100e
HH D2-101a
HH D2-101b
HH D2-101c
HH D2-101d
HH D2-102a
HH D2-102b
HH D2-102c
HH D2-102d
HH D2-102e
HH D2-102f
HH D2-103a
HH D2-108a
HH CH ₂ (D2-1a)
HH CH ₂ (D2-1b)
HH CH ₂ (D2-2a)
HH CH ₂ (D2-2b)
HH CH ₂ (D2-4a)
HH CH ₂ (D2-4b)
HH CH ₂ (D2-5a)
HH CH ₂ (D2-5b)
HH CH ₂ (D2-5c)
HH CH ₂ (D2-6a)
HH CH ₂ (D2-6b)
HH CH ₂ (D2-6c)
HH CH ₂ (D2-7a)
HH CH ₂ (D2-8a)
HH CH ₂ (D2-8b)
HH CH ₂ (D2-8c)
HH CH ₂ (D2-9a)
HH CH ₂ (D2-9b)
HH CH ₂ (D2-9c)
HH CH ₂ (D2-10a)
HH CH ₂ (D2-10b)
HH CH ₂ (D2-10c)
HH CH ₂ (D2-12a)
HH CH ₂ (D2-12b)
HH CH ₂ (D2-12c)
HH CH ₂ (D2-13a)
HH CH ₂ (D2-13b)
HH CH ₂ (D2-14a)
HH CH ₂ (D2-14b)
HH CH ₂ (D2-15a)
HH CH ₂ (D2-15b)
HH CH ₂ (D2-16a)
HH CH ₂ (D2-17a)
HH CH ₂ (D2-18a)
HH CH ₂ (D2-19a)
HH CH ₂ (D2-20a)
HH CH ₂ (D2-21a)
HH CH ₂ (D2-21b)
HH CH ₂ (D2-23a)
HH CH ₂ (D2-23b)
HH CH ₂ (D2-25a)
HH CH ₂ (D2-27a)
HH CH ₂ (D2-30a)
HH CH ₂ (D2-31a)
HH CH ₂ (D2-32a)
HH CH ₂ (D2-33a)
HH CH ₂ (D2-34a)
HH CH ₂ (D2-35a)
HH CH ₂ (D2-35b)
HH CH ₂ (D2-36a)
HH CH ₂ (D2-37a)
HH CH ₂ (D2-38a)
HH CH ₂ (D2-39a)
HH CH ₂ (D2-40a)
HH CH ₂ (D2-41a)
HH CH ₂ (D2-42a)
HH CH ₂ (D2-43a)
HH CH ₂ (D2-45a)
HH CH ₂ (D2-46a)
HH CH ₂ (D2-49a)
HH CH ₂ (D2-51a)
HH CH ₂ (D2-53a)
HH CH ₂ (D2-59a)
HH CH ₂ (D2-61a)
HH CH ₂ (D2-63a)
HH CH ₂ (D2-68a)
HH CH ₂ (D2-75a)
HH CH ₂ (D2-76a)
HH CH ₂ (D2-76b)
HH CH ₂ (D2-77a)
HH CH ₂ (D2-77b)
HH CH ₂ (D2-78a)
HH CH ₂ (D2-78b)
HH CH ₂ (D2-79a)
HH CH ₂ (D2-81a)
HH CH ₂ (D2-82a)
HH CH ₂ (D2-84a)
HH CH ₂ (D2-85a)
HH CH ₂ (D2-87a)
HH CH ₂ (D2-90a)
HH CH ₂ (D2-100a)
HH CH ₂ (D2-100b)
HH CH ₂ (D2-100c)
HH CH ₂ (D2-100d)
HH CH ₂ (D2-100e)
HH CH ₂ (D2-101a)
HH CH ₂ (D2-101b)
HH CH ₂ (D2-101c)
HH CH ₂ (D2-101d)
HH CH ₂ (D2-102a)
HH CH ₂ (D2-102b)
HH CH ₂ (D2-102c)
HH CH ₂ (D2-102d)
HH CH ₂ (D2-102e)
HH CH ₂ (D2-102f)
HH CH ₂ (D2-103a)
HH CH ₂ (D2-108a)
HH CH (Me) (D2-1a)
HH CH (Me) (D2-2a)
HH CH (Me) (D2-5a)
HH CH (Me) (D2-5c)
HH CH (Me) (D2-6c)
HH CH (Me) (D2-8c)
HH CH (Me) (D2-9b)
HH CH (Me) (D2-9c)
HH CH (Me) (D2-10b)
HH CH (Me) (D2-10c)
HH CH (Me) (D2-12b)
HH CH (Me) (D2-12c)
HH CH (Me) (D2-13b)
HH CH (Me) (D2-14a)
HH CH (Me) (D2-14b)
HH CH (Me) (D2-15a)
HH CH (Me) (D2-15b)
HH CH (Me) (D2-16a)
HH CH (Me) (D2-17a)
HH CH (Me) (D2-18a)
HH CH (Me) (D2-23b)
HH CH (Me) (D2-27a)
HH CH (Me) (D2-31a)
HH CH (Me) (D2-32a)
HH CH (Me) (D2-35a)
HH CH (Me) (D2-36a)
HH CH (Me) (D2-37a)
HH CH (Me) (D2-39a)
HH CH (Me) (D2-41a)
HH CH ₂ C (O) NH (D2-1a)
HH CH ₂ C (O) NH (D2-2a)
HH CH ₂ C (O) NH (D2-5a)
HH CH ₂ C (O) NH (D2-5c)
HH CH ₂ C (O) NH (D2-6c)
HH CH ₂ C (O) NH (D2-8c)
HH CH ₂ C (O) NH (D2-9b)
HH CH ₂ C (O) NH (D2-9c)
HH CH ₂ C (O) NH (D2-10b)
HH CH ₂ C (O) NH (D2-10c)
HH CH ₂ C (O) NH (D2-12b)
HH CH ₂ C (O) NH (D2-12c)
HH CH ₂ C (O) NH (D2-13b)
HH CH ₂ C (O) NH (D2-14a)
HH CH ₂ C (O) NH (D2-14b)
HH CH ₂ C (O) NH (D2-15a)
HH CH ₂ C (O) NH (D2-15b)
HH CH ₂ C (O) NH (D2-16a)
HH CH ₂ C (O) NH (D2-17a)
HH CH ₂ C (O) NH (D2-18a)
HH CH ₂ C (O) NH (D2-23b)
HH CH ₂ C (O) NH (D2-27a)
HH CH ₂ C (O) NH (D2-31a)
HH CH ₂ C (O) NH (D2-32a)
HH CH ₂ C (O) NH (D2-35a)
HH CH ₂ C (O) NH (D2-36a)
HH CH ₂ C (O) NH (D2-37a)
HH CH ₂ C (O) NH (D2-39a)
HH CH ₂ C (O) NH (D2-41a)
HH CH ₂ C (O) NH (D2-45a)
HH CH ₂ C (O) NH (D2-46a)
HH CH ₂ C (O) NH (D2-49a)
HH CH ₂ C (O) NH (D2-51a)
HH CH ₂ C (O) NH (D2-53a)
HH CH ₂ C (O) NH (D2-59a)
HH CH ₂ C (O) NH (D2-61a)
HH CH ₂ C (O) NH (D2-63a)
HH CH ₂ C (O) NH (D2-68a)
HH CH ₂ C (O) NH (D2-75a)
HH CH ₂ C (O) NH (D2-76a)
HH CH ₂ C (O) NH (D2-76b)
HH CH ₂ C (O) NH (D2-77a)
HH CH ₂ C (O) NH (D2-77b)
HH CH ₂ C (O) NH (D2-78a)
HH CH ₂ C (O) NH (D2-78b)
HH CH ₂ C (O) NH (D2-79a)
HH CH ₂ C (O) NH (D2-82a)
HH CH ₂ C (O) NH (D2-84a)
HH CH ₂ C (O) NH (D2-85a)
HH CH ₂ C (O) NH (D2-87a)
HH CH ₂ C (O) NH (D2-90a)
HH CH ₂ C (O) NH (D2-100a)
HH CH ₂ C (O) NH (D2-100b)
HH CH ₂ C (O) NH (D2-100c)
HH CH ₂ C (O) NH (D2-100d)
HH CH ₂ C (O) NH (D2-100e)
HH CH ₂ C (O) NH (D2-101a)
HH CH ₂ C (O) NH (D2-101b)
HH CH ₂ C (O) NH (D2-101c)
HH CH ₂ C (O) NH (D2-101d)
HH CH ₂ C (O) NH (D2-108a)
HH CH ₂ C (O) NHCH ₂ (D2-1a)
HH CH ₂ C (O) NHCH ₂ (D2-2a)
HH CH ₂ C (O) NHCH ₂ (D2-5a)
HH CH ₂ C (O) NHCH ₂ (D2-5c)
HH CH ₂ C (O) NHCH ₂ (D2-6c)
HH CH ₂ C (O) NHCH ₂ (D2-8c)
HH CH ₂ C (O) NHCH ₂ (D2-9b)
HH CH ₂ C (O) NHCH ₂ (D2-9c)
HH CH ₂ C (O) NHCH ₂ (D2-10b)
HH CH ₂ C (O) NHCH ₂ (D2-10c)
HH CH ₂ C (O) NHCH ₂ (D2-12b)
HH CH ₂ C (O) NHCH ₂ (D2-12c)
HH CH ₂ C (O) NHCH ₂ (D2-13b)
HH CH ₂ C (O) NHCH ₂ (D2-14a)
HH CH ₂ C (O) NHCH ₂ (D2-14b)
HH CH ₂ C (O) NHCH ₂ (D2-15a)
HH CH ₂ C (O) NHCH ₂ (D2-15b)
HH CH ₂ C (O) NHCH ₂ (D2-16a)
HH CH ₂ C (O) NHCH ₂ (D2-17a)
HH CH ₂ C (O) NHCH ₂ (D2-18a)
HH CH ₂ C (O) NHCH ₂ (D2-23b)
HH CH ₂ C (O) NHCH ₂ (D2-27a)
HH CH ₂ C (O) NHCH ₂ (D2-31a)
HH CH ₂ C (O) NHCH ₂ (D2-32a)
HH CH ₂ C (O) NHCH ₂ (D2-35a)
HH CH ₂ C (O) NHCH ₂ (D2-36a)
HH CH ₂ C (O) NHCH ₂ (D2-37a)
HH CH ₂ C (O) NHCH ₂ (D2-39a)
HH CH ₂ C (O) NHCH ₂ (D2-41a)
HH CH ₂ C (O) NHCH ₂ (D2-45a)
HH CH ₂ C (O) NHCH ₂ (D2-46a)
HH CH ₂ C (O) NHCH ₂ (D2-49a)
HH CH ₂ C (O) NHCH ₂ (D2-51a)
HH CH ₂ C (O) NHCH ₂ (D2-53a)
HH CH ₂ C (O) NHCH ₂ (D2-59a)
HH CH ₂ C (O) NHCH ₂ (D2-61a)
HH CH ₂ C (O) NHCH ₂ (D2-63a)
HH CH ₂ C (O) NHCH ₂ (D2-68a)
HH CH ₂ C (O) NHCH ₂ (D2-75a)
HH CH ₂ C (O) NHCH ₂ (D2-76a)
HH CH ₂ C (O) NHCH ₂ (D2-76b)
HH CH ₂ C (O) NHCH ₂ (D2-77a)
HH CH ₂ C (O) NHCH ₂ (D2-77b)
HH CH ₂ C (O) NHCH ₂ (D2-78a)
HH CH ₂ C (O) NHCH ₂ (D2-78b)
HH CH ₂ C (O) NHCH ₂ (D2-79a)
HH CH ₂ C (O) NHCH ₂ (D2-82a)
HH CH ₂ C (O) NHCH ₂ (D2-84a)
HH CH ₂ C (O) NHCH ₂ (D2-85a)
HH CH ₂ C (O) NHCH ₂ (D2-87a)
HH CH ₂ C (O) NHCH ₂ (D2-90a)
HH CH ₂ C (O) NHCH ₂ (D2-102a)
HH CH ₂ C (O) NHCH ₂ (D2-102b)
HH CH ₂ C (O) NHCH ₂ (D2-102c)
HH CH ₂ C (O) NHCH ₂ (D2-102d)
HH CH ₂ C (O) NHCH ₂ (D2-102e)
HH CH ₂ C (O) NHCH ₂ (D2-102f)
HH CH ₂ C (O) NHCH ₂ (D2-103a)
HH CH ₂ C (O) NHCH ₂ (D2-108a)
HH NH (D2-7a)
HH NH (D2-10c)
HH NH (D2-22a)
HH NH (D2-24a)
HH NH (D2-32a)
HH NC (O) Me (D2-32a)
HH NC (O) OMe (D2-32a)
HH NC (O) Et (D2-32a)
HH NC (O) OEt (D2-32a)
HH NC (O) CH ₂ CF ₃ (D2-32a)
HH NSO ₂ Me (D2-32a)
HH NSO ₂ CF ₃ (D2-32a)
HH NSO ₂ Ph (D2-32a)
HH NH (D2-35a)
HH NH (D2-36a)
HH NH (D2-37a)
HH NH (D2-39a)
HH NH (D2-43a)
HH NH (D2-45a)
HH NH (D2-49a)
HH NH (D2-51a)
HH NH (D2-53a)
HH NH (D2-59a)
HH NH (D2-61a)
HH NH (D2-63a)
HH NH (D2-108a)
HH NH {D2-32b (3-Cl)}
HH NH {D2-32b (4-Cl)}
HH NH {D2-32b (5-Cl)}
HH NH {D2-32b (6-Cl)}
HH NH {D2-32b (4-CF ₃ )}
HH NH {D2-108b (2-Cl)}
HH NH {D2-108b (3-Cl)}
HH NH {D2-108b (4-Cl)}
HH NH {D2-108b (2-Me)}
HH NH {D2-108b (3-Me)}
HH NH {D2-108b (4-Me)}
HH CH ₂ CH ₂ (D2-1a)
HH CH ₂ CH ₂ (D2-1b)
HH CH ₂ CH ₂ (D2-2a)
HH CH ₂ CH ₂ (D2-2b)
HH CH ₂ CH ₂ (D2-5c)
HH CH ₂ CH ₂ (D2-6c)
HH CH ₂ CH ₂ (D2-7a)
HH CH ₂ CH ₂ (D2-8c)
HH CH ₂ CH ₂ (D2-9b)
HH CH ₂ CH ₂ (D2-10b)
HH CH ₂ CH ₂ (D2-10c)
HH CH ₂ CH ₂ (D2-11a)
HH CH ₂ CH ₂ (D2-20a)
HH CH ₂ CH ₂ (D2-22a)
HH CH ₂ CH ₂ (D2-24a)
HH CH ₂ CH ₂ (D2-26a)
HH CH ₂ CH ₂ (D2-28a)
HH CH ₂ CH ₂ (D2-29a)
HH CH ₂ CH ₂ (D2-32a)
HH CH ₂ CH ₂ (D2-36a)
HH CH ₂ CH ₂ (D2-37a)
HH CH ₂ CH ₂ OCH ₂ (D2-1a)
HH CH ₂ CH ₂ OCH ₂ (D2-1b)
HH CH ₂ CH ₂ OCH ₂ (D2-2a)
HH CH ₂ CH ₂ OCH ₂ (D2-2b)
HH CH ₂ CH ₂ OCH ₂ (D2-4a)
HH CH ₂ CH ₂ OCH ₂ (D2-4b)
HH CH ₂ CH ₂ OCH ₂ (D2-5a)
HH CH ₂ CH ₂ OCH ₂ (D2-5b)
HH CH ₂ CH ₂ OCH ₂ (D2-5c)
HH CH ₂ CH ₂ OCH ₂ (D2-6a)
HH CH ₂ CH ₂ OCH ₂ (D2-6b)
HH CH ₂ CH ₂ OCH ₂ (D2-6c)
HH CH ₂ CH ₂ OCH ₂ (D2-7a)
HH CH ₂ CH ₂ OCH ₂ (D2-8a)
HH CH ₂ CH ₂ OCH ₂ (D2-8b)
HH CH ₂ CH ₂ OCH ₂ (D2-8c)
HH CH ₂ CH ₂ OCH ₂ (D2-9a)
HH CH ₂ CH ₂ OCH ₂ (D2-9b)
HH CH ₂ CH ₂ OCH ₂ (D2-9c)
HH CH ₂ CH ₂ OCH ₂ (D2-10a)
HH CH ₂ CH ₂ OCH ₂ (D2-10b)
HH CH ₂ CH ₂ OCH ₂ (D2-10c)
HH CH ₂ CH ₂ OCH ₂ (D2-12a)
HH CH ₂ CH ₂ OCH ₂ (D2-12b)
HH CH ₂ CH ₂ OCH ₂ (D2-12c)
HH CH ₂ CH ₂ OCH ₂ (D2-13a)
HH CH ₂ CH ₂ OCH ₂ (D2-13b)
HH CH ₂ CH ₂ OCH ₂ (D2-14a)
HH CH ₂ CH ₂ OCH ₂ (D2-14b)
HH CH ₂ CH ₂ OCH ₂ (D2-15a)
HH CH ₂ CH ₂ OCH ₂ (D2-15b)
HH CH ₂ CH ₂ OCH ₂ (D2-16a)
HH CH ₂ CH ₂ OCH ₂ (D2-17a)
HH CH ₂ CH ₂ OCH ₂ (D2-18a)
HH CH ₂ CH ₂ OCH ₂ (D2-19a)
HH CH ₂ CH ₂ OCH ₂ (D2-20a)
HH CH ₂ CH ₂ OCH ₂ (D2-21a)
HH CH ₂ CH ₂ OCH ₂ (D2-21b)
HH CH ₂ CH ₂ OCH ₂ (D2-23a)
HH CH ₂ CH ₂ OCH ₂ (D2-23b)
HH CH ₂ CH ₂ OCH ₂ (D2-25a)
HH CH ₂ CH ₂ OCH ₂ (D2-27a)
HH CH ₂ CH ₂ OCH ₂ (D2-30a)
HH CH ₂ CH ₂ OCH ₂ (D2-31a)
HH CH ₂ CH ₂ OCH ₂ (D2-32a)
HH CH ₂ CH ₂ OCH ₂ (D2-33a)
HH CH ₂ CH ₂ OCH ₂ (D2-34a)
HH CH ₂ CH ₂ OCH ₂ (D2-35a)
HH CH ₂ CH ₂ OCH ₂ (D2-35b)
HH CH ₂ CH ₂ OCH ₂ (D2-36a)
HH CH ₂ CH ₂ OCH ₂ (D2-37a)
HH CH ₂ CH ₂ OCH ₂ (D2-38a)
Me H CH ₂ CH ₂ OCH ₂ (D2-39a)
Me H CH ₂ CH ₂ OCH ₂ (D2-40a)
Me H CH ₂ CH ₂ OCH ₂ (D2-41a)
Me H CH ₂ CH ₂ OCH ₂ (D2-42a)
Me H CH ₂ CH ₂ OCH ₂ (D2-43a)
Me H CH ₂ CH ₂ OCH ₂ (D2-45a)
HH CH ₂ CH ₂ OCH ₂ (D2-46a)
HH CH ₂ CH ₂ OCH ₂ (D2-49a)
HH CH ₂ CH ₂ OCH ₂ (D2-51a)
HH CH ₂ CH ₂ OCH ₂ (D2-53a)
HH CH ₂ CH ₂ OCH ₂ (D2-59a)
HH CH ₂ CH ₂ OCH ₂ (D2-61a)
HH CH ₂ CH ₂ OCH ₂ (D2-63a)
HH CH ₂ CH ₂ OCH ₂ (D2-68a)
HH CH ₂ CH ₂ OCH ₂ (D2-75a)
HH CH ₂ CH ₂ OCH ₂ (D2-76a)
HH CH ₂ CH ₂ OCH ₂ (D2-76b)
HH CH ₂ CH ₂ OCH ₂ (D2-77a)
HH CH ₂ CH ₂ OCH ₂ (D2-77b)
HH CH ₂ CH ₂ OCH ₂ (D2-78a)
HH CH ₂ CH ₂ OCH ₂ (D2-78b)
HH CH ₂ CH ₂ OCH ₂ (D2-79a)
HH CH ₂ CH ₂ OCH ₂ (D2-81a)
HH CH ₂ CH ₂ OCH ₂ (D2-82a)
HH CH ₂ CH ₂ OCH ₂ (D2-84a)
HH CH ₂ CH ₂ OCH ₂ (D2-85a)
HH CH ₂ CH ₂ OCH ₂ (D2-87a)
HH CH ₂ CH ₂ OCH ₂ (D2-90a)
HH CH ₂ CH ₂ OCH ₂ (D2-100a)
HH CH ₂ CH ₂ OCH ₂ (D2-100b)
HH CH ₂ CH ₂ OCH ₂ (D2-100c)
HH CH ₂ CH ₂ OCH ₂ (D2-100d)
HH CH ₂ CH ₂ OCH ₂ (D2-100e)
HH CH ₂ CH ₂ OCH ₂ (D2-101a)
HH CH ₂ CH ₂ OCH ₂ (D2-101b)
HH CH ₂ CH ₂ OCH ₂ (D2-101c)
HH CH ₂ CH ₂ OCH ₂ (D2-101d)
HH CH ₂ CH ₂ OCH ₂ (D2-102a)
HH CH ₂ CH ₂ OCH ₂ (D2-102b)
HH CH ₂ CH ₂ OCH ₂ (D2-102c)
HH CH ₂ CH ₂ OCH ₂ (D2-102d)
HH CH ₂ CH ₂ OCH ₂ (D2-102e)
HH CH ₂ CH ₂ OCH ₂ (D2-102f)
HH CH ₂ CH ₂ OCH ₂ (D2-103a)
HH CH ₂ CH ₂ OCH ₂ (D2-108a)
HH CH ₂ CH ₂ SCH ₂ (D2-1a)
HH CH ₂ CH ₂ SCH ₂ (D2-1b)
HH CH ₂ CH ₂ SCH ₂ (D2-2a)
HH CH ₂ CH ₂ SCH ₂ (D2-2b)
HH CH ₂ CH ₂ SCH ₂ (D2-4a)
HH CH ₂ CH ₂ SCH ₂ (D2-4b)
HH CH ₂ CH ₂ SCH ₂ (D2-5a)
HH CH ₂ CH ₂ SCH ₂ (D2-5b)
HH CH ₂ CH ₂ SCH ₂ (D2-5c)
HH CH ₂ CH ₂ SCH ₂ (D2-6a)
HH CH ₂ CH ₂ SCH ₂ (D2-6b)
HH CH ₂ CH ₂ SCH ₂ (D2-6c)
HH CH ₂ CH ₂ SCH ₂ (D2-7a)
HH CH ₂ CH ₂ SCH ₂ (D2-8a)
HH CH ₂ CH ₂ SCH ₂ (D2-8b)
HH CH ₂ CH ₂ SCH ₂ (D2-8c)
HH CH ₂ CH ₂ SCH ₂ (D2-9a)
HH CH ₂ CH ₂ SCH ₂ (D2-9b)
HH CH ₂ CH ₂ SCH ₂ (D2-9c)
HH CH ₂ CH ₂ SCH ₂ (D2-10a)
HH CH ₂ CH ₂ SCH ₂ (D2-10b)
HH CH ₂ CH ₂ SCH ₂ (D2-10c)
HH CH ₂ CH ₂ SCH ₂ (D2-12a)
HH CH ₂ CH ₂ SCH ₂ (D2-12b)
HH CH ₂ CH ₂ SCH ₂ (D2-12c)
HH CH ₂ CH ₂ SCH ₂ (D2-13a)
HH CH ₂ CH ₂ SCH ₂ (D2-13b)
HH CH ₂ CH ₂ OCH ₂ (D2-14a)
HH CH ₂ CH ₂ SCH ₂ (D2-14b)
HH CH ₂ CH ₂ SCH ₂ (D2-15a)
HH CH ₂ CH ₂ SCH ₂ (D2-15b)
HH CH ₂ CH ₂ SCH ₂ (D2-16a)
HH CH ₂ CH ₂ SCH ₂ (D2-17a)
HH CH ₂ CH ₂ SCH ₂ (D2-18a)
HH CH ₂ CH ₂ SCH ₂ (D2-19a)
HH CH ₂ CH ₂ SCH ₂ (D2-20a)
HH CH ₂ CH ₂ SCH ₂ (D2-21a)
HH CH ₂ CH ₂ SCH ₂ (D2-21b)
HH CH ₂ CH ₂ SCH ₂ (D2-23a)
HH CH ₂ CH ₂ SCH ₂ (D2-23b)
HH CH ₂ CH ₂ SCH ₂ (D2-25a)
HH CH ₂ CH ₂ SCH ₂ (D2-27a)
HH CH ₂ CH ₂ SCH ₂ (D2-30a)
HH CH ₂ CH ₂ SCH ₂ (D2-31a)
HH CH ₂ CH ₂ SCH ₂ (D2-32a)
HH CH ₂ CH ₂ SCH ₂ (D2-33a)
HH CH ₂ CH ₂ SCH ₂ (D2-34a)
HH CH ₂ CH ₂ SCH ₂ (D2-35a)
HH CH ₂ CH ₂ SCH ₂ (D2-35b)
HH CH ₂ CH ₂ SCH ₂ (D2-36a)
HH CH ₂ CH ₂ SCH ₂ (D2-37a)
HH CH ₂ CH ₂ SCH ₂ (D2-38a)
HH CH ₂ CH ₂ SCH ₂ (D2-39a)
HH CH ₂ CH ₂ SCH ₂ (D2-40a)
HH CH ₂ CH ₂ SCH ₂ (D2-41a)
HH CH ₂ CH ₂ SCH ₂ (D2-42a)
HH CH ₂ CH ₂ SCH ₂ (D2-43a)
HH CH ₂ CH ₂ SCH ₂ (D2-45a)
HH CH ₂ CH ₂ SCH ₂ (D2-46a)
HH CH ₂ CH ₂ SCH ₂ (D2-49a)
HH CH ₂ CH ₂ SCH ₂ (D2-51a)
HH CH ₂ CH ₂ SCH ₂ (D2-53a)
HH CH ₂ CH ₂ SCH ₂ (D2-59a)
HH CH ₂ CH ₂ SCH ₂ (D2-61a)
HH CH ₂ CH ₂ SCH ₂ (D2-63a)
HH CH ₂ CH ₂ SCH ₂ (D2-68a)
HH CH ₂ CH ₂ SCH ₂ (D2-75a)
HH CH ₂ CH ₂ SCH ₂ (D2-76a)
HH CH ₂ CH ₂ SCH ₂ (D2-76b)
HH CH ₂ CH ₂ SCH ₂ (D2-77a)
HH CH ₂ CH ₂ SCH ₂ (D2-77b)
HH CH ₂ CH ₂ SCH ₂ (D2-78a)
HH CH ₂ CH ₂ SCH ₂ (D2-78b)
HH CH ₂ CH ₂ SCH ₂ (D2-79a)
HH CH ₂ CH ₂ SCH ₂ (D2-81a)
HH CH ₂ CH ₂ SCH ₂ (D2-82a)
HH CH ₂ CH ₂ SCH ₂ (D2-84a)
HH CH ₂ CH ₂ SCH ₂ (D2-85a)
HH CH ₂ CH ₂ SCH ₂ (D2-87a)
HH CH ₂ CH ₂ SCH ₂ (D2-90a)
HH CH ₂ CH ₂ SCH ₂ (D2-100a)
HH CH ₂ CH ₂ SCH ₂ (D2-100b)
HH CH ₂ CH ₂ SCH ₂ (D2-100c)
HH CH ₂ CH ₂ SCH ₂ (D2-100d)
HH CH ₂ CH ₂ SCH ₂ (D2-100e)
HH CH ₂ CH ₂ SCH ₂ (D2-101a)
HH CH ₂ CH ₂ SCH ₂ (D2-101b)
HH CH ₂ CH ₂ SCH ₂ (D2-101c)
HH CH ₂ CH ₂ SCH ₂ (D2-101d)
HH CH ₂ CH ₂ SCH ₂ (D2-102a)
HH CH ₂ CH ₂ SCH ₂ (D2-102b)
HH CH ₂ CH ₂ SCH ₂ (D2-102c)
HH CH ₂ CH ₂ SCH ₂ (D2-102d)
HH CH ₂ CH ₂ SCH ₂ (D2-102e)
HH CH ₂ CH ₂ SCH ₂ (D2-102f)
HH CH ₂ CH ₂ SCH ₂ (D2-103a)
HH CH ₂ CH ₂ SCH ₂ (D2-108a)
HH CH ₂ {D2-1c (3-Me)}
HH CH ₂ {D2-1d (5-Cl)}
HH CH ₂ {D2-2c (5-Br)}
HH CH ₂ {D2-2d (5-Cl)}
HH CH ₂ {D2-4c (5-Cl)}
HH CH ₂ {D2-4d (5-Cl)}
HH CH ₂ {D2-5d (3-Me)}
HH CH ₂ {D2-5e (3-Me)}
HH CH ₂ {D2-5f (5-Me)}
HH CH ₂ {D2-6d (3-Cl)}
HH CH ₂ {D2-6e (3-Me)}
HH CH ₂ {D2-6f (5-Me)}
HH CH ₂ {D2-7a (3-Me)}
HH CH ₂ {D2-8d (3-Cl)}
HH CH ₂ {D2-8e (3-CF ₃ )}
HH CH ₂ {D2-8f (5-Me)}
HH CH ₂ {D2-9d (2-Me)}
HH CH ₂ {D2-9e (2-Me)}
HH CH ₂ {D2-9f (4-Me)}
HH CH ₂ {D2-10e (2-Me)}
HH CH ₂ {D2-10f (2-Cl)}
HH CH ₂ {D2-10e (2-Br)}
HH CH ₂ {D2-12d (4-Me)}
HH CH ₂ {D2-12e (5-Me)}
HH CH ₂ {D2-12f (5-Cl)}
HH CH ₂ {D2-13c (Me)}
HH CH ₂ {D2-13d (Cl)}
HH CH ₂ {D2-14c (Me)}
HH CH ₂ {D2-14d (Me)}
HH CH ₂ {D2-15c (Cl)}
HH CH ₂ {D2-15d (Me)}
HH CH ₂ {D2-16b (Ph)}
HH CH ₂ {D2-17b (Ph)}
HH CH ₂ {D2-18b (Me)}
HH CH ₂ {D2-19b (Cl)}
HH CH ₂ {D2-20b (Me)}
HH CH ₂ {D2-21c (Me)}
HH CH ₂ {D2-21d (Me)}
HH CH ₂ {D2-23c (t-Bu)}
HH CH ₂ {D2-23d (Ph)}
HH CH ₂ {D2-25b (Me)}
HH CH ₂ {D2-27a (Me)}
HH CH ₂ {D2-32b (3-Cl)}
HH CH ₂ {D2-32b (4-Cl)}
HH CH ₂ {D2-32b (5-Cl)}
HH CH ₂ {D2-32b (6-Cl)}
HH CH ₂ {D2-32b (3-Me)}
HH CH ₂ {D2-32b (4-Me)}
HH CH ₂ {D2-32b (5-Me)}
HH CH ₂ {D2-32b (6-Me)}
HH CH ₂ {D2-32b (5-CF ₃ )}
HH CH ₂ {D2-33b (4-CF ₃ )}
HH CH ₂ {D2-34b (3-Cl)}
HH CH ₂ {D2-35c (3-Cl)}
HH CH ₂ {D2-35d (3-Cl)}
HH CH ₂ {D2-36b (2-Me)}
HH CH ₂ {D2-37b (4-Me)}
HH CH ₂ {D2-38b (2-Me)}
HH CH ₂ {D2-39b (5-Me)}
HH CH ₂ {D2-108b (2-Cl)}
HH CH ₂ {D2-108b (3-Cl)}
HH CH ₂ {D2-108b (4-Cl)}
HH CH ₂ {D2-108b (2-Me)}
HH CH ₂ {D2-108b (3-Me)}
HH CH ₂ {D2-108b (4-Me)}
HH CH ₂ {D2-108b (2-CF ₃ )}
HH CH ₂ {D2-108b (3-CF ₃ )}
HH CH ₂ {D2-108b (4-CF ₃ )}
HH CH ₂ {D2-108b (2-OMe)}
HH CH ₂ {D2-108b (3-OMe)}
HH CH ₂ {D2-108b (4-OMe)}
HH CH ₂ CH ₂ {D2-7b (4-Cl)}
HH CH ₂ CH ₂ {D2-10e (2-Cl)}
HH CH ₂ CH ₂ {D2-11b (2-Me)}
HH CH ₂ CH ₂ {D2-20b (4-Me)}
HH CH ₂ CH ₂ {D2-22b (3-SMe)}
HH CH ₂ CH ₂ {D2-24b (3-Me)}
HH CH ₂ CH ₂ {D2-26b (4-CO ₂ Me)}
HH CH ₂ CH ₂ {D2-28b (Me)}
HH CH ₂ CH ₂ {D2-29a (Ph)}
HH CH ₂ CH ₂ {D2-32b (3-Cl)}
HH CH ₂ CH ₂ {D2-36b (2-Me)}
HH CH ₂ CH ₂ (D2-37b (4-Me)
――――――――――――――――――――――――――
[Table 5]

第５表
―――――――――――――――――――
R^f2 R^f3
―――――――――――――――――――
H C(O)Me
H Me
H Et
H Pr-n
H Pr-i
H Pr-c
H Bu-n
H Bu-c
H Bu-i
H Bu-s
H Bu-t
H Pen-n
H Pen-c
H Hex-n
H Hex-c
H CH₂Br
H CH(Br)Me
H CH₂CH₂CH₂Cl
H CH(Br)CH₂CH₂CH₂Br
H CH₂CF₃
H CH₂CH(OH)CF₃
H CH₂CN
H CH₂C(O)OMe
H CH₂C(O)NHMe
H CH=CH₂
H CH=CHSMe
H CH=CHCF₃
H CH=C(Me)CF₃
H CH｛D2-108b(4-CF₃)｝
H C≡CH
H C≡CSiMe₃
H CH₂OMe
H CH₂OEt
H CH(Me)OCH₂CF₃
H CH(Me)ON=CHMe
H CH₂CH₂SC(O)Me
H CH₂OC(O)Me
H CH₂SMe
H CH₂S(O)Me
H CH₂S(O)₂Me
H CH₂SEt
H CH₂S(O)Et
H CH₂S(O)₂Et
H CH₂SCH₂CH=CH₂
H CH₂S(O)CH₂CH=CH₂
H CH₂S(O)₂CH₂CH=CH₂
H CH₂SCH₂CF₃
H CH₂S(O)CH₂CF₃
H CH₂S(O)₂CH₂CF₃
H CH(Me)SMe
H CH(Me)S(O)Me
H CH(Me)S(O)₂Me
H CH(Me)SEt
H CH(Me)S(O)Et
H CH(Me)S(O)₂Et
H CH(Me)S(=NCN)Et
H CH(Me)S(O)(=NCN)Et
H CH(Me)SPr-n
H CH(Me)S(O)Pr-n
H CH(Me)S(O)₂Pr-n
H CH(Me)SPr-i
H CH(Me)S(O)Pr-i
H CH(Me)S(O)₂Pr-i
H CH(Me)SBu-t
H CH(Me)S(O)Bu-t
H CH(Me)S(O)₂Bu-t
H CH(Me)SCH₂Pr-c
H CH(Me)S(O)CH₂Pr-c
H CH(Me)S(O)₂CH₂Pr-c
H CH(Me)SCH₂OMe
H CH(Me)SCH₂SMe
H CH(Me)S(O)CH₂SMe
H CH(Me)S(O)₂CH₂SMe
H CH(Me)SCH₂C≡CH
H CH(Me)S(O)CH₂C≡CH
H CH(Me)S(O)₂CH₂C≡CH
H CH(Me)SCH₂C(O)NHMe
H CH(Me)S(O)CH₂C(O)NHMe
H CH(Me)S(O)₂CH₂C(O)NHMe
H CH(Me)SCH₂C(O)OMe
H CH(Me)S(O)CH₂C(O)OMe
H CH(Me)S(O)₂CH₂C(O)OMe
H CH(Me)SCH₂CH₂CH₂Cl
H CH(Me)S(O)CH₂CH₂CH₂Cl
H CH(Me)S(O)₂CH₂CH₂CH₂Cl
H CH(Me)SCH₂CF₃
H CH(Me)S(O)CH₂CF₃
H CH(Me)S(O)₂CH₂CF₃
H CH(Me)SCH₂(D2-34a)
H CH(Me)S(O)CH₂(D2-34a)
H CH(Me)S(O)₂CH₂(D2-34a)
H CH(CH₃)SCH₂Si(CH₃)₃
H CH(Me)SCN
H CH(Me)SCH₂CN
H CH(Me)SC(O)Me
H CH(Me)S(D2-37a)
H CH(Et)SMe
H CH(Et)S(O)Me
H CH(Et)S(O)₂Me
H CH(Et)SEt
H CH(Et)S(O)Et
H CH(Et)S(O)₂Et
H CH(F)SMe
H CH(F)S(O)Me
H CH(F)S(O)₂Me
H CH(F)SEt
H CH(F)S(O)Et
H CH(F)S(O)₂Et
H CH{OC(O)Me}SMe
H CH{OC(O)Me}S(O)Me
H CH{OC(O)Me}S(O)₂Me
H CH(SMe)₂
H C(Me)₂SMe
H C(Me)₂S(O)Me
H C(Me)₂S(O)₂Me
H CH₂CH₂SH
H CH₂CH₂SMe
H CH₂CH₂S(O)Me
H CH₂CH₂S(O)₂Me
H CH₂CH₂SEt
H CH₂CH₂S(O)Et
H CH₂CH₂S(O)₂Et
H CH₂CH₂SPr-n
H CH₂CH₂S(O)Pr-n
H CH₂CH₂S(O)₂Pr-n
H CH₂CH₂SPr-i
H CH₂CH₂S(O)Pr-i
H CH₂CH₂S(O)₂Pr-i
H CH₂CH₂SCH₂CF₃
H CH₂CH₂S(O)CH₂CF₃
H CH₂CH₂S(O)₂CH₂CF₃
H CH₂CH₂SC(O)Me
H CH(Me)CH₂SMe
H CH(Me)CH₂S(O)Me
H CH(Me)CH₂S(O)₂Me
H CH(Me)CH₂SEt
H CH(Me)CH₂S(O)Et
H CH(Me)CH₂S(O)₂Et
H CH(Me)CH₂SPr-n
H CH(Me)CH₂S(O)Pr-n
H CH(Me)CH₂S(O)₂Pr-n
H CH(Me)CH₂SPr-i
H CH(Me)CH₂S(O)Pr-i
H CH(Me)CH₂S(O)₂Pr-i
H CH(Me)CH₂SCH₂CF₃
H CH(Me)CH₂S(O)CH₂CF₃
H CH(Me)CH₂S(O)₂CH₂CF₃
H CH(Me)CH₂SC(O)Me
H CH(Et)CH₂SMe
H CH(Et)CH₂S(O)Me
H CH(Et)CH₂S(O)₂Me
H CH(OMe)CH₂SMe
H CH(OMe)CH₂S(O)Me
H CH(OMe)CH₂S(O)₂Me
H CH(SMe)CH₂SMe
H CH(SMe)CH₂S(O)Me
H CH(SMe)CH₂S(O)₂Me
H CH(CH₂SMe)CH₂SMe
H CH(CH₂SMe)CH₂S(O)Me
H CH(CH₂SMe)CH₂S(O)₂Me
H CH(Cl)CH₂SMe
H CH(Cl)CH₂S(O)Me
H CH(Cl)CH₂S(O)₂Me
H CH(CN)CH₂SMe
H CH(CN)CH₂S(O)Me
H CH(CN)CH₂S(O)₂Me
H CH(CN)CH₂SEt
H CH(CN)CH₂S(O)Et
H CH(CN)CH₂S(O)₂Et
H CH{C(O)OMe}CH₂SMe
H CH{C(O)OMe}CH₂S(O)Me
H CH{C(O)OMe}CH₂S(O)₂Me
H CH{C(O)OMe}CH₂SEt
H CH{C(O)OMe}CH₂S(O)Et
H CH{C(O)OMe}CH₂S(O)₂Et
H CH(Ph)CH₂SMe
H CH(Ph)CH₂S(O)Me
H CH(Ph)CH₂S(O)₂Me
H C(Me)₂CH₂SMe
H C(Me)₂CH₂S(O)Me
H C(Me)₂CH₂S(O)₂Me
H C(=CH₂)CH₂SMe
H C(=CH₂)CH₂S(O)Me
H C(=CH₂)CH₂S(O)₂Me
H C(=CH₂)CH₂SEt
H C(=CH₂)CH₂S(O)Et
H C(=CH₂)CH₂S(O)₂Et
H CH₂CH₂CH₂SEt
H CH₂CH₂CH₂S(O)Et
H CH₂CH₂CH₂S(O)₂Et
H CH(Me)CH₂CH₂SEt
H CH(Me)CH₂CH₂S(O)Et
H CH(Me)CH₂CH₂S(O)₂Et
H CH₂CH(Me)CH₂SEt
H CH₂CH(Me)CH₂S(O)Et
H CH₂CH(Me)CH₂S(O)₂Et
H CH₂CH₂CH(Me)SEt
H CH₂CH₂CH(Me)S(O)Et
H CH₂CH₂CH(Me)S(O)₂Et
H CH₂CH₂CH₂SPr-n
H CH₂CH₂CH₂S(O)Pr-n
H CH₂CH₂CH₂S(O)₂Pr-n
H CH(Me)CH₂CH₂SPr-n
H CH(Me)CH₂CH₂S(O)Pr-n
H CH(Me)CH₂CH₂S(O)₂Pr-n
H CH₂CH(Me)CH₂SPr-n
H CH₂CH(Me)CH₂S(O)Pr-n
H CH₂CH(Me)CH₂S(O)₂Pr-n
H CH₂CH₂CH₂CH₂SMe
H CH₂CH₂CH₂CH₂S(O)Me
H CH₂CH₂CH₂CH₂S(O)₂Me
H CH₂CH₂CH₂CH₂SEt
H CH₂CH₂CH₂CH₂S(O)Et
H CH₂CH₂CH₂CH₂S(O)₂Et
H CH₂CH₂CH₂CH₂SPr-n
H CH₂CH₂CH₂CH₂S(O)Pr-n
H CH₂CH₂CH₂CH₂S(O)₂Pr-n
H CH₂CH(Me)SMe
H CH₂OCH₂SMe
H CH₂CH(SMe)₂
H C(=CH₂)CH₂C(O)OH
H C(=NOMe)CH₃
H C(=NOMe)Et
H C(=NOMe)Pr-n
H C(=NOEt)CH₃
H C(=NOPr-n)CH₃
H C(=NOPr-i)CH₃
H C(=NOBu-n)CH₃
H C(=NOCH₂Ph)CH₃
H C(=NOMe)CH₂OCH₂CF₃
H C(=NOMe)CH₂SMe
H C(=NOMe)CH₂S(O)Me
H C(=NOMe)CH₂S(O)₂Me
H C(=NOMe)CH₂SEt
H C(=NOMe)CH₂S(O)Et
H C(=NOMe)CH₂S(O)₂Et
H C(=NOMe)CH₂SCF₃
H C(=NOMe)CH₂S(O)CF₃
H C(=NOMe)CH₂S(O)₂CF₃
H C(=NOMe)CH₂SCH₂CF₃
H C(=NOMe)CH₂S(O)CH₂CF₃
H C(=NOMe)CH₂S(O)₂CH₂CF₃
H C(=NOEt)CH₂SMe
H C(=NOEt)CH₂S(O)Me
H C(=NOEt)CH₂S(O)₂Me
H C(=NOPr-n)CH₂SMe
H C(=NOPr-n)CH₂S(O)Me
H C(=NOPr-n)CH₂S(O)₂Me
H C(=NOPr-i)CH₂SMe
H C(=NOPr-i)CH₂S(O)Me
H C(=NOPr-i)CH₂S(O)₂Me
H C(=NOBu-n)CH₂SMe
H C(=NOBu-n)CH₂S(O)Me
H C(=NOBu-n)CH₂S(O)₂Me
H C(=NOCH₂Ph)CH₂SMe
H C(=NOCH₂Ph)CH₂S(O)Me
H C(=NOCH₂Ph)CH₂S(O)₂Me
H C(=NOCH₂CH=CH₂)CH₂SMe
H C(=NOCH₂OMe)CH₂SMe
H C(=NOCH₂CH₂OMe)CH₂SMe
H C{=NOCH₂CH₂Si(Me)₃}CH₂SMe
H CH₂CH(=NOMe)
H CH₂C(=NOMe)Me
H CH₂C(=NOMe)Et
H CH₂C(=NOMe)Pr-n
H CH₂C(=NOMe)Pr-i
H CH₂C(=NOMe)Bu-n
H CH₂C(=NOMe)Bu-i
H CH₂C(=NOMe)Bu-s
H CH₂C(=NOMe)Bu-t
H CH₂C(=NOMe)CF₃
H CH₂C(=NOCH₃)CH₂SCH₃
H CH(SMe)C(=NOMe)Me
H CH{S(O)Me}C(=NOMe)Me
H CH{S(O)₂Me}C(=NOMe)Me
H CH(SEt)C(=NOMe)Me
H CH{S(O)Et}C(=NOMe)Me
H CH{S(O)₂Et}C(=NOMe)Me
H CH₂NH₂
H CH₂NHC(O)Me
H CH₂NHC(O)OMe
H CH₂NHC(O)OBu-t
H CH₂NHSO₂Me
H CH₂N(Me)C(O)Me
H CH₂N(Me)C(O)OMe
H CH₂N(Me)C(O)OBu-t
H CH₂N(Me)SO₂Me
H CH(CH₂SMe)NH₂
H CH(CH₂SMe)NHC(O)Me
H CH(CH₂SMe)NHC(O)OMe
H CH(CH₂SMe)NHC(O)OBu-t
H CH(CH₂SMe)NHSO₂Me
H CH₂P(O)(OMe)₂
H CH₂P(O)(OEt)₂
H OBu-t
H O{D2-108b(4-NO₂)}
H SMe
H NH₂
H NHCH₂CH₂SMe
H N(Me)CH₂CH₂SMe
H NHCH₂CH₂CH₂SMe
H NHMe
H NHEt
H NPr-n
H NHCH(Me)₂
H NHCH₂C=CH₂
H NHCH₂C(O)OMe
H NHCH₂CF₃
H N(Me)CH₂CF₃
H NHC(O)OEt
H NHC(O)CCl₃
H NHC(O)CH₂SMe
H N(CH₂CH₃)C(O)CH₂SCH₃
H NHS(O)₂(D2-108a)
H NHCH=NOMe
H N=CHNMe₂
H NHPh
H NH(D2-1a)
H NH(D2-2a)
H NH(D2-2b)
H NH(D2-4a)
H NH(D2-5a)
H NH(D2-5b)
H NH(D2-5c)
H NH(D2-6a)
H NH(D2-6b)
H NH(D2-6c)
H NH(D2-7a)
H NH(D2-8a)
H NH(D2-8b)
H NH(D2-8c)
H NH(D2-9a)
H NH(D2-9b)
H NH(D2-9c)
H NH(D2-10a)
H NH(D2-10b)
H NH(D2-10c)
H NH(D2-11a)
H NH(D2-12a)
H NH(D2-12b)
H NH(D2-12c)
H NH(D2-13a)
H NH(D2-13b)
H NH(D2-14a)
H NH(D2-14b)
H NH(D2-15a)
H NH(D2-15b)
H NH(D2-16a)
H NH(D2-17a)
H NH(D2-18a)
H NH(D2-19a)
H NH(D2-20a)
H NH(D2-21a)
H NH(D2-21b)
H NH(D2-22a)
H NH(D2-23a)
H NH(D2-23b)
H NH(D2-24a)
H NH(D2-25a)
H NH(D2-26a)
H NH(D2-27a)
H NH(D2-28a)
H NH(D2-29a)
H NH(D2-30a)
H NH(D2-31a)
H NH(D2-32a)
H NH(D2-33a)
H NH(D2-34a)
H NH(D2-35a)
H NH(D2-35b)
H NH(D2-36a)
H NH(D2-37a)
H NH(D2-38a)
H NH(D2-39a)
H NH(D2-40a)
H NH(D2-40b)
H NH(D2-40c)
H NH(D2-41a)
H NH(D2-42a)
H NH(D2-43a)
H NH(D2-45a)
H NH(D2-50a)
H NH(D2-51a)
H NH(D2-59a)
H NH(D2-61a)
H NH(D2-79a)
H NH(D2-80a)
H NH{D2-108b(2-Cl)}
H NH{D2-108b(3-Cl)}
H NH{D2-108b(4-Cl)}
H NH{D2-108b(2-Me)}
H NH{D2-108b(3-Me)}
H NH{D2-108b(4-Me)}
H N(Me)Ph
H N(Me)(D2-1a)
H N(Me)(D2-2a)
H N(Me)(D2-2b)
H N(Me)(D2-4a)
H N(Me){D2-4b(Me)}
H N(Me)(D2-5a)
H N(Me)(D2-5b)
H N(Me)(D2-5c)
H N(Me)(D2-6a)
H N(Me)(D2-6b)
H N(Me)(D2-6c)
H N(Me)(D2-7a)
H N(Me)(D2-8a)
H N(Me)(D2-8b)
H N(Me)(D2-8c)
H N(Me)(D2-9a)
H N(Me)(D2-9b)
H N(Me)(D2-9c)
H N(Me)(D2-10a)
H N(Me)(D2-10b)
H N(Me)(D2-10c)
H N(Me)(D2-11a)
H N(Me)(D2-12a)
H N(Me)(D2-12b)
H N(Me)(D2-12c)
H N(Me)(D2-13a)
H N(Me)(D2-13b)
H N(Me)(D2-14a)
H N(Me)(D2-14b)
H N(Me)(D2-15a)
H N(Me)(D2-15b)
H N(Me)(D2-16a)
H N(Me)(D2-17a)
H N(Me)(D2-18a)
H N(Me)(D2-19a)
H N(Me)(D2-20a)
H N(Me)(D2-21a)
H N(Me)(D2-21b)
H N(Me)(D2-22a)
H N(Me)(D2-23a)
H N(Me)(D2-23b)
H N(Me)(D2-24a)
H N(Me)(D2-25a)
H N(Me)(D2-26a)
H N(Me)(D2-27a)
H N(Me)(D2-28a)
H N(Me)(D2-29a)
H N(Me)(D2-30a)
H N(Me)(D2-31a)
H N(Me)(D2-32a)
H N(Me)(D2-33a)
H N(Me)(D2-34a)
H N(Me)(D2-35a)
H N(Me)(D2-35b)
H N(Me)(D2-36a)
H N(Me)(D2-37a)
H N(Me)(D2-38a)
H N(Me)(D2-39a)
H N(Me)(D2-40a)
H N(Me)(D2-40b)
H N(Me)(D2-40c)
H N(Me)(D2-41a)
H N(Me)(D2-42a)
H N(Me)(D2-43a)
H N(Me)(D2-45a)
H N(Me)(D2-50a)
H N(Me)(D2-51a)
H N(Me)(D2-59a)
H N(Me)(D2-61a)
H N(Me)(D2-79a)
H N(Me)(D2-80a)
H N(Me){D2-108b(2-Cl)}
H N(Me){D2-108b(3-Cl)}
H N(Me){D2-108b(4-Cl)}
H N(Me){D2-108b(2-Me)}
H N(Me){D2-108b(3-Me)}
H N(Me){D2-108b(4-Me)}
H D2-8c(CH₂CF₃)
H D2-1b(5-Br)
H D2-2c(5-SMe)
H D2-2c{5-C(O)Me}
H D2-4a(Me)
H D2-5d｛5-（Pr-c）｝
H D2-5e(3,5-Me₂)
H D2-6d(4,5-Cl₂)
H D2-9b
H D2-10e(2-CF₃)
H D2-12f(4-NO₂)
H D2-13d(Me)
H D2-19a
H D2-32b(2-Br)
H D2-33b(2-OMe)
H D2-34a
H D2-35b
H D2-38b(4-SMe)
H D2-39b(5-Me)
H D2-82a
H D2-82b
H D2-87a
H D2-103b
H D2-103c
H D2-103d
H D2-103e
H CH₂(D2-2a)
H CH₂{D2-5f(3-Me)}
H CH₂(D2-28a)
H CH₂(D2-32a)
H CH₂(D2-33a)
H CH₂(D2-34a)
H CH₂{D2-33b(6-Cl)}
H CH₂(D2-34a)
Me C(O)Me
Me Me
Me Et
Me Pr-n
Me Pr-i
Me Pr-c
Me Bu-n
Me Bu-i
Me Bu-c
Me Bu-s
Me Bu-t
Me Pen-n
Me Pen-c
Me Hex-n
Me Hex-c
Me CH=CH₂
Me C≡CH
Me C≡CSiMe₃
Me CH₂Br
Me CH₂Br
Me CH(Br)Me
Me CH₂CF₃
Me CH₂CH(OH)CF₃
Me CH₂CN
Me CH(Me)CN
Me CH₂CH₂CN
Me CH(Me)CH₂CN
Me CH₂CH₂CH₂CN
Me CH(Me)CH₂CH₂CN
Me CH₂CH₂CH₂CH₂CN
Me CH(Me)CH₂CH₂CH₂CN
Me CH₂C(O)OMe
Me CH(Me)C(O)OMe
Me CH₂CH₂C(O)OMe
Me CH(Me)CH₂C(O)OMe
Me CH₂CH₂CH₂C(O)OMe
Me CH(Me)CH₂CH₂C(O)OMe
Me CH₂CH₂CH₂CH₂C(O)OMe
Me CH₂C(O)OEt
Me CH(Me)C(O)OEt
Me CH₂CH₂C(O)OEt
Me CH(Me)CH₂C(O)OEt
Me CH₂CH₂CH₂C(O)OEt
Me CH(Me)CH₂CH₂C(O)OEt
Me CH₂CH₂CH₂CH₂C(O)OEt
Me CH₂C(O)NHMe
Me CH₂OMe
Me CH₂OEt
Me CH₂OPr-n
Me CH₂OPr-i
Me CH₂OPr-c
Me CH₂OBu-n
Me CH₂OBu-i
Me CH₂OBu-s
Me CH₂OBu-t
Me CH₂OBu-c
Me CH₂OPen-n
Me CH₂OPen-c
Me CH₂OHex-n
Me CH₂OHex-c
Me CH₂OCH₂Pr-c
Me CH₂OCH₂CH=CH₂
Me CH₂OCH₂C≡CH
Me CH₂OCH₂OMe
Me CH₂OCH₂SMe
Me CH₂OCH₂Si(CH₃)₃
Me CH₂OCH₂(D2-34a)
Me CH₂OCF₃
Me CH₂OCF₂H
Me CH₂OCF₂Cl
Me CH₂OCF₂Br
Me CH₂OCH₂CF₃
Me CH₂OCH₂CF₂CF₃
Me CH₂OCH₂CN
Me CH₂OC(O)Me
Me CH₂OCH₂C(O)OMe
Me CH₂OCH₂C(O)OEt
Me CH₂ON=CHMe
Me CH₂ON=C(Me)₂
Me CH(Me)OMe
Me CH(Me)OEt
Me CH(Me)OPr-n
Me CH(Me)OPr-i
Me CH(Me)OPr-c
Me CH(Me)OBu-n
Me CH(Me)OBu-i
Me CH(Me)OBu-s
Me CH(Me)OBu-t
Me CH(Me)OBu-c
Me CH(Me)OPen-n
Me CH(Me)OPen-c
Me CH(Me)OHex-n
Me CH(Me)OHex-c
Me CH(Me)OCH₂Pr-c
Me CH(Me)OCH₂CH=CH₂
Me CH(Me)OCH₂C≡CH
Me CH(Me)OCH₂OMe
Me CH(Me)OCH₂SMe
Me CH(Me)OCH₂Si(CH₃)₃
Me CH(Me)OCH₂(D2-34a)
Me CH(Me)OCF₃
Me CH(Me)OCF₂H
Me CH(Me)OCF₂Cl
Me CH(Me)OCF₂Br
Me CH(Me)OCH₂CF₃
Me CH(Me)OCH₂CF₂CF₃
Me CH(Me)OCH₂CN
Me CH(Me)OC(O)Me
Me CH(Me)OCH₂C(O)OMe
Me CH(Me)OCH₂C(O)OEt
Me CH(Me)ON=CHMe
Me CH(Me)ON=C(Me)₂
Me CH₂SMe
Me CH₂S(O)Me
Me CH₂S(O)₂Me
Me CH₂SEt
Me CH₂S(O)Et
Me CH₂S(O)₂Et
Me CH₂SCH₂CH=CH₂
Me CH₂S(O)CH₂CH=CH₂
Me CH₂S(O)₂CH₂CH=CH₂
Me CH₂SCH₂CF₃
Me CH₂S(O)CH₂CF₃
Me CH₂S(O)₂CH₂CF₃
Me CH(Me)SMe
Me CH(Me)S(O)Me
Me CH(Me)S(O)₂Me
Me CH(Me)SEt
Me CH(Me)S(O)Et
Me CH(Me)S(O)₂Et
Me CH(Me)S(=NCN)Et
Me CH(Me)S(O)(=NCN)Et
Me CH(Me)SPr-n
Me CH(Me)S(O)Pr-n
Me CH(Me)S(O)₂Pr-n
Me CH(Me)SPr-i
Me CH(Me)S(O)Pr-i
Me CH(Me)S(O)₂Pr-i
Me CH(Me)SBu-t
Me CH(Me)S(O)Bu-t
Me CH(Me)S(O)₂Bu-t
Me CH(Me)SCH₂Pr-c
Me CH(Me)S(O)CH₂Pr-c
Me CH(Me)S(O)₂CH₂Pr-c
Me CH(Me)SCH₂OMe
Me CH(Me)SCH₂SMe
Me CH(Me)S(O)CH₂SMe
Me CH(Me)S(O)₂CH₂SMe
Me CH(Me)SCH₂C≡CH
Me CH(Me)S(O)CH₂C≡CH
Me CH(Me)S(O)₂CH₂C≡CH
Me CH(Me)SCH₂C(O)NHMe
Me CH(Me)S(O)CH₂C(O)NHMe
Me CH(Me)S(O)₂CH₂C(O)NHMe
Me CH(Me)SCH₂C(O)OMe
Me CH(Me)S(O)CH₂C(O)OMe
Me CH(Me)S(O)₂CH₂C(O)OMe
Me CH(Me)SCH₂CF₃
Me CH(Me)S(O)CH₂CF₃
Me CH(Me)S(O)₂CH₂CF₃
Me CH(Me)SCH₂(D2-34a)
Me CH(Me)S(O)CH₂(D2-34a)
Me CH(Me)S(O)₂CH₂(D2-34a)
Me CH(CH₃)SCH₂Si(CH₃)₃
Me CH(Me)SCN
Me CH(Me)SCH₂CN
Me CH(Me)SC(O)Me
Me CH(Me)S(D2-37a)
Me CH(Et)SMe
Me CH(Et)S(O)Me
Me CH(Et)S(O)₂Me
Me CH(Et)SEt
Me CH(Et)S(O)Et
Me CH(Et)S(O)₂Et
Me CH(Et)SCH₂CF₃
Me CH(Et)S(O)CH₂CF₃
Me CH(Et)S(O)₂CH₂CF₃
Me CH(F)SMe
Me CH(F)S(O)Me
Me CH(F)S(O)₂Me
Me CH(F)SEt
Me CH(F)S(O)Et
Me CH(F)S(O)₂Et
Me CH{OC(O)Me}SMe
Me CH{OC(O)Me}S(O)Me
Me CH{OC(O)Me}S(O)₂Me
Me CH(SMe)₂
Me C(Me)₂SMe
Me C(Me)₂S(O)Me
Me C(Me)₂S(O)₂Me
Me CH₂CH₂SH
Me CH₂CH₂SMe
Me CH₂CH₂S(O)Me
Me CH₂CH₂S(O)₂Me
Me CH₂CH₂SEt
Me CH₂CH₂S(O)Et
Me CH₂CH₂S(O)₂Et
Me CH₂CH₂SPr-n
Me CH₂CH₂S(O)Pr-n
Me CH₂CH₂S(O)₂Pr-n
Me CH₂CH₂SPr-i
Me CH₂CH₂S(O)Pr-i
Me CH₂CH₂S(O)₂Pr-i
Me CH(Me)SCH₂CH₂CH₂Cl
Me CH(Me)S(O)CH₂CH₂CH₂Cl
Me CH(Me)S(O)₂CH₂CH₂CH₂Cl
Me CH₂CH₂SCH₂CF₃
Me CH₂CH₂S(O)CH₂CF₃
Me CH₂CH₂S(O)₂CH₂CF₃
Me CH₂CH₂SC(O)Me
Me CH(Me)CH₂SMe
Me CH(Me)CH₂S(O)Me
Me CH(Me)CH₂S(O)₂Me
Me CH(Me)CH₂SEt
Me CH(Me)CH₂S(O)Et
Me CH(Me)CH₂S(O)₂Et
Me CH(Me)CH₂SPr-n
Me CH(Me)CH₂S(O)Pr-n
Me CH(Me)CH₂S(O)₂Pr-n
Me CH(Me)CH₂SPr-i
Me CH(Me)CH₂S(O)Pr-i
Me CH(Me)CH₂S(O)₂Pr-i
Me CH(Me)CH₂SCH₂CF₃
Me CH(Me)CH₂S(O)CH₂CF₃
Me CH(Me)CH₂S(O)₂CH₂CF₃
Me CH(Me)CH₂SC(O)Me
Me CH(Et)CH₂SMe
Me CH(Et)CH₂S(O)Me
Me CH(Et)CH₂S(O)₂Me
Me CH(OMe)CH₂SMe
Me CH(OMe)CH₂S(O)Me
Me CH(OMe)CH₂S(O)₂Me
Me CH(SMe)CH₂SMe
Me CH(SMe)CH₂S(O)Me
Me CH(SMe)CH₂S(O)₂Me
Me CH(CH₂SMe)CH₂SMe
Me CH(CH₂SMe)CH₂S(O)Me
Me CH(CH₂SMe)CH₂S(O)₂Me
Me CH(Cl)CH₂SMe
Me CH(Cl)CH₂S(O)Me
Me CH(Cl)CH₂S(O)₂Me
Me CH(CN)CH₂SMe
Me CH(CN)CH₂S(O)Me
Me CH(CN)CH₂S(O)₂Me
Me CH(CN)CH₂SEt
Me CH(CN)CH₂S(O)Et
Me CH(CN)CH₂S(O)₂Et
Me CH{C(O)OMe}CH₂SMe
Me CH{C(O)OMe}CH₂S(O)Me
Me CH{C(O)OMe}CH₂S(O)₂Me
Me CH{C(O)OMe}CH₂SEt
Me CH{C(O)OMe}CH₂S(O)Et
Me CH{C(O)OMe}CH₂S(O)₂Et
Me CH(Ph)CH₂SMe
Me CH(Ph)CH₂S(O)Me
Me CH(Ph)CH₂S(O)₂Me
Me C(Me)₂CH₂SMe
Me C(Me)₂CH₂S(O)Me
Me C(Me)₂CH₂S(O)₂Me
Me C(=CH₂)CH₂SMe
Me C(=CH₂)CH₂S(O)Me
Me C(=CH₂)CH₂S(O)₂Me
Me C(=CH₂)CH₂SEt
Me C(=CH₂)CH₂S(O)Et
Me C(=CH₂)CH₂S(O)₂Et
Me CH₂CH₂CH₂SEt
Me CH₂CH₂CH₂S(O)Et
Me CH₂CH₂CH₂S(O)₂Et
Me CH(Me)CH₂CH₂SEt
Me CH(Me)CH₂CH₂S(O)Et
Me CH(Me)CH₂CH₂S(O)₂Et
Me CH₂CH(Me)CH₂SEt
Me CH₂CH(Me)CH₂S(O)Et
Me CH₂CH(Me)CH₂S(O)₂Et
Me CH₂CH₂CH(Me)SEt
Me CH₂CH₂CH(Me)S(O)Et
Me CH₂CH₂CH(Me)S(O)₂Et
Me CH₂CH₂CH₂SPr-n
Me CH₂CH₂CH₂S(O)Pr-n
Me CH₂CH₂CH₂S(O)₂Pr-n
Me CH(Me)CH₂CH₂SPr-n
Me CH(Me)CH₂CH₂S(O)Pr-n
Me CH(Me)CH₂CH₂S(O)₂Pr-n
Me CH₂CH(Me)CH₂SPr-n
Me CH₂CH(Me)CH₂S(O)Pr-n
Me CH₂CH(Me)CH₂S(O)₂Pr-n
Me CH₂CH₂CH₂CH₂SMe
Me CH₂CH₂CH₂CH₂S(O)Me
Me CH₂CH₂CH₂CH₂S(O)₂Me
Me CH₂CH₂CH₂CH₂SEt
Me CH₂CH₂CH₂CH₂S(O)Et
Me CH₂CH₂CH₂CH₂S(O)₂Et
Me CH₂CH₂CH₂CH₂SPr-n
Me CH₂CH₂CH₂CH₂S(O)Pr-n
Me CH₂CH₂CH₂CH₂S(O)₂Pr-n
Me CH₂CH(Me)SMe
Me CH₂OCH₂SMe
Me CH=CHSMe
Me CH₂CH(SMe)₂
Me CH₂CH₂SC(O)Me
Me C(=CH₂)CH₂C(O)OH
Me C(=NOMe)CH₃
Me C(=NOMe)Et
Me C(=NOMe)Pr-n
Me C(=NOEt)CH₃
Me C(=NOPr-n)CH₃
Me C(=NOPr-i)CH₃
Me C(=NOBu-n)CH₃
Me C(=NOCH₂Ph)CH₃
Me C(=NOMe)CH₂OCH₂CF₃
Me C(=NOMe)CH₂SMe
Me C(=NOMe)CH₂S(O)Me
Me C(=NOMe)CH₂S(O)₂Me
Me C(=NOMe)CH₂SEt
Me C(=NOMe)CH₂S(O)Et
Me C(=NOMe)CH₂S(O)₂Et
Me C(=NOMe)CH₂SCF₃
Me C(=NOMe)CH₂S(O)CF₃
Me C(=NOMe)CH₂S(O)₂CF₃
Me C(=NOMe)CH₂SCH₂CF₃
Me C(=NOMe)CH₂S(O)CH₂CF₃
Me C(=NOMe)CH₂S(O)₂CH₂CF₃
Me C(=NOEt)CH₂SMe
Me C(=NOEt)CH₂S(O)Me
Me C(=NOEt)CH₂S(O)₂Me
Me C(=NOPr-n)CH₂SMe
Me C(=NOPr-n)CH₂S(O)Me
Me C(=NOPr-n)CH₂S(O)₂Me
Me C(=NOPr-i)CH₂SMe
Me C(=NOPr-i)CH₂S(O)Me
Me C(=NOPr-i)CH₂S(O)₂Me
Me C(=NOBu-n)CH₂SMe
Me C(=NOBu-n)CH₂S(O)Me
Me C(=NOBu-n)CH₂S(O)₂Me
Me C(=NOCH₂Ph)CH₂SMe
Me C(=NOCH₂Ph)CH₂S(O)Me
Me C(=NOCH₂Ph)CH₂S(O)₂Me
Me C(=NOCH₂CH=CH₂)CH₂SMe
Me C(=NOCH₂OMe)CH₂SMe
Me C(=NOCH₂CH₂OMe)CH₂SMe
Me C{=NOCH₂CH₂Si(Me)₃}CH₂SMe
Me CH₂CH(=NOMe)
Me CH₂C(=NOMe)Me
Me CH₂C(=NOMe)Et
Me CH₂C(=NOMe)Pr-n
Me CH₂C(=NOMe)Pr-i
Me CH₂C(=NOMe)Bu-n
Me CH₂C(=NOMe)Bu-i
Me CH₂C(=NOMe)Bu-s
Me CH₂C(=NOMe)Bu-t
Me CH₂C(=NOMe)CF₃
Me CH₂C(=NOCH₃)CH₂SCH₃
Me CH(SMe)C(=NOMe)Me
Me CH{S(O)Me}C(=NOMe)Me
Me CH{S(O)₂Me}C(=NOMe)Me
Me CH(SEt)C(=NOMe)Me
Me CH{S(O)Et}C(=NOMe)Me
Me CH{S(O)₂Et}C(=NOMe)Me
Me CH₂NH₂
Me CH₂NHC(O)Me
Me CH₂NHC(O)OMe
Me CH₂NHC(O)OBu-t
Me CH₂NHSO₂Me
Me CH₂N(Me)C(O)Me
Me CH₂N(Me)C(O)OMe
Me CH₂N(Me)C(O)OBu-t
Me CH₂N(Me)SO₂Me
Me CH(CH₂SMe)NH₂
Me CH(CH₂SMe)NHC(O)Me
Me CH(CH₂SMe)NHC(O)OMe
Me CH(CH₂SMe)NHC(O)OBu-t
Me CH(CH₂SMe)NHSO₂Me
Me CH₂P(O)(OMe)₂
Me CH₂P(O)(OEt)₂
Me OBu-t
Me SMe
Me NH₂
Me NHCH₂CH₂SMe
Me N(Me)CH₂CH₂SMe
Me NHCH₂CH₂CH₂SMe
Me NHMe
Me NHEt
Me NPr-n
Me NHCH(Me)₂
Me NHCH₂C(O)OMe
Me NHCH₂CF₃
Me N(Me)CH₂CF₃
Me NHC(O)OEt
Me NHC(O)CCl₃
Me NHC(O)CH₂SMe
Me N(CH₂CH₃)C(O)CH₂SCH₃
Me NHS(O)₂(D2-108a)
Me NHPh
Me NH(D2-1a)
Me NH(D2-2a)
Me NH(D2-2b)
Me NH(D2-4a)
Me NH{D2-4b}
Me NH(D2-5a)
Me NH(D2-5b)
Me NH(D2-5c)
Me NH(D2-6a)
Me NH(D2-6b)
Me NH(D2-6c)
Me NH(D2-7a)
Me NH(D2-8a)
Me NH(D2-8b)
Me NH(D2-8c)
Me NH(D2-9a)
Me NH(D2-9b)
Me NH(D2-9c)
Me NH(D2-10a)
Me NH(D2-10b)
Me NH(D2-10c)
Me NH(D2-11a)
Me NH(D2-12a)
Me NH(D2-12b)
Me NH(D2-12c)
Me NH(D2-13a)
Me NH(D2-13b)
Me NH(D2-14a)
Me NH(D2-14b)
Me NH(D2-15a)
Me NH(D2-15b)
Me NH(D2-16a)
Me NH(D2-17a)
Me NH(D2-18a)
Me NH(D2-19a)
Me NH(D2-20a)
Me NH(D2-21a)
Me NH(D2-21b)
Me NH(D2-22a)
Me NH(D2-23a)
Me NH(D2-23b)
Me NH(D2-24a)
Me NH(D2-25a)
Me NH(D2-26a)
Me NH(D2-27a)
Me NH(D2-28a)
Me NH(D2-29a)
Me NH(D2-30a)
Me NH(D2-31a)
Me NH(D2-32a)
Me NH(D2-33a)
Me NH(D2-34a)
Me NH(D2-35a)
Me NH(D2-35b)
Me NH(D2-36a)
Me NH(D2-37a)
Me NH(D2-38a)
Me NH(D2-39a)
Me NH(D2-40a)
Me NH(D2-40b)
Me NH(D2-40c)
Me NH(D2-41a)
Me NH(D2-42a)
Me NH(D2-43a)
Me NH(D2-45a)
Me NH(D2-50a)
Me NH(D2-51a)
Me NH(D2-59a)
Me NH(D2-61a)
Me NH(D2-79a)
Me NH(D2-80a)
Me NH{D2-108b(2-Cl)}
Me NH{D2-108b(3-Cl)}
Me NH{D2-108b(4-Cl)}
Me NH{D2-108b(2-Me)}
Me NH{D2-108b(3-Me)}
Me NH{D2-108b(4-Me)}
Me N(Me)Ph
Me N(Me)(D2-1a)
Me N(Me)(D2-2a)
Me N(Me)(D2-2b)
Me N(Me)(D2-4a)
Me N(Me){D2-4b}
Me N(Me)(D2-5a)
Me N(Me)(D2-5b)
Me N(Me)(D2-5c)
Me N(Me)(D2-6a)
Me N(Me)(D2-6b)
Me N(Me)(D2-6c)
Me N(Me)(D2-7a)
Me N(Me)(D2-8a)
Me N(Me)(D2-8b)
Me N(Me)(D2-8c)
Me N(Me)(D2-9a)
Me N(Me)(D2-9b)
Me N(Me)(D2-9c)
Me N(Me)(D2-10a)
Me N(Me)(D2-10b)
Me N(Me)(D2-10c)
Me N(Me)(D2-11a)
Me N(Me)(D2-12a)
Me N(Me)(D2-12b)
Me N(Me)(D2-12c)
Me N(Me)(D2-13a)
Me N(Me)(D2-13b)
Me N(Me)(D2-14a)
Me N(Me)(D2-14b)
Me N(Me)(D2-15a)
Me N(Me)(D2-15b)
Me N(Me)(D2-16a)
Me N(Me)(D2-17a)
Me N(Me)(D2-18a)
Me N(Me)(D2-19a)
Me N(Me)(D2-20a)
Me N(Me)(D2-21a)
Me N(Me)(D2-21b)
Me N(Me)(D2-22a)
Me N(Me)(D2-23a)
Me N(Me)(D2-23b)
Me N(Me)(D2-24a)
Me N(Me)(D2-25a)
Me N(Me)(D2-26a)
Me N(Me)(D2-27a)
Me N(Me)(D2-28a)
Me N(Me)(D2-29a)
Me N(Me)(D2-30a)
Me N(Me)(D2-31a)
Me N(Me)(D2-32a)
Me N(Me)(D2-33a)
Me N(Me)(D2-34a)
Me N(Me)(D2-35a)
Me N(Me)(D2-35b)
Me N(Me)(D2-36a)
Me N(Me)(D2-37a)
Me N(Me)(D2-38a)
Me N(Me)(D2-39a)
Me N(Me)(D2-40a)
Me N(Me)(D2-40b)
Me N(Me)(D2-40c)
Me N(Me)(D2-41a)
Me N(Me)(D2-42a)
Me N(Me)(D2-43a)
Me N(Me)(D2-45a)
Me N(Me)(D2-50a)
Me N(Me)(D2-51a)
Me N(Me)(D2-59a)
Me N(Me)(D2-61a)
Me N(Me)(D2-79a)
Me N(Me)(D2-80a)
Me N(Me){D2-108b(2-Cl)}
Me N(Me){D2-108b(3-Cl)}
Me N(Me){D2-108b(4-Cl)}
Me N(Me){D2-108b(2-Me)}
Me N(Me){D2-108b(3-Me)}
Me N(Me){D2-108b(4-Me)}
Me D2-19a
Me D2-32b(2-Br)
Me D2-33b(2-OMe)
Me D2-35b
Me D2-38b(4-SMe)
Me D2-39b(5-Me)
Me D2-82a
Me D2-82b
Me D2-87a
Me D2-103b
Me D2-103c
Me D2-103d
Me D2-103e
Me CH₂(D2-2a)
Me CH₂{D2-5f(3-Me)}
Me CH₂(D2-28a)
Me CH₂(D2-32a)
Me CH₂(D2-33a)
Me CH₂{D2-33b(6-Cl)}
Me CH₂(D2-34a)
Et C(O)(D2-2a)
Et C(O)Me
Et C(O)Et
Et C(O)Pr-n
Et C(O)Pr-i
Et C(O)Pr-c
Et C(O)Bu-n
Et C(O)Bu-i
Et C(O)Bu-s
Et C(O)Bu-t
Et C(O)Pen-n
Et C(O)Pen-c
Et C(O)Hex-n
Et C(O)Hex-c
Et C(O)CF₃
Et C(O)OMe
Et C(O)OEt
Et C(O)NHPh
Et Me
Et Et
Et Pr-n
Et Pr-i
Et Pr-c
Et Bu-n
Et Bu-i
Et Bu-c
Et Bu-s
Et Bu-t
Et Pen-n
Et Pen-c
Et Hex-n
Et Hex-c
Et (CH₂)_６CH₃
Et (CH₂)₇CH₃
Et (CH₂)_８CH₃
Et (CH₂)_９CH₃
Et (CH₂)₁₀CH₃
Et (CH₂)_1１CH₃
Et CH(Me)(CH₂)₂CH₃
Et CH(Me)(CH₂)_３CH₃
Et CH(Me)(CH₂)_４CH₃
Et CH(Me)(CH₂)_５CH₃
Et CH(Me)(CH₂)_６CH₃
Et CH(Me)(CH₂)_７CH₃
Et CH(Me)(CH₂)_８CH₃
Et CH₂Pr-c
Et CH₂Bu-t
Et CH=CH₂
Et C(Me)=CH₂
Et CH=CH(D2-1a)
Et CH=CH(D2-2a)
Et CH=CH(D2-33a）
Et CH=CH｛D2-108b(4-CF₃)｝
Et C≡CH
Et C≡CSiMe₃
Et CHCl₂
Et CH₂Br
Et CH(Br)Me
Et CH₂CH₂CH₂CH₂Br
Et CH(Br)Bu-t
Et CH₂CF₃
Et CF₂CF₂Cl
Et CH₂CH(CF₃)₂
Et CH₂CH(OH)CF₃
Et CH₂CH₂C(F)=CF₂
Et CH₂CN
Et CH(Me)CN
Et CH₂CH₂CN
Et CH(Me)CH₂CN
Et CH₂CH₂CH₂CN
Et CH(Me)CH₂CH₂CN
Et CH₂CH₂CH₂CH₂CN
Et CH(Me)CH₂CH₂CH₂CN
Et CH₂C(O)OMe
Et CH(Me)C(O)OMe
Et CH₂CH₂C(O)OMe
Et CH(Me)CH₂C(O)OMe
Et CH₂CH₂CH₂C(O)OMe
Et CH(Me)CH₂CH₂C(O)OMe
Et CH₂CH₂CH₂CH₂C(O)OMe
Et CH₂C(O)OEt
Et CH(Me)C(O)OEt
Et CH₂CH₂C(O)OEt
Et CH(Me)CH₂C(O)OEt
Et CH₂CH₂CH₂C(O)OEt
Et CH(Me)CH₂CH₂C(O)OEt
Et CH₂CH₂CH₂CH₂C(O)OEt
Et CH₂C(O)NHMe
Et CH₂C(O)NHCH₂CF₃
Et CH₂OMe
Et CH₂OEt
Et CH₂OPr-n
Et CH₂OPr-i
Et CH₂OPr-c
Et CH₂OBu-n
Et CH₂OBu-i
Et CH₂OBu-s
Et CH₂OBu-t
Et CH₂OBu-c
Et CH₂OPen-n
Et CH₂OPen-c
Et CH₂OHex-n
Et CH₂OHex-c
Et CH₂OCH₂Pr-c
Et CH₂OCH₂CH=CH₂
Et CH₂OCH₂C≡CH
Et CH₂OCH₂OMe
Et CH₂OCH₂SMe
Et CH₂OCH₂Si(CH₃)₃
Et CH₂OCH₂(D2-34a)
Et CH₂OCF₃
Et CH₂OCF₂H
Et CH₂OCF₂Cl
Et CH₂OCF₂Br
Et CH₂OCH₂CF₃
Et CH₂OCH₂CF₂CF₃
Et CH₂OCH₂CN
Et CH₂OC(O)Me
Et CH₂OCH₂C(O)OMe
Et CH₂OCH₂C(O)OEt
Et CH₂ON=CHMe
Et CH₂ON=C(Me)₂
Et CH(Me)OMe
Et CH(Me)OEt
Et CH(Me)OPr-n
Et CH(Me)OPr-i
Et CH(Me)OPr-c
Et CH(Me)OBu-n
Et CH(Me)OBu-i
Et CH(Me)OBu-s
Et CH(Me)OBu-t
Et CH(Me)OBu-c
Et CH(Me)OPen-n
Et CH(Me)OPen-c
Et CH(Me)OHex-n
Et CH(Me)OHex-c
Et CH(Me)OCH₂Pr-c
Et CH(Me)OCH₂CH=CH₂
Et CH(Me)OCH₂C≡CH
Et CH(Me)OCH₂OMe
Et CH(Me)OCH₂SMe
Et CH(Me)OCH₂Si(CH₃)₃
Et CH(Me)OCH₂(D2-34a)
Et CH(Me)OCF₃
Et CH(Me)OCF₂H
Et CH(Me)OCF₂Cl
Et CH(Me)OCF₂Br
Et CH(Me)OCH₂CF₃
Et CH(Me)OCH₂CF₂CF₃
Et CH(Me)OCH₂CN
Et CH(Me)OC(O)Me
Et CH(Me)OCH₂C(O)OMe
Et CH(Me)OCH₂C(O)OEt
Et CH(Me)ON=CHMe
Et CH(Me)ON=C(Me)₂
Et C(Me)₂OC(O)Me
Et CH₂SMe
Et CH₂S(O)Me
Et CH₂S(O)₂Me
Et CH₂SEt
Et CH₂S(O)Et
Et CH₂S(O)₂Et
Et CH₂SPr-n
Et CH₂S(O)Pr-n
Et CH₂S(O)₂Pr-n
Et CH₂SPr-i
Et CH₂S(O)Pr-i
Et CH₂S(O)₂Pr-i
Et CH₂SPr-c
Et CH₂S(O)Pr-c
Et CH₂S(O)₂Pr-c
Et CH₂SCH₂CH=CH₂
Et CH₂S(O)CH₂CH=CH₂
Et CH₂S(O)₂CH₂CH=CH₂
Et CH₂SCH₂C≡CH
Et CH₂S(O)CH₂C≡CH
Et CH₂S(O)₂CH₂C≡CH
Et CH₂SCH₂CF₃
Et CH₂S(O)CH₂CF₃
Et CH₂S(O)₂CH₂CF₃
Et CH₂SCH₂CH(OMe)₂
Et CH₂SCH₂CH(=NOMe)
Et CH(Me)SMe
Et CH(Me)S(O)Me
Et CH(Me)S(O)₂Me
Et CH(Me)SEt
Et CH(Me)S(O)Et
Et CH(Me)S(O)₂Et
Et CH(Me)S(=NCN)Et
Et CH(Me)S(O)(=NCN)Et
Et CH(Me)SPr-n
Et CH(Me)S(O)Pr-n
Et CH(Me)S(O)₂Pr-n
Et CH(Me)SPr-i
Et CH(Me)S(O)Pr-i
Et CH(Me)S(O)₂Pr-i
Et CH(Me)SBu-t
Et CH(Me)S(O)Bu-t
Et CH(Me)S(O)₂Bu-t
Et CH(Me)SCH₂Pr-c
Et CH(Me)S(O)CH₂Pr-c
Et CH(Me)S(O)₂CH₂Pr-c
Et CH(Me)SCH₂OMe
Et CH(Me)SCH₂SMe
Et CH(Me)S(O)CH₂SMe
Et CH(Me)S(O)₂CH₂SMe
Et CH(Me)SCH₂C=CH₂
Et CH(Me)S(O)CH₂C=CH₂
Et CH(Me)S(O)₂CH₂C=CH₂
Et CH(Me)SCH₂C≡CH
Et CH(Me)S(O)CH₂C≡CH
Et CH(Me)S(O)₂CH₂C≡CH
Et CH(Me)SCH₂C(O)NHMe
Et CH(Me)S(O)CH₂C(O)NHMe
Et CH(Me)S(O)₂CH₂C(O)NHMe
Et CH(Me)SCH₂C(O)OMe
Et CH(Me)S(O)CH₂C(O)OMe
Et CH(Me)S(O)₂CH₂C(O)OMe
Et CH(Me)SCH₂CH₂CH₂Cl
Et CH(Me)S(O)CH₂CH₂CH₂Cl
Et CH(Me)S(O)₂CH₂CH₂CH₂Cl
Et CH(Me)SCH₂CF₃
Et CH(Me)S(O)CH₂CF₃
Et CH(Me)S(O)₂CH₂CF₃
Et CH(Me)SCH₂Ph
Et CH(Me)S(O)CH₂Ph
Et CH(Me)S(O)₂CH₂Ph
Et CH(Me)SCH₂(D2-34a)
Et CH(Me)S(O)CH₂(D2-34a)
Et CH(Me)S(O)₂CH₂(D2-34a)
Et CH(CH₃)SCH₂Si(CH₃)₃
Et CH(Me)SCN
Et CH(Me)SCH₂CN
Et CH(Me)SC(O)Me
Et CH(Me)S(D2-12a)
Et CH(Me)S(D2-32a)
Et CH(Me)S{D2-32b(3-NO₂)}
Et CH(Me)S{D2-32b(3-CF₃)}
Et CH(Me)S(D2-37a)
Et CH(Me)S(D2-51a)
Et CH(Et)SMe
Et CH(Et)S(O)Me
Et CH(Et)S(O)₂Me
Et CH(Et)SEt
Et CH(Et)S(O)Et
Et CH(Et)S(O)₂Et
Et CH(Et)SCH₂CF₃
Et CH(Et)S(O)CH₂CF₃
Et CH(Et)S(O)₂CH₂CF₃
Et CH(Pr-n)SMe
Et CH(Pr-n)S(O)Me
Et CH(Pr-n)S(O)₂Me
Et CH(Pr-n)SEt
Et CH(Pr-n)S(O)Et
Et CH(Pr-n)S(O)₂Et
Et CH(Pr-n)S(=NCN)Et
Et CH(Pr-n)S(O)(=NCN)Et
Et CH(Pr-n)SPr-n
Et CH(Pr-n)S(O)Pr-n
Et CH(Pr-n)S(O)₂Pr-n
Et CH(Pr-n)SPr-i
Et CH(Pr-n)S(O)Pr-i
Et CH(Pr-n)S(O)₂Pr-i
Et CH(Pr-n)SPr-c
Et CH(Pr-n)S(O)Pr-c
Et CH(Pr-n)S(O)₂Pr-c
Et CH(Pr-n)SCH₂CF₃
Et CH(Pr-n)S(O)CH₂CF₃
Et CH(Pr-n)S(O)₂CH₂CF₃
Et CH(Pr-i)SMe
Et CH(Pr-i)S(O)Me
Et CH(Pr-i)S(O)₂Me
Et CH(Pr-i)SEt
Et CH(Pr-i)S(O)Et
Et CH(Pr-i)S(O)₂Et
Et CH(Pr-i)S(=NCN)Et
Et CH(Pr-i)S(O)(=NCN)Et
Et CH(Pr-i)SPr-n
Et CH(Pr-i)S(O)Pr-n
Et CH(Pr-i)S(O)₂Pr-n
Et CH(Pr-i)SPr-i
Et CH(Pr-i)S(O)Pr-i
Et CH(Pr-i)S(O)₂Pr-i
Et CH(Pr-i)SPr-c
Et CH(Pr-i)S(O)Pr-c
Et CH(Pr-i)S(O)₂Pr-c
Et CH(Pr-i)SCH₂CF₃
Et CH(Pr-i)S(O)CH₂CF₃
Et CH(Pr-i)S(O)₂CH₂CF₃
Et CH(Pr-c)SMe
Et CH(Pr-c)S(O)Me
Et CH(Pr-c)S(O)₂Me
Et CH(Pr-c)SEt
Et CH(Pr-c)S(O)Et
Et CH(Pr-c)S(O)₂Et
Et CH(Pr-c)S(=NCN)Et
Et CH(Pr-c)S(O)(=NCN)Et
Et CH(Pr-c)SPr-n
Et CH(Pr-c)S(O)Pr-n
Et CH(Pr-c)S(O)₂Pr-n
Et CH(Pr-c)SPr-i
Et CH(Pr-c)S(O)Pr-i
Et CH(Pr-c)S(O)₂Pr-i
Et CH(Pr-c)SPr-c
Et CH(Pr-c)S(O)Pr-c
Et CH(Pr-c)S(O)₂Pr-c
Et CH(Pr-c)SCH₂CF₃
Et CH(Pr-c)S(O)CH₂CF₃
Et CH(Pr-c)S(O)₂CH₂CF₃
Et CH(Bu-n)SMe
Et CH(Bu-n)S(O)Me
Et CH(Bu-n)S(O)₂Me
Et CH(Bu-n)SEt
Et CH(Bu-n)S(O)Et
Et CH(Bu-n)S(O)₂Et
Et CH(Bu-n)S(=NCN)Et
Et CH(Bu-n)S(O)(=NCN)Et
Et CH(Bu-n)SPr-n
Et CH(Bu-n)S(O)Pr-n
Et CH(Bu-n)S(O)₂Pr-n
Et CH(Bu-n)SPr-i
Et CH(Bu-n)S(O)Pr-i
Et CH(Bu-n)S(O)₂Pr-i
Et CH(Bu-n)SPr-c
Et CH(Bu-n)S(O)Pr-c
Et CH(Bu-n)S(O)₂Pr-c
Et CH(Bu-n)SCH₂CF₃
Et CH(Bu-n)S(O)CH₂CF₃
Et CH(Bu-n)S(O)₂CH₂CF₃
Et CH(F)SMe
Et CH(F)S(O)Me
Et CH(F)S(O)₂Me
Et CH(F)SEt
Et CH(F)S(O)Et
Et CH(F)S(O)₂Et
Et CH(F)S(=NCN)Et
Et CH(F)S(O)(=NCN)Et
Et CH(F)SCH₂CF₃
Et CH(F)S(O)CH₂CF₃
Et CH(F)S(O)₂CH₂CF₃
Et C(F)₂SMe
Et C(F)₂S(O)Me
Et C(F)₂S(O)₂Me
Et C(F)₂SEt
Et C(F)₂S(O)Et
Et C(F)₂S(O)₂Et
Et C(F)₂S(=NCN)Et
Et C(F)₂S(O)(=NCN)Et
Et C(F)₂SCH₂CF₃
Et C(F)₂S(O)CH₂CF₃
Et C(F)₂S(O)₂CH₂CF₃
Et CH(Cl)SMe
Et CH(Cl)S(O)Me
Et CH(Cl)S(O)₂Me
Et CH(Cl)SEt
Et CH(Cl)S(O)Et
Et CH(Cl)S(O)₂Et
Et CH(Cl)S(=NCN)Et
Et CH(Cl)S(O)(=NCN)Et
Et CH(Cl)SCH₂CF₃
Et CH(Cl)S(O)CH₂CF₃
Et CH(Cl)S(O)₂CH₂CF₃
Et C(Cl)₂SMe
Et C(Cl)₂S(O)Me
Et C(Cl)₂S(O)₂Me
Et C(Cl)₂SEt
Et C(Cl)₂S(O)Et
Et C(Cl)₂S(O)₂Et
Et C(Cl)₂S(=NCN)Et
Et C(Cl)₂S(O)(=NCN)Et
Et C(Cl)₂SCH₂CF₃
Et C(Cl)₂S(O)CH₂CF₃
Et C(Cl)₂S(O)₂CH₂CF₃
Et CH(Br)SMe
Et CH(Br)S(O)Me
Et CH(Br)S(O)₂Me
Et CH(Br)SEt
Et CH(Br)S(O)Et
Et CH(Br)S(O)₂Et
Et CH(Br)S(=NCN)Et
Et CH(Br)S(O)(=NCN)Et
Et CH(Br)SCH₂CF₃
Et CH(Br)S(O)CH₂CF₃
Et CH(Br)S(O)₂CH₂CF₃
Et CH(I)SMe
Et CH(I)S(O)Me
Et CH(I)S(O)₂Me
Et CH(I)SEt
Et CH(I)S(O)Et
Et CH(I)S(O)₂Et
Et CH(I)S(=NCN)Et
Et CH(I)S(O)(=NCN)Et
Et CH(I)SCH₂CF₃
Et CH(I)S(O)CH₂CF₃
Et CH(I)S(O)₂CH₂CF₃
Et CH{OC(O)Me}SMe
Et CH{OC(O)Me}S(O)Me
Et CH{OC(O)Me}S(O)₂Me
Et CH{OC(O)OMe}SEt
Et CH{OC(O)OMe}S(O)Et
Et CH{OC(O)OMe}S(O)₂Et
Et CH{OC(O)OMe}S(=NCN)Et
Et CH{OC(O)OMe}S(O)(=NCN)Et
Et CH{OC(O)OEt}SMe
Et CH{OC(O)OEt}S(O)Me
Et CH{OC(O)OEt}S(O)₂Me
Et CH{OC(O)OEt}SEt
Et CH{OC(O)OEt}S(O)Et
Et CH{OC(O)OEt}S(O)₂Et
Et CH{OC(O)OEt}S(=NCN)Et
Et CH{OC(O)OEt}S(O)(=NCN)Et
Et CH(OMe)SMe
Et CH(OMe)S(O)Me
Et CH(OMe)S(O)₂Me
Et CH(OMe)SEt
Et CH(OMe)S(O)Et
Et CH(OMe)S(O)₂Et
Et CH(OMe)S(=NCN)Et
Et CH(OMe)S(O)(=NCN)Et
Et CH(OEt)SMe
Et CH(OEt)S(O)Me
Et CH(OEt)S(O)₂Me
Et CH(OEt)SEt
Et CH(OEt)S(O)Et
Et CH(OEt)S(O)₂Et
Et CH(OEt)S(=NCN)Et
Et CH(OEt)S(O)(=NCN)Et
Et CH(SMe)₂
Et CH(SMe)S(O)Me
Et CH(SMe)S(O)₂Me
Et CH(SMe)SEt
Et CH(SMe)S(O)Et
Et CH(SMe)S(O)₂Et
Et CH(SMe)S(=NCN)Et
Et CH(SMe)S(O)(=NCN)Et
Et CH(SEt)SMe
Et CH(SEt)S(O)Me
Et CH(SEt)S(O)₂Me
Et CH(SEt)SEt
Et CH(SEt)S(O)Et
Et CH(SEt)S(O)₂Et
Et CH(SEt)S(=NCN)Et
Et CH(SEt)S(O)(=NCN)Et
Et CH(CN)SMe
Et CH(CN)S(O)Me
Et CH(CN)S(O)₂Me
Et CH(CN)SEt
Et CH(CN)S(O)Et
Et CH(CN)S(O)₂Et
Et CH(CN)S(=NCN)Et
Et CH(CN)S(O)(=NCN)Et
Et CH{C(O)OMe}SMe
Et CH{C(O)OMe}S(O)Me
Et CH{C(O)OMe}S(O)₂Me
Et CH{C(O)OMe}SMe
Et CH{C(O)OMe}S(O)Me
Et CH{C(O)OMe}S(O)₂Me
Et CH{C(O)OMe}SEt
Et CH{C(O)OMe}S(O)Et
Et CH{C(O)OMe}S(O)₂Et
Et CH{C(O)OMe}S(=NCN)Et
Et CH{C(O)OMe}S(O)(=NCN)Et
Et CH{C(O)OEt}SMe
Et CH{C(O)OEt}S(O)Me
Et CH{C(O)OEt}S(O)₂Me
Et CH{C(O)OEt}SEt
Et CH{C(O)OEt}S(O)Et
Et CH{C(O)OEt}S(O)Et
Et CH{C(O)OEt}S(=NCN)Et
Et CH{C(O)OEt}S(O)(=NCN)Et
Et C(Me)₂SMe
Et C(Me)₂S(O)Me
Et C(Me)₂S(O)₂Me
Et CH₂CH₂SH
Et CH₂CH₂SMe
Et CH₂CH₂S(O)Me
Et CH₂CH₂S(O)₂Me
Et CH₂CH₂SEt
Et CH₂CH₂S(O)Et
Et CH₂CH₂S(O)₂Et
Et CH₂CH₂SPr-n
Et CH₂CH₂S(O)Pr-n
Et CH₂CH₂S(O)₂Pr-n
Et CH₂CH₂SPr-i
Et CH₂CH₂S(O)Pr-i
Et CH₂CH₂S(O)₂Pr-i
Et CH₂CH₂SCH₂CF₃
Et CH₂CH₂S(O)CH₂CF₃
Et CH₂CH₂S(O)₂CH₂CF₃
Et CH₂CH₂SC(O)Me
Et CH(Me)CH₂SMe
Et CH(Me)CH₂S(O)Me
Et CH(Me)CH₂S(O)₂Me
Et CH(Me)CH₂SEt
Et CH(Me)CH₂S(O)Et
Et CH(Me)CH₂S(O)₂Et
Et CH(Me)CH₂SPr-n
Et CH(Me)CH₂S(O)Pr-n
Et CH(Me)CH₂S(O)₂Pr-n
Et CH(Me)CH₂SPr-i
Et CH(Me)CH₂S(O)Pr-i
Et CH(Me)CH₂S(O)₂Pr-i
Et CH(Me)CH₂SCH₂CF₃
Et CH(Me)CH₂S(O)CH₂CF₃
Et CH(Me)CH₂S(O)₂CH₂CF₃
Et CH(Me)CH₂SC(O)Me
Et CH(Et)CH₂SMe
Et CH(Et)CH₂S(O)Me
Et CH(Et)CH₂S(O)₂Me
Et CH(Et)CH₂SEt
Et CH(Et)CH₂S(O)Et
Et CH(Et)CH₂S(O)₂Et
Et CH(Pr-n)CH₂SMe
Et CH(Pr-n)CH₂S(O)Me
Et CH(Pr-n)CH₂S(O)₂Me
Et CH(Pr-n)CH₂SEt
Et CH(Pr-n)CH₂S(O)Et
Et CH(Pr-n)CH₂S(O)₂Et
Et CH(Pr-i)CH₂SMe
Et CH(Pr-i)CH₂S(O)Me
Et CH(Pr-i)CH₂S(O)₂Me
Et CH(Pr-i)CH₂SEt
Et CH(Pr-i)CH₂S(O)Et
Et CH(Pr-i)CH₂S(O)₂Et
Et CH(Pr-c)CH₂SMe
Et CH(Pr-c)CH₂S(O)Me
Et CH(Pr-c)CH₂S(O)₂Me
Et CH(Pr-c)CH₂SEt
Et CH(Pr-c)CH₂S(O)Et
Et CH(Pr-c)CH₂S(O)₂Et
Et CH(Bu-n)CH₂SMe
Et CH(Bu-n)CH₂S(O)Me
Et CH(Bu-n)CH₂S(O)₂Me
Et CH(Bu-n)CH₂SEt
Et CH(Bu-n)CH₂S(O)Et
Et CH(Bu-n)CH₂S(O)₂Et
Et CH(Bu-i)CH₂SMe
Et CH(Bu-i)CH₂S(O)Me
Et CH(Bu-i)CH₂S(O)₂Me
Et CH(Bu-i)CH₂SEt
Et CH(Bu-i)CH₂S(O)Et
Et CH(Bu-i)CH₂S(O)₂Et
Et CH(Bu-s)CH₂SMe
Et CH(Bu-s)CH₂S(O)Me
Et CH(Bu-s)CH₂S(O)₂Me
Et CH(Bu-s)CH₂SEt
Et CH(Bu-s)CH₂S(O)Et
Et CH(Bu-s)CH₂S(O)₂Et
Et CH(Bu-t)CH₂SMe
Et CH(Bu-t)CH₂S(O)Me
Et CH(Bu-t)CH₂S(O)₂Me
Et CH(Bu-t)CH₂SEt
Et CH(Bu-t)CH₂S(O)Et
Et CH(Bu-t)CH₂S(O)₂Et
Et CH(OMe)CH₂SMe
Et CH(OMe)CH₂S(O)Me
Et CH(OMe)CH₂S(O)₂Me
Et CH(OMe)CH₂SEt
Et CH(OMe)CH₂S(O)Et
Et CH(OMe)CH₂S(O)₂Et
Et CH(SMe)CH₂SMe
Et CH(SMe)CH₂S(O)Me
Et CH(SMe)CH₂S(O)₂Me
Et CH(SMe)CH₂SEt
Et CH(SMe)CH₂S(O)Et
Et CH(SMe)CH₂S(O)₂Et
Et CH(CH₂OMe)CH₂SMe
Et CH(CH₂OMe)CH₂S(O)Me
Et CH(CH₂OMe)CH₂S(O)₂Me
Et CH(CH₂OMe)CH₂SEt
Et CH(CH₂OMe)CH₂S(O)Et
Et CH(CH₂OMe)CH₂S(O)₂Et
Et CH(CH₂SMe)CH₂SMe
Et CH(CH₂SMe)CH₂S(O)Me
Et CH(CH₂SMe)CH₂S(O)₂Me
Et CH(CH₂SMe)CH₂SEt
Et CH(CH₂SMe)CH₂S(O)Et
Et CH(CH₂SMe)CH₂S(O)₂Et
Et CH(F)CH₂SMe
Et CH(F)CH₂S(O)Me
Et CH(F)CH₂S(O)₂Me
Et CH(F)CH₂SEt
Et CH(F)CH₂S(O)Et
Et CH(F)CH₂S(O)₂Et
Et C(F)₂CH₂SMe
Et C(F)₂CH₂S(O)Me
Et C(F)₂CH₂S(O)₂Me
Et C(F)₂CH₂SEt
Et C(F)₂CH₂S(O)Et
Et C(F)₂CH₂S(O)₂Et
Et CH(Cl)CH₂SMe
Et CH(Cl)CH₂S(O)Me
Et CH(Cl)CH₂S(O)₂Me
Et CH(Cl)CH₂SEt
Et CH(Cl)CH₂S(O)Et
Et CH(Cl)CH₂S(O)₂Et
Et C(Cl)₂CH₂SMe
Et C(Cl)₂CH₂S(O)Me
Et C(Cl)₂CH₂S(O)₂Me
Et C(Cl)₂CH₂SEt
Et C(Cl)₂CH₂S(O)Et
Et C(Cl)₂CH₂S(O)₂Et
Et CH(Br)CH₂SMe
Et CH(Br)CH₂S(O)Me
Et CH(Br)CH₂S(O)₂Me
Et CH(Br)CH₂SEt
Et CH(Br)CH₂S(O)Et
Et CH(Br)CH₂S(O)₂Et
Et CH(I)CH₂SMe
Et CH(I)CH₂S(O)Me
Et CH(I)CH₂S(O)₂Me
Et CH(I)CH₂SEt
Et CH(I)CH₂S(O)Et
Et CH(I)CH₂S(O)₂Et
Et CH(CN)CH₂SMe
Et CH(CN)CH₂S(O)Me
Et CH(CN)CH₂S(O)₂Me
Et CH(CN)CH₂SEt
Et CH(CN)CH₂S(O)Et
Et CH(CN)CH₂S(O)₂Et
Et CH{C(O)OMe}CH₂SMe
Et CH{C(O)OMe}CH₂S(O)Me
Et CH{C(O)OMe}CH₂S(O)₂Me
Et CH{C(O)OMe}CH₂SEt
Et CH{C(O)OMe}CH₂S(O)Et
Et CH{C(O)OMe}CH₂S(O)₂Et
Et CH{C(O)OEt}CH₂SMe
Et CH{C(O)OEt}CH₂S(O)Me
Et CH{C(O)OEt}CH₂S(O)₂Me
Et CH{C(O)OEt}CH₂SEt
Et CH{C(O)OEt}CH₂S(O)Et
Et CH{C(O)OEt}CH₂S(O)₂Et
Et CH(Ph)CH₂SMe
Et CH(Ph)CH₂S(O)Me
Et CH(Ph)CH₂S(O)₂Me
Et CH(Ph)CH₂SEt
Et CH(Ph)CH₂S(O)Et
Et CH(Ph)CH₂S(O)₂Et
Et C(Me)₂CH₂SMe
Et C(Me)₂CH₂S(O)Me
Et C(Me)₂CH₂S(O)₂Me
Et C(Me)₂CH₂SEt
Et C(Me)₂CH₂S(O)Et
Et C(Me)₂CH₂S(O)₂Et
Et C(Et)₂CH₂SMe
Et C(Et)₂CH₂S(O)Me
Et C(Et)₂CH₂S(O)₂Me
Et C(Et)₂CH₂SEt
Et C(Et)₂CH₂S(O)Et
Et C(Et)₂CH₂S(O)₂Et
Et C(=CH₂)CH₂SMe
Et C(=CH₂)CH₂S(O)Me
Et C(=CH₂)CH₂S(O)₂Me
Et C(=CH₂)CH₂SEt
Et C(=CH₂)CH₂S(O)Et
Et C(=CH₂)CH₂S(O)₂Et
Et CH₂CH₂CH₂SEt
Et CH₂CH₂CH₂S(O)Et
Et CH₂CH₂CH₂S(O)₂Et
Et CH(Me)CH₂CH₂SEt
Et CH(Me)CH₂CH₂S(O)Et
Et CH(Me)CH₂CH₂S(O)₂Et
Et CH₂CH(Me)CH₂SEt
Et CH₂CH(Me)CH₂S(O)Et
Et CH₂CH(Me)CH₂S(O)₂Et
Et CH₂CH₂CH(Me)SEt
Et CH₂CH₂CH(Me)S(O)Et
Et CH₂CH₂CH(Me)S(O)₂Et
Et CH₂CH₂CH₂SPr-n
Et CH₂CH₂CH₂S(O)Pr-n
Et CH₂CH₂CH₂S(O)₂Pr-n
Et CH(Me)CH₂CH₂SPr-n
Et CH(Me)CH₂CH₂S(O)Pr-n
Et CH(Me)CH₂CH₂S(O)₂Pr-n
Et CH₂CH(Me)CH₂SPr-n
Et CH₂CH(Me)CH₂S(O)Pr-n
Et CH₂CH(Me)CH₂S(O)₂Pr-n
Et CH₂CH₂CH₂CH₂SMe
Et CH₂CH₂CH₂CH₂S(O)Me
Et CH₂CH₂CH₂CH₂S(O)₂Me
Et CH₂CH₂CH₂CH₂SEt
Et CH₂CH₂CH₂CH₂S(O)Et
Et CH₂CH₂CH₂CH₂S(O)₂Et
Et CH₂CH₂CH₂CH₂SPr-n
Et CH₂CH₂CH₂CH₂S(O)Pr-n
Et CH₂CH₂CH₂CH₂S(O)₂Pr-n
Et CH₂CH(Me)SMe
Et CH₂CH(Me)S(O)Me
Et CH₂CH(Me)S(O)₂Me
Et CH₂CH(Me)SEt
Et CH₂CH(Me)S(O)Et
Et CH₂CH(Me)S(O)₂Et
Et CH₂CH(Et)SMe
Et CH₂CH(Et)S(O)Me
Et CH₂CH(Et)S(O)₂Me
Et CH₂CH(Et)SEt
Et CH₂CH(Et)S(O)Et
Et CH₂CH(Et)S(O)₂Et
Et CH₂CH(Pr-n)SMe
Et CH₂CH(Pr-n)S(O)Me
Et CH₂CH(Pr-n)S(O)₂Me
Et CH₂CH(Pr-n)SEt
Et CH₂CH(Pr-n)S(O)Et
Et CH₂CH(Pr-n)S(O)₂Et
Et CH₂CH(Pr-i)SMe
Et CH₂CH(Pr-i)S(O)Me
Et CH₂CH(Pr-i)S(O)₂Me
Et CH₂CH(Pr-i)SEt
Et CH₂CH(Pr-i)S(O)Et
Et CH₂CH(Pr-i)S(O)₂Et
Et CH₂CH(Pr-c)SMe
Et CH₂CH(Pr-c)S(O)Me
Et CH₂CH(Pr-c)S(O)₂Me
Et CH₂CH(Pr-c)SEt
Et CH₂CH(Pr-c)S(O)Et
Et CH₂CH(Pr-c)S(O)₂Et
Et CH₂CH(Bu-n)SMe
Et CH₂CH(Bu-n)S(O)Me
Et CH₂CH(Bu-n)S(O)₂Me
Et CH₂CH(Bu-n)SEt
Et CH₂CH(Bu-n)S(O)Et
Et CH₂CH(Bu-n)S(O)₂Et
Et CH₂CH(Bu-i)SMe
Et CH₂CH(Bu-i)S(O)Me
Et CH₂CH(Bu-i)S(O)₂Me
Et CH₂CH(Bu-i)SEt
Et CH₂CH(Bu-i)S(O)Et
Et CH₂CH(Bu-i)S(O)₂Et
Et CH₂CH(Bu-s)SMe
Et CH₂CH(Bu-s)S(O)Me
Et CH₂CH(Bu-s)S(O)₂Me
Et CH₂CH(Bu-s)SEt
Et CH₂CH(Bu-s)S(O)Et
Et CH₂CH(Bu-s)S(O)₂Et
Et CH₂CH(Bu-t)SMe
Et CH₂CH(Bu-t)S(O)Me
Et CH₂CH(Bu-t)S(O)₂Me
Et CH₂CH(Bu-t)SEt
Et CH₂CH(Bu-t)S(O)Et
Et CH₂CH(Bu-t)S(O)₂Et
Et CH₂C(Et)₂SMe
Et CH₂C(Et)₂S(O)Me
Et CH₂C(Et)₂S(O)₂Me
Et CH₂C(Et)₂SEt
Et CH₂C(Et)₂S(O)Et
Et CH₂C(Et)₂S(O)₂Et
Et CH(Et)CH(Me)SMe
Et CH(Et)CH(Me)S(O)Me
Et CH(Et)CH(Me)S(O)₂Me
Et CH(Et)CH(Me)SEt
Et CH(Et)CH(Me)S(O)Et
Et CH(Et)CH(Me)S(O)₂Et
Et CH(Et)CH(Et)SMe
Et CH(Et)CH(Et)S(O)Me
Et CH(Et)CH(Et)S(O)₂Me
Et CH(Et)CH(Et)SEt
Et CH(Et)CH(Et)S(O)Et
Et CH(Et)CH(Et)S(O)₂Et
Et CH=CHSMe
Et CH₂CH(SMe)₂
Et CH₂CH₂SC(O)Me
Et C(CH₂)CH₂C(O)OH
Et C(=NOMe)Me
Et C(=NOMe)Et
Et C(=NOMe)Pr-n
Et C(=NOEt)Me
Et C(=NOPr-n)Me
Et C(=NOPr-i)Me
Et C(=NOBu-n)Me
Et C(=NOCH₂Ph)Me
Et C(=NOMe)C(=NOMe)Me
Et C(=NOMe)CH₂OCH₂CF₃
Et C(=NOMe)CH₂SMe
Et C(=NOMe)CH₂S(O)Me
Et C(=NOMe)CH₂S(O)₂Me
Et C(=NOMe)CH₂SEt
Et C(=NOMe)CH₂S(O)Et
Et C(=NOMe)CH₂S(O)₂Et
Et C(=NOMe)CH₂SCF₃
Et C(=NOMe)CH₂S(O)CF₃
Et C(=NOMe)CH₂S(O)₂CF₃
Et C(=NOMe)CH₂SCH₂CF₃
Et C(=NOMe)CH₂S(O)CH₂CF₃
Et C(=NOMe)CH₂S(O)₂CH₂CF₃
Et C(=NOEt)CH₂SMe
Et C(=NOEt)CH₂S(O)Me
Et C(=NOEt)CH₂S(O)₂Me
Et C(=NOPr-n)CH₂SMe
Et C(=NOPr-n)CH₂S(O)Me
Et C(=NOPr-n)CH₂S(O)₂Me
Et C(=NOPr-i)CH₂SMe
Et C(=NOPr-i)CH₂S(O)Me
Et C(=NOPr-i)CH₂S(O)₂Me
Et C(=NOBu-n)CH₂SMe
Et C(=NOBu-n)CH₂S(O)Me
Et C(=NOBu-n)CH₂S(O)₂Me
Et C(=NOCH₂Ph)CH₂SMe
Et C(=NOCH₂Ph)CH₂S(O)Me
Et C(=NOCH₂Ph)CH₂S(O)₂Me
Et C(=NOCH₂CH=CH₂)CH₂SMe
Et C(=NOCH₂OMe)CH₂SMe
Et C(=NOCH₂CH₂OMe)CH₂SMe
Et C{=NOCH₂CH₂Si(Me)₃}CH₂SMe
Et CH₂CH(=NOMe)
Et CH₂C(=NOMe)Me
Et CH₂C(=NOMe)Et
Et CH₂C(=NOMe)Pr-n
Et CH₂C(=NOMe)Pr-i
Et CH₂C(=NOMe)Bu-n
Et CH₂C(=NOMe)Bu-i
Et CH₂C(=NOMe)Bu-s
Et CH₂C(=NOMe)Bu-t
Et CH₂C(=NOMe)CF₃
Et CH₂C(=NOCH₃)CH₂SCH₃
Et CH(SMe)C(=NOMe)Me
Et CH{S(O)Me}C(=NOMe)Me
Et CH{S(O)₂Me}C(=NOMe)Me
Et CH(SEt)C(=NOMe)Me
Et CH{S(O)Et}C(=NOMe)Me
Et CH{S(O)₂Et}C(=NOMe)Me
Et CH₂NH₂
Et CH₂NMe₂
Et CH₂NHC(O)Me
Et CH₂NHC(O)CF₃
Et CH₂NHC(O)CH₂OMe
Et CH₂NHC(O)CH₂SMe
Et CH₂NHC(O)OMe
Et CH₂NHC(O)OBu-t
Et CH₂NHSO₂Me
Et CH₂NHSO₂NMe₂
Et CH₂NHSO₂CF₃
Et CH₂N(Me)C(O)Me
Et CH₂N(Me)C(O)OMe
Et CH₂N(Me)C(O)OBu-t
Et CH₂N(Me)SO₂Me
Et CH(Me)NHC(O)OBu-t
Et CH(CH₂SMe)NH₂
Et CH(CH₂SMe)NHC(O)Me
Et CH(CH₂SMe)NHC(O)OMe
Et CH(CH₂SMe)NHC(O)OBu-t
Et CH(CH₂SMe)NHSO₂Me
Et CH₂NHC(O)NHMe
Et CH₂NHC(O)NHEt
Et CH₂NHC(O)NHPr-n
Et CH₂NHC(O)NHPr-i
Et CH₂NHC(O)NHPr-c
Et CH₂NHC(S)NHMe
Et CH₂NHC(S)NHEt
Et CH₂NHC(S)NHPr-n
Et CH₂NHC(S)NHPr-i
Et CH₂NHC(S)NHPr-c
Et CH₂CH₂NHC(O)OBu-t
Et CH₂P(O)(OMe)₂
Et CH₂P(O)(OEt)₂
Et SMe
Et OBu-t
Et O{D2-108(4-NO₂)}
Et NH₂
Et NHCH₂SMe
Et NHCH₂CH₂SMe
Et N(Me)CH₂SMe
Et N(Me)CH₂CH₂SMe
Et NHCH₂CH₂CH₂SMe
Et NHMe
Et NHEt
Et NPr-n
Et NHPr-i
Et NHCH₂C(O)OMe
Et NHCH₂CF₃
Et N(Me)CH₂CF₃
Et NHC(O)OEt
Et NHC(O)CCl₃
Et NHC(O)CH₂SMe
Et N(CH₂CH₃)C(O)CH₂SCH₃
Et NHS(O)₂(D2-108a)
Et NHPh
Et NH(D2-1a)
Et NH(D2-2a)
Et NH(D2-2b)
Et NH(D2-4a)
Et NH{D2-4b}
Et NH(D2-5a)
Et NH(D2-5b)
Et NH(D2-5c)
Et NH(D2-6a)
Et NH(D2-6b)
Et NH(D2-6c)
Et NH(D2-7a)
Et NH(D2-8a)
Et NH(D2-8b)
Et NH(D2-8c)
Et NH(D2-9a)
Et NH(D2-9b)
Et NH(D2-9c)
Et NH(D2-10a)
Et NH(D2-10b)
Et NH(D2-10c)
Et NH(D2-11a)
Et NH(D2-12a)
Et NH(D2-12b)
Et NH(D2-12c)
Et NH(D2-13a)
Et NH(D2-13b)
Et NH(D2-14a)
Et NH(D2-14b)
Et NH(D2-15a)
Et NH(D2-15b)
Et NH(D2-16a)
Et NH(D2-17a)
Et NH(D2-18a)
Et NH(D2-19a)
Et NH(D2-20a)
Et NH(D2-21a)
Et NH(D2-21b)
Et NH(D2-22a)
Et NH(D2-23a)
Et NH(D2-23b)
Et NH(D2-24a)
Et NH(D2-25a)
Et NH(D2-26a)
Et NH(D2-27a)
Et NH(D2-28a)
Et NH(D2-29a)
Et NH(D2-30a)
Et NH(D2-31a)
Et NH(D2-32a)
Et NH(D2-33a)
Et NH(D2-34a)
Et NH(D2-35a)
Et NH(D2-35b)
Et NH(D2-36a)
Et NH(D2-37a)
Et NH(D2-38a)
Et NH(D2-39a)
Et NH(D2-40a)
Et NH(D2-40b)
Et NH(D2-40c)
Et NH(D2-41a)
Et NH(D2-42a)
Et NH(D2-43a)
Et NH(D2-45a)
Et NH(D2-49a)
Et NH(D2-51a)
Et NH(D2-59a)
Et NH(D2-61a)
Et NH(D2-79a)
Et NH(D2-80a)
Et NH{D2-108b(2-Cl)}
Et NH{D2-108b(3-Cl)}
Et NH{D2-108b(4-Cl)}
Et NH{D2-108b(2-Me)}
Et NH{D2-108b(3-Me)}
Et NH{D2-108b(4-Me)}
Et N(Me)Ph
Et N(Me)(D2-1a)
Et N(Me)(D2-2a)
Et N(Me)(D2-2b)
Et N(Me)(D2-4a)
Et N(Me){D2-4b}
Et N(Me)(D2-5a)
Et N(Me)(D2-5b)
Et N(Me)(D2-5c)
Et N(Me)(D2-6a)
Et N(Me)(D2-6b)
Et N(Me)(D2-6c)
Et N(Me)(D2-7a)
Et N(Me)(D2-8a)
Et N(Me)(D2-8b)
Et N(Me)(D2-8c)
Et N(Me)(D2-9a)
Et N(Me)(D2-9b)
Et N(Me)(D2-9c)
Et N(Me)(D2-10a)
Et N(Me)(D2-10b)
Et N(Me)(D2-10c)
Et N(Me)(D2-11a)
Et N(Me)(D2-12a)
Et N(Me)(D2-12b)
Et N(Me)(D2-12c)
Et N(Me)(D2-13a)
Et N(Me)(D2-13b)
Et N(Me)(D2-14a)
Et N(Me)(D2-14b)
Et N(Me)(D2-15a)
Et N(Me)(D2-15b)
Et N(Me)(D2-16a)
Et N(Me)(D2-17a)
Et N(Me)(D2-18a)
Et N(Me)(D2-19a)
Et N(Me)(D2-20a)
Et N(Me)(D2-21a)
Et N(Me)(D2-21b)
Et N(Me)(D2-22a)
Et N(Me)(D2-23a)
Et N(Me)(D2-23b)
Et N(Me)(D2-24a)
Et N(Me)(D2-25a)
Et N(Me)(D2-26a)
Et N(Me)(D2-27a)
Et N(Me)(D2-28a)
Et N(Me)(D2-29a)
Et N(Me)(D2-30a)
Et N(Me)(D2-31a)
Et N(Me)(D2-32a)
Et N(Me)(D2-33a)
Et N(Me)(D2-34a)
Et N(Me)(D2-35a)
Et N(Me)(D2-35b)
Et N(Me)(D2-36a)
Et N(Me)(D2-37a)
Et N(Me)(D2-38a)
Et N(Me)(D2-39a)
Et N(Me)(D2-40a)
Et N(Me)(D2-40b)
Et N(Me)(D2-40c)
Et N(Me)(D2-41a)
Et N(Me)(D2-42a)
Et N(Me)(D2-43a)
Et N(Me)(D2-45a)
Et N(Me)(D2-49a)
Et N(Me)(D2-51a)
Et N(Me)(D2-59a)
Et N(Me)(D2-61a)
Et N(Me)(D2-79a)
Et N(Me)(D2-80a)
Et N(Me){D2-108b(2-Cl)}
Et N(Me){D2-108b(3-Cl)}
Et N(Me){D2-108b(4-Cl)}
Et N(Me){D2-108b(2-Me)}
Et N(Me){D2-108b(3-Me)}
Et N(Me){D2-108b(4-Me)}
Et D2-4a
Et D2-9b
Et D2-19a
Et D2-32b(2-Br)
Et D2-33a
Et D2-33b(2-OMe)
Et D2-33b(6-CN)
Et D2-34a
Et D2-35b
Et D2-38b(4-SMe)
Et D2-39b(5-Me)
Et D2-81a
Et D2-81b
Et D2-82a
Et D2-82b
Et D2-87a
Et D2-103b
Et D2-103c
Et D2-103d
Et D2-103e
Et D2-103f
Et D2-103g
Et D2-103h
Et D2-103i
Et D2-108b(2-Cl)
Et D2-108b(3-Cl)
Et D2-108b(4-Cl)
Et D2-108b(2-SMe)
Et D2-108b(3-SMe)
Et D2-108b(4-SMe)
Et D2-108b(3-SCF₃)
Et D2-108b(3,4-OCF₂O-)
Et CH₂(D2-2a)
Et CH₂(D2-28a)
Et CH₂(D2-32a)
Et CH₂(D2-33a)
Et CH₂{D2-33b(6-Cl)}
Et CH₂(D2-34a)
Et CH₂(D2-87a)
Et CH₂(D2-93a)
Et CH₂(D2-98a)
Et CH₂{D2-108b(2,3-OCH₂O-)}
n-Pr CH(Me)SMe
n-Pr CH(Me)S(O)Me
n-Pr CH(Me)S(O)₂Me
n-Pr CH(Me)SEt
n-Pr CH(Me)S(O)Et
n-Pr CH(Me)S(O)₂Et
n-Pr CH₂CH₂SMe
n-Pr CH₂CH₂S(O)Me
n-Pr CH₂CH₂S(O)₂Me
n-Pr CH(Me)CH₂SMe
n-Pr CH(Me)CH₂S(O)Me
n-Pr CH(Me)CH₂S(O)₂Me
n-Pr OBu-t
i-Pr CH(Me)SMe
i-Pr CH(Me)S(O)Me
i-Pr CH(Me)S(O)₂Me
i-Pr CH(Me)SEt
i-Pr CH(Me)S(O)Et
i-Pr CH(Me)S(O)₂Et
i-Pr CH₂CH₂SMe
i-Pr CH₂CH₂S(O)Me
i-Pr CH₂CH₂S(O)₂Me
i-Pr CH(Me)CH₂SMe
i-Pr CH(Me)CH₂S(O)Me
i-Pr CH(Me)CH₂S(O)₂Me
i-Pr OBu-t
CH₂Pr-c CH(Me)SMe
CH₂Pr-c CH(Me)S(O)Me
CH₂Pr-c CH(Me)S(O)₂Me
CH₂Pr-c CH(Me)SEt
CH₂Pr-c CH(Me)S(O)Et
CH₂Pr-c CH(Me)S(O)₂Et
CH₂Pr-c CH₂CH₂SMe
CH₂Pr-c CH₂CH₂S(O)Me
CH₂Pr-c CH₂CH₂S(O)₂Me
CH₂Pr-c CH(Me)CH₂SMe
CH₂Pr-c CH(Me)CH₂S(O)Me
CH₂Pr-c CH(Me)CH₂S(O)₂Me
CH₂Pr-c OBu-t
CH₂CH=CH₂ CH(Me)SMe
CH₂CH=CH₂ CH(Me)S(O)Me
CH₂CH=CH₂ CH(Me)S(O)₂Me
CH₂CH=CH₂ CH(Me)SEt
CH₂CH=CH₂ CH(Me)S(O)Et
CH₂CH=CH₂ CH(Me)S(O)₂Et
CH₂CH=CH₂ CH₂CH₂SMe
CH₂CH=CH₂ CH₂CH₂S(O)Me
CH₂CH=CH₂ CH₂CH₂S(O)₂Me
CH₂CH=CH₂ CH(Me)CH₂SMe
CH₂CH=CH₂ CH(Me)CH₂S(O)Me
CH₂CH=CH₂ CH(Me)CH₂S(O)₂Me
CH₂C≡CH CH(Me)SMe
CH₂C≡CH CH(Me)S(O)Me
CH₂C≡CH CH(Me)S(O)₂Me
CH₂C≡CH CH(Me)SEt
CH₂C≡CH CH(Me)S(O)Et
CH₂C≡CH CH(Me)S(O)₂Et
CH₂C≡CH CH₂CH₂SMe
CH₂C≡CH CH₂CH₂S(O)Me
CH₂C≡CH CH₂CH₂S(O)₂Me
CH₂C≡CH CH(Me)CH₂SMe
CH₂C≡CH CH(Me)CH₂S(O)Me
CH₂C≡CH CH(Me)CH₂S(O)₂Me
CH₂OMe CH(Me)SMe
CH₂OMe CH(Me)S(O)Me
CH₂OMe CH(Me)S(O)₂Me
CH₂OMe CH(Me)SEt
CH₂OMe CH(Me)S(O)Et
CH₂OMe CH(Me)S(O)₂Et
CH₂OMe CH₂CH₂SMe
CH₂OMe CH₂CH₂S(O)Me
CH₂OMe CH₂CH₂S(O)₂Me
CH₂OMe CH(Me)CH₂SMe
CH₂OMe CH(Me)CH₂S(O)Me
CH₂OMe CH(Me)CH₂S(O)₂Me
CH₂OEt CH(Me)SEt
CH₂OEt CH(Me)S(O)Et
CH₂OEt CH(Me)S(O)₂Et
CH₂CH₂OMe CH(Me)SEt
CH₂CH₂OMe CH(Me)S(O)Et
CH₂CH₂OMe CH(Me)S(O)₂Et
CH₂CN CH(Me)SMe
CH₂CN CH(Me)S(O)Me
CH₂CN CH(Me)S(O)₂Me
CH₂CN CH(Me)SEt
CH₂CN CH(Me)S(O)Et
CH₂CN CH(Me)S(O)₂Et
CH₂CN CH₂CH₂SMe
CH₂CN CH₂CH₂S(O)Me
CH₂CN CH₂CH₂S(O)₂Me
CH₂CN CH(Me)CH₂SMe
CH₂CN CH(Me)CH₂S(O)Me
CH₂CN CH(Me)CH₂S(O)₂Me
CH₂C(O)OMe CH₂SMe
CH₂C(O)OMe CH₂S(O)Me
CH₂C(O)OMe CH₂S(O)₂Me
CH₂C(O)OMe CH₂SEt
CH₂C(O)OMe CH₂S(O)Et
CH₂C(O)OMe CH₂S(O)₂Et
CH₂C(O)OMe CH₂SPr-n
CH₂C(O)OMe CH₂S(O)Pr-n
CH₂C(O)OMe CH₂S(O)₂Pr-n
CH₂C(O)OMe CH₂SPr-i
CH₂C(O)OMe CH₂S(O)Pr-i
CH₂C(O)OMe CH₂S(O)₂Pr-i
CH₂C(O)OMe CH₂SPr-c
CH₂C(O)OMe CH₂S(O)Pr-c
CH₂C(O)OMe CH₂S(O)₂Pr-c
CH₂C(O)OMe CH₂SCH₂CH=CH₂
CH₂C(O)OMe CH₂S(O)CH₂CH=CH₂
CH₂C(O)OMe CH₂S(O)₂CH₂CH=CH₂
CH₂C(O)OMe CH₂SCH₂C≡CH
CH₂C(O)OMe CH₂S(O)CH₂C≡CH
CH₂C(O)OMe CH₂S(O)₂CH₂C≡CH
CH₂C(O)OMe CH₂SCH₂CF₃
CH₂C(O)OMe CH₂S(O)CH₂CF₃
CH₂C(O)OMe CH₂S(O)₂CH₂CF₃
CH₂C(O)OMe CH₂SCH₂CH(OMe)₂
CH₂C(O)OMe CH₂SCH₂CH(=NOMe)
CH₂C(O)OMe CH(Me)SMe
CH₂C(O)OMe CH(Me)S(O)Me
CH₂C(O)OMe CH(Me)S(O)₂Me
CH₂C(O)OMe CH(Me)SEt
CH₂C(O)OMe CH(Me)S(O)Et
CH₂C(O)OMe CH(Me)S(O)₂Et
CH₂C(O)OMe CH(Me)S(=NCN)Et
CH₂C(O)OMe CH(Me)S(O)(=NCN)Et
CH₂C(O)OMe CH(Me)SPr-n
CH₂C(O)OMe CH(Me)S(O)Pr-n
CH₂C(O)OMe CH(Me)S(O)₂Pr-n
CH₂C(O)OMe CH(Me)SPr-i
CH₂C(O)OMe CH(Me)S(O)Pr-i
CH₂C(O)OMe CH(Me)S(O)₂Pr-i
CH₂C(O)OMe CH(Me)SBu-t
CH₂C(O)OMe CH(Me)S(O)Bu-t
CH₂C(O)OMe CH(Me)S(O)₂Bu-t
CH₂C(O)OMe CH(Me)SCH₂Pr-c
CH₂C(O)OMe CH(Me)S(O)CH₂Pr-c
CH₂C(O)OMe CH(Me)S(O)₂CH₂Pr-c
CH₂C(O)OMe CH(Me)SCH₂OMe
CH₂C(O)OMe CH(Me)SCH₂SMe
CH₂C(O)OMe CH(Me)S(O)CH₂SMe
CH₂C(O)OMe CH(Me)S(O)₂CH₂SMe
CH₂C(O)OMe CH(Me)SCH₂C=CH₂
CH₂C(O)OMe CH(Me)S(O)CH₂C=CH₂
CH₂C(O)OMe CH(Me)S(O)₂CH₂C=CH₂
CH₂C(O)OMe CH(Me)SCH₂C≡CH
CH₂C(O)OMe CH(Me)S(O)CH₂C≡CH
CH₂C(O)OMe CH(Me)S(O)₂CH₂C≡CH
CH₂C(O)OMe CH(Me)SCH₂C(O)NHMe
CH₂C(O)OMe CH(Me)S(O)CH₂C(O)NHMe
CH₂C(O)OMe CH(Me)S(O)₂CH₂C(O)NHMe
CH₂C(O)OMe CH(Me)SCH₂C(O)OMe
CH₂C(O)OMe CH(Me)S(O)CH₂C(O)OMe
CH₂C(O)OMe CH(Me)S(O)₂CH₂C(O)OMe
CH₂C(O)OMe CH(Me)SCH₂CH₂CH₂Cl
CH₂C(O)OMe CH(Me)S(O)CH₂CH₂CH₂Cl
CH₂C(O)OMe CH(Me)S(O)₂CH₂CH₂CH₂Cl
CH₂C(O)OMe CH(Me)SCH₂CF₃
CH₂C(O)OMe CH(Me)S(O)CH₂CF₃
CH₂C(O)OMe CH(Me)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Me)SCH₂Ph
CH₂C(O)OMe CH(Me)S(O)CH₂Ph
CH₂C(O)OMe CH(Me)S(O)₂CH₂Ph
CH₂C(O)OMe CH(Me)SCH₂(D2-34a)
CH₂C(O)OMe H(Me)S(O)CH₂(D2-34a)
CH₂C(O)OMe H(Me)S(O)₂CH₂(D2-34a)
CH₂C(O)OMe CH(CH₃)SCH₂Si(CH₃)₃
CH₂C(O)OMe CH(Me)SCN
CH₂C(O)OMe CH(Me)SCH₂CN
CH₂C(O)OMe CH(Me)SC(O)Me
CH₂C(O)OMe CH(Me)S(D2-12a)
CH₂C(O)OMe CH(Me)S(D2-32a)
CH₂C(O)OMe CH(Me)S{D2-32b(3-NO₂)}
CH₂C(O)OMe CH(Me)S{D2-32b(3-CF₃)}
CH₂C(O)OMe CH(Me)S(D2-37a)
CH₂C(O)OMe CH(Me)S(D2-51a)
CH₂C(O)OMe CH(Et)SMe
CH₂C(O)OMe CH(Et)S(O)Me
CH₂C(O)OMe CH(Et)S(O)₂Me
CH₂C(O)OMe CH(Et)SEt
CH₂C(O)OMe CH(Et)S(O)Et
CH₂C(O)OMe CH(Et)S(O)₂Et
CH₂C(O)OMe CH(Et)SCH₂CF₃
CH₂C(O)OMe CH(Et)S(O)CH₂CF₃
CH₂C(O)OMe CH(Et)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Pr-n)SMe
CH₂C(O)OMe CH(Pr-n)S(O)Me
CH₂C(O)OMe CH(Pr-n)S(O)₂Me
CH₂C(O)OMe CH(Pr-n)SEt
CH₂C(O)OMe CH(Pr-n)S(O)Et
CH₂C(O)OMe CH(Pr-n)S(O)₂Et
CH₂C(O)OMe CH(Pr-n)S(=NCN)Et
CH₂C(O)OMe CH(Pr-n)S(O)(=NCN)Et
CH₂C(O)OMe CH(Pr-n)SPr-n
CH₂C(O)OMe CH(Pr-n)S(O)Pr-n
CH₂C(O)OMe CH(Pr-n)S(O)₂Pr-n
CH₂C(O)OMe CH(Pr-n)SPr-i
CH₂C(O)OMe CH(Pr-n)S(O)Pr-i
CH₂C(O)OMe CH(Pr-n)S(O)₂Pr-i
CH₂C(O)OMe CH(Pr-n)SPr-c
CH₂C(O)OMe CH(Pr-n)S(O)Pr-c
CH₂C(O)OMe CH(Pr-n)S(O)₂Pr-c
CH₂C(O)OMe CH(Pr-n)SCH₂CF₃
CH₂C(O)OMe CH(Pr-n)S(O)CH₂CF₃
CH₂C(O)OMe CH(Pr-n)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Pr-i)SMe
CH₂C(O)OMe CH(Pr-i)S(O)Me
CH₂C(O)OMe CH(Pr-i)S(O)₂Me
CH₂C(O)OMe CH(Pr-i)SEt
CH₂C(O)OMe CH(Pr-i)S(O)Et
CH₂C(O)OMe CH(Pr-i)S(O)₂Et
CH₂C(O)OMe CH(Pr-i)S(=NCN)Et
CH₂C(O)OMe CH(Pr-i)S(O)(=NCN)Et
CH₂C(O)OMe CH(Pr-i)SPr-n
CH₂C(O)OMe CH(Pr-i)S(O)Pr-n
CH₂C(O)OMe CH(Pr-i)S(O)₂Pr-n
CH₂C(O)OMe CH(Pr-i)SPr-i
CH₂C(O)OMe CH(Pr-i)S(O)Pr-i
CH₂C(O)OMe CH(Pr-i)S(O)₂Pr-i
CH₂C(O)OMe CH(Pr-i)SPr-c
CH₂C(O)OMe CH(Pr-i)S(O)Pr-c
CH₂C(O)OMe CH(Pr-i)S(O)₂Pr-c
CH₂C(O)OMe CH(Pr-i)SCH₂CF₃
CH₂C(O)OMe CH(Pr-i)S(O)CH₂CF₃
CH₂C(O)OMe CH(Pr-i)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Pr-c)SMe
CH₂C(O)OMe CH(Pr-c)S(O)Me
CH₂C(O)OMe CH(Pr-c)S(O)₂Me
CH₂C(O)OMe CH(Pr-c)SEt
CH₂C(O)OMe CH(Pr-c)S(O)Et
CH₂C(O)OMe CH(Pr-c)S(O)₂Et
CH₂C(O)OMe CH(Pr-c)S(=NCN)Et
CH₂C(O)OMe CH(Pr-c)S(O)(=NCN)Et
CH₂C(O)OMe CH(Pr-c)SPr-n
CH₂C(O)OMe CH(Pr-c)S(O)Pr-n
CH₂C(O)OMe CH(Pr-c)S(O)₂Pr-n
CH₂C(O)OMe CH(Pr-c)SPr-i
CH₂C(O)OMe CH(Pr-c)S(O)Pr-i
CH₂C(O)OMe CH(Pr-c)S(O)₂Pr-i
CH₂C(O)OMe CH(Pr-c)SPr-c
CH₂C(O)OMe CH(Pr-c)S(O)Pr-c
CH₂C(O)OMe CH(Pr-c)S(O)₂Pr-c
CH₂C(O)OMe CH(Pr-c)SCH₂CF₃
CH₂C(O)OMe CH(Pr-c)S(O)CH₂CF₃
CH₂C(O)OMe CH(Pr-c)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Bu-n)SMe
CH₂C(O)OMe CH(Bu-n)S(O)Me
CH₂C(O)OMe CH(Bu-n)S(O)₂Me
CH₂C(O)OMe CH(Bu-n)SEt
CH₂C(O)OMe CH(Bu-n)S(O)Et
CH₂C(O)OMe CH(Bu-n)S(O)₂Et
CH₂C(O)OMe CH(Bu-n)S(=NCN)Et
CH₂C(O)OMe CH(Bu-n)S(O)(=NCN)Et
CH₂C(O)OMe CH(Bu-n)SPr-n
CH₂C(O)OMe CH(Bu-n)S(O)Pr-n
CH₂C(O)OMe CH(Bu-n)S(O)₂Pr-n
CH₂C(O)OMe CH(Bu-n)SPr-i
CH₂C(O)OMe CH(Bu-n)S(O)Pr-i
CH₂C(O)OMe CH(Bu-n)S(O)₂Pr-i
CH₂C(O)OMe CH(Bu-n)SPr-c
CH₂C(O)OMe CH(Bu-n)S(O)Pr-c
CH₂C(O)OMe CH(Bu-n)S(O)₂Pr-c
CH₂C(O)OMe CH(Bu-n)SCH₂CF₃
CH₂C(O)OMe CH(Bu-n)S(O)CH₂CF₃
CH₂C(O)OMe CH(Bu-n)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(F)SMe
CH₂C(O)OMe CH(F)S(O)Me
CH₂C(O)OMe CH(F)S(O)₂Me
CH₂C(O)OMe CH(F)SEt
CH₂C(O)OMe CH(F)S(O)Et
CH₂C(O)OMe CH(F)S(O)₂Et
CH₂C(O)OMe CH(F)S(=NCN)Et
CH₂C(O)OMe CH(F)S(O)(=NCN)Et
CH₂C(O)OMe CH(F)SCH₂CF₃
CH₂C(O)OMe CH(F)S(O)CH₂CF₃
CH₂C(O)OMe CH(F)S(O)₂CH₂CF₃
CH₂C(O)OMe C(F)₂SMe
CH₂C(O)OMe C(F)₂S(O)Me
CH₂C(O)OMe C(F)₂S(O)₂Me
CH₂C(O)OMe C(F)₂SEt
CH₂C(O)OMe C(F)₂S(O)Et
CH₂C(O)OMe C(F)₂S(O)₂Et
CH₂C(O)OMe C(F)₂S(=NCN)Et
CH₂C(O)OMe C(F)₂S(O)(=NCN)Et
CH₂C(O)OMe C(F)₂SCH₂CF₃
CH₂C(O)OMe C(F)₂S(O)CH₂CF₃
CH₂C(O)OMe C(F)₂S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Cl)SMe
CH₂C(O)OMe CH(Cl)S(O)Me
CH₂C(O)OMe CH(Cl)S(O)₂Me
CH₂C(O)OMe CH(Cl)SEt
CH₂C(O)OMe CH(Cl)S(O)Et
CH₂C(O)OMe CH(Cl)S(O)₂Et
CH₂C(O)OMe CH(Cl)S(=NCN)Et
CH₂C(O)OMe CH(Cl)S(O)(=NCN)Et
CH₂C(O)OMe CH(Cl)SCH₂CF₃
CH₂C(O)OMe CH(Cl)S(O)CH₂CF₃
CH₂C(O)OMe CH(Cl)S(O)₂CH₂CF₃
CH₂C(O)OMe C(Cl)₂SMe
CH₂C(O)OMe C(Cl)₂S(O)Me
CH₂C(O)OMe C(Cl)₂S(O)₂Me
CH₂C(O)OMe C(Cl)₂SEt
CH₂C(O)OMe C(Cl)₂S(O)Et
CH₂C(O)OMe C(Cl)₂S(O)₂Et
CH₂C(O)OMe C(Cl)₂S(=NCN)Et
CH₂C(O)OMe C(Cl)₂S(O)(=NCN)Et
CH₂C(O)OMe C(Cl)₂SCH₂CF₃
CH₂C(O)OMe C(Cl)₂S(O)CH₂CF₃
CH₂C(O)OMe C(Cl)₂S(O)₂CH₂CF₃
CH₂C(O)OMe CH(Br)SMe
CH₂C(O)OMe CH(Br)S(O)Me
CH₂C(O)OMe CH(Br)S(O)₂Me
CH₂C(O)OMe CH(Br)SEt
CH₂C(O)OMe CH(Br)S(O)Et
CH₂C(O)OMe CH(Br)S(O)₂Et
CH₂C(O)OMe CH(Br)S(=NCN)Et
CH₂C(O)OMe CH(Br)S(O)(=NCN)Et
CH₂C(O)OMe CH(Br)SCH₂CF₃
CH₂C(O)OMe CH(Br)S(O)CH₂CF₃
CH₂C(O)OMe CH(Br)S(O)₂CH₂CF₃
CH₂C(O)OMe CH(I)SMe
CH₂C(O)OMe CH(I)S(O)Me
CH₂C(O)OMe CH(I)S(O)₂Me
CH₂C(O)OMe CH(I)SEt
CH₂C(O)OMe CH(I)S(O)Et
CH₂C(O)OMe CH(I)S(O)₂Et
CH₂C(O)OMe CH(I)S(=NCN)Et
CH₂C(O)OMe CH(I)S(O)(=NCN)Et
CH₂C(O)OMe CH(I)SCH₂CF₃
CH₂C(O)OMe CH(I)S(O)CH₂CF₃
CH₂C(O)OMe CH(I)S(O)₂CH₂CF₃
CH₂C(O)OMe CH{OC(O)Me}SMe
CH₂C(O)OMe CH{OC(O)Me}S(O)Me
CH₂C(O)OMe CH{OC(O)Me}S(O)₂Me
CH₂C(O)OMe CH{OC(O)OMe}SEt
CH₂C(O)OMe CH{OC(O)OMe}S(O)Et
CH₂C(O)OMe CH{OC(O)OMe}S(O)₂Et
CH₂C(O)OMe CH{OC(O)OMe}S(=NCN)Et
CH₂C(O)OMe CH{OC(O)OMe}S(O)(=NCN)Et
CH₂C(O)OMe CH{OC(O)OEt}SMe
CH₂C(O)OMe CH{OC(O)OEt}S(O)Me
CH₂C(O)OMe CH{OC(O)OEt}S(O)₂Me
CH₂C(O)OMe CH{OC(O)OEt}SEt
CH₂C(O)OMe CH{OC(O)OEt}S(O)Et
CH₂C(O)OMe CH{OC(O)OEt}S(O)₂Et
CH₂C(O)OMe CH{OC(O)OEt}S(=NCN)Et
CH₂C(O)OMe CH{OC(O)OEt}S(O)(=NCN)Et
CH₂C(O)OMe CH(OMe)SMe
CH₂C(O)OMe CH(OMe)S(O)Me
CH₂C(O)OMe CH(OMe)S(O)₂Me
CH₂C(O)OMe CH(OMe)SEt
CH₂C(O)OMe CH(OMe)S(O)Et
CH₂C(O)OMe CH(OMe)S(O)₂Et
CH₂C(O)OMe CH(OMe)S(=NCN)Et
CH₂C(O)OMe CH(OMe)S(O)(=NCN)Et
CH₂C(O)OMe CH(OEt)SMe
CH₂C(O)OMe CH(OEt)S(O)Me
CH₂C(O)OMe CH(OEt)S(O)₂Me
CH₂C(O)OMe CH(OEt)SEt
CH₂C(O)OMe CH(OEt)S(O)Et
CH₂C(O)OMe CH(OEt)S(O)₂Et
CH₂C(O)OMe CH(OEt)S(=NCN)Et
CH₂C(O)OMe CH(OEt)S(O)(=CN)Et
CH₂C(O)OMe CH(SMe)₂
CH₂C(O)OMe CH(SMe)S(O)Me
CH₂C(O)OMe CH(SMe)S(O)₂Me
CH₂C(O)OMe CH(SMe)SEt
CH₂C(O)OMe CH(SMe)S(O)Et
CH₂C(O)OMe CH(SMe)S(O)₂Et
CH₂C(O)OMe CH(SMe)S(=NCN)Et
CH₂C(O)OMe CH(SMe)S(O)(=NCN)Et
CH₂C(O)OMe CH(SEt)SMe
CH₂C(O)OMe CH(SEt)S(O)Me
CH₂C(O)OMe CH(SEt)S(O)₂Me
CH₂C(O)OMe CH(SEt)SEt
CH₂C(O)OMe CH(SEt)S(O)Et
CH₂C(O)OMe CH(SEt)S(O)₂Et
CH₂C(O)OMe CH(SEt)S(=NCN)Et
CH₂C(O)OMe CH(SEt)S(O)(=NCN)Et
CH₂C(O)OMe CH(CN)SMe
CH₂C(O)OMe CH(CN)S(O)Me
CH₂C(O)OMe CH(CN)S(O)₂Me
CH₂C(O)OMe CH(CN)SEt
CH₂C(O)OMe CH(CN)S(O)Et
CH₂C(O)OMe CH(CN)S(O)₂Et
CH₂C(O)OMe CH(CN)S(=NCN)Et
CH₂C(O)OMe CH(CN)S(O)(=NCN)Et
CH₂C(O)OMe CH{C(O)OMe}SMe
CH₂C(O)OMe CH{C(O)OMe}S(O)Me
CH₂C(O)OMe CH{C(O)OMe}S(O)₂Me
CH₂C(O)OMe CH{C(O)OMe}SMe
CH₂C(O)OMe CH{C(O)OMe}S(O)Me
CH₂C(O)OMe CH{C(O)OMe}S(O)₂Me
CH₂C(O)OMe CH{C(O)OMe}SEt
CH₂C(O)OMe CH{C(O)OMe}S(O)Et
CH₂C(O)OMe CH{C(O)OMe}S(O)₂Et
CH₂C(O)OMe CH{C(O)OMe}S(=NCN)Et
CH₂C(O)OMe CH{C(O)OMe}S(O)(=NCN)Et
CH₂C(O)OMe CH{C(O)OEt}SMe
CH₂C(O)OMe CH{C(O)OEt}S(O)Me
CH₂C(O)OMe CH{C(O)OEt}S(O)₂Me
CH₂C(O)OMe CH{C(O)OEt}SEt
CH₂C(O)OMe CH{C(O)OEt}S(O)Et
CH₂C(O)OMe CH{C(O)OEt}S(O)₂Et
CH₂C(O)OMe CH{C(O)OEt}S(=NCN)Et
CH₂C(O)OMe CH{C(O)OEt}S(O)(=NCN)Et
CH₂C(O)OMe C(Me)₂SMe
CH₂C(O)OMe C(Me)₂S(O)Me
CH₂C(O)OMe C(Me)₂S(O)₂Me
CH₂C(O)OMe CH₂CH₂SMe
CH₂C(O)OMe CH₂CH₂S(O)Me
CH₂C(O)OMe CH₂CH₂S(O)₂Me
CH₂C(O)OMe CH(Me)CH₂SMe
CH₂C(O)OMe CH(Me)CH₂S(O)Me
CH₂C(O)OMe CH(Me)CH₂S(O)₂Me
CH₂C(O)OMe NHPh
CH₂C(O)OMe NH(D2-1a)
CH₂C(O)OMe NH(D2-2a)
CH₂C(O)OMe NH(D2-2b)
CH₂C(O)OMe NH(D2-5a)
CH₂C(O)OMe NH(D2-5b)
CH₂C(O)OMe NH(D2-5c)
CH₂C(O)OMe NH(D2-6a)
CH₂C(O)OMe NH(D2-6b)
CH₂C(O)OMe NH(D2-6c)
CH₂C(O)OMe NH(D2-7a)
CH₂C(O)OMe NH(D2-8a)
CH₂C(O)OMe NH(D2-8b)
CH₂C(O)OMe NH(D2-8c)
CH₂C(O)OMe NH(D2-9a)
CH₂C(O)OMe NH(D2-9b)
CH₂C(O)OMe NH(D2-9c)
CH₂C(O)OMe NH(D2-10a)
CH₂C(O)OMe NH(D2-10b)
CH₂C(O)OMe NH(D2-10c)
CH₂C(O)OMe NH(D2-11a)
CH₂C(O)OMe NH(D2-12a)
CH₂C(O)OMe NH(D2-12b)
CH₂C(O)OMe NH(D2-12c)
CH₂C(O)OMe NH(D2-13a)
CH₂C(O)OMe NH(D2-13b)
CH₂C(O)OMe NH(D2-14a)
CH₂C(O)OMe NH(D2-14b)
CH₂C(O)OMe NH(D2-15a)
CH₂C(O)OMe NH(D2-15b)
CH₂C(O)OMe NH(D2-16a)
CH₂C(O)OMe NH(D2-17a)
CH₂C(O)OMe NH(D2-18a)
CH₂C(O)OMe NH(D2-19a)
CH₂C(O)OMe NH(D2-20a)
CH₂C(O)OMe NH(D2-21a)
CH₂C(O)OMe NH(D2-21b)
CH₂C(O)OMe NH(D2-22a)
CH₂C(O)OMe NH(D2-23a)
CH₂C(O)OMe NH(D2-23b)
CH₂C(O)OMe NH(D2-24a)
CH₂C(O)OMe NH(D2-25a)
CH₂C(O)OMe NH(D2-26a)
CH₂C(O)OMe NH(D2-27a)
CH₂C(O)OMe NH(D2-28a)
CH₂C(O)OMe NH(D2-29a)
CH₂C(O)OMe NH(D2-30a)
CH₂C(O)OMe NH(D2-31a)
CH₂C(O)OMe NH(D2-32a)
CH₂C(O)OMe NH(D2-33a)
CH₂C(O)OMe NH(D2-34a)
CH₂C(O)OMe NH(D2-35a)
CH₂C(O)OMe NH(D2-35b)
CH₂C(O)OMe NH(D2-36a)
CH₂C(O)OMe NH(D2-37a)
CH₂C(O)OMe NH(D2-38a)
CH₂C(O)OMe NH(D2-39a)
CH₂C(O)OMe NH(D2-40a)
CH₂C(O)OMe NH(D2-40b)
CH₂C(O)OMe NH(D2-40c)
CH₂C(O)OMe NH(D2-41a)
CH₂C(O)OMe NH(D2-42a)
CH₂C(O)OMe NH(D2-43a)
CH₂C(O)OMe NH(D2-45a)
CH₂C(O)OMe NH(D2-49a)
CH₂C(O)OMe NH(D2-51a)
CH₂C(O)OMe NH(D2-59a)
CH₂C(O)OMe NH(D2-61a)
CH₂C(O)OMe NH(D2-79a)
CH₂C(O)OMe NH(D2-80a)
CH₂C(O)OMe NH{D2-108b(2-Cl)}
CH₂C(O)OMe NH{D2-108b(3-Cl)}
CH₂C(O)OMe NH{D2-108b(4-Cl)}
CH₂C(O)OMe NH{D2-108b(2-Me)}
CH₂C(O)OMe NH{D2-108b(3-Me)}
CH₂C(O)OMe NH{D2-108b(4-Me)}
CH₂C(O)OMe N(Me)Ph
CH₂C(O)OMe N(Me)(D2-1a)
CH₂C(O)OMe N(Me)(D2-2a)
CH₂C(O)OMe N(Me)(D2-2b)
CH₂C(O)OMe N(Me)(D2-4a)
CH₂C(O)OMe N(Me)(D2-5a)
CH₂C(O)OMe N(Me)(D2-5b)
CH₂C(O)OMe N(Me)(D2-5c)
CH₂C(O)OMe N(Me)(D2-6a)
CH₂C(O)OMe N(Me)(D2-6b)
CH₂C(O)OMe N(Me)(D2-6c)
CH₂C(O)OMe N(Me)(D2-7a)
CH₂C(O)OMe N(Me)(D2-8a)
CH₂C(O)OMe N(Me)(D2-8b)
CH₂C(O)OMe N(Me)(D2-8c)
CH₂C(O)OMe N(Me)(D2-9a)
CH₂C(O)OMe N(Me)(D2-9b)
CH₂C(O)OMe N(Me)(D2-9c)
CH₂C(O)OMe N(Me)(D2-10a)
CH₂C(O)OMe N(Me)(D2-10b)
CH₂C(O)OMe N(Me)(D2-10c)
CH₂C(O)OMe N(Me)(D2-11a)
CH₂C(O)OMe N(Me)(D2-12a)
CH₂C(O)OMe N(Me)(D2-12b)
CH₂C(O)OMe N(Me)(D2-12c)
CH₂C(O)OMe N(Me)(D2-13a)
CH₂C(O)OMe N(Me)(D2-13b)
CH₂C(O)OMe N(Me)(D2-14a)
CH₂C(O)OMe N(Me)(D2-14b)
CH₂C(O)OMe N(Me)(D2-15a)
CH₂C(O)OMe N(Me)(D2-15b)
CH₂C(O)OMe N(Me)(D2-16a)
CH₂C(O)OMe N(Me)(D2-17a)
CH₂C(O)OMe N(Me)(D2-18a)
CH₂C(O)OMe N(Me)(D2-19a)
CH₂C(O)OMe N(Me)(D2-20a)
CH₂C(O)OMe N(Me)(D2-21a)
CH₂C(O)OMe N(Me)(D2-21b)
CH₂C(O)OMe N(Me)(D2-22a)
CH₂C(O)OMe N(Me)(D2-23a)
CH₂C(O)OMe N(Me)(D2-23b)
CH₂C(O)OMe N(Me)(D2-24a)
CH₂C(O)OMe N(Me)(D2-25a)
CH₂C(O)OMe N(Me)(D2-26a)
CH₂C(O)OMe N(Me)(D2-27a)
CH₂C(O)OMe N(Me)(D2-28a)
CH₂C(O)OMe N(Me)(D2-29a)
CH₂C(O)OMe N(Me)(D2-30a)
CH₂C(O)OMe N(Me)(D2-31a)
CH₂C(O)OMe N(Me)(D2-32a)
CH₂C(O)OMe N(Me)(D2-34a)
CH₂C(O)OMe N(Me)(D2-35a)
CH₂C(O)OMe N(Me)(D2-35b)
CH₂C(O)OMe N(Me)(D2-36a)
CH₂C(O)OMe N(Me)(D2-37a)
CH₂C(O)OMe N(Me)(D2-38a)
CH₂C(O)OMe N(Me)(D2-39a)
CH₂C(O)OMe N(Me)(D2-40a)
CH₂C(O)OMe N(Me)(D2-40b)
CH₂C(O)OMe N(Me)(D2-40c)
CH₂C(O)OMe N(Me)(D2-41a)
CH₂C(O)OMe N(Me)(D2-42a)
CH₂C(O)OMe N(Me)(D2-43a)
CH₂C(O)OMe N(Me)(D2-45a)
CH₂C(O)OMe N(Me)(D2-49a)
CH₂C(O)OMe N(Me)(D2-51a)
CH₂C(O)OMe N(Me)(D2-59a)
CH₂C(O)OMe N(Me)(D2-61a)
CH₂C(O)OMe N(Me)(D2-79a)
CH₂C(O)OMe N(Me)(D2-80a)
CH₂C(O)OMe N(Me){D2-108b(2-Cl)}
CH₂C(O)OMe N(Me){D2-108b(3-Cl)}
CH₂C(O)OMe N(Me){D2-108b(4-Cl)}
CH₂C(O)OMe N(Me){D2-108b(2-Me)}
CH₂C(O)OMe N(Me){D2-108b(3-Me)}
CH₂C(O)OMe N(Me){D2-108b(4-Me)}
CH₂C(O)OEt CH₂SMe
CH₂C(O)OEt CH₂S(O)Me
CH₂C(O)OEt CH₂S(O)₂Me
CH₂C(O)OEt CH₂SEt
CH₂C(O)OEt CH₂S(O)Et
CH₂C(O)OEt CH₂S(O)₂Et
CH₂C(O)OEt CH₂SPr-n
CH₂C(O)OEt CH₂S(O)Pr-n
CH₂C(O)OEt CH₂S(O)₂Pr-n
CH₂C(O)OEt CH₂SPr-i
CH₂C(O)OEt CH₂S(O)Pr-i
CH₂C(O)OEt CH₂S(O)₂Pr-i
CH₂C(O)OEt CH₂SPr-c
CH₂C(O)OEt CH₂S(O)Pr-c
CH₂C(O)OEt CH₂S(O)₂Pr-c
CH₂C(O)OEt CH₂SCH₂CH=CH₂
CH₂C(O)OEt CH₂S(O)CH₂CH=CH₂
CH₂C(O)OEt CH₂S(O)₂CH₂CH=CH₂
CH₂C(O)OEt CH₂SCH₂C≡CH
CH₂C(O)OEt CH₂S(O)CH₂C≡CH
CH₂C(O)OEt CH₂S(O)₂CH₂C≡CH
CH₂C(O)OEt CH₂SCH₂CF₃
CH₂C(O)OEt CH₂S(O)CH₂CF₃
CH₂C(O)OEt CH₂S(O)₂CH₂CF₃
CH₂C(O)OEt CH₂SCH₂CH(OMe)₂
CH₂C(O)OEt CH₂SCH₂CH(=NOMe)
CH₂C(O)OEt CH(Me)SMe
CH₂C(O)OEt CH(Me)S(O)Me
CH₂C(O)OEt CH(Me)S(O)₂Me
CH₂C(O)OEt CH(Me)SEt
CH₂C(O)OEt CH(Me)S(O)Et
CH₂C(O)OEt CH(Me)S(O)₂Et
CH₂C(O)OEt CH(Me)S(=NCN)Et
CH₂C(O)OEt CH(Me)S(O)(=NCN)Et
CH₂C(O)OEt CH(Me)SPr-n
CH₂C(O)OEt CH(Me)S(O)Pr-n
CH₂C(O)OEt CH(Me)S(O)₂Pr-n
CH₂C(O)OEt CH(Me)SPr-i
CH₂C(O)OEt CH(Me)S(O)Pr-i
CH₂C(O)OEt CH(Me)S(O)₂Pr-i
CH₂C(O)OEt CH(Me)SBu-t
CH₂C(O)OEt CH(Me)S(O)Bu-t
CH₂C(O)OEt CH(Me)S(O)₂Bu-t
CH₂C(O)OEt CH(Me)SCH₂Pr-c
CH₂C(O)OEt CH(Me)S(O)CH₂Pr-c
CH₂C(O)OEt CH(Me)S(O)₂CH₂Pr-c
CH₂C(O)OEt CH(Me)SCH₂OMe
CH₂C(O)OEt CH(Me)SCH₂SMe
CH₂C(O)OEt CH(Me)S(O)CH₂SMe
CH₂C(O)OEt CH(Me)S(O)₂CH₂SMe
CH₂C(O)OEt CH(Me)SCH₂C=CH₂
CH₂C(O)OEt CH(Me)S(O)CH₂C=CH₂
CH₂C(O)OEt CH(Me)S(O)₂CH₂C=CH₂
CH₂C(O)OEt CH(Me)SCH₂C≡CH
CH₂C(O)OEt CH(Me)S(O)CH₂C≡CH
CH₂C(O)OEt CH(Me)S(O)₂CH₂C≡CH
CH₂C(O)OEt CH(Me)SCH₂C(O)NHMe
CH₂C(O)OEt CH(Me)S(O)CH₂C(O)NHMe
CH₂C(O)OEt CH(Me)S(O)₂CH₂C(O)NHMe
CH₂C(O)OEt CH(Me)SCH₂C(O)OMe
CH₂C(O)OEt CH(Me)S(O)CH₂C(O)OMe
CH₂C(O)OEt CH(Me)S(O)₂CH₂C(O)OMe
CH₂C(O)OEt CH(Me)SCH₂CH₂CH₂Cl
CH₂C(O)OEt CH(Me)S(O)CH₂CH₂CH₂Cl
CH₂C(O)OEt CH(Me)S(O)₂CH₂CH₂CH₂Cl
CH₂C(O)OEt CH(Me)SCH₂CF₃
CH₂C(O)OEt CH(Me)S(O)CH₂CF₃
CH₂C(O)OEt CH(Me)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Me)SCH₂Ph
CH₂C(O)OEt CH(Me)S(O)CH₂Ph
CH₂C(O)OEt CH(Me)S(O)₂CH₂Ph
CH₂C(O)OEt CH(Me)SCH₂(D2-34a)
CH₂C(O)OEt CH(Me)S(O)CH₂(D2-34a)
CH₂C(O)OEt CH(Me)S(O)₂CH₂(D2-34a)
CH₂C(O)OEt CH(CH₃)SCH₂Si(CH₃)₃
CH₂C(O)OEt CH(Me)SCN
CH₂C(O)OEt CH(Me)SCH₂CN
CH₂C(O)OEt CH(Me)SC(O)Me
CH₂C(O)OEt CH(Me)S(D2-12a)
CH₂C(O)OEt CH(Me)S(D2-32a)
CH₂C(O)OEt CH(Me)S{D2-32b(3-NO₂)}
CH₂C(O)OEt CH(Me)S{D2-32b(3-CF₃)}
CH₂C(O)OEt CH(Me)S(D2-37a)
CH₂C(O)OEt CH(Me)S(D2-51a)
CH₂C(O)OEt CH(Et)SMe
CH₂C(O)OEt CH(Et)S(O)Me
CH₂C(O)OEt CH(Et)S(O)₂Me
CH₂C(O)OEt CH(Et)SEt
CH₂C(O)OEt CH(Et)S(O)Et
CH₂C(O)OEt CH(Et)S(O)₂Et
CH₂C(O)OEt CH(Et)SCH₂CF₃
CH₂C(O)OEt CH(Et)S(O)CH₂CF₃
CH₂C(O)OEt CH(Et)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Pr-n)SMe
CH₂C(O)OEt CH(Pr-n)S(O)Me
CH₂C(O)OEt CH(Pr-n)S(O)₂Me
CH₂C(O)OEt CH(Pr-n)SEt
CH₂C(O)OEt CH(Pr-n)S(O)Et
CH₂C(O)OEt CH(Pr-n)S(O)₂Et
CH₂C(O)OEt CH(Pr-n)S(=NCN)Et
CH₂C(O)OEt CH(Pr-n)S(O)(=NCN)Et
CH₂C(O)OEt CH(Pr-n)SPr-n
CH₂C(O)OEt CH(Pr-n)S(O)Pr-n
CH₂C(O)OEt CH(Pr-n)S(O)₂Pr-n
CH₂C(O)OEt CH(Pr-n)SPr-i
CH₂C(O)OEt CH(Pr-n)S(O)Pr-i
CH₂C(O)OEt CH(Pr-n)S(O)₂Pr-i
CH₂C(O)OEt CH(Pr-n)SPr-c
CH₂C(O)OEt CH(Pr-n)S(O)Pr-c
CH₂C(O)OEt CH(Pr-n)S(O)₂Pr-c
CH₂C(O)OEt CH(Pr-n)SCH₂CF₃
CH₂C(O)OEt CH(Pr-n)S(O)CH₂CF₃
CH₂C(O)OEt CH(Pr-n)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Pr-i)SMe
CH₂C(O)OEt CH(Pr-i)S(O)Me
CH₂C(O)OEt CH(Pr-i)S(O)₂Me
CH₂C(O)OEt CH(Pr-i)SEt
CH₂C(O)OEt CH(Pr-i)S(O)Et
CH₂C(O)OEt CH(Pr-i)S(O)₂Et
CH₂C(O)OEt CH(Pr-i)S(=NCN)Et
CH₂C(O)OEt CH(Pr-i)S(O)(=NCN)Et
CH₂C(O)OEt CH(Pr-i)SPr-n
CH₂C(O)OEt CH(Pr-i)S(O)Pr-n
CH₂C(O)OEt CH(Pr-i)S(O)₂Pr-n
CH₂C(O)OEt CH(Pr-i)SPr-i
CH₂C(O)OEt CH(Pr-i)S(O)Pr-i
CH₂C(O)OEt CH(Pr-i)S(O)₂Pr-i
CH₂C(O)OEt CH(Pr-i)SPr-c
CH₂C(O)OEt CH(Pr-i)S(O)Pr-c
CH₂C(O)OEt CH(Pr-i)S(O)₂Pr-c
CH₂C(O)OEt CH(Pr-i)SCH₂CF₃
CH₂C(O)OEt CH(Pr-i)S(O)CH₂CF₃
CH₂C(O)OEt CH(Pr-i)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Pr-c)SMe
CH₂C(O)OEt CH(Pr-c)S(O)Me
CH₂C(O)OEt CH(Pr-c)S(O)₂Me
CH₂C(O)OEt CH(Pr-c)SEt
CH₂C(O)OEt CH(Pr-c)S(O)Et
CH₂C(O)OEt CH(Pr-c)S(O)₂Et
CH₂C(O)OEt CH(Pr-c)S(=NCN)Et
CH₂C(O)OEt CH(Pr-c)S(O)(=NCN)Et
CH₂C(O)OEt CH(Pr-c)SPr-n
CH₂C(O)OEt CH(Pr-c)S(O)Pr-n
CH₂C(O)OEt CH(Pr-c)S(O)₂Pr-n
CH₂C(O)OEt CH(Pr-c)SPr-i
CH₂C(O)OEt CH(Pr-c)S(O)Pr-i
CH₂C(O)OEt CH(Pr-c)S(O)₂Pr-i
CH₂C(O)OEt CH(Pr-c)SPr-c
CH₂C(O)OEt CH(Pr-c)S(O)Pr-c
CH₂C(O)OEt CH(Pr-c)S(O)₂Pr-c
CH₂C(O)OEt CH(Pr-c)SCH₂CF₃
CH₂C(O)OEt CH(Pr-c)S(O)CH₂CF₃
CH₂C(O)OEt CH(Pr-c)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Bu-n)SMe
CH₂C(O)OEt CH(Bu-n)S(O)Me
CH₂C(O)OEt CH(Bu-n)S(O)₂Me
CH₂C(O)OEt CH(Bu-n)SEt
CH₂C(O)OEt CH(Bu-n)S(O)Et
CH₂C(O)OEt CH(Bu-n)S(O)₂Et
CH₂C(O)OEt CH(Bu-n)S(=NCN)Et
CH₂C(O)OEt CH(Bu-n)S(O)(=NCN)Et
CH₂C(O)OEt CH(Bu-n)SPr-n
CH₂C(O)OEt CH(Bu-n)S(O)Pr-n
CH₂C(O)OEt CH(Bu-n)S(O)₂Pr-n
CH₂C(O)OEt CH(Bu-n)SPr-i
CH₂C(O)OEt CH(Bu-n)S(O)Pr-i
CH₂C(O)OEt CH(Bu-n)S(O)₂Pr-i
CH₂C(O)OEt CH(Bu-n)SPr-c
CH₂C(O)OEt CH(Bu-n)S(O)Pr-c
CH₂C(O)OEt CH(Bu-n)S(O)₂Pr-c
CH₂C(O)OEt CH(Bu-n)SCH₂CF₃
CH₂C(O)OEt CH(Bu-n)S(O)CH₂CF₃
CH₂C(O)OEt CH(Bu-n)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(F)SMe
CH₂C(O)OEt CH(F)S(O)Me
CH₂C(O)OEt CH(F)S(O)₂Me
CH₂C(O)OEt CH(F)SEt
CH₂C(O)OEt CH(F)S(O)Et
CH₂C(O)OEt CH(F)S(O)₂Et
CH₂C(O)OEt CH(F)S(=NCN)Et
CH₂C(O)OEt CH(F)S(O)(=NCN)Et
CH₂C(O)OEt CH(F)SCH₂CF₃
CH₂C(O)OEt CH(F)S(O)CH₂CF₃
CH₂C(O)OEt CH(F)S(O)₂CH₂CF₃
CH₂C(O)OEt C(F)₂SMe
CH₂C(O)OEt C(F)₂S(O)Me
CH₂C(O)OEt C(F)₂S(O)₂Me
CH₂C(O)OEt C(F)₂SEt
CH₂C(O)OEt C(F)₂S(O)Et
CH₂C(O)OEt C(F)₂S(O)₂Et
CH₂C(O)OEt C(F)₂S(=NCN)Et
CH₂C(O)OEt C(F)₂S(O)(=NCN)Et
CH₂C(O)OEt C(F)₂SCH₂CF₃
CH₂C(O)OEt C(F)₂S(O)CH₂CF₃
CH₂C(O)OEt C(F)₂S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Cl)SMe
CH₂C(O)OEt CH(Cl)S(O)Me
CH₂C(O)OEt CH(Cl)S(O)₂Me
CH₂C(O)OEt CH(Cl)SEt
CH₂C(O)OEt CH(Cl)S(O)Et
CH₂C(O)OEt CH(Cl)S(O)₂Et
CH₂C(O)OEt CH(Cl)S(=NCN)Et
CH₂C(O)OEt CH(Cl)S(O)(=NCN)Et
CH₂C(O)OEt CH(Cl)SCH₂CF₃
CH₂C(O)OEt CH(Cl)S(O)CH₂CF₃
CH₂C(O)OEt CH(Cl)S(O)₂CH₂CF₃
CH₂C(O)OEt C(Cl)₂SMe
CH₂C(O)OEt C(Cl)₂S(O)Me
CH₂C(O)OEt C(Cl)₂S(O)₂Me
CH₂C(O)OEt C(Cl)₂SEt
CH₂C(O)OEt C(Cl)₂S(O)Et
CH₂C(O)OEt C(Cl)₂S(O)₂Et
CH₂C(O)OEt C(Cl)₂S(=NCN)Et
CH₂C(O)OEt C(Cl)₂S(O)(=NCN)Et
CH₂C(O)OEt C(Cl)₂SCH₂CF₃
CH₂C(O)OEt C(Cl)₂S(O)CH₂CF₃
CH₂C(O)OEt C(Cl)₂S(O)₂CH₂CF₃
CH₂C(O)OEt CH(Br)SMe
CH₂C(O)OEt CH(Br)S(O)Me
CH₂C(O)OEt CH(Br)S(O)₂Me
CH₂C(O)OEt CH(Br)SEt
CH₂C(O)OEt CH(Br)S(O)Et
CH₂C(O)OEt CH(Br)S(O)₂Et
CH₂C(O)OEt CH(Br)S(=NCN)Et
CH₂C(O)OEt CH(Br)S(O)(=NCN)Et
CH₂C(O)OEt CH(Br)SCH₂CF₃
CH₂C(O)OEt CH(Br)S(O)CH₂CF₃
CH₂C(O)OEt CH(Br)S(O)₂CH₂CF₃
CH₂C(O)OEt CH(I)SMe
CH₂C(O)OEt CH(I)S(O)Me
CH₂C(O)OEt CH(I)S(O)₂Me
CH₂C(O)OEt CH(I)SEt
CH₂C(O)OEt CH(I)S(O)Et
CH₂C(O)OEt CH(I)S(O)₂Et
CH₂C(O)OEt CH(I)S(=NCN)Et
CH₂C(O)OEt CH(I)S(O)(=NCN)Et
CH₂C(O)OEt CH(I)SCH₂CF₃
CH₂C(O)OEt CH(I)S(O)CH₂CF₃
CH₂C(O)OEt CH(I)S(O)₂CH₂CF₃
CH₂C(O)OEt CH{OC(O)Me}SMe
CH₂C(O)OEt CH{OC(O)Me}S(O)Me
CH₂C(O)OEt CH{OC(O)Me}S(O)₂Me
CH₂C(O)OEt CH{OC(O)OMe}SEt
CH₂C(O)OEt CH{OC(O)OMe}S(O)Et
CH₂C(O)OEt CH{OC(O)OMe}S(O)₂Et
CH₂C(O)OEt CH{OC(O)OMe}S(=NCN)Et
CH₂C(O)OEt CH{OC(O)OMe}S(O)(=NCN)Et
CH₂C(O)OEt CH{OC(O)OEt}SMe
CH₂C(O)OEt CH{OC(O)OEt}S(O)Me
CH₂C(O)OEt CH{OC(O)OEt}S(O)₂Me
CH₂C(O)OEt CH{OC(O)OEt}SEt
CH₂C(O)OEt CH{OC(O)OEt}S(O)Et
CH₂C(O)OEt CH{OC(O)OEt}S(O)₂Et
CH₂C(O)OEt CH{OC(O)OEt}S(=NCN)Et
CH₂C(O)OEt CH{OC(O)OEt}S(O)(=NCN)Et
CH₂C(O)OEt CH(OMe)SMe
CH₂C(O)OEt CH(OMe)S(O)Me
CH₂C(O)OEt CH(OMe)S(O)₂Me
CH₂C(O)OEt CH(OMe)SEt
CH₂C(O)OEt CH(OMe)S(O)Et
CH₂C(O)OEt CH(OMe)S(O)₂Et
CH₂C(O)OEt CH(OMe)S(=NCN)Et
CH₂C(O)OEt CH(OMe)S(O)(=NCN)Et
CH₂C(O)OEt CH(OEt)SMe
CH₂C(O)OEt CH(OEt)S(O)Me
CH₂C(O)OEt CH(OEt)S(O)₂Me
CH₂C(O)OEt CH(OEt)SEt
CH₂C(O)OEt CH(OEt)S(O)Et
CH₂C(O)OEt CH(OEt)S(O)₂Et
CH₂C(O)OEt CH(OEt)S(=NCN)Et
CH₂C(O)OEt CH(OEt)S(O)(=NCN)Et
CH₂C(O)OEt CH(SMe)₂
CH₂C(O)OEt CH(SMe)S(O)Me
CH₂C(O)OEt CH(SMe)S(O)₂Me
CH₂C(O)OEt CH(SMe)SEt
CH₂C(O)OEt CH(SMe)S(O)Et
CH₂C(O)OEt CH(SMe)S(O)₂Et
CH₂C(O)OEt CH(SMe)S(=NCN)Et
CH₂C(O)OEt CH(SMe)S(O)(=NCN)Et
CH₂C(O)OEt CH(SEt)SMe
CH₂C(O)OEt CH(SEt)S(O)Me
CH₂C(O)OEt CH(SEt)S(O)₂Me
CH₂C(O)OEt CH(SEt)SEt
CH₂C(O)OEt CH(SEt)S(O)Et
CH₂C(O)OEt CH(SEt)S(O)₂Et
CH₂C(O)OEt CH(SEt)S(=NCN)Et
CH₂C(O)OEt CH(SEt)S(O)(=NCN)Et
CH₂C(O)OEt CH(CN)SMe
CH₂C(O)OEt CH(CN)S(O)Me
CH₂C(O)OEt CH(CN)S(O)₂Me
CH₂C(O)OEt CH(CN)SEt
CH₂C(O)OEt CH(CN)S(O)Et
CH₂C(O)OEt CH(CN)S(O)₂Et
CH₂C(O)OEt CH(CN)S(=NCN)Et
CH₂C(O)OEt CH(CN)S(O)(=NCN)Et
CH₂C(O)OEt CH{C(O)OMe}SMe
CH₂C(O)OEt CH{C(O)OMe}S(O)Me
CH₂C(O)OEt CH{C(O)OMe}S(O)₂Me
CH₂C(O)OEt CH{C(O)OMe}SMe
CH₂C(O)OEt CH{C(O)OMe}S(O)Me
CH₂C(O)OEt CH{C(O)OMe}S(O)₂Me
CH₂C(O)OEt CH{C(O)OMe}SEt
CH₂C(O)OEt CH{C(O)OMe}S(O)Et
CH₂C(O)OEt CH{C(O)OMe}S(O)₂Et
CH₂C(O)OEt CH{C(O)OMe}S(=NCN)Et
CH₂C(O)OEt CH{C(O)OMe}S(O)(=NCN)Et
CH₂C(O)OEt CH{C(O)OEt}SMe
CH₂C(O)OEt CH{C(O)OEt}S(O)Me
CH₂C(O)OEt CH{C(O)OEt}S(O)₂Me
CH₂C(O)OEt CH{C(O)OEt}SEt
CH₂C(O)OEt CH{C(O)OEt}S(O)Et
CH₂C(O)OEt CH{C(O)OEt}S(O)₂Et
CH₂C(O)OEt CH{C(O)OEt}S(=NCN)Et
CH₂C(O)OEt CH{C(O)OEt}S(O)(=NCN)Et
CH₂C(O)OEt C(Me)₂SMe
CH₂C(O)OEt C(Me)₂S(O)Me
CH₂C(O)OEt C(Me)₂S(O)₂Me
CH₂C(O)OEt CH₂CH₂SMe
CH₂C(O)OEt CH₂CH₂S(O)Me
CH₂C(O)OEt CH₂CH₂S(O)₂Me
CH₂C(O)OEt CH(Me)CH₂SMe
CH₂C(O)OEt CH(Me)CH₂S(O)Me
CH₂C(O)OEt CH(Me)CH₂S(O)₂Me
C(O)OMe CH₂SMe
C(O)OMe CH₂S(O)Me
C(O)OMe CH₂S(O)₂Me
C(O)OMe CH₂SEt
C(O)OMe CH₂S(O)Et
C(O)OMe CH₂S(O)₂Et
C(O)OMe CH₂SPr-n
C(O)OMe CH₂S(O)Pr-n
C(O)OMe CH₂S(O)₂Pr-n
C(O)OMe CH₂SPr-i
C(O)OMe CH₂S(O)Pr-i
C(O)OMe CH₂S(O)₂Pr-i
C(O)OMe CH₂SPr-c
C(O)OMe CH₂S(O)Pr-c
C(O)OMe CH₂S(O)₂Pr-c
C(O)OMe CH₂SCH₂CH=CH₂
C(O)OMe CH₂S(O)CH₂CH=CH₂
C(O)OMe CH₂S(O)₂CH₂CH=CH₂
C(O)OMe CH₂SCH₂C≡CH
C(O)OMe CH₂S(O)CH₂C≡CH
C(O)OMe CH₂S(O)₂CH₂C≡CH
C(O)OMe CH₂SCH₂CF₃
C(O)OMe CH₂S(O)CH₂CF₃
C(O)OMe CH₂S(O)₂CH₂CF₃
C(O)OMe CH₂SCH₂CH(OMe)₂
C(O)OMe CH₂SCH₂CH(=NOMe)
C(O)OMe CH(Me)SMe
C(O)OMe CH(Me)S(O)Me
C(O)OMe CH(Me)S(O)₂Me
C(O)OMe CH(Me)SEt
C(O)OMe CH(Me)S(O)Et
C(O)OMe CH(Me)S(O)₂Et
C(O)OMe CH(Me)S(=NCN)Et
C(O)OMe CH(Me)S(O)(=NCN)Et
C(O)OMe CH(Me)SPr-n
C(O)OMe CH(Me)S(O)Pr-n
C(O)OMe CH(Me)S(O)₂Pr-n
C(O)OMe CH(Me)SPr-i
C(O)OMe CH(Me)S(O)Pr-i
C(O)OMe CH(Me)S(O)₂Pr-i
C(O)OMe CH(Me)SBu-t
C(O)OMe CH(Me)S(O)Bu-t
C(O)OMe CH(Me)S(O)₂Bu-t
C(O)OMe CH(Me)SCH₂Pr-c
C(O)OMe CH(Me)S(O)CH₂Pr-c
C(O)OMe CH(Me)S(O)₂CH₂Pr-c
C(O)OMe CH(Me)SCH₂OMe
C(O)OMe CH(Me)SCH₂SMe
C(O)OMe CH(Me)S(O)CH₂SMe
C(O)OMe CH(Me)S(O)₂CH₂SMe
C(O)OMe CH(Me)SCH₂C=CH₂
C(O)OMe CH(Me)S(O)CH₂C=CH₂
C(O)OMe CH(Me)S(O)₂CH₂C=CH₂
C(O)OMe CH(Me)SCH₂C≡CH
C(O)OMe CH(Me)S(O)CH₂C≡CH
C(O)OMe CH(Me)S(O)₂CH₂C≡CH
C(O)OMe CH(Me)SCH₂C(O)NHMe
C(O)OMe CH(Me)S(O)CH₂C(O)NHMe
C(O)OMe CH(Me)S(O)₂CH₂C(O)NHMe
C(O)OMe CH(Me)SCH₂C(O)OMe
C(O)OMe CH(Me)S(O)CH₂C(O)OMe
C(O)OMe CH(Me)S(O)₂CH₂C(O)OMe
C(O)OMe CH(Me)SCH₂CH₂CH₂Cl
C(O)OMe CH(Me)S(O)CH₂CH₂CH₂Cl
C(O)OMe CH(Me)S(O)₂CH₂CH₂CH₂Cl
C(O)OMe CH(Me)SCH₂CF₃
C(O)OMe CH(Me)S(O)CH₂CF₃
C(O)OMe CH(Me)S(O)₂CH₂CF₃
C(O)OMe CH(Me)SCH₂Ph
C(O)OMe CH(Me)S(O)CH₂Ph
C(O)OMe CH(Me)S(O)₂CH₂Ph
C(O)OMe CH(Me)SCH₂(D2-34a)
C(O)OMe CH(Me)S(O)CH₂(D2-34a)
C(O)OMe CH(Me)S(O)₂CH₂(D2-34a)
C(O)OMe CH(CH₃)SCH₂Si(CH₃)₃
C(O)OMe CH(Me)SCN
C(O)OMe CH(Me)SCH₂CN
C(O)OMe CH(Me)SC(O)Me
C(O)OMe CH(Me)S(D2-12a)
C(O)OMe CH(Me)S(D2-32a)
C(O)OMe CH(Me)S{D2-32b(3-NO₂)}
C(O)OMe CH(Me)S{D2-32b(3-CF₃)}
C(O)OMe CH(Me)S(D2-37a)
C(O)OMe CH(Me)S(D2-51a)
C(O)OMe CH(Et)SMe
C(O)OMe CH(Et)S(O)Me
C(O)OMe CH(Et)S(O)₂Me
C(O)OMe CH(Et)SEt
C(O)OMe CH(Et)S(O)Et
C(O)OMe CH(Et)S(O)₂Et
C(O)OMe CH(Et)SCH₂CF₃
C(O)OMe CH(Et)S(O)CH₂CF₃
C(O)OMe CH(Et)S(O)₂CH₂CF₃
C(O)OMe CH(Pr-n)SMe
C(O)OMe CH(Pr-n)S(O)Me
C(O)OMe CH(Pr-n)S(O)₂Me
C(O)OMe CH(Pr-n)SEt
C(O)OMe CH(Pr-n)S(O)Et
C(O)OMe CH(Pr-n)S(O)₂Et
C(O)OMe CH(Pr-n)S(=NCN)Et
C(O)OMe CH(Pr-n)S(O)(=NCN)Et
C(O)OMe CH(Pr-n)SPr-n
C(O)OMe CH(Pr-n)S(O)Pr-n
C(O)OMe CH(Pr-n)S(O)₂Pr-n
C(O)OMe CH(Pr-n)SPr-i
C(O)OMe CH(Pr-n)S(O)Pr-i
C(O)OMe CH(Pr-n)S(O)₂Pr-i
C(O)OMe CH(Pr-n)SPr-c
C(O)OMe CH(Pr-n)S(O)Pr-c
C(O)OMe CH(Pr-n)S(O)₂Pr-c
C(O)OMe CH(Pr-n)SCH₂CF₃
C(O)OMe CH(Pr-n)S(O)CH₂CF₃
C(O)OMe CH(Pr-n)S(O)₂CH₂CF₃
C(O)OMe CH(Pr-i)SMe
C(O)OMe CH(Pr-i)S(O)Me
C(O)OMe CH(Pr-i)S(O)₂Me
C(O)OMe CH(Pr-i)SEt
C(O)OMe CH(Pr-i)S(O)Et
C(O)OMe CH(Pr-i)S(O)₂Et
C(O)OMe CH(Pr-i)S(=NCN)Et
C(O)OMe CH(Pr-i)S(O)(=NCN)Et
C(O)OMe CH(Pr-i)SPr-n
C(O)OMe CH(Pr-i)S(O)Pr-n
C(O)OMe CH(Pr-i)S(O)₂Pr-n
C(O)OMe CH(Pr-i)SPr-i
C(O)OMe CH(Pr-i)S(O)Pr-i
C(O)OMe CH(Pr-i)S(O)₂Pr-i
C(O)OMe CH(Pr-i)SPr-c
C(O)OMe CH(Pr-i)S(O)Pr-c
C(O)OMe CH(Pr-i)S(O)₂Pr-c
C(O)OMe CH(Pr-i)SCH₂CF₃
C(O)OMe CH(Pr-i)S(O)CH₂CF₃
C(O)OMe CH(Pr-i)S(O)₂CH₂CF₃
C(O)OMe CH(Pr-c)SMe
C(O)OMe CH(Pr-c)S(O)Me
C(O)OMe CH(Pr-c)S(O)₂Me
C(O)OMe CH(Pr-c)SEt
C(O)OMe CH(Pr-c)S(O)Et
C(O)OMe CH(Pr-c)S(O)₂Et
C(O)OMe CH(Pr-c)S(=NCN)Et
C(O)OMe CH(Pr-c)S(O)(=NCN)Et
C(O)OMe CH(Pr-c)SPr-n
C(O)OMe CH(Pr-c)S(O)Pr-n
C(O)OMe CH(Pr-c)S(O)₂Pr-n
C(O)OMe CH(Pr-c)SPr-i
C(O)OMe CH(Pr-c)S(O)Pr-i
C(O)OMe CH(Pr-c)S(O)₂Pr-i
C(O)OMe CH(Pr-c)SPr-c
C(O)OMe CH(Pr-c)S(O)Pr-c
C(O)OMe CH(Pr-c)S(O)₂Pr-c
C(O)OMe CH(Pr-c)SCH₂CF₃
C(O)OMe CH(Pr-c)S(O)CH₂CF₃
C(O)OMe CH(Pr-c)S(O)₂CH₂CF₃
C(O)OMe CH(Bu-n)SMe
C(O)OMe CH(Bu-n)S(O)Me
C(O)OMe CH(Bu-n)S(O)₂Me
C(O)OMe CH(Bu-n)SEt
C(O)OMe CH(Bu-n)S(O)Et
C(O)OMe CH(Bu-n)S(O)₂Et
C(O)OMe CH(Bu-n)S(=NCN)Et
C(O)OMe CH(Bu-n)S(O)(=NCN)Et
C(O)OMe CH(Bu-n)SPr-n
C(O)OMe CH(Bu-n)S(O)Pr-n
C(O)OMe CH(Bu-n)S(O)₂Pr-n
C(O)OMe CH(Bu-n)SPr-i
C(O)OMe CH(Bu-n)S(O)Pr-i
C(O)OMe CH(Bu-n)S(O)₂Pr-i
C(O)OMe CH(Bu-n)SPr-c
C(O)OMe CH(Bu-n)S(O)Pr-c
C(O)OMe CH(Bu-n)S(O)₂Pr-c
C(O)OMe CH(Bu-n)SCH₂CF₃
C(O)OMe CH(Bu-n)S(O)CH₂CF₃
C(O)OMe CH(Bu-n)S(O)₂CH₂CF₃
C(O)OMe CH(F)SMe
C(O)OMe CH(F)S(O)Me
C(O)OMe CH(F)S(O)₂Me
C(O)OMe CH(F)SEt
C(O)OMe CH(F)S(O)Et
C(O)OMe CH(F)S(O)₂Et
C(O)OMe CH(F)S(=NCN)Et
C(O)OMe CH(F)S(O)(=NCN)Et
C(O)OMe CH(F)SCH₂CF₃
C(O)OMe CH(F)S(O)CH₂CF₃
C(O)OMe CH(F)S(O)₂CH₂CF₃
C(O)OMe C(F)₂SMe
C(O)OMe C(F)₂S(O)Me
C(O)OMe C(F)₂S(O)₂Me
C(O)OMe C(F)₂SEt
C(O)OMe C(F)₂S(O)Et
C(O)OMe C(F)₂S(O)₂Et
C(O)OMe C(F)₂S(=NCN)Et
C(O)OMe C(F)₂S(O)(=NCN)Et
C(O)OMe C(F)₂SCH₂CF₃
C(O)OMe C(F)₂S(O)CH₂CF₃
C(O)OMe C(F)₂S(O)₂CH₂CF₃
C(O)OMe CH(Cl)SMe
C(O)OMe CH(Cl)S(O)Me
C(O)OMe CH(Cl)S(O)₂Me
C(O)OMe CH(Cl)SEt
C(O)OMe CH(Cl)S(O)Et
C(O)OMe CH(Cl)S(O)₂Et
C(O)OMe CH(Cl)S(=NCN)Et
C(O)OMe CH(Cl)S(O)(=NCN)Et
C(O)OMe CH(Cl)SCH₂CF₃
C(O)OMe CH(Cl)S(O)CH₂CF₃
C(O)OMe CH(Cl)S(O)₂CH₂CF₃
C(O)OMe C(Cl)₂SMe
C(O)OMe C(Cl)₂S(O)Me
C(O)OMe C(Cl)₂S(O)₂Me
C(O)OMe C(Cl)₂SEt
C(O)OMe C(Cl)₂S(O)Et
C(O)OMe C(Cl)₂S(O)₂Et
C(O)OMe C(Cl)₂S(=NCN)Et
C(O)OMe C(Cl)₂S(O)(=NCN)Et
C(O)OMe C(Cl)₂SCH₂CF₃
C(O)OMe C(Cl)₂S(O)CH₂CF₃
C(O)OMe C(Cl)₂S(O)₂CH₂CF₃
C(O)OMe CH(Br)SMe
C(O)OMe CH(Br)S(O)Me
C(O)OMe CH(Br)S(O)₂Me
C(O)OMe CH(Br)SEt
C(O)OMe CH(Br)S(O)Et
C(O)OMe CH(Br)S(O)₂Et
C(O)OMe CH(Br)S(=NCN)Et
C(O)OMe CH(Br)S(O)(=NCN)Et
C(O)OMe CH(Br)SCH₂CF₃
C(O)OMe CH(Br)S(O)CH₂CF₃
C(O)OMe CH(Br)S(O)₂CH₂CF₃
C(O)OMe CH(I)SMe
C(O)OMe CH(I)S(O)Me
C(O)OMe CH(I)S(O)₂Me
C(O)OMe CH(I)SEt
C(O)OMe CH(I)S(O)Et
C(O)OMe CH(I)S(O)₂Et
C(O)OMe CH(I)S(=NCN)Et
C(O)OMe CH(I)S(O)(=NCN)Et
C(O)OMe CH(I)SCH₂CF₃
C(O)OMe CH(I)S(O)CH₂CF₃
C(O)OMe CH(I)S(O)₂CH₂CF₃
C(O)OMe CH{OC(O)Me}SMe
C(O)OMe CH{OC(O)Me}S(O)Me
C(O)OMe CH{OC(O)Me}S(O)₂Me
C(O)OMe CH{OC(O)OMe}SEt
C(O)OMe CH{OC(O)OMe}S(O)Et
C(O)OMe CH{OC(O)OMe}S(O)₂Et
C(O)OMe CH{OC(O)OMe}S(=NCN)Et
C(O)OMe CH{OC(O)OMe}S(O)(=NCN)Et
C(O)OMe CH{OC(O)OEt}SMe
C(O)OMe CH{OC(O)OEt}S(O)Me
C(O)OMe CH{OC(O)OEt}S(O)₂Me
C(O)OMe CH{OC(O)OEt}SEt
C(O)OMe CH{OC(O)OEt}S(O)Et
C(O)OMe CH{OC(O)OEt}S(O)₂Et
C(O)OMe CH{OC(O)OEt}S(=NCN)Et
C(O)OMe CH{OC(O)OEt}S(O)(=NCN)Et
C(O)OMe CH(OMe)SMe
C(O)OMe CH(OMe)S(O)Me
C(O)OMe CH(OMe)S(O)₂Me
C(O)OMe CH(OMe)SEt
C(O)OMe CH(OMe)S(O)Et
C(O)OMe CH(OMe)S(O)₂Et
C(O)OMe CH(OMe)S(=NCN)Et
C(O)OMe CH(OMe)S(O)(=NCN)Et
C(O)OMe CH(OEt)SMe
C(O)OMe CH(OEt)S(O)Me
C(O)OMe CH(OEt)S(O)₂Me
C(O)OMe CH(OEt)SEt
C(O)OMe CH(OEt)S(O)Et
C(O)OMe CH(OEt)S(O)₂Et
C(O)OMe CH(OEt)S(=NCN)Et
C(O)OMe CH(OEt)S(O)(=NCN)Et
C(O)OMe CH(SMe)₂
C(O)OMe CH(SMe)S(O)Me
C(O)OMe CH(SMe)S(O)₂Me
C(O)OMe CH(SMe)SEt
C(O)OMe CH(SMe)S(O)Et
C(O)OMe CH(SMe)S(O)₂Et
C(O)OMe CH(SMe)S(=NCN)Et
C(O)OMe CH(SMe)S(O)(=NCN)Et
C(O)OMe CH(SEt)SMe
C(O)OMe CH(SEt)S(O)Me
C(O)OMe CH(SEt)S(O)₂Me
C(O)OMe CH(SEt)SEt
C(O)OMe CH(SEt)S(O)Et
C(O)OMe CH(SEt)S(O)₂Et
C(O)OMe CH(SEt)S(=NCN)Et
C(O)OMe CH(SEt)S(O)(=NCN)Et
C(O)OMe CH(CN)SMe
C(O)OMe CH(CN)S(O)Me
C(O)OMe CH(CN)S(O)₂Me
C(O)OMe CH(CN)SEt
C(O)OMe CH(CN)S(O)Et
C(O)OMe CH(CN)S(O)₂Et
C(O)OMe CH(CN)S(=NCN)Et
C(O)OMe CH(CN)S(O)(=NCN)Et
C(O)OMe CH{C(O)OMe}SMe
C(O)OMe CH{C(O)OMe}S(O)Me
C(O)OMe CH{C(O)OMe}S(O)₂Me
C(O)OMe CH{C(O)OMe}SMe
C(O)OMe CH{C(O)OMe}S(O)Me
C(O)OMe CH{C(O)OMe}S(O)₂Me
C(O)OMe CH{C(O)OMe}SEt
C(O)OMe CH{C(O)OMe}S(O)Et
C(O)OMe CH{C(O)OMe}S(O)₂Et
C(O)OMe CH{C(O)OMe}S(=NCN)Et
C(O)OMe CH{C(O)OMe}S(O)(=NCN)Et
C(O)OMe CH{C(O)OEt}SMe
C(O)OMe CH{C(O)OEt}S(O)Me
C(O)OMe CH{C(O)OEt}S(O)₂Me
C(O)OMe CH{C(O)OEt}SEt
C(O)OMe CH{C(O)OEt}S(O)Et
C(O)OMe CH{C(O)OEt}S(O)₂Et
C(O)OMe CH{C(O)OEt}S(=NCN)Et
C(O)OMe CH{C(O)OEt}S(O)(=NCN)Et
C(O)OMe C(Me)₂SMe
C(O)OMe C(Me)₂S(O)Me
C(O)OMe C(Me)₂S(O)₂Me
C(O)OMe CH₂CH₂SMe
C(O)OMe CH₂CH₂S(O)Me
C(O)OMe CH₂CH₂S(O)₂Me
C(O)OMe CH(Me)CH₂SMe
C(O)OMe CH(Me)CH₂S(O)Me
C(O)OMe CH(Me)CH₂S(O)₂Me
C(O)OEt CH₂SMe
C(O)OEt CH₂S(O)Me
C(O)OEt CH₂S(O)₂Me
C(O)OEt CH₂SEt
C(O)OEt CH₂S(O)Et
C(O)OEt CH₂S(O)₂Et
C(O)OEt CH₂SPr-n
C(O)OEt CH₂S(O)Pr-n
C(O)OEt CH₂S(O)₂Pr-n
C(O)OEt CH₂SPr-i
C(O)OEt CH₂S(O)Pr-i
C(O)OEt CH₂S(O)₂Pr-i
C(O)OEt CH₂SPr-c
C(O)OEt CH₂S(O)Pr-c
C(O)OEt CH₂S(O)₂Pr-c
C(O)OEt CH₂SCH₂CH=CH₂
C(O)OEt CH₂S(O)CH₂CH=CH₂
C(O)OEt CH₂S(O)₂CH₂CH=CH₂
C(O)OEt CH₂SCH₂C≡CH
C(O)OEt CH₂S(O)CH₂C≡CH
C(O)OEt CH₂S(O)₂CH₂C≡CH
C(O)OEt CH₂SCH₂CF₃
C(O)OEt CH₂S(O)CH₂CF₃
C(O)OEt CH₂S(O)₂CH₂CF₃
C(O)OEt CH₂SCH₂CH(OMe)₂
C(O)OEt CH₂SCH₂CH(=NOMe)
C(O)OEt CH(Me)SMe
C(O)OEt CH(Me)S(O)Me
C(O)OEt CH(Me)S(O)₂Me
C(O)OEt CH(Me)SEt
C(O)OEt CH(Me)S(O)Et
C(O)OEt CH(Me)S(O)₂Et
C(O)OEt CH(Me)S(=NCN)Et
C(O)OEt CH(Me)S(O)(=NCN)Et
C(O)OEt CH(Me)SPr-n
C(O)OEt CH(Me)S(O)Pr-n
C(O)OEt CH(Me)S(O)₂Pr-n
C(O)OEt CH(Me)SPr-i
C(O)OEt CH(Me)S(O)Pr-i
C(O)OEt CH(Me)S(O)₂Pr-i
C(O)OEt CH(Me)SBu-t
C(O)OEt CH(Me)S(O)Bu-t
C(O)OEt CH(Me)S(O)₂Bu-t
C(O)OEt CH(Me)SCH₂Pr-c
C(O)OEt CH(Me)S(O)CH₂Pr-c
C(O)OEt CH(Me)S(O)₂CH₂Pr-c
C(O)OEt CH(Me)SCH₂OMe
C(O)OEt CH(Me)SCH₂SMe
C(O)OEt CH(Me)S(O)CH₂SMe
C(O)OEt CH(Me)S(O)₂CH₂SMe
C(O)OEt CH(Me)SCH₂C=CH₂
C(O)OEt CH(Me)S(O)CH₂C=CH₂
C(O)OEt CH(Me)S(O)₂CH₂C=CH₂
C(O)OEt CH(Me)SCH₂C≡CH
C(O)OEt CH(Me)S(O)CH₂C≡CH
C(O)OEt CH(Me)S(O)₂CH₂C≡CH
C(O)OEt CH(Me)SCH₂C(O)NHMe
C(O)OEt CH(Me)S(O)CH₂C(O)NHMe
C(O)OEt CH(Me)S(O)₂CH₂C(O)NHMe
C(O)OEt CH(Me)SCH₂C(O)OMe
C(O)OEt CH(Me)S(O)CH₂C(O)OMe
C(O)OEt CH(Me)S(O)₂CH₂C(O)OMe
C(O)OEt CH(Me)SCH₂CH₂CH₂Cl
C(O)OEt CH(Me)S(O)CH₂CH₂CH₂Cl
C(O)OEt CH(Me)S(O)₂CH₂CH₂CH₂Cl
C(O)OEt CH(Me)SCH₂CF₃
C(O)OEt CH(Me)S(O)CH₂CF₃
C(O)OEt CH(Me)S(O)₂CH₂CF₃
C(O)OEt CH(Me)SCH₂Ph
C(O)OEt CH(Me)S(O)CH₂Ph
C(O)OEt CH(Me)S(O)₂CH₂Ph
C(O)OEt CH(Me)SCH₂(D2-34a)
C(O)OEt CH(Me)S(O)CH₂(D2-34a)
C(O)OEt CH(Me)S(O)₂CH₂(D2-34a)
C(O)OEt CH(CH₃)SCH₂Si(CH₃)₃
C(O)OEt CH(Me)SCN
C(O)OEt CH(Me)SCH₂CN
C(O)OEt CH(Me)SC(O)Me
C(O)OEt CH(Me)S(D2-12a)
C(O)OEt CH(Me)S(D2-32a)
C(O)OEt CH(Me)S{D2-32b(3-NO₂)}
C(O)OEt CH(Me)S{D2-32b(3-CF₃)}
C(O)OEt CH(Me)S(D2-37a)
C(O)OEt CH(Me)S(D2-51a)
C(O)OEt CH(Et)SMe
C(O)OEt CH(Et)S(O)Me
C(O)OEt CH(Et)S(O)₂Me
C(O)OEt CH(Et)SEt
C(O)OEt CH(Et)S(O)Et
C(O)OEt CH(Et)S(O)₂Et
C(O)OEt CH(Et)SCH₂CF₃
C(O)OEt CH(Et)S(O)CH₂CF₃
C(O)OEt CH(Et)S(O)₂CH₂CF₃
C(O)OEt CH(Pr-n)SMe
C(O)OEt CH(Pr-n)S(O)Me
C(O)OEt CH(Pr-n)S(O)₂Me
C(O)OEt CH(Pr-n)SEt
C(O)OEt CH(Pr-n)S(O)Et
C(O)OEt CH(Pr-n)S(O)₂Et
C(O)OEt CH(Pr-n)S(=NCN)Et
C(O)OEt CH(Pr-n)S(O)(=NCN)Et
C(O)OEt CH(Pr-n)SPr-n
C(O)OEt CH(Pr-n)S(O)Pr-n
C(O)OEt CH(Pr-n)S(O)₂Pr-n
C(O)OEt CH(Pr-n)SPr-i
C(O)OEt CH(Pr-n)S(O)Pr-i
C(O)OEt CH(Pr-n)S(O)₂Pr-i
C(O)OEt CH(Pr-n)SPr-c
C(O)OEt CH(Pr-n)S(O)Pr-c
C(O)OEt CH(Pr-n)S(O)₂Pr-c
C(O)OEt CH(Pr-n)SCH₂CF₃
C(O)OEt CH(Pr-n)S(O)CH₂CF₃
C(O)OEt CH(Pr-n)S(O)₂CH₂CF₃
C(O)OEt CH(Pr-i)SMe
C(O)OEt CH(Pr-i)S(O)Me
C(O)OEt CH(Pr-i)S(O)₂Me
C(O)OEt CH(Pr-i)SEt
C(O)OEt CH(Pr-i)S(O)Et
C(O)OEt CH(Pr-i)S(O)₂Et
C(O)OEt CH(Pr-i)S(=NCN)Et
C(O)OEt CH(Pr-i)S(O)(=NCN)Et
C(O)OEt CH(Pr-i)SPr-n
C(O)OEt CH(Pr-i)S(O)Pr-n
C(O)OEt CH(Pr-i)S(O)₂Pr-n
C(O)OEt CH(Pr-i)SPr-i
C(O)OEt CH(Pr-i)S(O)Pr-i
C(O)OEt CH(Pr-i)S(O)₂Pr-i
C(O)OEt CH(Pr-i)SPr-c
C(O)OEt CH(Pr-i)S(O)Pr-c
C(O)OEt CH(Pr-i)S(O)₂Pr-c
C(O)OEt CH(Pr-i)SCH₂CF₃
C(O)OEt CH(Pr-i)S(O)CH₂CF₃
C(O)OEt CH(Pr-i)S(O)₂CH₂CF₃
C(O)OEt CH(Pr-c)SMe
C(O)OEt CH(Pr-c)S(O)Me
C(O)OEt CH(Pr-c)S(O)₂Me
C(O)OEt CH(Pr-c)SEt
C(O)OEt CH(Pr-c)S(O)Et
C(O)OEt CH(Pr-c)S(O)₂Et
C(O)OEt CH(Pr-c)S(=NCN)Et
C(O)OEt CH(Pr-c)S(O)(=NCN)Et
C(O)OEt CH(Pr-c)SPr-n
C(O)OEt CH(Pr-c)S(O)Pr-n
C(O)OEt CH(Pr-c)S(O)₂Pr-n
C(O)OEt CH(Pr-c)SPr-i
C(O)OEt CH(Pr-c)S(O)Pr-i
C(O)OEt CH(Pr-c)S(O)₂Pr-i
C(O)OEt CH(Pr-c)SPr-c
C(O)OEt CH(Pr-c)S(O)Pr-c
C(O)OEt CH(Pr-c)S(O)₂Pr-c
C(O)OEt CH(Pr-c)SCH₂CF₃
C(O)OEt CH(Pr-c)S(O)CH₂CF₃
C(O)OEt CH(Pr-c)S(O)₂CH₂CF₃
C(O)OEt CH(Bu-n)SMe
C(O)OEt CH(Bu-n)S(O)Me
C(O)OEt CH(Bu-n)S(O)₂Me
C(O)OEt CH(Bu-n)SEt
C(O)OEt CH(Bu-n)S(O)Et
C(O)OEt CH(Bu-n)S(O)₂Et
C(O)OEt CH(Bu-n)S(=NCN)Et
C(O)OEt CH(Bu-n)S(O)(=NCN)Et
C(O)OEt CH(Bu-n)SPr-n
C(O)OEt CH(Bu-n)S(O)Pr-n
C(O)OEt CH(Bu-n)S(O)₂Pr-n
C(O)OEt CH(Bu-n)SPr-i
C(O)OEt CH(Bu-n)S(O)Pr-i
C(O)OEt CH(Bu-n)S(O)₂Pr-i
C(O)OEt CH(Bu-n)SPr-c
C(O)OEt CH(Bu-n)S(O)Pr-c
C(O)OEt CH(Bu-n)S(O)₂Pr-c
C(O)OEt CH(Bu-n)SCH₂CF₃
C(O)OEt CH(Bu-n)S(O)CH₂CF₃
C(O)OEt CH(Bu-n)S(O)₂CH₂CF₃
C(O)OEt CH(F)SMe
C(O)OEt CH(F)S(O)Me
C(O)OEt CH(F)S(O)₂Me
C(O)OEt CH(F)SEt
C(O)OEt CH(F)S(O)Et
C(O)OEt CH(F)S(O)₂Et
C(O)OEt CH(F)S(=NCN)Et
C(O)OEt CH(F)S(O)(=NCN)Et
C(O)OEt CH(F)SCH₂CF₃
C(O)OEt CH(F)S(O)CH₂CF₃
C(O)OEt CH(F)S(O)₂CH₂CF₃
C(O)OEt C(F)₂SMe
C(O)OEt C(F)₂S(O)Me
C(O)OEt C(F)₂S(O)₂Me
C(O)OEt C(F)₂SEt
C(O)OEt C(F)₂S(O)Et
C(O)OEt C(F)₂S(O)₂Et
C(O)OEt C(F)₂S(=NCN)Et
C(O)OEt C(F)₂S(O)(=NCN)Et
C(O)OEt C(F)₂SCH₂CF₃
C(O)OEt C(F)₂S(O)CH₂CF₃
C(O)OEt C(F)₂S(O)₂CH₂CF₃
C(O)OEt CH(Cl)SMe
C(O)OEt CH(Cl)S(O)Me
C(O)OEt CH(Cl)S(O)₂Me
C(O)OEt CH(Cl)SEt
C(O)OEt CH(Cl)S(O)Et
C(O)OEt CH(Cl)S(O)₂Et
C(O)OEt CH(Cl)S(=NCN)Et
C(O)OEt CH(Cl)S(O)(=NCN)Et
C(O)OEt CH(Cl)SCH₂CF₃
C(O)OEt CH(Cl)S(O)CH₂CF₃
C(O)OEt CH(Cl)S(O)₂CH₂CF₃
C(O)OEt C(Cl)₂SMe
C(O)OEt C(Cl)₂S(O)Me
C(O)OEt C(Cl)₂S(O)₂Me
C(O)OEt C(Cl)₂SEt
C(O)OEt C(Cl)₂S(O)Et
C(O)OEt C(Cl)₂S(O)₂Et
C(O)OEt C(Cl)₂S(=NCN)Et
C(O)OEt C(Cl)₂S(O)(=NCN)Et
C(O)OEt C(Cl)₂SCH₂CF₃
C(O)OEt C(Cl)₂S(O)CH₂CF₃
C(O)OEt C(Cl)₂S(O)₂CH₂CF₃
C(O)OEt CH(Br)SMe
C(O)OEt CH(Br)S(O)Me
C(O)OEt CH(Br)S(O)₂Me
C(O)OEt CH(Br)SEt
C(O)OEt CH(Br)S(O)Et
C(O)OEt CH(Br)S(O)₂Et
C(O)OEt CH(Br)S(=NCN)Et
C(O)OEt CH(Br)S(O)(=NCN)Et
C(O)OEt CH(Br)SCH₂CF₃
C(O)OEt CH(Br)S(O)CH₂CF₃
C(O)OEt CH(Br)S(O)₂CH₂CF₃
C(O)OEt CH(I)SMe
C(O)OEt CH(I)S(O)Me
C(O)OEt CH(I)S(O)₂Me
C(O)OEt CH(I)SEt
C(O)OEt CH(I)S(O)Et
C(O)OEt CH(I)S(O)₂Et
C(O)OEt CH(I)S(=NCN)Et
C(O)OEt CH(I)S(O)(=NCN)Et
C(O)OEt CH(I)SCH₂CF₃
C(O)OEt CH(I)S(O)CH₂CF₃
C(O)OEt CH(I)S(O)₂CH₂CF₃
C(O)OEt CH{OC(O)Me}SMe
C(O)OEt CH{OC(O)Me}S(O)Me
C(O)OEt CH{OC(O)Me}S(O)₂Me
C(O)OEt CH{OC(O)OMe}SEt
C(O)OEt CH{OC(O)OMe}S(O)Et
C(O)OEt CH{OC(O)OMe}S(O)₂Et
C(O)OEt CH{OC(O)OMe}S(=NCN)Et
C(O)OEt CH{OC(O)OMe}S(O)(=NCN)Et
C(O)OEt CH{OC(O)OEt}SMe
C(O)OEt CH{OC(O)OEt}S(O)Me
C(O)OEt CH{OC(O)OEt}S(O)₂Me
C(O)OEt CH{OC(O)OEt}SEt
C(O)OEt CH{OC(O)OEt}S(O)Et
C(O)OEt CH{OC(O)OEt}S(O)₂Et
C(O)OEt CH{OC(O)OEt}S(=NCN)Et
C(O)OEt CH{OC(O)OEt}S(O)(=NCN)Et
C(O)OEt CH(OMe)SMe
C(O)OEt CH(OMe)S(O)Me
C(O)OEt CH(OMe)S(O)₂Me
C(O)OEt CH(OMe)SEt
C(O)OEt CH(OMe)S(O)Et
C(O)OEt CH(OMe)S(O)₂Et
C(O)OEt CH(OMe)S(=NCN)Et
C(O)OEt CH(OMe)S(O)(=NCN)Et
C(O)OEt CH(OEt)SMe
C(O)OEt CH(OEt)S(O)Me
C(O)OEt CH(OEt)S(O)₂Me
C(O)OEt CH(OEt)SEt
C(O)OEt CH(OEt)S(O)Et
C(O)OEt CH(OEt)S(O)₂Et
C(O)OEt CH(OEt)S(=NCN)Et
C(O)OEt CH(OEt)S(O)(=NCN)Et
C(O)OEt CH(SMe)₂
C(O)OEt CH(SMe)S(O)Me
C(O)OEt CH(SMe)S(O)₂Me
C(O)OEt CH(SMe)SEt
C(O)OEt CH(SMe)S(O)Et
C(O)OEt CH(SMe)S(O)₂Et
C(O)OEt CH(SMe)S(=NCN)Et
C(O)OEt CH(SMe)S(O)(=NCN)Et
C(O)OEt CH(SEt)SMe
C(O)OEt CH(SEt)S(O)Me
C(O)OEt CH(SEt)S(O)₂Me
C(O)OEt CH(SEt)SEt
C(O)OEt CH(SEt)S(O)Et
C(O)OEt CH(SEt)S(O)₂Et
C(O)OEt CH(SEt)S(=NCN)Et
C(O)OEt CH(SEt)S(O)(=NCN)Et
C(O)OEt CH(CN)SMe
C(O)OEt CH(CN)S(O)Me
C(O)OEt CH(CN)S(O)₂Me
C(O)OEt CH(CN)SEt
C(O)OEt CH(CN)S(O)Et
C(O)OEt CH(CN)S(O)₂Et
C(O)OEt CH(CN)S(=NCN)Et
C(O)OEt CH(CN)S(O)(=NCN)Et
C(O)OEt CH{C(O)OMe}SMe
C(O)OEt CH{C(O)OMe}S(O)Me
C(O)OEt CH{C(O)OMe}S(O)₂Me
C(O)OEt CH{C(O)OMe}SMe
C(O)OEt CH{C(O)OMe}S(O)Me
C(O)OEt CH{C(O)OMe}S(O)₂Me
C(O)OEt CH{C(O)OMe}SEt
C(O)OEt CH{C(O)OMe}S(O)Et
C(O)OEt CH{C(O)OMe}S(O)₂Et
C(O)OEt CH{C(O)OMe}S(=NCN)Et
C(O)OEt CH{C(O)OMe}S(O)(=NCN)Et
C(O)OEt CH{C(O)OEt}SMe
C(O)OEt CH{C(O)OEt}S(O)Me
C(O)OEt CH{C(O)OEt}S(O)₂Me
C(O)OEt CH{C(O)OEt}SEt
C(O)OEt CH{C(O)OEt}S(O)Et
C(O)OEt CH{C(O)OEt}S(O)₂Et
C(O)OEt CH{C(O)OEt}S(=NCN)Et
C(O)OEt CH{C(O)OEt}S(O)(=NCN)Et
C(O)OEt C(Me)₂SMe
C(O)OEt C(Me)₂S(O)Me
C(O)OEt C(Me)₂S(O)₂Me
C(O)OEt CH₂CH₂SMe
C(O)OEt CH₂CH₂S(O)Me
C(O)OEt CH₂CH₂S(O)₂Me
C(O)OEt CH(Me)CH₂SMe
C(O)OEt CH(Me)CH₂S(O)Me
C(O)OEt CH(Me)CH₂S(O)₂Me
CH₂CF₃ CH₂SMe
CH₂CF₃ CH₂S(O)Me
CH₂CF₃ CH₂S(O)₂Me
CH₂CF₃ CH₂SEt
CH₂CF₃ CH₂S(O)Et
CH₂CF₃ CH₂S(O)₂Et
CH₂CF₃ CH₂SPr-n
CH₂CF₃ CH₂S(O)Pr-n
CH₂CF₃ CH₂S(O)₂Pr-n
CH₂CF₃ CH₂SPr-i
CH₂CF₃ CH₂S(O)Pr-i
CH₂CF₃ CH₂S(O)₂Pr-i
CH₂CF₃ CH₂SPr-c
CH₂CF₃ CH₂S(O)Pr-c
CH₂CF₃ CH₂S(O)₂Pr-c
CH₂CF₃ CH₂SCH₂CH=CH₂
CH₂CF₃ CH₂S(O)CH₂CH=CH₂
CH₂CF₃ CH₂S(O)₂CH₂CH=CH₂
CH₂CF₃ CH₂SCH₂C≡CH
CH₂CF₃ CH₂S(O)CH₂C≡CH
CH₂CF₃ CH₂S(O)₂CH₂C≡CH
CH₂CF₃ CH₂SCH₂CF₃
CH₂CF₃ CH₂S(O)CH₂CF₃
CH₂CF₃ CH₂S(O)₂CH₂CF₃
CH₂CF₃ CH₂SCH₂CH(OMe)₂
CH₂CF₃ CH₂SCH₂CH(=NOMe)
CH₂CF₃ CH(Me)SMe
CH₂CF₃ CH(Me)S(O)Me
CH₂CF₃ CH(Me)S(O)₂Me
CH₂CF₃ CH(Me)SEt
CH₂CF₃ CH(Me)S(O)Et
CH₂CF₃ CH(Me)S(O)₂Et
CH₂CF₃ CH(Me)S(=NCN)Et
CH₂CF₃ CH(Me)S(O)(=NCN)Et
CH₂CF₃ CH(Me)SPr-n
CH₂CF₃ CH(Me)S(O)Pr-n
CH₂CF₃ CH(Me)S(O)₂Pr-n
CH₂CF₃ CH(Me)SPr-i
CH₂CF₃ CH(Me)S(O)Pr-i
CH₂CF₃ CH(Me)S(O)₂Pr-i
CH₂CF₃ CH(Me)SBu-t
CH₂CF₃ CH(Me)S(O)Bu-t
CH₂CF₃ CH(Me)S(O)₂Bu-t
CH₂CF₃ CH(Me)SCH₂Pr-c
CH₂CF₃ CH(Me)S(O)CH₂Pr-c
CH₂CF₃ CH(Me)S(O)₂CH₂Pr-c
CH₂CF₃ CH(Me)SCH₂OMe
CH₂CF₃ CH(Me)SCH₂SMe
CH₂CF₃ CH(Me)S(O)CH₂SMe
CH₂CF₃ CH(Me)S(O)₂CH₂SMe
CH₂CF₃ CH(Me)SCH₂C=CH₂
CH₂CF₃ CH(Me)S(O)CH₂C=CH₂
CH₂CF₃ CH(Me)S(O)₂CH₂C=CH₂
CH₂CF₃ CH(Me)SCH₂C≡CH
CH₂CF₃ CH(Me)S(O)CH₂C≡CH
CH₂CF₃ CH(Me)S(O)₂CH₂C≡CH
CH₂CF₃ CH(Me)SCH₂C(O)NHMe
CH₂CF₃ CH(Me)S(O)CH₂C(O)NHMe
CH₂CF₃ CH(Me)S(O)₂CH₂C(O)NHMe
CH₂CF₃ CH(Me)SCH₂C(O)OMe
CH₂CF₃ CH(Me)S(O)CH₂C(O)OMe
CH₂CF₃ CH(Me)S(O)₂CH₂C(O)OMe
CH₂CF₃ CH(Me)SCH₂CH₂CH₂Cl
CH₂CF₃ CH(Me)S(O)CH₂CH₂CH₂Cl
CH₂CF₃ CH(Me)S(O)₂CH₂CH₂CH₂Cl
CH₂CF₃ CH(Me)SCH₂CF₃
CH₂CF₃ CH(Me)S(O)CH₂CF₃
CH₂CF₃ CH(Me)S(O)₂CH₂CF₃
CH₂CF₃ CH(Me)SCH₂Ph
CH₂CF₃ CH(Me)S(O)CH₂Ph
CH₂CF₃ CH(Me)S(O)₂CH₂Ph
CH₂CF₃ CH(Me)SCH₂(D2-34a)
CH₂CF₃ CH(Me)S(O)CH₂(D2-34a)
CH₂CF₃ CH(Me)S(O)₂CH₂(D2-34a)
CH₂CF₃ CH(CH₃)SCH₂Si(CH₃)₃
CH₂CF₃ CH(Me)SCN
CH₂CF₃ CH(Me)SCH₂CN
CH₂CF₃ CH(Me)SC(O)Me
CH₂CF₃ CH(Me)S(D2-12a)
CH₂CF₃ CH(Me)S(D2-32a)
CH₂CF₃ CH(Me)S{D2-32b(3-NO₂)}
CH₂CF₃ CH(Me)S{D2-32b(3-CF₃)}
CH₂CF₃ CH(Me)S(D2-37a)
CH₂CF₃ CH(Me)S(D2-51a)
CH₂CF₃ CH(Et)SMe
CH₂CF₃ CH(Et)S(O)Me
CH₂CF₃ CH(Et)S(O)₂Me
CH₂CF₃ CH(Et)SEt
CH₂CF₃ CH(Et)S(O)Et
CH₂CF₃ CH(Et)S(O)₂Et
CH₂CF₃ CH(Et)SCH₂CF₃
CH₂CF₃ CH(Et)S(O)CH₂CF₃
CH₂CF₃ CH(Et)S(O)₂CH₂CF₃
CH₂CF₃ CH(Pr-n)SMe
CH₂CF₃ CH(Pr-n)S(O)Me
CH₂CF₃ CH(Pr-n)S(O)₂Me
CH₂CF₃ CH(Pr-n)SEt
CH₂CF₃ CH(Pr-n)S(O)Et
CH₂CF₃ CH(Pr-n)S(O)₂Et
CH₂CF₃ CH(Pr-n)S(=NCN)Et
CH₂CF₃ CH(Pr-n)S(O)(=NCN)Et
CH₂CF₃ CH(Pr-n)SPr-n
CH₂CF₃ CH(Pr-n)S(O)Pr-n
CH₂CF₃ CH(Pr-n)S(O)₂Pr-n
CH₂CF₃ CH(Pr-n)SPr-i
CH₂CF₃ CH(Pr-n)S(O)Pr-i
CH₂CF₃ CH(Pr-n)S(O)₂Pr-i
CH₂CF₃ CH(Pr-n)SPr-c
CH₂CF₃ CH(Pr-n)S(O)Pr-c
CH₂CF₃ CH(Pr-n)S(O)₂Pr-c
CH₂CF₃ CH(Pr-n)SCH₂CF₃
CH₂CF₃ CH(Pr-n)S(O)CH₂CF₃
CH₂CF₃ CH(Pr-n)S(O)₂CH₂CF₃
CH₂CF₃ CH(Pr-i)SMe
CH₂CF₃ CH(Pr-i)S(O)Me
CH₂CF₃ CH(Pr-i)S(O)₂Me
CH₂CF₃ CH(Pr-i)SEt
CH₂CF₃ CH(Pr-i)S(O)Et
CH₂CF₃ CH(Pr-i)S(O)₂Et
CH₂CF₃ CH(Pr-i)S(=NCN)Et
CH₂CF₃ CH(Pr-i)S(O)(=NCN)Et
CH₂CF₃ CH(Pr-i)SPr-n
CH₂CF₃ CH(Pr-i)S(O)Pr-n
CH₂CF₃ CH(Pr-i)S(O)₂Pr-n
CH₂CF₃ CH(Pr-i)SPr-i
CH₂CF₃ CH(Pr-i)S(O)Pr-i
CH₂CF₃ CH(Pr-i)S(O)₂Pr-i
CH₂CF₃ CH(Pr-i)SPr-c
CH₂CF₃ CH(Pr-i)S(O)Pr-c
CH₂CF₃ CH(Pr-i)S(O)₂Pr-c
CH₂CF₃ CH(Pr-i)SCH₂CF₃
CH₂CF₃ CH(Pr-i)S(O)CH₂CF₃
CH₂CF₃ CH(Pr-i)S(O)₂CH₂CF₃
CH₂CF₃ CH(Pr-c)SMe
CH₂CF₃ CH(Pr-c)S(O)Me
CH₂CF₃ CH(Pr-c)S(O)₂Me
CH₂CF₃ CH(Pr-c)SEt
CH₂CF₃ CH(Pr-c)S(O)Et
CH₂CF₃ CH(Pr-c)S(O)₂Et
CH₂CF₃ CH(Pr-c)S(=NCN)Et
CH₂CF₃ CH(Pr-c)S(O)(=NCN)Et
CH₂CF₃ CH(Pr-c)SPr-n
CH₂CF₃ CH(Pr-c)S(O)Pr-n
CH₂CF₃ CH(Pr-c)S(O)₂Pr-n
CH₂CF₃ CH(Pr-c)SPr-i
CH₂CF₃ CH(Pr-c)S(O)Pr-i
CH₂CF₃ CH(Pr-c)S(O)₂Pr-i
CH₂CF₃ CH(Pr-c)SPr-c
CH₂CF₃ CH(Pr-c)S(O)Pr-c
CH₂CF₃ CH(Pr-c)S(O)₂Pr-c
CH₂CF₃ CH(Pr-c)SCH₂CF₃
CH₂CF₃ CH(Pr-c)S(O)CH₂CF₃
CH₂CF₃ CH(Pr-c)S(O)₂CH₂CF₃
CH₂CF₃ CH(Bu-n)SMe
CH₂CF₃ CH(Bu-n)S(O)Me
CH₂CF₃ CH(Bu-n)S(O)₂Me
CH₂CF₃ CH(Bu-n)SEt
CH₂CF₃ CH(Bu-n)S(O)Et
CH₂CF₃ CH(Bu-n)S(O)₂Et
CH₂CF₃ CH(Bu-n)S(=NCN)Et
CH₂CF₃ CH(Bu-n)S(O)(=NCN)Et
CH₂CF₃ CH(Bu-n)SPr-n
CH₂CF₃ CH(Bu-n)S(O)Pr-n
CH₂CF₃ CH(Bu-n)S(O)₂Pr-n
CH₂CF₃ CH(Bu-n)SPr-i
CH₂CF₃ CH(Bu-n)S(O)Pr-i
CH₂CF₃ CH(Bu-n)S(O)₂Pr-i
CH₂CF₃ CH(Bu-n)SPr-c
CH₂CF₃ CH(Bu-n)S(O)Pr-c
CH₂CF₃ CH(Bu-n)S(O)₂Pr-c
CH₂CF₃ CH(Bu-n)SCH₂CF₃
CH₂CF₃ CH(Bu-n)S(O)CH₂CF₃
CH₂CF₃ CH(Bu-n)S(O)₂CH₂CF₃
CH₂CF₃ CH(F)SMe
CH₂CF₃ CH(F)S(O)Me
CH₂CF₃ CH(F)S(O)₂Me
CH₂CF₃ CH(F)SEt
CH₂CF₃ CH(F)S(O)Et
CH₂CF₃ CH(F)S(O)₂Et
CH₂CF₃ CH(F)S(=NCN)Et
CH₂CF₃ CH(F)S(O)(=NCN)Et
CH₂CF₃ CH(F)SCH₂CF₃
CH₂CF₃ CH(F)S(O)CH₂CF₃
CH₂CF₃ CH(F)S(O)₂CH₂CF₃
CH₂CF₃ C(F)₂SMe
CH₂CF₃ C(F)₂S(O)Me
CH₂CF₃ C(F)₂S(O)₂Me
CH₂CF₃ C(F)₂SEt
CH₂CF₃ C(F)₂S(O)Et
CH₂CF₃ C(F)₂S(O)₂Et
CH₂CF₃ C(F)₂S(=NCN)Et
CH₂CF₃ C(F)₂S(O)(=NCN)Et
CH₂CF₃ C(F)₂SCH₂CF₃
CH₂CF₃ C(F)₂S(O)CH₂CF₃
CH₂CF₃ C(F)₂S(O)₂CH₂CF₃
CH₂CF₃ CH(Cl)SMe
CH₂CF₃ CH(Cl)S(O)Me
CH₂CF₃ CH(Cl)S(O)₂Me
CH₂CF₃ CH(Cl)SEt
CH₂CF₃ CH(Cl)S(O)Et
CH₂CF₃ CH(Cl)S(O)₂Et
CH₂CF₃ CH(Cl)S(=NCN)Et
CH₂CF₃ CH(Cl)S(O)(=NCN)Et
CH₂CF₃ CH(Cl)SCH₂CF₃
CH₂CF₃ CH(Cl)S(O)CH₂CF₃
CH₂CF₃ CH(Cl)S(O)₂CH₂CF₃
CH₂CF₃ C(Cl)₂SMe
CH₂CF₃ C(Cl)₂S(O)Me
CH₂CF₃ C(Cl)₂S(O)₂Me
CH₂CF₃ C(Cl)₂SEt
CH₂CF₃ C(Cl)₂S(O)Et
CH₂CF₃ C(Cl)₂S(O)₂Et
CH₂CF₃ C(Cl)₂S(=NCN)Et
CH₂CF₃ C(Cl)₂S(O)(=NCN)Et
CH₂CF₃ C(Cl)₂SCH₂CF₃
CH₂CF₃ C(Cl)₂S(O)CH₂CF₃
CH₂CF₃ C(Cl)₂S(O)₂CH₂CF₃
CH₂CF₃ CH(Br)SMe
CH₂CF₃ CH(Br)S(O)Me
CH₂CF₃ CH(Br)S(O)₂Me
CH₂CF₃ CH(Br)SEt
CH₂CF₃ CH(Br)S(O)Et
CH₂CF₃ CH(Br)S(O)₂Et
CH₂CF₃ CH(Br)S(=NCN)Et
CH₂CF₃ CH(Br)S(O)(=NCN)Et
CH₂CF₃ CH(Br)SCH₂CF₃
CH₂CF₃ CH(Br)S(O)CH₂CF₃
CH₂CF₃ CH(Br)S(O)₂CH₂CF₃
CH₂CF₃ CH(I)SMe
CH₂CF₃ CH(I)S(O)Me
CH₂CF₃ CH(I)S(O)₂Me
CH₂CF₃ CH(I)SEt
CH₂CF₃ CH(I)S(O)Et
CH₂CF₃ CH(I)S(O)₂Et
CH₂CF₃ CH(I)S(=NCN)Et
CH₂CF₃ CH(I)S(O)(=NCN)Et
CH₂CF₃ CH(I)SCH₂CF₃
CH₂CF₃ CH(I)S(O)CH₂CF₃
CH₂CF₃ CH(I)S(O)₂CH₂CF₃
CH₂CF₃ CH{OC(O)Me}SMe
CH₂CF₃ CH{OC(O)Me}S(O)Me
CH₂CF₃ CH{OC(O)Me}S(O)₂Me
CH₂CF₃ CH{OC(O)OMe}SEt
CH₂CF₃ CH{OC(O)OMe}S(O)Et
CH₂CF₃ CH{OC(O)OMe}S(O)₂Et
CH₂CF₃ CH{OC(O)OMe}S(=NCN)Et
CH₂CF₃ CH{OC(O)OMe}S(O)(=NCN)Et
CH₂CF₃ CH{OC(O)OEt}SMe
CH₂CF₃ CH{OC(O)OEt}S(O)Me
CH₂CF₃ CH{OC(O)OEt}S(O)₂Me
CH₂CF₃ CH{OC(O)OEt}SEt
CH₂CF₃ CH{OC(O)OEt}S(O)Et
CH₂CF₃ CH{OC(O)OEt}S(O)₂Et
CH₂CF₃ CH{OC(O)OEt}S(=NCN)Et
CH₂CF₃ CH{OC(O)OEt}S(O)(=NCN)Et
CH₂CF₃ CH(OMe)SMe
CH₂CF₃ CH(OMe)S(O)Me
CH₂CF₃ CH(OMe)S(O)₂Me
CH₂CF₃ CH(OMe)SEt
CH₂CF₃ CH(OMe)S(O)Et
CH₂CF₃ CH(OMe)S(O)₂Et
CH₂CF₃ CH(OMe)S(=NCN)Et
CH₂CF₃ CH(OMe)S(O)(=NCN)Et
CH₂CF₃ CH(OEt)SMe
CH₂CF₃ CH(OEt)S(O)Me
CH₂CF₃ CH(OEt)S(O)₂Me
CH₂CF₃ CH(OEt)SEt
CH₂CF₃ CH(OEt)S(O)Et
CH₂CF₃ CH(OEt)S(O)₂Et
CH₂CF₃ CH(OEt)S(=NCN)Et
CH₂CF₃ CH(OEt)S(O)(=NCN)Et
CH₂CF₃ CH(SMe)₂
CH₂CF₃ CH(SMe)S(O)Me
CH₂CF₃ CH(SMe)S(O)₂Me
CH₂CF₃ CH(SMe)SEt
CH₂CF₃ CH(SMe)S(O)Et
CH₂CF₃ CH(SMe)S(O)₂Et
CH₂CF₃ CH(SMe)S(=NCN)Et
CH₂CF₃ CH(SMe)S(O)(=NCN)Et
CH₂CF₃ CH(SEt)SMe
CH₂CF₃ CH(SEt)S(O)Me
CH₂CF₃ CH(SEt)S(O)₂Me
CH₂CF₃ CH(SEt)SEt
CH₂CF₃ CH(SEt)S(O)Et
CH₂CF₃ CH(SEt)S(O)₂Et
CH₂CF₃ CH(SEt)S(=NCN)Et
CH₂CF₃ CH(SEt)S(O)(=NCN)Et
CH₂CF₃ CH(CN)SMe
CH₂CF₃ CH(CN)S(O)Me
CH₂CF₃ CH(CN)S(O)₂Me
CH₂CF₃ CH(CN)SEt
CH₂CF₃ CH(CN)S(O)Et
CH₂CF₃ CH(CN)S(O)₂Et
CH₂CF₃ CH(CN)S(=NCN)Et
CH₂CF₃ CH(CN)S(O)(=NCN)Et
CH₂CF₃ CH{C(O)OMe}SMe
CH₂CF₃ CH{C(O)OMe}S(O)Me
CH₂CF₃ CH{C(O)OMe}S(O)₂Me
CH₂CF₃ CH{C(O)OMe}SMe
CH₂CF₃ CH{C(O)OMe}S(O)Me
CH₂CF₃ CH{C(O)OMe}S(O)₂Me
CH₂CF₃ CH{C(O)OMe}SEt
CH₂CF₃ CH{C(O)OMe}S(O)Et
CH₂CF₃ CH{C(O)OMe}S(O)₂Et
CH₂CF₃ CH{C(O)OMe}S(=NCN)Et
CH₂CF₃ CH{C(O)OMe}S(O)(=NCN)Et
CH₂CF₃ CH{C(O)OEt}SMe
CH₂CF₃ CH{C(O)OEt}S(O)Me
CH₂CF₃ CH{C(O)OEt}S(O)₂Me
CH₂CF₃ CH{C(O)OEt}SEt
CH₂CF₃ CH{C(O)OEt}S(O)Et
CH₂CF₃ CH{C(O)OEt}S(O)₂Et
CH₂CF₃ CH{C(O)OEt}S(=NCN)Et
CH₂CF₃ CH{C(O)OEt}S(O)(=NCN)Et
CH₂CF₃ C(Me)₂SMe
CH₂CF₃ C(Me)₂S(O)Me
CH₂CF₃ C(Me)₂S(O)₂Me
CH₂CF₃ OBu-t
S(O)₂Me CH₂SMe
S(O)₂Me CH₂S(O)Me
S(O)₂Me CH₂S(O)₂Me
S(O)₂Me CH₂SEt
S(O)₂Me CH₂S(O)Et
S(O)₂Me CH₂S(O)₂Et
S(O)₂Me CH₂SPr-n
S(O)₂Me CH₂S(O)Pr-n
S(O)₂Me CH₂S(O)₂Pr-n
S(O)₂Me CH₂SPr-i
S(O)₂Me CH₂S(O)Pr-i
S(O)₂Me CH₂S(O)₂Pr-i
S(O)₂Me CH₂SPr-c
S(O)₂Me CH₂S(O)Pr-c
S(O)₂Me CH₂S(O)₂Pr-c
S(O)₂Me CH₂SCH₂CH=CH₂
S(O)₂Me CH₂S(O)CH₂CH=CH₂
S(O)₂Me CH₂S(O)₂CH₂CH=CH₂
S(O)₂Me CH₂SCH₂C≡CH
S(O)₂Me CH₂S(O)CH₂C≡CH
S(O)₂Me CH₂S(O)₂CH₂C≡CH
S(O)₂Me CH₂SCH₂CF₃
S(O)₂Me CH₂S(O)CH₂CF₃
S(O)₂Me CH₂S(O)₂CH₂CF₃
S(O)₂Me CH₂SCH₂CH(OMe)₂
S(O)₂Me CH₂SCH₂CH(=NOMe)
S(O)₂Me CH(Me)SMe
S(O)₂Me CH(Me)S(O)Me
S(O)₂Me CH(Me)S(O)₂Me
S(O)₂Me CH(Me)SEt
S(O)₂Me CH(Me)S(O)Et
S(O)₂Me CH(Me)S(O)₂Et
S(O)₂Me CH(Me)S(=NCN)Et
S(O)₂Me CH(Me)S(O)(=NCN)Et
S(O)₂Me CH(Me)SPr-n
S(O)₂Me CH(Me)S(O)Pr-n
S(O)₂Me CH(Me)S(O)₂Pr-n
S(O)₂Me CH(Me)SPr-i
S(O)₂Me CH(Me)S(O)Pr-i
S(O)₂Me CH(Me)S(O)₂Pr-i
S(O)₂Me CH(Me)SBu-t
S(O)₂Me CH(Me)S(O)Bu-t
S(O)₂Me CH(Me)S(O)₂Bu-t
S(O)₂Me CH(Me)SCH₂Pr-c
S(O)₂Me CH(Me)S(O)CH₂Pr-c
S(O)₂Me CH(Me)S(O)₂CH₂Pr-c
S(O)₂Me CH(Me)SCH₂OMe
S(O)₂Me CH(Me)SCH₂SMe
S(O)₂Me CH(Me)S(O)CH₂SMe
S(O)₂Me CH(Me)S(O)₂CH₂SMe
S(O)₂Me CH(Me)SCH₂C=CH₂
S(O)₂Me CH(Me)S(O)CH₂C=CH₂
S(O)₂Me CH(Me)S(O)₂CH₂C=CH₂
S(O)₂Me CH(Me)SCH₂C≡CH
S(O)₂Me CH(Me)S(O)CH₂C≡CH
S(O)₂Me CH(Me)S(O)₂CH₂C≡CH
S(O)₂Me CH(Me)SCH₂C(O)NHMe
S(O)₂Me CH(Me)S(O)CH₂C(O)NHMe
S(O)₂Me CH(Me)S(O)₂CH₂C(O)NHMe
S(O)₂Me CH(Me)SCH₂C(O)OMe
S(O)₂Me CH(Me)S(O)CH₂C(O)OMe
S(O)₂Me CH(Me)S(O)₂CH₂C(O)OMe
S(O)₂Me CH(Me)SCH₂CH₂CH₂Cl
S(O)₂Me CH(Me)S(O)CH₂CH₂CH₂Cl
S(O)₂Me CH(Me)S(O)₂CH₂CH₂CH₂Cl
S(O)₂Me CH(Me)SCH₂CF₃
S(O)₂Me CH(Me)S(O)CH₂CF₃
S(O)₂Me CH(Me)S(O)₂CH₂CF₃
S(O)₂Me CH(Me)SCH₂Ph
S(O)₂Me CH(Me)S(O)CH₂Ph
S(O)₂Me CH(Me)S(O)₂CH₂Ph
S(O)₂Me CH(Me)SCH₂(D2-34a)
S(O)₂Me CH(Me)S(O)CH₂(D2-34a)
S(O)₂Me CH(Me)S(O)₂CH₂(D2-34a)
S(O)₂Me CH(CH₃)SCH₂Si(CH₃)₃
S(O)₂Me CH(Me)SCN
S(O)₂Me CH(Me)SCH₂CN
S(O)₂Me CH(Me)SC(O)Me
S(O)₂Me CH(Me)S(D2-12a)
S(O)₂Me CH(Me)S(D2-32a)
S(O)₂Me CH(Me)S{D2-32b(3-NO₂)}
S(O)₂Me CH(Me)S{D2-32b(3-CF₃)}
S(O)₂Me CH(Me)S(D2-37a)
S(O)₂Me CH(Me)S(D2-51a)
S(O)₂Me CH(Et)SMe
S(O)₂Me CH(Et)S(O)Me
S(O)₂Me CH(Et)S(O)₂Me
S(O)₂Me CH(Et)SEt
S(O)₂Me CH(Et)S(O)Et
S(O)₂Me CH(Et)S(O)₂Et
S(O)₂Me CH(Et)SCH₂CF₃
S(O)₂Me CH(Et)S(O)CH₂CF₃
S(O)₂Me CH(Et)S(O)₂CH₂CF₃
S(O)₂Me CH(Pr-n)SMe
S(O)₂Me CH(Pr-n)S(O)Me
S(O)₂Me CH(Pr-n)S(O)₂Me
S(O)₂Me CH(Pr-n)SEt
S(O)₂Me CH(Pr-n)S(O)Et
S(O)₂Me CH(Pr-n)S(O)₂Et
S(O)₂Me CH(Pr-n)S(=NCN)Et
S(O)₂Me CH(Pr-n)S(O)(=NCN)Et
S(O)₂Me CH(Pr-n)SPr-n
S(O)₂Me CH(Pr-n)S(O)Pr-n
S(O)₂Me CH(Pr-n)S(O)₂Pr-n
S(O)₂Me CH(Pr-n)SPr-i
S(O)₂Me CH(Pr-n)S(O)Pr-i
S(O)₂Me CH(Pr-n)S(O)₂Pr-i
S(O)₂Me CH(Pr-n)SPr-c
S(O)₂Me CH(Pr-n)S(O)Pr-c
S(O)₂Me CH(Pr-n)S(O)₂Pr-c
S(O)₂Me CH(Pr-n)SCH₂CF₃
S(O)₂Me CH(Pr-n)S(O)CH₂CF₃
S(O)₂Me CH(Pr-n)S(O)₂CH₂CF₃
S(O)₂Me CH(Pr-i)SMe
S(O)₂Me CH(Pr-i)S(O)Me
S(O)₂Me CH(Pr-i)S(O)₂Me
S(O)₂Me CH(Pr-i)SEt
S(O)₂Me CH(Pr-i)S(O)Et
S(O)₂Me CH(Pr-i)S(O)₂Et
S(O)₂Me CH(Pr-i)S(=NCN)Et
S(O)₂Me CH(Pr-i)S(O)(=NCN)Et
S(O)₂Me CH(Pr-i)SPr-n
S(O)₂Me CH(Pr-i)S(O)Pr-n
S(O)₂Me CH(Pr-i)S(O)₂Pr-n
S(O)₂Me CH(Pr-i)SPr-i
S(O)₂Me CH(Pr-i)S(O)Pr-i
S(O)₂Me CH(Pr-i)S(O)₂Pr-i
S(O)₂Me CH(Pr-i)SPr-c
S(O)₂Me CH(Pr-i)S(O)Pr-c
S(O)₂Me CH(Pr-i)S(O)₂Pr-c
S(O)₂Me CH(Pr-i)SCH₂CF₃
S(O)₂Me CH(Pr-i)S(O)CH₂CF₃
S(O)₂Me CH(Pr-i)S(O)₂CH₂CF₃
S(O)₂Me CH(Pr-c)SMe
S(O)₂Me CH(Pr-c)S(O)Me
S(O)₂Me CH(Pr-c)S(O)₂Me
S(O)₂Me CH(Pr-c)SEt
S(O)₂Me CH(Pr-c)S(O)Et
S(O)₂Me CH(Pr-c)S(O)₂Et
S(O)₂Me CH(Pr-c)S(=NCN)Et
S(O)₂Me CH(Pr-c)S(O)(=NCN)Et
S(O)₂Me CH(Pr-c)SPr-n
S(O)₂Me CH(Pr-c)S(O)Pr-n
S(O)₂Me CH(Pr-c)S(O)₂Pr-n
S(O)₂Me CH(Pr-c)SPr-i
S(O)₂Me CH(Pr-c)S(O)Pr-i
S(O)₂Me CH(Pr-c)S(O)₂Pr-i
S(O)₂Me CH(Pr-c)SPr-c
S(O)₂Me CH(Pr-c)S(O)Pr-c
S(O)₂Me CH(Pr-c)S(O)₂Pr-c
S(O)₂Me CH(Pr-c)SCH₂CF₃
S(O)₂Me CH(Pr-c)S(O)CH₂CF₃
S(O)₂Me CH(Pr-c)S(O)₂CH₂CF₃
S(O)₂Me CH(Bu-n)SMe
S(O)₂Me CH(Bu-n)S(O)Me
S(O)₂Me CH(Bu-n)S(O)₂Me
S(O)₂Me CH(Bu-n)SEt
S(O)₂Me CH(Bu-n)S(O)Et
S(O)₂Me CH(Bu-n)S(O)₂Et
S(O)₂Me CH(Bu-n)S(=NCN)Et
S(O)₂Me CH(Bu-n)S(O)(=NCN)Et
S(O)₂Me CH(Bu-n)SPr-n
S(O)₂Me CH(Bu-n)S(O)Pr-n
S(O)₂Me CH(Bu-n)S(O)₂Pr-n
S(O)₂Me CH(Bu-n)SPr-i
S(O)₂Me CH(Bu-n)S(O)Pr-i
S(O)₂Me CH(Bu-n)S(O)₂Pr-i
S(O)₂Me CH(Bu-n)SPr-c
S(O)₂Me CH(Bu-n)S(O)Pr-c
S(O)₂Me CH(Bu-n)S(O)₂Pr-c
S(O)₂Me CH(Bu-n)SCH₂CF₃
S(O)₂Me CH(Bu-n)S(O)CH₂CF₃
S(O)₂Me CH(Bu-n)S(O)₂CH₂CF₃
S(O)₂Me CH(F)SMe
S(O)₂Me CH(F)S(O)Me
S(O)₂Me CH(F)S(O)₂Me
S(O)₂Me CH(F)SEt
S(O)₂Me CH(F)S(O)Et
S(O)₂Me CH(F)S(O)₂Et
S(O)₂Me CH(F)S(=NCN)Et
S(O)₂Me CH(F)S(O)(=NCN)Et
S(O)₂Me CH(F)SCH₂CF₃
S(O)₂Me CH(F)S(O)CH₂CF₃
S(O)₂Me CH(F)S(O)₂CH₂CF₃
S(O)₂Me C(F)₂SMe
S(O)₂Me C(F)₂S(O)Me
S(O)₂Me C(F)₂S(O)₂Me
S(O)₂Me C(F)₂SEt
S(O)₂Me C(F)₂S(O)Et
S(O)₂Me C(F)₂S(O)₂Et
S(O)₂Me C(F)₂S(=NCN)Et
S(O)₂Me C(F)₂S(O)(=NCN)Et
S(O)₂Me C(F)₂SCH₂CF₃
S(O)₂Me C(F)₂S(O)CH₂CF₃
S(O)₂Me C(F)₂S(O)₂CH₂CF₃
S(O)₂Me CH(Cl)SMe
S(O)₂Me CH(Cl)S(O)Me
S(O)₂Me CH(Cl)S(O)₂Me
S(O)₂Me CH(Cl)SEt
S(O)₂Me CH(Cl)S(O)Et
S(O)₂Me CH(Cl)S(O)₂Et
S(O)₂Me CH(Cl)S(=NCN)Et
S(O)₂Me CH(Cl)S(O)(=NCN)Et
S(O)₂Me CH(Cl)SCH₂CF₃
S(O)₂Me CH(Cl)S(O)CH₂CF₃
S(O)₂Me CH(Cl)S(O)₂CH₂CF₃
S(O)₂Me C(Cl)₂SMe
S(O)₂Me C(Cl)₂S(O)Me
S(O)₂Me C(Cl)₂S(O)₂Me
S(O)₂Me C(Cl)₂SEt
S(O)₂Me C(Cl)₂S(O)Et
S(O)₂Me C(Cl)₂S(O)₂Et
S(O)₂Me C(Cl)₂S(=NCN)Et
S(O)₂Me C(Cl)₂S(O)(=NCN)Et
S(O)₂Me C(Cl)₂SCH₂CF₃
S(O)₂Me C(Cl)₂S(O)CH₂CF₃
S(O)₂Me C(Cl)₂S(O)₂CH₂CF₃
S(O)₂Me CH(Br)SMe
S(O)₂Me CH(Br)S(O)Me
S(O)₂Me CH(Br)S(O)₂Me
S(O)₂Me CH(Br)SEt
S(O)₂Me CH(Br)S(O)Et
S(O)₂Me CH(Br)S(O)₂Et
S(O)₂Me CH(Br)S(=NCN)Et
S(O)₂Me CH(Br)S(O)(=NCN)Et
S(O)₂Me CH(Br)SCH₂CF₃
S(O)₂Me CH(Br)S(O)CH₂CF₃
S(O)₂Me CH(Br)S(O)₂CH₂CF₃
S(O)₂Me CH(I)SMe
S(O)₂Me CH(I)S(O)Me
S(O)₂Me CH(I)S(O)₂Me
S(O)₂Me CH(I)SEt
S(O)₂Me CH(I)S(O)Et
S(O)₂Me CH(I)S(O)₂Et
S(O)₂Me CH(I)S(=NCN)Et
S(O)₂Me CH(I)S(O)(=NCN)Et
S(O)₂Me CH(I)SCH₂CF₃
S(O)₂Me CH(I)S(O)CH₂CF₃
S(O)₂Me CH(I)S(O)₂CH₂CF₃
S(O)₂Me CH{OC(O)Me}SMe
S(O)₂Me CH{OC(O)Me}S(O)Me
S(O)₂Me CH{OC(O)Me}S(O)₂Me
S(O)₂Me CH{OC(O)OMe}SEt
S(O)₂Me CH{OC(O)OMe}S(O)Et
S(O)₂Me CH{OC(O)OMe}S(O)₂Et
S(O)₂Me CH{OC(O)OMe}S(=NCN)Et
S(O)₂Me CH{OC(O)OMe}S(O)(=NCN)Et
S(O)₂Me CH{OC(O)OEt}SMe
S(O)₂Me CH{OC(O)OEt}S(O)Me
S(O)₂Me CH{OC(O)OEt}S(O)₂Me
S(O)₂Me CH{OC(O)OEt}SEt
S(O)₂Me CH{OC(O)OEt}S(O)Et
S(O)₂Me CH{OC(O)OEt}S(O)₂Et
S(O)₂Me CH{OC(O)OEt}S(=NCN)Et
S(O)₂Me CH{OC(O)OEt}S(O)(=NCN)Et
S(O)₂Me CH(OMe)SMe
S(O)₂Me CH(OMe)S(O)Me
S(O)₂Me CH(OMe)S(O)₂Me
S(O)₂Me CH(OMe)SEt
S(O)₂Me CH(OMe)S(O)Et
S(O)₂Me CH(OMe)S(O)₂Et
S(O)₂Me CH(OMe)S(=NCN)Et
S(O)₂Me CH(OMe)S(O)(=NCN)Et
S(O)₂Me CH(OEt)SMe
S(O)₂Me CH(OEt)S(O)Me
S(O)₂Me CH(OEt)S(O)₂Me
S(O)₂Me CH(OEt)SEt
S(O)₂Me CH(OEt)S(O)Et
S(O)₂Me CH(OEt)S(O)₂Et
S(O)₂Me CH(OEt)S(=NCN)Et
S(O)₂Me CH(OEt)S(O)(=NCN)Et
S(O)₂Me CH(SMe)₂
S(O)₂Me CH(SMe)S(O)Me
S(O)₂Me CH(SMe)S(O)₂Me
S(O)₂Me CH(SMe)SEt
S(O)₂Me CH(SMe)S(O)Et
S(O)₂Me CH(SMe)S(O)₂Et
S(O)₂Me CH(SMe)S(=NCN)Et
S(O)₂Me CH(SMe)S(O)(=NCN)Et
S(O)₂Me CH(SEt)SMe
S(O)₂Me CH(SEt)S(O)Me
S(O)₂Me CH(SEt)S(O)₂Me
S(O)₂Me CH(SEt)SEt
S(O)₂Me CH(SEt)S(O)Et
S(O)₂Me CH(SEt)S(O)₂Et
S(O)₂Me CH(SEt)S(=NCN)Et
S(O)₂Me CH(SEt)S(O)(=NCN)Et
S(O)₂Me CH(CN)SMe
S(O)₂Me CH(CN)S(O)Me
S(O)₂Me CH(CN)S(O)₂Me
S(O)₂Me CH(CN)SEt
S(O)₂Me CH(CN)S(O)Et
S(O)₂Me CH(CN)S(O)₂Et
S(O)₂Me CH(CN)S(=NCN)Et
S(O)₂Me CH(CN)S(O)(=NCN)Et
S(O)₂Me CH{C(O)OMe}SMe
S(O)₂Me CH{C(O)OMe}S(O)Me
S(O)₂Me CH{C(O)OMe}S(O)₂Me
S(O)₂Me CH{C(O)OMe}SMe
S(O)₂Me CH{C(O)OMe}S(O
S(O)₂Me CH{C(O)OMe}S(O)₂Me
S(O)₂Me CH{C(O)OMe}SEt
S(O)₂Me CH{C(O)OMe}S(O)Et
S(O)₂Me CH{C(O)OMe}S(O)₂Et
S(O)₂Me CH{C(O)OMe}S(=NCN)Et
S(O)₂Me CH{C(O)OMe}S(O)(=NCN)Et
S(O)₂Me CH{C(O)OEt}SMe
S(O)₂Me CH{C(O)OEt}S(O)Me
S(O)₂Me CH{C(O)OEt}S(O)₂Me
S(O)₂Me CH{C(O)OEt}SEt
S(O)₂Me CH{C(O)OEt}S(O)Et
S(O)₂Me CH{C(O)OEt}S(O)₂Et
S(O)₂Me CH{C(O)OEt}S(=NCN)Et
S(O)₂Me CH{C(O)OEt}S(O)(=NCN)Et
S(O)₂Me C(Me)₂SMe
S(O)₂Me C(Me)₂S(O)Me
S(O)₂Me C(Me)₂S(O)₂Me
SC(Cl)₃ CH(Me)SMe
SC(Cl)₃ CH(Me)S(O)Me
SC(Cl)₃ CH(Me)S(O)₂Me
SC(Cl)₃ CH(Me)SEt
SC(Cl)₃ CH(Me)S(O)Et
SC(Cl)₃ CH(Me)S(O)₂Et
SC(Cl)₃ CH(Me)CH₂SMe
CH₂CH₂CH₂SMe Me
CH₂CH₂SMe Me
NH₂ OBu-t
NHC(O)CH₂SMe OBu-t
N(Me)C(O)CH₂SMe OBu-t
NHC(O)CH(Me)SMe OBu-t
N(Me)C(O)CH(Me)SMe OBu-t
NHC(O)CH₂CH₂SMe OBu-t
N{C(O)OBu-t}₂ OBu-t
NHC(O)OBu-t OBu-t
―――――――――――――――――――
〔第６表〕 Table 5
―――――――――――――――――――
R^f2                       R^f3
―――――――――――――――――――
H C (O) Me
H Me
H Et
H Pr-n
H Pr-i
H Pr-c
H Bu-n
H Bu-c
H Bu-i
H Bu-s
H Bu-t
H Pen-n
H Pen-c
H Hex-n
H Hex-c
H CH₂Br
H CH (Br) Me
H CH₂CH₂CH₂Cl
H CH (Br) CH₂CH₂CH₂Br
H CH₂CF_Three
H CH₂CH (OH) CF_Three
H CH₂CN
H CH₂C (O) OMe
H CH₂C (O) NHMe
H CH = CH₂
H CH = CHSMe
H CH = CHCF_Three
H CH = C (Me) CF_Three
H CH {D2-108b (4-CF_Three)}
H C≡CH
H C≡CSiMe_Three
H CH₂OMe
H CH₂OEt
H CH (Me) OCH₂CF_Three
H CH (Me) ON = CHMe
H CH₂CH₂SC (O) Me
H CH₂OC (O) Me
H CH₂SMe
H CH₂S (O) Me
H CH₂S (O)₂Me
H CH₂SEt
H CH₂S (O) Et
H CH₂S (O)₂Et
H CH₂SCH₂CH = CH₂
H CH₂S (O) CH₂CH = CH₂
H CH₂S (O)₂CH₂CH = CH₂
H CH₂SCH₂CF_Three
H CH₂S (O) CH₂CF_Three
H CH₂S (O)₂CH₂CF_Three
H CH (Me) SMe
H CH (Me) S (O) Me
H CH (Me) S (O)₂Me
H CH (Me) SEt
H CH (Me) S (O) Et
H CH (Me) S (O)₂Et
H CH (Me) S (= NCN) Et
H CH (Me) S (O) (= NCN) Et
H CH (Me) SPr-n
H CH (Me) S (O) Pr-n
H CH (Me) S (O)₂Pr-n
H CH (Me) SPr-i
H CH (Me) S (O) Pr-i
H CH (Me) S (O)₂Pr-i
H CH (Me) SBu-t
H CH (Me) S (O) Bu-t
H CH (Me) S (O)₂Bu-t
H CH (Me) SCH₂Pr-c
H CH (Me) S (O) CH₂Pr-c
H CH (Me) S (O)₂CH₂Pr-c
H CH (Me) SCH₂OMe
H CH (Me) SCH₂SMe
H CH (Me) S (O) CH₂SMe
H CH (Me) S (O)₂CH₂SMe
H CH (Me) SCH₂C≡CH
H CH (Me) S (O) CH₂C≡CH
H CH (Me) S (O)₂CH₂C≡CH
H CH (Me) SCH₂C (O) NHMe
H CH (Me) S (O) CH₂C (O) NHMe
H CH (Me) S (O)₂CH₂C (O) NHMe
H CH (Me) SCH₂C (O) OMe
H CH (Me) S (O) CH₂C (O) OMe
H CH (Me) S (O)₂CH₂C (O) OMe
H CH (Me) SCH₂CH₂CH₂Cl
H CH (Me) S (O) CH₂CH₂CH₂Cl
H CH (Me) S (O)₂CH₂CH₂CH₂Cl
H CH (Me) SCH₂CF_Three
H CH (Me) S (O) CH₂CF_Three
H CH (Me) S (O)₂CH₂CF_Three
H CH (Me) SCH₂(D2-34a)
H CH (Me) S (O) CH₂(D2-34a)
H CH (Me) S (O)₂CH₂(D2-34a)
H CH (CH_Three) SCH₂Si (CH_Three)_Three
H CH (Me) SCN
H CH (Me) SCH₂CN
H CH (Me) SC (O) Me
H CH (Me) S (D2-37a)
H CH (Et) SMe
H CH (Et) S (O) Me
H CH (Et) S (O)₂Me
H CH (Et) SEt
H CH (Et) S (O) Et
H CH (Et) S (O)₂Et
H CH (F) SMe
H CH (F) S (O) Me
H CH (F) S (O)₂Me
H CH (F) SEt
H CH (F) S (O) Et
H CH (F) S (O)₂Et
H CH {OC (O) Me} SMe
H CH {OC (O) Me} S (O) Me
H CH {OC (O) Me} S (O)₂Me
H CH (SMe)₂
H C (Me)₂SMe
H C (Me)₂S (O) Me
H C (Me)₂S (O)₂Me
H CH₂CH₂SH
H CH₂CH₂SMe
H CH₂CH₂S (O) Me
H CH₂CH₂S (O)₂Me
H CH₂CH₂SEt
H CH₂CH₂S (O) Et
H CH₂CH₂S (O)₂Et
H CH₂CH₂SPr-n
H CH₂CH₂S (O) Pr-n
H CH₂CH₂S (O)₂Pr-n
H CH₂CH₂SPr-i
H CH₂CH₂S (O) Pr-i
H CH₂CH₂S (O)₂Pr-i
H CH₂CH₂SCH₂CF_Three
H CH₂CH₂S (O) CH₂CF_Three
H CH₂CH₂S (O)₂CH₂CF_Three
H CH₂CH₂SC (O) Me
H CH (Me) CH₂SMe
H CH (Me) CH₂S (O) Me
H CH (Me) CH₂S (O)₂Me
H CH (Me) CH₂SEt
H CH (Me) CH₂S (O) Et
H CH (Me) CH₂S (O)₂Et
H CH (Me) CH₂SPr-n
H CH (Me) CH₂S (O) Pr-n
H CH (Me) CH₂S (O)₂Pr-n
H CH (Me) CH₂SPr-i
H CH (Me) CH₂S (O) Pr-i
H CH (Me) CH₂S (O)₂Pr-i
H CH (Me) CH₂SCH₂CF_Three
H CH (Me) CH₂S (O) CH₂CF_Three
H CH (Me) CH₂S (O)₂CH₂CF_Three
H CH (Me) CH₂SC (O) Me
H CH (Et) CH₂SMe
H CH (Et) CH₂S (O) Me
H CH (Et) CH₂S (O)₂Me
H CH (OMe) CH₂SMe
H CH (OMe) CH₂S (O) Me
H CH (OMe) CH₂S (O)₂Me
H CH (SMe) CH₂SMe
H CH (SMe) CH₂S (O) Me
H CH (SMe) CH₂S (O)₂Me
H CH (CH₂SMe) CH₂SMe
H CH (CH₂SMe) CH₂S (O) Me
H CH (CH₂SMe) CH₂S (O)₂Me
H CH (Cl) CH₂SMe
H CH (Cl) CH₂S (O) Me
H CH (Cl) CH₂S (O)₂Me
H CH (CN) CH₂SMe
H CH (CN) CH₂S (O) Me
H CH (CN) CH₂S (O)₂Me
H CH (CN) CH₂SEt
H CH (CN) CH₂S (O) Et
H CH (CN) CH₂S (O)₂Et
H CH {C (O) OMe} CH₂SMe
H CH {C (O) OMe} CH₂S (O) Me
H CH {C (O) OMe} CH₂S (O)₂Me
H CH {C (O) OMe} CH₂SEt
H CH {C (O) OMe} CH₂S (O) Et
H CH {C (O) OMe} CH₂S (O)₂Et
H CH (Ph) CH₂SMe
H CH (Ph) CH₂S (O) Me
H CH (Ph) CH₂S (O)₂Me
H C (Me)₂CH₂SMe
H C (Me)₂CH₂S (O) Me
H C (Me)₂CH₂S (O)₂Me
H C (= CH₂) CH₂SMe
H C (= CH₂) CH₂S (O) Me
H C (= CH₂) CH₂S (O)₂Me
H C (= CH₂) CH₂SEt
H C (= CH₂) CH₂S (O) Et
H C (= CH₂) CH₂S (O)₂Et
H CH₂CH₂CH₂SEt
H CH₂CH₂CH₂S (O) Et
H CH₂CH₂CH₂S (O)₂Et
H CH (Me) CH₂CH₂SEt
H CH (Me) CH₂CH₂S (O) Et
H CH (Me) CH₂CH₂S (O)₂Et
H CH₂CH (Me) CH₂SEt
H CH₂CH (Me) CH₂S (O) Et
H CH₂CH (Me) CH₂S (O)₂Et
H CH₂CH₂CH (Me) SEt
H CH₂CH₂CH (Me) S (O) Et
H CH₂CH₂CH (Me) S (O)₂Et
H CH₂CH₂CH₂SPr-n
H CH₂CH₂CH₂S (O) Pr-n
H CH₂CH₂CH₂S (O)₂Pr-n
H CH (Me) CH₂CH₂SPr-n
H CH (Me) CH₂CH₂S (O) Pr-n
H CH (Me) CH₂CH₂S (O)₂Pr-n
H CH₂CH (Me) CH₂SPr-n
H CH₂CH (Me) CH₂S (O) Pr-n
H CH₂CH (Me) CH₂S (O)₂Pr-n
H CH₂CH₂CH₂CH₂SMe
H CH₂CH₂CH₂CH₂S (O) Me
H CH₂CH₂CH₂CH₂S (O)₂Me
H CH₂CH₂CH₂CH₂SEt
H CH₂CH₂CH₂CH₂S (O) Et
H CH₂CH₂CH₂CH₂S (O)₂Et
H CH₂CH₂CH₂CH₂SPr-n
H CH₂CH₂CH₂CH₂S (O) Pr-n
H CH₂CH₂CH₂CH₂S (O)₂Pr-n
H CH₂CH (Me) SMe
H CH₂OCH₂SMe
H CH₂CH (SMe)₂
H C (= CH₂) CH₂C (O) OH
H C (= NOMe) CH_Three
H C (= NOMe) Et
H C (= NOMe) Pr-n
H C (= NOEt) CH_Three
H C (= NOPr-n) CH_Three
H C (= NOPr-i) CH_Three
H C (= NOBu-n) CH_Three
H C (= NOCH₂Ph) CH_Three
H C (= NOMe) CH₂OCH₂CF_Three
H C (= NOMe) CH₂SMe
H C (= NOMe) CH₂S (O) Me
H C (= NOMe) CH₂S (O)₂Me
H C (= NOMe) CH₂SEt
H C (= NOMe) CH₂S (O) Et
H C (= NOMe) CH₂S (O)₂Et
H C (= NOMe) CH₂SCF_Three
H C (= NOMe) CH₂S (O) CF_Three
H C (= NOMe) CH₂S (O)₂CF_Three
H C (= NOMe) CH₂SCH₂CF_Three
H C (= NOMe) CH₂S (O) CH₂CF_Three
H C (= NOMe) CH₂S (O)₂CH₂CF_Three
H C (= NOEt) CH₂SMe
H C (= NOEt) CH₂S (O) Me
H C (= NOEt) CH₂S (O)₂Me
H C (= NOPr-n) CH₂SMe
H C (= NOPr-n) CH₂S (O) Me
H C (= NOPr-n) CH₂S (O)₂Me
H C (= NOPr-i) CH₂SMe
H C (= NOPr-i) CH₂S (O) Me
H C (= NOPr-i) CH₂S (O)₂Me
H C (= NOBu-n) CH₂SMe
H C (= NOBu-n) CH₂S (O) Me
H C (= NOBu-n) CH₂S (O)₂Me
H C (= NOCH₂Ph) CH₂SMe
H C (= NOCH₂Ph) CH₂S (O) Me
H C (= NOCH₂Ph) CH₂S (O)₂Me
H C (= NOCH₂CH = CH₂) CH₂SMe
H C (= NOCH₂OMe) CH₂SMe
H C (= NOCH₂CH₂OMe) CH₂SMe
H C {= NOCH₂CH₂Si (Me)_Three} CH₂SMe
H CH₂CH (= NOMe)
H CH₂C (= NOMe) Me
H CH₂C (= NOMe) Et
H CH₂C (= NOMe) Pr-n
H CH₂C (= NOMe) Pr-i
H CH₂C (= NOMe) Bu-n
H CH₂C (= NOMe) Bu-i
H CH₂C (= NOMe) Bu-s
H CH₂C (= NOMe) Bu-t
H CH₂C (= NOMe) CF_Three
H CH₂C (= NOCH_Three) CH₂SCH_Three
H CH (SMe) C (= NOMe) Me
H CH {S (O) Me} C (= NOMe) Me
H CH {S (O)₂Me} C (= NOMe) Me
H CH (SEt) C (= NOMe) Me
H CH {S (O) Et} C (= NOMe) Me
H CH {S (O)₂Et} C (= NOMe) Me
H CH₂NH₂
H CH₂NHC (O) Me
H CH₂NHC (O) OMe
H CH₂NHC (O) OBu-t
H CH₂NHSO₂Me
H CH₂N (Me) C (O) Me
H CH₂N (Me) C (O) OMe
H CH₂N (Me) C (O) OBu-t
H CH₂N (Me) SO₂Me
H CH (CH₂SMe) NH₂
H CH (CH₂SMe) NHC (O) Me
H CH (CH₂SMe) NHC (O) OMe
H CH (CH₂SMe) NHC (O) OBu-t
H CH (CH₂SMe) NHSO₂Me
H CH₂P (O) (OMe)₂
H CH₂P (O) (OEt)₂
H OBu-t
H O {D2-108b (4-NO₂)}
H SMe
H NH₂
H NHCH₂CH₂SMe
H N (Me) CH₂CH₂SMe
H NHCH₂CH₂CH₂SMe
H NHMe
H NHEt
H NPr-n
H NHCH (Me)₂
H NHCH₂C = CH₂
H NHCH₂C (O) OMe
H NHCH₂CF_Three
H N (Me) CH₂CF_Three
H NHC (O) OEt
H NHC (O) CCl_Three
H NHC (O) CH₂SMe
H N (CH₂CH_Three) C (O) CH₂SCH_Three
H NHS (O)₂(D2-108a)
H NHCH = NOMe
H N = CHNMe₂
H NHPh
H NH (D2-1a)
H NH (D2-2a)
H NH (D2-2b)
H NH (D2-4a)
H NH (D2-5a)
H NH (D2-5b)
H NH (D2-5c)
H NH (D2-6a)
H NH (D2-6b)
H NH (D2-6c)
H NH (D2-7a)
H NH (D2-8a)
H NH (D2-8b)
H NH (D2-8c)
H NH (D2-9a)
H NH (D2-9b)
H NH (D2-9c)
H NH (D2-10a)
H NH (D2-10b)
H NH (D2-10c)
H NH (D2-11a)
H NH (D2-12a)
H NH (D2-12b)
H NH (D2-12c)
H NH (D2-13a)
H NH (D2-13b)
H NH (D2-14a)
H NH (D2-14b)
H NH (D2-15a)
H NH (D2-15b)
H NH (D2-16a)
H NH (D2-17a)
H NH (D2-18a)
H NH (D2-19a)
H NH (D2-20a)
H NH (D2-21a)
H NH (D2-21b)
H NH (D2-22a)
H NH (D2-23a)
H NH (D2-23b)
H NH (D2-24a)
H NH (D2-25a)
H NH (D2-26a)
H NH (D2-27a)
H NH (D2-28a)
H NH (D2-29a)
H NH (D2-30a)
H NH (D2-31a)
H NH (D2-32a)
H NH (D2-33a)
H NH (D2-34a)
H NH (D2-35a)
H NH (D2-35b)
H NH (D2-36a)
H NH (D2-37a)
H NH (D2-38a)
H NH (D2-39a)
H NH (D2-40a)
H NH (D2-40b)
H NH (D2-40c)
H NH (D2-41a)
H NH (D2-42a)
H NH (D2-43a)
H NH (D2-45a)
H NH (D2-50a)
H NH (D2-51a)
H NH (D2-59a)
H NH (D2-61a)
H NH (D2-79a)
H NH (D2-80a)
H NH {D2-108b (2-Cl)}
H NH {D2-108b (3-Cl)}
H NH {D2-108b (4-Cl)}
H NH {D2-108b (2-Me)}
H NH {D2-108b (3-Me)}
H NH {D2-108b (4-Me)}
H N (Me) Ph
H N (Me) (D2-1a)
H N (Me) (D2-2a)
H N (Me) (D2-2b)
H N (Me) (D2-4a)
H N (Me) {D2-4b (Me)}
H N (Me) (D2-5a)
H N (Me) (D2-5b)
H N (Me) (D2-5c)
H N (Me) (D2-6a)
H N (Me) (D2-6b)
H N (Me) (D2-6c)
H N (Me) (D2-7a)
H N (Me) (D2-8a)
H N (Me) (D2-8b)
H N (Me) (D2-8c)
H N (Me) (D2-9a)
H N (Me) (D2-9b)
H N (Me) (D2-9c)
H N (Me) (D2-10a)
H N (Me) (D2-10b)
H N (Me) (D2-10c)
H N (Me) (D2-11a)
H N (Me) (D2-12a)
H N (Me) (D2-12b)
H N (Me) (D2-12c)
H N (Me) (D2-13a)
H N (Me) (D2-13b)
H N (Me) (D2-14a)
H N (Me) (D2-14b)
H N (Me) (D2-15a)
H N (Me) (D2-15b)
H N (Me) (D2-16a)
H N (Me) (D2-17a)
H N (Me) (D2-18a)
H N (Me) (D2-19a)
H N (Me) (D2-20a)
H N (Me) (D2-21a)
H N (Me) (D2-21b)
H N (Me) (D2-22a)
H N (Me) (D2-23a)
H N (Me) (D2-23b)
H N (Me) (D2-24a)
H N (Me) (D2-25a)
H N (Me) (D2-26a)
H N (Me) (D2-27a)
H N (Me) (D2-28a)
H N (Me) (D2-29a)
H N (Me) (D2-30a)
H N (Me) (D2-31a)
H N (Me) (D2-32a)
H N (Me) (D2-33a)
H N (Me) (D2-34a)
H N (Me) (D2-35a)
H N (Me) (D2-35b)
H N (Me) (D2-36a)
H N (Me) (D2-37a)
H N (Me) (D2-38a)
H N (Me) (D2-39a)
H N (Me) (D2-40a)
H N (Me) (D2-40b)
H N (Me) (D2-40c)
H N (Me) (D2-41a)
H N (Me) (D2-42a)
H N (Me) (D2-43a)
H N (Me) (D2-45a)
H N (Me) (D2-50a)
H N (Me) (D2-51a)
H N (Me) (D2-59a)
H N (Me) (D2-61a)
H N (Me) (D2-79a)
H N (Me) (D2-80a)
H N (Me) {D2-108b (2-Cl)}
H N (Me) {D2-108b (3-Cl)}
H N (Me) {D2-108b (4-Cl)}
H N (Me) {D2-108b (2-Me)}
H N (Me) {D2-108b (3-Me)}
H N (Me) {D2-108b (4-Me)}
H D2-8c (CH₂CF_Three)
H D2-1b (5-Br)
H D2-2c (5-SMe)
H D2-2c {5-C (O) Me}
H D2-4a (Me)
H D2-5d {5- (Pr-c)}
H D2-5e (3,5-Me₂)
H D2-6d (4,5-Cl₂)
H D2-9b
H D2-10e (2-CF_Three)
H D2-12f (4-NO₂)
H D2-13d (Me)
H D2-19a
H D2-32b (2-Br)
H D2-33b (2-OMe)
H D2-34a
H D2-35b
H D2-38b (4-SMe)
H D2-39b (5-Me)
H D2-82a
H D2-82b
H D2-87a
H D2-103b
H D2-103c
H D2-103d
H D2-103e
H CH₂(D2-2a)
H CH₂{D2-5f (3-Me)}
H CH₂(D2-28a)
H CH₂(D2-32a)
H CH₂(D2-33a)
H CH₂(D2-34a)
H CH₂{D2-33b (6-Cl)}
H CH₂(D2-34a)
Me C (O) Me
Me Me
Me Et
Me Pr-n
Me Pr-i
Me Pr-c
Me Bu-n
Me Bu-i
Me Bu-c
Me Bu-s
Me Bu-t
Me Pen-n
Me Pen-c
Me Hex-n
Me Hex-c
Me CH = CH₂
Me C≡CH
Me C≡CSiMe_Three
Me CH₂Br
Me CH₂Br
Me CH (Br) Me
Me CH₂CF_Three
Me CH₂CH (OH) CF_Three
Me CH₂CN
Me CH (Me) CN
Me CH₂CH₂CN
Me CH (Me) CH₂CN
Me CH₂CH₂CH₂CN
Me CH (Me) CH₂CH₂CN
Me CH₂CH₂CH₂CH₂CN
Me CH (Me) CH₂CH₂CH₂CN
Me CH₂C (O) OMe
Me CH (Me) C (O) OMe
Me CH₂CH₂C (O) OMe
Me CH (Me) CH₂C (O) OMe
Me CH₂CH₂CH₂C (O) OMe
Me CH (Me) CH₂CH₂C (O) OMe
Me CH₂CH₂CH₂CH₂C (O) OMe
Me CH₂C (O) OEt
Me CH (Me) C (O) OEt
Me CH₂CH₂C (O) OEt
Me CH (Me) CH₂C (O) OEt
Me CH₂CH₂CH₂C (O) OEt
Me CH (Me) CH₂CH₂C (O) OEt
Me CH₂CH₂CH₂CH₂C (O) OEt
Me CH₂C (O) NHMe
Me CH₂OMe
Me CH₂OEt
Me CH₂OPr-n
Me CH₂OPr-i
Me CH₂OPr-c
Me CH₂OBu-n
Me CH₂OBu-i
Me CH₂OBu-s
Me CH₂OBu-t
Me CH₂OBu-c
Me CH₂OPen-n
Me CH₂OPen-c
Me CH₂OHex-n
Me CH₂OHex-c
Me CH₂OCH₂Pr-c
Me CH₂OCH₂CH = CH₂
Me CH₂OCH₂C≡CH
Me CH₂OCH₂OMe
Me CH₂OCH₂SMe
Me CH₂OCH₂Si (CH_Three)_Three
Me CH₂OCH₂(D2-34a)
Me CH₂OCF_Three
Me CH₂OCF₂H
Me CH₂OCF₂Cl
Me CH₂OCF₂Br
Me CH₂OCH₂CF_Three
Me CH₂OCH₂CF₂CF_Three
Me CH₂OCH₂CN
Me CH₂OC (O) Me
Me CH₂OCH₂C (O) OMe
Me CH₂OCH₂C (O) OEt
Me CH₂ON = CHMe
Me CH₂ON = C (Me)₂
Me CH (Me) OMe
Me CH (Me) OEt
Me CH (Me) OPr-n
Me CH (Me) OPr-i
Me CH (Me) OPr-c
Me CH (Me) OBu-n
Me CH (Me) OBu-i
Me CH (Me) OBu-s
Me CH (Me) OBu-t
Me CH (Me) OBu-c
Me CH (Me) OPen-n
Me CH (Me) OPen-c
Me CH (Me) OHex-n
Me CH (Me) OHex-c
Me CH (Me) OCH₂Pr-c
Me CH (Me) OCH₂CH = CH₂
Me CH (Me) OCH₂C≡CH
Me CH (Me) OCH₂OMe
Me CH (Me) OCH₂SMe
Me CH (Me) OCH₂Si (CH_Three)_Three
Me CH (Me) OCH₂(D2-34a)
Me CH (Me) OCF_Three
Me CH (Me) OCF₂H
Me CH (Me) OCF₂Cl
Me CH (Me) OCF₂Br
Me CH (Me) OCH₂CF_Three
Me CH (Me) OCH₂CF₂CF_Three
Me CH (Me) OCH₂CN
Me CH (Me) OC (O) Me
Me CH (Me) OCH₂C (O) OMe
Me CH (Me) OCH₂C (O) OEt
Me CH (Me) ON = CHMe
Me CH (Me) ON = C (Me)₂
Me CH₂SMe
Me CH₂S (O) Me
Me CH₂S (O)₂Me
Me CH₂SEt
Me CH₂S (O) Et
Me CH₂S (O)₂Et
Me CH₂SCH₂CH = CH₂
Me CH₂S (O) CH₂CH = CH₂
Me CH₂S (O)₂CH₂CH = CH₂
Me CH₂SCH₂CF_Three
Me CH₂S (O) CH₂CF_Three
Me CH₂S (O)₂CH₂CF_Three
Me CH (Me) SMe
Me CH (Me) S (O) Me
Me CH (Me) S (O)₂Me
Me CH (Me) SEt
Me CH (Me) S (O) Et
Me CH (Me) S (O)₂Et
Me CH (Me) S (= NCN) Et
Me CH (Me) S (O) (= NCN) Et
Me CH (Me) SPr-n
Me CH (Me) S (O) Pr-n
Me CH (Me) S (O)₂Pr-n
Me CH (Me) SPr-i
Me CH (Me) S (O) Pr-i
Me CH (Me) S (O)₂Pr-i
Me CH (Me) SBu-t
Me CH (Me) S (O) Bu-t
Me CH (Me) S (O)₂Bu-t
Me CH (Me) SCH₂Pr-c
Me CH (Me) S (O) CH₂Pr-c
Me CH (Me) S (O)₂CH₂Pr-c
Me CH (Me) SCH₂OMe
Me CH (Me) SCH₂SMe
Me CH (Me) S (O) CH₂SMe
Me CH (Me) S (O)₂CH₂SMe
Me CH (Me) SCH₂C≡CH
Me CH (Me) S (O) CH₂C≡CH
Me CH (Me) S (O)₂CH₂C≡CH
Me CH (Me) SCH₂C (O) NHMe
Me CH (Me) S (O) CH₂C (O) NHMe
Me CH (Me) S (O)₂CH₂C (O) NHMe
Me CH (Me) SCH₂C (O) OMe
Me CH (Me) S (O) CH₂C (O) OMe
Me CH (Me) S (O)₂CH₂C (O) OMe
Me CH (Me) SCH₂CF_Three
Me CH (Me) S (O) CH₂CF_Three
Me CH (Me) S (O)₂CH₂CF_Three
Me CH (Me) SCH₂(D2-34a)
Me CH (Me) S (O) CH₂(D2-34a)
Me CH (Me) S (O)₂CH₂(D2-34a)
Me CH (CH_Three) SCH₂Si (CH_Three)_Three
Me CH (Me) SCN
Me CH (Me) SCH₂CN
Me CH (Me) SC (O) Me
Me CH (Me) S (D2-37a)
Me CH (Et) SMe
Me CH (Et) S (O) Me
Me CH (Et) S (O)₂Me
Me CH (Et) SEt
Me CH (Et) S (O) Et
Me CH (Et) S (O)₂Et
Me CH (Et) SCH₂CF_Three
Me CH (Et) S (O) CH₂CF_Three
Me CH (Et) S (O)₂CH₂CF_Three
Me CH (F) SMe
Me CH (F) S (O) Me
Me CH (F) S (O)₂Me
Me CH (F) SEt
Me CH (F) S (O) Et
Me CH (F) S (O)₂Et
Me CH {OC (O) Me} SMe
Me CH {OC (O) Me} S (O) Me
Me CH {OC (O) Me} S (O)₂Me
Me CH (SMe)₂
Me C (Me)₂SMe
Me C (Me)₂S (O) Me
Me C (Me)₂S (O)₂Me
Me CH₂CH₂SH
Me CH₂CH₂SMe
Me CH₂CH₂S (O) Me
Me CH₂CH₂S (O)₂Me
Me CH₂CH₂SEt
Me CH₂CH₂S (O) Et
Me CH₂CH₂S (O)₂Et
Me CH₂CH₂SPr-n
Me CH₂CH₂S (O) Pr-n
Me CH₂CH₂S (O)₂Pr-n
Me CH₂CH₂SPr-i
Me CH₂CH₂S (O) Pr-i
Me CH₂CH₂S (O)₂Pr-i
Me CH (Me) SCH₂CH₂CH₂Cl
Me CH (Me) S (O) CH₂CH₂CH₂Cl
Me CH (Me) S (O)₂CH₂CH₂CH₂Cl
Me CH₂CH₂SCH₂CF_Three
Me CH₂CH₂S (O) CH₂CF_Three
Me CH₂CH₂S (O)₂CH₂CF_Three
Me CH₂CH₂SC (O) Me
Me CH (Me) CH₂SMe
Me CH (Me) CH₂S (O) Me
Me CH (Me) CH₂S (O)₂Me
Me CH (Me) CH₂SEt
Me CH (Me) CH₂S (O) Et
Me CH (Me) CH₂S (O)₂Et
Me CH (Me) CH₂SPr-n
Me CH (Me) CH₂S (O) Pr-n
Me CH (Me) CH₂S (O)₂Pr-n
Me CH (Me) CH₂SPr-i
Me CH (Me) CH₂S (O) Pr-i
Me CH (Me) CH₂S (O)₂Pr-i
Me CH (Me) CH₂SCH₂CF_Three
Me CH (Me) CH₂S (O) CH₂CF_Three
Me CH (Me) CH₂S (O)₂CH₂CF_Three
Me CH (Me) CH₂SC (O) Me
Me CH (Et) CH₂SMe
Me CH (Et) CH₂S (O) Me
Me CH (Et) CH₂S (O)₂Me
Me CH (OMe) CH₂SMe
Me CH (OMe) CH₂S (O) Me
Me CH (OMe) CH₂S (O)₂Me
Me CH (SMe) CH₂SMe
Me CH (SMe) CH₂S (O) Me
Me CH (SMe) CH₂S (O)₂Me
Me CH (CH₂SMe) CH₂SMe
Me CH (CH₂SMe) CH₂S (O) Me
Me CH (CH₂SMe) CH₂S (O)₂Me
Me CH (Cl) CH₂SMe
Me CH (Cl) CH₂S (O) Me
Me CH (Cl) CH₂S (O)₂Me
Me CH (CN) CH₂SMe
Me CH (CN) CH₂S (O) Me
Me CH (CN) CH₂S (O)₂Me
Me CH (CN) CH₂SEt
Me CH (CN) CH₂S (O) Et
Me CH (CN) CH₂S (O)₂Et
Me CH {C (O) OMe} CH₂SMe
Me CH {C (O) OMe} CH₂S (O) Me
Me CH {C (O) OMe} CH₂S (O)₂Me
Me CH {C (O) OMe} CH₂SEt
Me CH {C (O) OMe} CH₂S (O) Et
Me CH {C (O) OMe} CH₂S (O)₂Et
Me CH (Ph) CH₂SMe
Me CH (Ph) CH₂S (O) Me
Me CH (Ph) CH₂S (O)₂Me
Me C (Me)₂CH₂SMe
Me C (Me)₂CH₂S (O) Me
Me C (Me)₂CH₂S (O)₂Me
Me C (= CH₂) CH₂SMe
Me C (= CH₂) CH₂S (O) Me
Me C (= CH₂) CH₂S (O)₂Me
Me C (= CH₂) CH₂SEt
Me C (= CH₂) CH₂S (O) Et
Me C (= CH₂) CH₂S (O)₂Et
Me CH₂CH₂CH₂SEt
Me CH₂CH₂CH₂S (O) Et
Me CH₂CH₂CH₂S (O)₂Et
Me CH (Me) CH₂CH₂SEt
Me CH (Me) CH₂CH₂S (O) Et
Me CH (Me) CH₂CH₂S (O)₂Et
Me CH₂CH (Me) CH₂SEt
Me CH₂CH (Me) CH₂S (O) Et
Me CH₂CH (Me) CH₂S (O)₂Et
Me CH₂CH₂CH (Me) SEt
Me CH₂CH₂CH (Me) S (O) Et
Me CH₂CH₂CH (Me) S (O)₂Et
Me CH₂CH₂CH₂SPr-n
Me CH₂CH₂CH₂S (O) Pr-n
Me CH₂CH₂CH₂S (O)₂Pr-n
Me CH (Me) CH₂CH₂SPr-n
Me CH (Me) CH₂CH₂S (O) Pr-n
Me CH (Me) CH₂CH₂S (O)₂Pr-n
Me CH₂CH (Me) CH₂SPr-n
Me CH₂CH (Me) CH₂S (O) Pr-n
Me CH₂CH (Me) CH₂S (O)₂Pr-n
Me CH₂CH₂CH₂CH₂SMe
Me CH₂CH₂CH₂CH₂S (O) Me
Me CH₂CH₂CH₂CH₂S (O)₂Me
Me CH₂CH₂CH₂CH₂SEt
Me CH₂CH₂CH₂CH₂S (O) Et
Me CH₂CH₂CH₂CH₂S (O)₂Et
Me CH₂CH₂CH₂CH₂SPr-n
Me CH₂CH₂CH₂CH₂S (O) Pr-n
Me CH₂CH₂CH₂CH₂S (O)₂Pr-n
Me CH₂CH (Me) SMe
Me CH₂OCH₂SMe
Me CH = CHSMe
Me CH₂CH (SMe)₂
Me CH₂CH₂SC (O) Me
Me C (= CH₂) CH₂C (O) OH
Me C (= NOMe) CH_Three
Me C (= NOMe) Et
Me C (= NOMe) Pr-n
Me C (= NOEt) CH_Three
Me C (= NOPr-n) CH_Three
Me C (= NOPr-i) CH_Three
Me C (= NOBu-n) CH_Three
Me C (= NOCH₂Ph) CH_Three
Me C (= NOMe) CH₂OCH₂CF_Three
Me C (= NOMe) CH₂SMe
Me C (= NOMe) CH₂S (O) Me
Me C (= NOMe) CH₂S (O)₂Me
Me C (= NOMe) CH₂SEt
Me C (= NOMe) CH₂S (O) Et
Me C (= NOMe) CH₂S (O)₂Et
Me C (= NOMe) CH₂SCF_Three
Me C (= NOMe) CH₂S (O) CF_Three
Me C (= NOMe) CH₂S (O)₂CF_Three
Me C (= NOMe) CH₂SCH₂CF_Three
Me C (= NOMe) CH₂S (O) CH₂CF_Three
Me C (= NOMe) CH₂S (O)₂CH₂CF_Three
Me C (= NOEt) CH₂SMe
Me C (= NOEt) CH₂S (O) Me
Me C (= NOEt) CH₂S (O)₂Me
Me C (= NOPr-n) CH₂SMe
Me C (= NOPr-n) CH₂S (O) Me
Me C (= NOPr-n) CH₂S (O)₂Me
Me C (= NOPr-i) CH₂SMe
Me C (= NOPr-i) CH₂S (O) Me
Me C (= NOPr-i) CH₂S (O)₂Me
Me C (= NOBu-n) CH₂SMe
Me C (= NOBu-n) CH₂S (O) Me
Me C (= NOBu-n) CH₂S (O)₂Me
Me C (= NOCH₂Ph) CH₂SMe
Me C (= NOCH₂Ph) CH₂S (O) Me
Me C (= NOCH₂Ph) CH₂S (O)₂Me
Me C (= NOCH₂CH = CH₂) CH₂SMe
Me C (= NOCH₂OMe) CH₂SMe
Me C (= NOCH₂CH₂OMe) CH₂SMe
Me C {= NOCH₂CH₂Si (Me)_Three} CH₂SMe
Me CH₂CH (= NOMe)
Me CH₂C (= NOMe) Me
Me CH₂C (= NOMe) Et
Me CH₂C (= NOMe) Pr-n
Me CH₂C (= NOMe) Pr-i
Me CH₂C (= NOMe) Bu-n
Me CH₂C (= NOMe) Bu-i
Me CH₂C (= NOMe) Bu-s
Me CH₂C (= NOMe) Bu-t
Me CH₂C (= NOMe) CF_Three
Me CH₂C (= NOCH_Three) CH₂SCH_Three
Me CH (SMe) C (= NOMe) Me
Me CH {S (O) Me} C (= NOMe) Me
Me CH {S (O)₂Me} C (= NOMe) Me
Me CH (SEt) C (= NOMe) Me
Me CH {S (O) Et} C (= NOMe) Me
Me CH {S (O)₂Et} C (= NOMe) Me
Me CH₂NH₂
Me CH₂NHC (O) Me
Me CH₂NHC (O) OMe
Me CH₂NHC (O) OBu-t
Me CH₂NHSO₂Me
Me CH₂N (Me) C (O) Me
Me CH₂N (Me) C (O) OMe
Me CH₂N (Me) C (O) OBu-t
Me CH₂N (Me) SO₂Me
Me CH (CH₂SMe) NH₂
Me CH (CH₂SMe) NHC (O) Me
Me CH (CH₂SMe) NHC (O) OMe
Me CH (CH₂SMe) NHC (O) OBu-t
Me CH (CH₂SMe) NHSO₂Me
Me CH₂P (O) (OMe)₂
Me CH₂P (O) (OEt)₂
Me OBu-t
Me SMe
Me NH₂
Me NHCH₂CH₂SMe
Me N (Me) CH₂CH₂SMe
Me NHCH₂CH₂CH₂SMe
Me NHMe
Me NHEt
Me NPr-n
Me NHCH (Me)₂
Me NHCH₂C (O) OMe
Me NHCH₂CF_Three
Me N (Me) CH₂CF_Three
Me NHC (O) OEt
Me NHC (O) CCl_Three
Me NHC (O) CH₂SMe
Me N (CH₂CH_Three) C (O) CH₂SCH_Three
Me NHS (O)₂(D2-108a)
Me NHPh
Me NH (D2-1a)
Me NH (D2-2a)
Me NH (D2-2b)
Me NH (D2-4a)
Me NH {D2-4b}
Me NH (D2-5a)
Me NH (D2-5b)
Me NH (D2-5c)
Me NH (D2-6a)
Me NH (D2-6b)
Me NH (D2-6c)
Me NH (D2-7a)
Me NH (D2-8a)
Me NH (D2-8b)
Me NH (D2-8c)
Me NH (D2-9a)
Me NH (D2-9b)
Me NH (D2-9c)
Me NH (D2-10a)
Me NH (D2-10b)
Me NH (D2-10c)
Me NH (D2-11a)
Me NH (D2-12a)
Me NH (D2-12b)
Me NH (D2-12c)
Me NH (D2-13a)
Me NH (D2-13b)
Me NH (D2-14a)
Me NH (D2-14b)
Me NH (D2-15a)
Me NH (D2-15b)
Me NH (D2-16a)
Me NH (D2-17a)
Me NH (D2-18a)
Me NH (D2-19a)
Me NH (D2-20a)
Me NH (D2-21a)
Me NH (D2-21b)
Me NH (D2-22a)
Me NH (D2-23a)
Me NH (D2-23b)
Me NH (D2-24a)
Me NH (D2-25a)
Me NH (D2-26a)
Me NH (D2-27a)
Me NH (D2-28a)
Me NH (D2-29a)
Me NH (D2-30a)
Me NH (D2-31a)
Me NH (D2-32a)
Me NH (D2-33a)
Me NH (D2-34a)
Me NH (D2-35a)
Me NH (D2-35b)
Me NH (D2-36a)
Me NH (D2-37a)
Me NH (D2-38a)
Me NH (D2-39a)
Me NH (D2-40a)
Me NH (D2-40b)
Me NH (D2-40c)
Me NH (D2-41a)
Me NH (D2-42a)
Me NH (D2-43a)
Me NH (D2-45a)
Me NH (D2-50a)
Me NH (D2-51a)
Me NH (D2-59a)
Me NH (D2-61a)
Me NH (D2-79a)
Me NH (D2-80a)
Me NH {D2-108b (2-Cl)}
Me NH {D2-108b (3-Cl)}
Me NH {D2-108b (4-Cl)}
Me NH {D2-108b (2-Me)}
Me NH {D2-108b (3-Me)}
Me NH {D2-108b (4-Me)}
Me N (Me) Ph
Me N (Me) (D2-1a)
Me N (Me) (D2-2a)
Me N (Me) (D2-2b)
Me N (Me) (D2-4a)
Me N (Me) {D2-4b}
Me N (Me) (D2-5a)
Me N (Me) (D2-5b)
Me N (Me) (D2-5c)
Me N (Me) (D2-6a)
Me N (Me) (D2-6b)
Me N (Me) (D2-6c)
Me N (Me) (D2-7a)
Me N (Me) (D2-8a)
Me N (Me) (D2-8b)
Me N (Me) (D2-8c)
Me N (Me) (D2-9a)
Me N (Me) (D2-9b)
Me N (Me) (D2-9c)
Me N (Me) (D2-10a)
Me N (Me) (D2-10b)
Me N (Me) (D2-10c)
Me N (Me) (D2-11a)
Me N (Me) (D2-12a)
Me N (Me) (D2-12b)
Me N (Me) (D2-12c)
Me N (Me) (D2-13a)
Me N (Me) (D2-13b)
Me N (Me) (D2-14a)
Me N (Me) (D2-14b)
Me N (Me) (D2-15a)
Me N (Me) (D2-15b)
Me N (Me) (D2-16a)
Me N (Me) (D2-17a)
Me N (Me) (D2-18a)
Me N (Me) (D2-19a)
Me N (Me) (D2-20a)
Me N (Me) (D2-21a)
Me N (Me) (D2-21b)
Me N (Me) (D2-22a)
Me N (Me) (D2-23a)
Me N (Me) (D2-23b)
Me N (Me) (D2-24a)
Me N (Me) (D2-25a)
Me N (Me) (D2-26a)
Me N (Me) (D2-27a)
Me N (Me) (D2-28a)
Me N (Me) (D2-29a)
Me N (Me) (D2-30a)
Me N (Me) (D2-31a)
Me N (Me) (D2-32a)
Me N (Me) (D2-33a)
Me N (Me) (D2-34a)
Me N (Me) (D2-35a)
Me N (Me) (D2-35b)
Me N (Me) (D2-36a)
Me N (Me) (D2-37a)
Me N (Me) (D2-38a)
Me N (Me) (D2-39a)
Me N (Me) (D2-40a)
Me N (Me) (D2-40b)
Me N (Me) (D2-40c)
Me N (Me) (D2-41a)
Me N (Me) (D2-42a)
Me N (Me) (D2-43a)
Me N (Me) (D2-45a)
Me N (Me) (D2-50a)
Me N (Me) (D2-51a)
Me N (Me) (D2-59a)
Me N (Me) (D2-61a)
Me N (Me) (D2-79a)
Me N (Me) (D2-80a)
Me N (Me) {D2-108b (2-Cl)}
Me N (Me) {D2-108b (3-Cl)}
Me N (Me) {D2-108b (4-Cl)}
Me N (Me) {D2-108b (2-Me)}
Me N (Me) {D2-108b (3-Me)}
Me N (Me) {D2-108b (4-Me)}
Me D2-19a
Me D2-32b (2-Br)
Me D2-33b (2-OMe)
Me D2-35b
Me D2-38b (4-SMe)
Me D2-39b (5-Me)
Me D2-82a
Me D2-82b
Me D2-87a
Me D2-103b
Me D2-103c
Me D2-103d
Me D2-103e
Me CH₂(D2-2a)
Me CH₂{D2-5f (3-Me)}
Me CH₂(D2-28a)
Me CH₂(D2-32a)
Me CH₂(D2-33a)
Me CH₂{D2-33b (6-Cl)}
Me CH₂(D2-34a)
Et C (O) (D2-2a)
Et C (O) Me
Et C (O) Et
Et C (O) Pr-n
Et C (O) Pr-i
Et C (O) Pr-c
Et C (O) Bu-n
Et C (O) Bu-i
Et C (O) Bu-s
Et C (O) Bu-t
Et C (O) Pen-n
Et C (O) Pen-c
Et C (O) Hex-n
Et C (O) Hex-c
Et C (O) CF_Three
Et C (O) OMe
Et C (O) OEt
Et C (O) NHPh
Et Me
Et Et
Et Pr-n
Et Pr-i
Et Pr-c
Et Bu-n
Et Bu-i
Et Bu-c
Et Bu-s
Et Bu-t
Et Pen-n
Et Pen-c
Et Hex-n
Et Hex-c
Et (CH₂)₆CH_Three
Et (CH₂)₇CH_Three
Et (CH₂)₈CH_Three
Et (CH₂)₉CH_Three
Et (CH₂)_TenCH_Three
Et (CH₂)₁₁CH_Three
Et CH (Me) (CH₂)₂CH_Three
Et CH (Me) (CH₂)₃CH_Three
Et CH (Me) (CH₂)₄CH_Three
Et CH (Me) (CH₂)₅CH_Three
Et CH (Me) (CH₂)₆CH_Three
Et CH (Me) (CH₂)₇CH_Three
Et CH (Me) (CH₂)₈CH_Three
Et CH₂Pr-c
Et CH₂Bu-t
Et CH = CH₂
Et C (Me) = CH₂
Et CH = CH (D2-1a)
Et CH = CH (D2-2a)
Et CH = CH (D2-33a)
Et CH = CH {D2-108b (4-CF_Three)}
Et C≡CH
Et C≡CSiMe_Three
Et CHCl₂
Et CH₂Br
Et CH (Br) Me
Et CH₂CH₂CH₂CH₂Br
Et CH (Br) Bu-t
Et CH₂CF_Three
Et CF₂CF₂Cl
Et CH₂CH (CF_Three)₂
Et CH₂CH (OH) CF_Three
Et CH₂CH₂C (F) = CF₂
Et CH₂CN
Et CH (Me) CN
Et CH₂CH₂CN
Et CH (Me) CH₂CN
Et CH₂CH₂CH₂CN
Et CH (Me) CH₂CH₂CN
Et CH₂CH₂CH₂CH₂CN
Et CH (Me) CH₂CH₂CH₂CN
Et CH₂C (O) OMe
Et CH (Me) C (O) OMe
Et CH₂CH₂C (O) OMe
Et CH (Me) CH₂C (O) OMe
Et CH₂CH₂CH₂C (O) OMe
Et CH (Me) CH₂CH₂C (O) OMe
Et CH₂CH₂CH₂CH₂C (O) OMe
Et CH₂C (O) OEt
Et CH (Me) C (O) OEt
Et CH₂CH₂C (O) OEt
Et CH (Me) CH₂C (O) OEt
Et CH₂CH₂CH₂C (O) OEt
Et CH (Me) CH₂CH₂C (O) OEt
Et CH₂CH₂CH₂CH₂C (O) OEt
Et CH₂C (O) NHMe
Et CH₂C (O) NHCH₂CF_Three
Et CH₂OMe
Et CH₂OEt
Et CH₂OPr-n
Et CH₂OPr-i
Et CH₂OPr-c
Et CH₂OBu-n
Et CH₂OBu-i
Et CH₂OBu-s
Et CH₂OBu-t
Et CH₂OBu-c
Et CH₂OPen-n
Et CH₂OPen-c
Et CH₂OHex-n
Et CH₂OHex-c
Et CH₂OCH₂Pr-c
Et CH₂OCH₂CH = CH₂
Et CH₂OCH₂C≡CH
Et CH₂OCH₂OMe
Et CH₂OCH₂SMe
Et CH₂OCH₂Si (CH_Three)_Three
Et CH₂OCH₂(D2-34a)
Et CH₂OCF_Three
Et CH₂OCF₂H
Et CH₂OCF₂Cl
Et CH₂OCF₂Br
Et CH₂OCH₂CF_Three
Et CH₂OCH₂CF₂CF_Three
Et CH₂OCH₂CN
Et CH₂OC (O) Me
Et CH₂OCH₂C (O) OMe
Et CH₂OCH₂C (O) OEt
Et CH₂ON = CHMe
Et CH₂ON = C (Me)₂
Et CH (Me) OMe
Et CH (Me) OEt
Et CH (Me) OPr-n
Et CH (Me) OPr-i
Et CH (Me) OPr-c
Et CH (Me) OBu-n
Et CH (Me) OBu-i
Et CH (Me) OBu-s
Et CH (Me) OBu-t
Et CH (Me) OBu-c
Et CH (Me) OPen-n
Et CH (Me) OPen-c
Et CH (Me) OHex-n
Et CH (Me) OHex-c
Et CH (Me) OCH₂Pr-c
Et CH (Me) OCH₂CH = CH₂
Et CH (Me) OCH₂C≡CH
Et CH (Me) OCH₂OMe
Et CH (Me) OCH₂SMe
Et CH (Me) OCH₂Si (CH_Three)_Three
Et CH (Me) OCH₂(D2-34a)
Et CH (Me) OCF_Three
Et CH (Me) OCF₂H
Et CH (Me) OCF₂Cl
Et CH (Me) OCF₂Br
Et CH (Me) OCH₂CF_Three
Et CH (Me) OCH₂CF₂CF_Three
Et CH (Me) OCH₂CN
Et CH (Me) OC (O) Me
Et CH (Me) OCH₂C (O) OMe
Et CH (Me) OCH₂C (O) OEt
Et CH (Me) ON = CHMe
Et CH (Me) ON = C (Me)₂
Et C (Me)₂OC (O) Me
Et CH₂SMe
Et CH₂S (O) Me
Et CH₂S (O)₂Me
Et CH₂SEt
Et CH₂S (O) Et
Et CH₂S (O)₂Et
Et CH₂SPr-n
Et CH₂S (O) Pr-n
Et CH₂S (O)₂Pr-n
Et CH₂SPr-i
Et CH₂S (O) Pr-i
Et CH₂S (O)₂Pr-i
Et CH₂SPr-c
Et CH₂S (O) Pr-c
Et CH₂S (O)₂Pr-c
Et CH₂SCH₂CH = CH₂
Et CH₂S (O) CH₂CH = CH₂
Et CH₂S (O)₂CH₂CH = CH₂
Et CH₂SCH₂C≡CH
Et CH₂S (O) CH₂C≡CH
Et CH₂S (O)₂CH₂C≡CH
Et CH₂SCH₂CF_Three
Et CH₂S (O) CH₂CF_Three
Et CH₂S (O)₂CH₂CF_Three
Et CH₂SCH₂CH (OMe)₂
Et CH₂SCH₂CH (= NOMe)
Et CH (Me) SMe
Et CH (Me) S (O) Me
Et CH (Me) S (O)₂Me
Et CH (Me) SEt
Et CH (Me) S (O) Et
Et CH (Me) S (O)₂Et
Et CH (Me) S (= NCN) Et
Et CH (Me) S (O) (= NCN) Et
Et CH (Me) SPr-n
Et CH (Me) S (O) Pr-n
Et CH (Me) S (O)₂Pr-n
Et CH (Me) SPr-i
Et CH (Me) S (O) Pr-i
Et CH (Me) S (O)₂Pr-i
Et CH (Me) SBu-t
Et CH (Me) S (O) Bu-t
Et CH (Me) S (O)₂Bu-t
Et CH (Me) SCH₂Pr-c
Et CH (Me) S (O) CH₂Pr-c
Et CH (Me) S (O)₂CH₂Pr-c
Et CH (Me) SCH₂OMe
Et CH (Me) SCH₂SMe
Et CH (Me) S (O) CH₂SMe
Et CH (Me) S (O)₂CH₂SMe
Et CH (Me) SCH₂C = CH₂
Et CH (Me) S (O) CH₂C = CH₂
Et CH (Me) S (O)₂CH₂C = CH₂
Et CH (Me) SCH₂C≡CH
Et CH (Me) S (O) CH₂C≡CH
Et CH (Me) S (O)₂CH₂C≡CH
Et CH (Me) SCH₂C (O) NHMe
Et CH (Me) S (O) CH₂C (O) NHMe
Et CH (Me) S (O)₂CH₂C (O) NHMe
Et CH (Me) SCH₂C (O) OMe
Et CH (Me) S (O) CH₂C (O) OMe
Et CH (Me) S (O)₂CH₂C (O) OMe
Et CH (Me) SCH₂CH₂CH₂Cl
Et CH (Me) S (O) CH₂CH₂CH₂Cl
Et CH (Me) S (O)₂CH₂CH₂CH₂Cl
Et CH (Me) SCH₂CF_Three
Et CH (Me) S (O) CH₂CF_Three
Et CH (Me) S (O)₂CH₂CF_Three
Et CH (Me) SCH₂Ph
Et CH (Me) S (O) CH₂Ph
Et CH (Me) S (O)₂CH₂Ph
Et CH (Me) SCH₂(D2-34a)
Et CH (Me) S (O) CH₂(D2-34a)
Et CH (Me) S (O)₂CH₂(D2-34a)
Et CH (CH_Three) SCH₂Si (CH_Three)_Three
Et CH (Me) SCN
Et CH (Me) SCH₂CN
Et CH (Me) SC (O) Me
Et CH (Me) S (D2-12a)
Et CH (Me) S (D2-32a)
Et CH (Me) S {D2-32b (3-NO₂)}
Et CH (Me) S {D2-32b (3-CF_Three)}
Et CH (Me) S (D2-37a)
Et CH (Me) S (D2-51a)
Et CH (Et) SMe
Et CH (Et) S (O) Me
Et CH (Et) S (O)₂Me
Et CH (Et) SEt
Et CH (Et) S (O) Et
Et CH (Et) S (O)₂Et
Et CH (Et) SCH₂CF_Three
Et CH (Et) S (O) CH₂CF_Three
Et CH (Et) S (O)₂CH₂CF_Three
Et CH (Pr-n) SMe
Et CH (Pr-n) S (O) Me
Et CH (Pr-n) S (O)₂Me
Et CH (Pr-n) SEt
Et CH (Pr-n) S (O) Et
Et CH (Pr-n) S (O)₂Et
Et CH (Pr-n) S (= NCN) Et
Et CH (Pr-n) S (O) (= NCN) Et
Et CH (Pr-n) SPr-n
Et CH (Pr-n) S (O) Pr-n
Et CH (Pr-n) S (O)₂Pr-n
Et CH (Pr-n) SPr-i
Et CH (Pr-n) S (O) Pr-i
Et CH (Pr-n) S (O)₂Pr-i
Et CH (Pr-n) SPr-c
Et CH (Pr-n) S (O) Pr-c
Et CH (Pr-n) S (O)₂Pr-c
Et CH (Pr-n) SCH₂CF_Three
Et CH (Pr-n) S (O) CH₂CF_Three
Et CH (Pr-n) S (O)₂CH₂CF_Three
Et CH (Pr-i) SMe
Et CH (Pr-i) S (O) Me
Et CH (Pr-i) S (O)₂Me
Et CH (Pr-i) SEt
Et CH (Pr-i) S (O) Et
Et CH (Pr-i) S (O)₂Et
Et CH (Pr-i) S (= NCN) Et
Et CH (Pr-i) S (O) (= NCN) Et
Et CH (Pr-i) SPr-n
Et CH (Pr-i) S (O) Pr-n
Et CH (Pr-i) S (O)₂Pr-n
Et CH (Pr-i) SPr-i
Et CH (Pr-i) S (O) Pr-i
Et CH (Pr-i) S (O)₂Pr-i
Et CH (Pr-i) SPr-c
Et CH (Pr-i) S (O) Pr-c
Et CH (Pr-i) S (O)₂Pr-c
Et CH (Pr-i) SCH₂CF_Three
Et CH (Pr-i) S (O) CH₂CF_Three
Et CH (Pr-i) S (O)₂CH₂CF_Three
Et CH (Pr-c) SMe
Et CH (Pr-c) S (O) Me
Et CH (Pr-c) S (O)₂Me
Et CH (Pr-c) SEt
Et CH (Pr-c) S (O) Et
Et CH (Pr-c) S (O)₂Et
Et CH (Pr-c) S (= NCN) Et
Et CH (Pr-c) S (O) (= NCN) Et
Et CH (Pr-c) SPr-n
Et CH (Pr-c) S (O) Pr-n
Et CH (Pr-c) S (O)₂Pr-n
Et CH (Pr-c) SPr-i
Et CH (Pr-c) S (O) Pr-i
Et CH (Pr-c) S (O)₂Pr-i
Et CH (Pr-c) SPr-c
Et CH (Pr-c) S (O) Pr-c
Et CH (Pr-c) S (O)₂Pr-c
Et CH (Pr-c) SCH₂CF_Three
Et CH (Pr-c) S (O) CH₂CF_Three
Et CH (Pr-c) S (O)₂CH₂CF_Three
Et CH (Bu-n) SMe
Et CH (Bu-n) S (O) Me
Et CH (Bu-n) S (O)₂Me
Et CH (Bu-n) SEt
Et CH (Bu-n) S (O) Et
Et CH (Bu-n) S (O)₂Et
Et CH (Bu-n) S (= NCN) Et
Et CH (Bu-n) S (O) (= NCN) Et
Et CH (Bu-n) SPr-n
Et CH (Bu-n) S (O) Pr-n
Et CH (Bu-n) S (O)₂Pr-n
Et CH (Bu-n) SPr-i
Et CH (Bu-n) S (O) Pr-i
Et CH (Bu-n) S (O)₂Pr-i
Et CH (Bu-n) SPr-c
Et CH (Bu-n) S (O) Pr-c
Et CH (Bu-n) S (O)₂Pr-c
Et CH (Bu-n) SCH₂CF_Three
Et CH (Bu-n) S (O) CH₂CF_Three
Et CH (Bu-n) S (O)₂CH₂CF_Three
Et CH (F) SMe
Et CH (F) S (O) Me
Et CH (F) S (O)₂Me
Et CH (F) SEt
Et CH (F) S (O) Et
Et CH (F) S (O)₂Et
Et CH (F) S (= NCN) Et
Et CH (F) S (O) (= NCN) Et
Et CH (F) SCH₂CF_Three
Et CH (F) S (O) CH₂CF_Three
Et CH (F) S (O)₂CH₂CF_Three
Et C (F)₂SMe
Et C (F)₂S (O) Me
Et C (F)₂S (O)₂Me
Et C (F)₂SEt
Et C (F)₂S (O) Et
Et C (F)₂S (O)₂Et
Et C (F)₂S (= NCN) Et
Et C (F)₂S (O) (= NCN) Et
Et C (F)₂SCH₂CF_Three
Et C (F)₂S (O) CH₂CF_Three
Et C (F)₂S (O)₂CH₂CF_Three
Et CH (Cl) SMe
Et CH (Cl) S (O) Me
Et CH (Cl) S (O)₂Me
Et CH (Cl) SEt
Et CH (Cl) S (O) Et
Et CH (Cl) S (O)₂Et
Et CH (Cl) S (= NCN) Et
Et CH (Cl) S (O) (= NCN) Et
Et CH (Cl) SCH₂CF_Three
Et CH (Cl) S (O) CH₂CF_Three
Et CH (Cl) S (O)₂CH₂CF_Three
Et C (Cl)₂SMe
Et C (Cl)₂S (O) Me
Et C (Cl)₂S (O)₂Me
Et C (Cl)₂SEt
Et C (Cl)₂S (O) Et
Et C (Cl)₂S (O)₂Et
Et C (Cl)₂S (= NCN) Et
Et C (Cl)₂S (O) (= NCN) Et
Et C (Cl)₂SCH₂CF_Three
Et C (Cl)₂S (O) CH₂CF_Three
Et C (Cl)₂S (O)₂CH₂CF_Three
Et CH (Br) SMe
Et CH (Br) S (O) Me
Et CH (Br) S (O)₂Me
Et CH (Br) SEt
Et CH (Br) S (O) Et
Et CH (Br) S (O)₂Et
Et CH (Br) S (= NCN) Et
Et CH (Br) S (O) (= NCN) Et
Et CH (Br) SCH₂CF_Three
Et CH (Br) S (O) CH₂CF_Three
Et CH (Br) S (O)₂CH₂CF_Three
Et CH (I) SMe
Et CH (I) S (O) Me
Et CH (I) S (O)₂Me
Et CH (I) SEt
Et CH (I) S (O) Et
Et CH (I) S (O)₂Et
Et CH (I) S (= NCN) Et
Et CH (I) S (O) (= NCN) Et
Et CH (I) SCH₂CF_Three
Et CH (I) S (O) CH₂CF_Three
Et CH (I) S (O)₂CH₂CF_Three
Et CH {OC (O) Me} SMe
Et CH {OC (O) Me} S (O) Me
Et CH {OC (O) Me} S (O)₂Me
Et CH {OC (O) OMe} SEt
Et CH {OC (O) OMe} S (O) Et
Et CH {OC (O) OMe} S (O)₂Et
Et CH {OC (O) OMe} S (= NCN) Et
Et CH {OC (O) OMe} S (O) (= NCN) Et
Et CH {OC (O) OEt} SMe
Et CH {OC (O) OEt} S (O) Me
Et CH {OC (O) OEt} S (O)₂Me
Et CH {OC (O) OEt} SEt
Et CH {OC (O) OEt} S (O) Et
Et CH {OC (O) OEt} S (O)₂Et
Et CH {OC (O) OEt} S (= NCN) Et
Et CH {OC (O) OEt} S (O) (= NCN) Et
Et CH (OMe) SMe
Et CH (OMe) S (O) Me
Et CH (OMe) S (O)₂Me
Et CH (OMe) SEt
Et CH (OMe) S (O) Et
Et CH (OMe) S (O)₂Et
Et CH (OMe) S (= NCN) Et
Et CH (OMe) S (O) (= NCN) Et
Et CH (OEt) SMe
Et CH (OEt) S (O) Me
Et CH (OEt) S (O)₂Me
Et CH (OEt) SEt
Et CH (OEt) S (O) Et
Et CH (OEt) S (O)₂Et
Et CH (OEt) S (= NCN) Et
Et CH (OEt) S (O) (= NCN) Et
Et CH (SMe)₂
Et CH (SMe) S (O) Me
Et CH (SMe) S (O)₂Me
Et CH (SMe) SEt
Et CH (SMe) S (O) Et
Et CH (SMe) S (O)₂Et
Et CH (SMe) S (= NCN) Et
Et CH (SMe) S (O) (= NCN) Et
Et CH (SEt) SMe
Et CH (SEt) S (O) Me
Et CH (SEt) S (O)₂Me
Et CH (SEt) SEt
Et CH (SEt) S (O) Et
Et CH (SEt) S (O)₂Et
Et CH (SEt) S (= NCN) Et
Et CH (SEt) S (O) (= NCN) Et
Et CH (CN) SMe
Et CH (CN) S (O) Me
Et CH (CN) S (O)₂Me
Et CH (CN) SEt
Et CH (CN) S (O) Et
Et CH (CN) S (O)₂Et
Et CH (CN) S (= NCN) Et
Et CH (CN) S (O) (= NCN) Et
Et CH {C (O) OMe} SMe
Et CH {C (O) OMe} S (O) Me
Et CH {C (O) OMe} S (O)₂Me
Et CH {C (O) OMe} SMe
Et CH {C (O) OMe} S (O) Me
Et CH {C (O) OMe} S (O)₂Me
Et CH {C (O) OMe} SEt
Et CH {C (O) OMe} S (O) Et
Et CH {C (O) OMe} S (O)₂Et
Et CH {C (O) OMe} S (= NCN) Et
Et CH {C (O) OMe} S (O) (= NCN) Et
Et CH {C (O) OEt} SMe
Et CH {C (O) OEt} S (O) Me
Et CH {C (O) OEt} S (O)₂Me
Et CH {C (O) OEt} SEt
Et CH {C (O) OEt} S (O) Et
Et CH {C (O) OEt} S (O) Et
Et CH {C (O) OEt} S (= NCN) Et
Et CH {C (O) OEt} S (O) (= NCN) Et
Et C (Me)₂SMe
Et C (Me)₂S (O) Me
Et C (Me)₂S (O)₂Me
Et CH₂CH₂SH
Et CH₂CH₂SMe
Et CH₂CH₂S (O) Me
Et CH₂CH₂S (O)₂Me
Et CH₂CH₂SEt
Et CH₂CH₂S (O) Et
Et CH₂CH₂S (O)₂Et
Et CH₂CH₂SPr-n
Et CH₂CH₂S (O) Pr-n
Et CH₂CH₂S (O)₂Pr-n
Et CH₂CH₂SPr-i
Et CH₂CH₂S (O) Pr-i
Et CH₂CH₂S (O)₂Pr-i
Et CH₂CH₂SCH₂CF_Three
Et CH₂CH₂S (O) CH₂CF_Three
Et CH₂CH₂S (O)₂CH₂CF_Three
Et CH₂CH₂SC (O) Me
Et CH (Me) CH₂SMe
Et CH (Me) CH₂S (O) Me
Et CH (Me) CH₂S (O)₂Me
Et CH (Me) CH₂SEt
Et CH (Me) CH₂S (O) Et
Et CH (Me) CH₂S (O)₂Et
Et CH (Me) CH₂SPr-n
Et CH (Me) CH₂S (O) Pr-n
Et CH (Me) CH₂S (O)₂Pr-n
Et CH (Me) CH₂SPr-i
Et CH (Me) CH₂S (O) Pr-i
Et CH (Me) CH₂S (O)₂Pr-i
Et CH (Me) CH₂SCH₂CF_Three
Et CH (Me) CH₂S (O) CH₂CF_Three
Et CH (Me) CH₂S (O)₂CH₂CF_Three
Et CH (Me) CH₂SC (O) Me
Et CH (Et) CH₂SMe
Et CH (Et) CH₂S (O) Me
Et CH (Et) CH₂S (O)₂Me
Et CH (Et) CH₂SEt
Et CH (Et) CH₂S (O) Et
Et CH (Et) CH₂S (O)₂Et
Et CH (Pr-n) CH₂SMe
Et CH (Pr-n) CH₂S (O) Me
Et CH (Pr-n) CH₂S (O)₂Me
Et CH (Pr-n) CH₂SEt
Et CH (Pr-n) CH₂S (O) Et
Et CH (Pr-n) CH₂S (O)₂Et
Et CH (Pr-i) CH₂SMe
Et CH (Pr-i) CH₂S (O) Me
Et CH (Pr-i) CH₂S (O)₂Me
Et CH (Pr-i) CH₂SEt
Et CH (Pr-i) CH₂S (O) Et
Et CH (Pr-i) CH₂S (O)₂Et
Et CH (Pr-c) CH₂SMe
Et CH (Pr-c) CH₂S (O) Me
Et CH (Pr-c) CH₂S (O)₂Me
Et CH (Pr-c) CH₂SEt
Et CH (Pr-c) CH₂S (O) Et
Et CH (Pr-c) CH₂S (O)₂Et
Et CH (Bu-n) CH₂SMe
Et CH (Bu-n) CH₂S (O) Me
Et CH (Bu-n) CH₂S (O)₂Me
Et CH (Bu-n) CH₂SEt
Et CH (Bu-n) CH₂S (O) Et
Et CH (Bu-n) CH₂S (O)₂Et
Et CH (Bu-i) CH₂SMe
Et CH (Bu-i) CH₂S (O) Me
Et CH (Bu-i) CH₂S (O)₂Me
Et CH (Bu-i) CH₂SEt
Et CH (Bu-i) CH₂S (O) Et
Et CH (Bu-i) CH₂S (O)₂Et
Et CH (Bu-s) CH₂SMe
Et CH (Bu-s) CH₂S (O) Me
Et CH (Bu-s) CH₂S (O)₂Me
Et CH (Bu-s) CH₂SEt
Et CH (Bu-s) CH₂S (O) Et
Et CH (Bu-s) CH₂S (O)₂Et
Et CH (Bu-t) CH₂SMe
Et CH (Bu-t) CH₂S (O) Me
Et CH (Bu-t) CH₂S (O)₂Me
Et CH (Bu-t) CH₂SEt
Et CH (Bu-t) CH₂S (O) Et
Et CH (Bu-t) CH₂S (O)₂Et
Et CH (OMe) CH₂SMe
Et CH (OMe) CH₂S (O) Me
Et CH (OMe) CH₂S (O)₂Me
Et CH (OMe) CH₂SEt
Et CH (OMe) CH₂S (O) Et
Et CH (OMe) CH₂S (O)₂Et
Et CH (SMe) CH₂SMe
Et CH (SMe) CH₂S (O) Me
Et CH (SMe) CH₂S (O)₂Me
Et CH (SMe) CH₂SEt
Et CH (SMe) CH₂S (O) Et
Et CH (SMe) CH₂S (O)₂Et
Et CH (CH₂OMe) CH₂SMe
Et CH (CH₂OMe) CH₂S (O) Me
Et CH (CH₂OMe) CH₂S (O)₂Me
Et CH (CH₂OMe) CH₂SEt
Et CH (CH₂OMe) CH₂S (O) Et
Et CH (CH₂OMe) CH₂S (O)₂Et
Et CH (CH₂SMe) CH₂SMe
Et CH (CH₂SMe) CH₂S (O) Me
Et CH (CH₂SMe) CH₂S (O)₂Me
Et CH (CH₂SMe) CH₂SEt
Et CH (CH₂SMe) CH₂S (O) Et
Et CH (CH₂SMe) CH₂S (O)₂Et
Et CH (F) CH₂SMe
Et CH (F) CH₂S (O) Me
Et CH (F) CH₂S (O)₂Me
Et CH (F) CH₂SEt
Et CH (F) CH₂S (O) Et
Et CH (F) CH₂S (O)₂Et
Et C (F)₂CH₂SMe
Et C (F)₂CH₂S (O) Me
Et C (F)₂CH₂S (O)₂Me
Et C (F)₂CH₂SEt
Et C (F)₂CH₂S (O) Et
Et C (F)₂CH₂S (O)₂Et
Et CH (Cl) CH₂SMe
Et CH (Cl) CH₂S (O) Me
Et CH (Cl) CH₂S (O)₂Me
Et CH (Cl) CH₂SEt
Et CH (Cl) CH₂S (O) Et
Et CH (Cl) CH₂S (O)₂Et
Et C (Cl)₂CH₂SMe
Et C (Cl)₂CH₂S (O) Me
Et C (Cl)₂CH₂S (O)₂Me
Et C (Cl)₂CH₂SEt
Et C (Cl)₂CH₂S (O) Et
Et C (Cl)₂CH₂S (O)₂Et
Et CH (Br) CH₂SMe
Et CH (Br) CH₂S (O) Me
Et CH (Br) CH₂S (O)₂Me
Et CH (Br) CH₂SEt
Et CH (Br) CH₂S (O) Et
Et CH (Br) CH₂S (O)₂Et
Et CH (I) CH₂SMe
Et CH (I) CH₂S (O) Me
Et CH (I) CH₂S (O)₂Me
Et CH (I) CH₂SEt
Et CH (I) CH₂S (O) Et
Et CH (I) CH₂S (O)₂Et
Et CH (CN) CH₂SMe
Et CH (CN) CH₂S (O) Me
Et CH (CN) CH₂S (O)₂Me
Et CH (CN) CH₂SEt
Et CH (CN) CH₂S (O) Et
Et CH (CN) CH₂S (O)₂Et
Et CH {C (O) OMe} CH₂SMe
Et CH {C (O) OMe} CH₂S (O) Me
Et CH {C (O) OMe} CH₂S (O)₂Me
Et CH {C (O) OMe} CH₂SEt
Et CH {C (O) OMe} CH₂S (O) Et
Et CH {C (O) OMe} CH₂S (O)₂Et
Et CH {C (O) OEt} CH₂SMe
Et CH {C (O) OEt} CH₂S (O) Me
Et CH {C (O) OEt} CH₂S (O)₂Me
Et CH {C (O) OEt} CH₂SEt
Et CH {C (O) OEt} CH₂S (O) Et
Et CH {C (O) OEt} CH₂S (O)₂Et
Et CH (Ph) CH₂SMe
Et CH (Ph) CH₂S (O) Me
Et CH (Ph) CH₂S (O)₂Me
Et CH (Ph) CH₂SEt
Et CH (Ph) CH₂S (O) Et
Et CH (Ph) CH₂S (O)₂Et
Et C (Me)₂CH₂SMe
Et C (Me)₂CH₂S (O) Me
Et C (Me)₂CH₂S (O)₂Me
Et C (Me)₂CH₂SEt
Et C (Me)₂CH₂S (O) Et
Et C (Me)₂CH₂S (O)₂Et
Et C (Et)₂CH₂SMe
Et C (Et)₂CH₂S (O) Me
Et C (Et)₂CH₂S (O)₂Me
Et C (Et)₂CH₂SEt
Et C (Et)₂CH₂S (O) Et
Et C (Et)₂CH₂S (O)₂Et
Et C (= CH₂) CH₂SMe
Et C (= CH₂) CH₂S (O) Me
Et C (= CH₂) CH₂S (O)₂Me
Et C (= CH₂) CH₂SEt
Et C (= CH₂) CH₂S (O) Et
Et C (= CH₂) CH₂S (O)₂Et
Et CH₂CH₂CH₂SEt
Et CH₂CH₂CH₂S (O) Et
Et CH₂CH₂CH₂S (O)₂Et
Et CH (Me) CH₂CH₂SEt
Et CH (Me) CH₂CH₂S (O) Et
Et CH (Me) CH₂CH₂S (O)₂Et
Et CH₂CH (Me) CH₂SEt
Et CH₂CH (Me) CH₂S (O) Et
Et CH₂CH (Me) CH₂S (O)₂Et
Et CH₂CH₂CH (Me) SEt
Et CH₂CH₂CH (Me) S (O) Et
Et CH₂CH₂CH (Me) S (O)₂Et
Et CH₂CH₂CH₂SPr-n
Et CH₂CH₂CH₂S (O) Pr-n
Et CH₂CH₂CH₂S (O)₂Pr-n
Et CH (Me) CH₂CH₂SPr-n
Et CH (Me) CH₂CH₂S (O) Pr-n
Et CH (Me) CH₂CH₂S (O)₂Pr-n
Et CH₂CH (Me) CH₂SPr-n
Et CH₂CH (Me) CH₂S (O) Pr-n
Et CH₂CH (Me) CH₂S (O)₂Pr-n
Et CH₂CH₂CH₂CH₂SMe
Et CH₂CH₂CH₂CH₂S (O) Me
Et CH₂CH₂CH₂CH₂S (O)₂Me
Et CH₂CH₂CH₂CH₂SEt
Et CH₂CH₂CH₂CH₂S (O) Et
Et CH₂CH₂CH₂CH₂S (O)₂Et
Et CH₂CH₂CH₂CH₂SPr-n
Et CH₂CH₂CH₂CH₂S (O) Pr-n
Et CH₂CH₂CH₂CH₂S (O)₂Pr-n
Et CH₂CH (Me) SMe
Et CH₂CH (Me) S (O) Me
Et CH₂CH (Me) S (O)₂Me
Et CH₂CH (Me) SEt
Et CH₂CH (Me) S (O) Et
Et CH₂CH (Me) S (O)₂Et
Et CH₂CH (Et) SMe
Et CH₂CH (Et) S (O) Me
Et CH₂CH (Et) S (O)₂Me
Et CH₂CH (Et) SEt
Et CH₂CH (Et) S (O) Et
Et CH₂CH (Et) S (O)₂Et
Et CH₂CH (Pr-n) SMe
Et CH₂CH (Pr-n) S (O) Me
Et CH₂CH (Pr-n) S (O)₂Me
Et CH₂CH (Pr-n) SEt
Et CH₂CH (Pr-n) S (O) Et
Et CH₂CH (Pr-n) S (O)₂Et
Et CH₂CH (Pr-i) SMe
Et CH₂CH (Pr-i) S (O) Me
Et CH₂CH (Pr-i) S (O)₂Me
Et CH₂CH (Pr-i) SEt
Et CH₂CH (Pr-i) S (O) Et
Et CH₂CH (Pr-i) S (O)₂Et
Et CH₂CH (Pr-c) SMe
Et CH₂CH (Pr-c) S (O) Me
Et CH₂CH (Pr-c) S (O)₂Me
Et CH₂CH (Pr-c) SEt
Et CH₂CH (Pr-c) S (O) Et
Et CH₂CH (Pr-c) S (O)₂Et
Et CH₂CH (Bu-n) SMe
Et CH₂CH (Bu-n) S (O) Me
Et CH₂CH (Bu-n) S (O)₂Me
Et CH₂CH (Bu-n) SEt
Et CH₂CH (Bu-n) S (O) Et
Et CH₂CH (Bu-n) S (O)₂Et
Et CH₂CH (Bu-i) SMe
Et CH₂CH (Bu-i) S (O) Me
Et CH₂CH (Bu-i) S (O)₂Me
Et CH₂CH (Bu-i) SEt
Et CH₂CH (Bu-i) S (O) Et
Et CH₂CH (Bu-i) S (O)₂Et
Et CH₂CH (Bu-s) SMe
Et CH₂CH (Bu-s) S (O) Me
Et CH₂CH (Bu-s) S (O)₂Me
Et CH₂CH (Bu-s) SEt
Et CH₂CH (Bu-s) S (O) Et
Et CH₂CH (Bu-s) S (O)₂Et
Et CH₂CH (Bu-t) SMe
Et CH₂CH (Bu-t) S (O) Me
Et CH₂CH (Bu-t) S (O)₂Me
Et CH₂CH (Bu-t) SEt
Et CH₂CH (Bu-t) S (O) Et
Et CH₂CH (Bu-t) S (O)₂Et
Et CH₂C (Et)₂SMe
Et CH₂C (Et)₂S (O) Me
Et CH₂C (Et)₂S (O)₂Me
Et CH₂C (Et)₂SEt
Et CH₂C (Et)₂S (O) Et
Et CH₂C (Et)₂S (O)₂Et
Et CH (Et) CH (Me) SMe
Et CH (Et) CH (Me) S (O) Me
Et CH (Et) CH (Me) S (O)₂Me
Et CH (Et) CH (Me) SEt
Et CH (Et) CH (Me) S (O) Et
Et CH (Et) CH (Me) S (O)₂Et
Et CH (Et) CH (Et) SMe
Et CH (Et) CH (Et) S (O) Me
Et CH (Et) CH (Et) S (O)₂Me
Et CH (Et) CH (Et) SEt
Et CH (Et) CH (Et) S (O) Et
Et CH (Et) CH (Et) S (O)₂Et
Et CH = CHSMe
Et CH₂CH (SMe)₂
Et CH₂CH₂SC (O) Me
Et C (CH₂) CH₂C (O) OH
Et C (= NOMe) Me
Et C (= NOMe) Et
Et C (= NOMe) Pr-n
Et C (= NOEt) Me
Et C (= NOPr-n) Me
Et C (= NOPr-i) Me
Et C (= NOBu-n) Me
Et C (= NOCH₂Ph) Me
Et C (= NOMe) C (= NOMe) Me
Et C (= NOMe) CH₂OCH₂CF_Three
Et C (= NOMe) CH₂SMe
Et C (= NOMe) CH₂S (O) Me
Et C (= NOMe) CH₂S (O)₂Me
Et C (= NOMe) CH₂SEt
Et C (= NOMe) CH₂S (O) Et
Et C (= NOMe) CH₂S (O)₂Et
Et C (= NOMe) CH₂SCF_Three
Et C (= NOMe) CH₂S (O) CF_Three
Et C (= NOMe) CH₂S (O)₂CF_Three
Et C (= NOMe) CH₂SCH₂CF_Three
Et C (= NOMe) CH₂S (O) CH₂CF_Three
Et C (= NOMe) CH₂S (O)₂CH₂CF_Three
Et C (= NOEt) CH₂SMe
Et C (= NOEt) CH₂S (O) Me
Et C (= NOEt) CH₂S (O)₂Me
Et C (= NOPr-n) CH₂SMe
Et C (= NOPr-n) CH₂S (O) Me
Et C (= NOPr-n) CH₂S (O)₂Me
Et C (= NOPr-i) CH₂SMe
Et C (= NOPr-i) CH₂S (O) Me
Et C (= NOPr-i) CH₂S (O)₂Me
Et C (= NOBu-n) CH₂SMe
Et C (= NOBu-n) CH₂S (O) Me
Et C (= NOBu-n) CH₂S (O)₂Me
Et C (= NOCH₂Ph) CH₂SMe
Et C (= NOCH₂Ph) CH₂S (O) Me
Et C (= NOCH₂Ph) CH₂S (O)₂Me
Et C (= NOCH₂CH = CH₂) CH₂SMe
Et C (= NOCH₂OMe) CH₂SMe
Et C (= NOCH₂CH₂OMe) CH₂SMe
Et C {= NOCH₂CH₂Si (Me)_Three} CH₂SMe
Et CH₂CH (= NOMe)
Et CH₂C (= NOMe) Me
Et CH₂C (= NOMe) Et
Et CH₂C (= NOMe) Pr-n
Et CH₂C (= NOMe) Pr-i
Et CH₂C (= NOMe) Bu-n
Et CH₂C (= NOMe) Bu-i
Et CH₂C (= NOMe) Bu-s
Et CH₂C (= NOMe) Bu-t
Et CH₂C (= NOMe) CF_Three
Et CH₂C (= NOCH_Three) CH₂SCH_Three
Et CH (SMe) C (= NOMe) Me
Et CH {S (O) Me} C (= NOMe) Me
Et CH {S (O)₂Me} C (= NOMe) Me
Et CH (SEt) C (= NOMe) Me
Et CH {S (O) Et} C (= NOMe) Me
Et CH {S (O)₂Et} C (= NOMe) Me
Et CH₂NH₂
Et CH₂NMe₂
Et CH₂NHC (O) Me
Et CH₂NHC (O) CF_Three
Et CH₂NHC (O) CH₂OMe
Et CH₂NHC (O) CH₂SMe
Et CH₂NHC (O) OMe
Et CH₂NHC (O) OBu-t
Et CH₂NHSO₂Me
Et CH₂NHSO₂NMe₂
Et CH₂NHSO₂CF_Three
Et CH₂N (Me) C (O) Me
Et CH₂N (Me) C (O) OMe
Et CH₂N (Me) C (O) OBu-t
Et CH₂N (Me) SO₂Me
Et CH (Me) NHC (O) OBu-t
Et CH (CH₂SMe) NH₂
Et CH (CH₂SMe) NHC (O) Me
Et CH (CH₂SMe) NHC (O) OMe
Et CH (CH₂SMe) NHC (O) OBu-t
Et CH (CH₂SMe) NHSO₂Me
Et CH₂NHC (O) NHMe
Et CH₂NHC (O) NHEt
Et CH₂NHC (O) NHPr-n
Et CH₂NHC (O) NHPr-i
Et CH₂NHC (O) NHPr-c
Et CH₂NHC (S) NHMe
Et CH₂NHC (S) NHEt
Et CH₂NHC (S) NHPr-n
Et CH₂NHC (S) NHPr-i
Et CH₂NHC (S) NHPr-c
Et CH₂CH₂NHC (O) OBu-t
Et CH₂P (O) (OMe)₂
Et CH₂P (O) (OEt)₂
Et SMe
Et OBu-t
Et O {D2-108 (4-NO₂)}
Et NH₂
Et NHCH₂SMe
Et NHCH₂CH₂SMe
Et N (Me) CH₂SMe
Et N (Me) CH₂CH₂SMe
Et NHCH₂CH₂CH₂SMe
Et NHMe
Et NHEt
Et NPr-n
Et NHPr-i
Et NHCH₂C (O) OMe
Et NHCH₂CF_Three
Et N (Me) CH₂CF_Three
Et NHC (O) OEt
Et NHC (O) CCl_Three
Et NHC (O) CH₂SMe
Et N (CH₂CH_Three) C (O) CH₂SCH_Three
Et NHS (O)₂(D2-108a)
Et NHPh
Et NH (D2-1a)
Et NH (D2-2a)
Et NH (D2-2b)
Et NH (D2-4a)
Et NH {D2-4b}
Et NH (D2-5a)
Et NH (D2-5b)
Et NH (D2-5c)
Et NH (D2-6a)
Et NH (D2-6b)
Et NH (D2-6c)
Et NH (D2-7a)
Et NH (D2-8a)
Et NH (D2-8b)
Et NH (D2-8c)
Et NH (D2-9a)
Et NH (D2-9b)
Et NH (D2-9c)
Et NH (D2-10a)
Et NH (D2-10b)
Et NH (D2-10c)
Et NH (D2-11a)
Et NH (D2-12a)
Et NH (D2-12b)
Et NH (D2-12c)
Et NH (D2-13a)
Et NH (D2-13b)
Et NH (D2-14a)
Et NH (D2-14b)
Et NH (D2-15a)
Et NH (D2-15b)
Et NH (D2-16a)
Et NH (D2-17a)
Et NH (D2-18a)
Et NH (D2-19a)
Et NH (D2-20a)
Et NH (D2-21a)
Et NH (D2-21b)
Et NH (D2-22a)
Et NH (D2-23a)
Et NH (D2-23b)
Et NH (D2-24a)
Et NH (D2-25a)
Et NH (D2-26a)
Et NH (D2-27a)
Et NH (D2-28a)
Et NH (D2-29a)
Et NH (D2-30a)
Et NH (D2-31a)
Et NH (D2-32a)
Et NH (D2-33a)
Et NH (D2-34a)
Et NH (D2-35a)
Et NH (D2-35b)
Et NH (D2-36a)
Et NH (D2-37a)
Et NH (D2-38a)
Et NH (D2-39a)
Et NH (D2-40a)
Et NH (D2-40b)
Et NH (D2-40c)
Et NH (D2-41a)
Et NH (D2-42a)
Et NH (D2-43a)
Et NH (D2-45a)
Et NH (D2-49a)
Et NH (D2-51a)
Et NH (D2-59a)
Et NH (D2-61a)
Et NH (D2-79a)
Et NH (D2-80a)
Et NH {D2-108b (2-Cl)}
Et NH {D2-108b (3-Cl)}
Et NH {D2-108b (4-Cl)}
Et NH {D2-108b (2-Me)}
Et NH {D2-108b (3-Me)}
Et NH {D2-108b (4-Me)}
Et N (Me) Ph
Et N (Me) (D2-1a)
Et N (Me) (D2-2a)
Et N (Me) (D2-2b)
Et N (Me) (D2-4a)
Et N (Me) {D2-4b}
Et N (Me) (D2-5a)
Et N (Me) (D2-5b)
Et N (Me) (D2-5c)
Et N (Me) (D2-6a)
Et N (Me) (D2-6b)
Et N (Me) (D2-6c)
Et N (Me) (D2-7a)
Et N (Me) (D2-8a)
Et N (Me) (D2-8b)
Et N (Me) (D2-8c)
Et N (Me) (D2-9a)
Et N (Me) (D2-9b)
Et N (Me) (D2-9c)
Et N (Me) (D2-10a)
Et N (Me) (D2-10b)
Et N (Me) (D2-10c)
Et N (Me) (D2-11a)
Et N (Me) (D2-12a)
Et N (Me) (D2-12b)
Et N (Me) (D2-12c)
Et N (Me) (D2-13a)
Et N (Me) (D2-13b)
Et N (Me) (D2-14a)
Et N (Me) (D2-14b)
Et N (Me) (D2-15a)
Et N (Me) (D2-15b)
Et N (Me) (D2-16a)
Et N (Me) (D2-17a)
Et N (Me) (D2-18a)
Et N (Me) (D2-19a)
Et N (Me) (D2-20a)
Et N (Me) (D2-21a)
Et N (Me) (D2-21b)
Et N (Me) (D2-22a)
Et N (Me) (D2-23a)
Et N (Me) (D2-23b)
Et N (Me) (D2-24a)
Et N (Me) (D2-25a)
Et N (Me) (D2-26a)
Et N (Me) (D2-27a)
Et N (Me) (D2-28a)
Et N (Me) (D2-29a)
Et N (Me) (D2-30a)
Et N (Me) (D2-31a)
Et N (Me) (D2-32a)
Et N (Me) (D2-33a)
Et N (Me) (D2-34a)
Et N (Me) (D2-35a)
Et N (Me) (D2-35b)
Et N (Me) (D2-36a)
Et N (Me) (D2-37a)
Et N (Me) (D2-38a)
Et N (Me) (D2-39a)
Et N (Me) (D2-40a)
Et N (Me) (D2-40b)
Et N (Me) (D2-40c)
Et N (Me) (D2-41a)
Et N (Me) (D2-42a)
Et N (Me) (D2-43a)
Et N (Me) (D2-45a)
Et N (Me) (D2-49a)
Et N (Me) (D2-51a)
Et N (Me) (D2-59a)
Et N (Me) (D2-61a)
Et N (Me) (D2-79a)
Et N (Me) (D2-80a)
Et N (Me) {D2-108b (2-Cl)}
Et N (Me) {D2-108b (3-Cl)}
Et N (Me) {D2-108b (4-Cl)}
Et N (Me) {D2-108b (2-Me)}
Et N (Me) {D2-108b (3-Me)}
Et N (Me) {D2-108b (4-Me)}
Et D2-4a
Et D2-9b
Et D2-19a
Et D2-32b (2-Br)
Et D2-33a
Et D2-33b (2-OMe)
Et D2-33b (6-CN)
Et D2-34a
Et D2-35b
Et D2-38b (4-SMe)
Et D2-39b (5-Me)
Et D2-81a
Et D2-81b
Et D2-82a
Et D2-82b
Et D2-87a
Et D2-103b
Et D2-103c
Et D2-103d
Et D2-103e
Et D2-103f
Et D2-103g
Et D2-103h
Et D2-103i
Et D2-108b (2-Cl)
Et D2-108b (3-Cl)
Et D2-108b (4-Cl)
Et D2-108b (2-SMe)
Et D2-108b (3-SMe)
Et D2-108b (4-SMe)
Et D2-108b (3-SCF_Three)
Et D2-108b (3,4-OCF₂O-)
Et CH₂(D2-2a)
Et CH₂(D2-28a)
Et CH₂(D2-32a)
Et CH₂(D2-33a)
Et CH₂{D2-33b (6-Cl)}
Et CH₂(D2-34a)
Et CH₂(D2-87a)
Et CH₂(D2-93a)
Et CH₂(D2-98a)
Et CH₂{D2-108b (2,3-OCH₂O-)}
n-Pr CH (Me) SMe
n-Pr CH (Me) S (O) Me
n-Pr CH (Me) S (O)₂Me
n-Pr CH (Me) SEt
n-Pr CH (Me) S (O) Et
n-Pr CH (Me) S (O)₂Et
n-Pr CH₂CH₂SMe
n-Pr CH₂CH₂S (O) Me
n-Pr CH₂CH₂S (O)₂Me
n-Pr CH (Me) CH₂SMe
n-Pr CH (Me) CH₂S (O) Me
n-Pr CH (Me) CH₂S (O)₂Me
n-Pr OBu-t
i-Pr CH (Me) SMe
i-Pr CH (Me) S (O) Me
i-Pr CH (Me) S (O)₂Me
i-Pr CH (Me) SEt
i-Pr CH (Me) S (O) Et
i-Pr CH (Me) S (O)₂Et
i-Pr CH₂CH₂SMe
i-Pr CH₂CH₂S (O) Me
i-Pr CH₂CH₂S (O)₂Me
i-Pr CH (Me) CH₂SMe
i-Pr CH (Me) CH₂S (O) Me
i-Pr CH (Me) CH₂S (O)₂Me
i-Pr OBu-t
CH₂Pr-c CH (Me) SMe
CH₂Pr-c CH (Me) S (O) Me
CH₂Pr-c CH (Me) S (O)₂Me
CH₂Pr-c CH (Me) SEt
CH₂Pr-c CH (Me) S (O) Et
CH₂Pr-c CH (Me) S (O)₂Et
CH₂Pr-c CH₂CH₂SMe
CH₂Pr-c CH₂CH₂S (O) Me
CH₂Pr-c CH₂CH₂S (O)₂Me
CH₂Pr-c CH (Me) CH₂SMe
CH₂Pr-c CH (Me) CH₂S (O) Me
CH₂Pr-c CH (Me) CH₂S (O)₂Me
CH₂Pr-c OBu-t
CH₂CH = CH₂                 CH (Me) SMe
CH₂CH = CH₂                 CH (Me) S (O) Me
CH₂CH = CH₂                 CH (Me) S (O)₂Me
CH₂CH = CH₂                 CH (Me) SEt
CH₂CH = CH₂                 CH (Me) S (O) Et
CH₂CH = CH₂                 CH (Me) S (O)₂Et
CH₂CH = CH₂                 CH₂CH₂SMe
CH₂CH = CH₂                 CH₂CH₂S (O) Me
CH₂CH = CH₂                 CH₂CH₂S (O)₂Me
CH₂CH = CH₂                 CH (Me) CH₂SMe
CH₂CH = CH₂               CH (Me) CH₂S (O) Me
CH₂CH = CH₂              CH (Me) CH₂S (O)₂Me
CH₂C≡CH CH (Me) SMe
CH₂C≡CH CH (Me) S (O) Me
CH₂C≡CH CH (Me) S (O)₂Me
CH₂C≡CH CH (Me) SEt
CH₂C≡CH CH (Me) S (O) Et
CH₂C≡CH CH (Me) S (O)₂Et
CH₂C≡CH CH₂CH₂SMe
CH₂C≡CH CH₂CH₂S (O) Me
CH₂C≡CH CH₂CH₂S (O)₂Me
CH₂C≡CH CH (Me) CH₂SMe
CH₂C≡CH CH (Me) CH₂S (O) Me
CH₂C≡CH CH (Me) CH₂S (O)₂Me
CH₂OMe CH (Me) SMe
CH₂OMe CH (Me) S (O) Me
CH₂OMe CH (Me) S (O)₂Me
CH₂OMe CH (Me) SEt
CH₂OMe CH (Me) S (O) Et
CH₂OMe CH (Me) S (O)₂Et
CH₂OMe CH₂CH₂SMe
CH₂OMe CH₂CH₂S (O) Me
CH₂OMe CH₂CH₂S (O)₂Me
CH₂OMe CH (Me) CH₂SMe
CH₂OMe CH (Me) CH₂S (O) Me
CH₂OMe CH (Me) CH₂S (O)₂Me
CH₂OEt CH (Me) SEt
CH₂OEt CH (Me) S (O) Et
CH₂OEt CH (Me) S (O)₂Et
CH₂CH₂OMe CH (Me) SEt
CH₂CH₂OMe CH (Me) S (O) Et
CH₂CH₂OMe CH (Me) S (O)₂Et
CH₂CN CH (Me) SMe
CH₂CN CH (Me) S (O) Me
CH₂CN CH (Me) S (O)₂Me
CH₂CN CH (Me) SEt
CH₂CN CH (Me) S (O) Et
CH₂CN CH (Me) S (O)₂Et
CH₂CN CH₂CH₂SMe
CH₂CN CH₂CH₂S (O) Me
CH₂CN CH₂CH₂S (O)₂Me
CH₂CN CH (Me) CH₂SMe
CH₂CN CH (Me) CH₂S (O) Me
CH₂CN CH (Me) CH₂S (O)₂Me
CH₂C (O) OMe CH₂SMe
CH₂C (O) OMe CH₂S (O) Me
CH₂C (O) OMe CH₂S (O)₂Me
CH₂C (O) OMe CH₂SEt
CH₂C (O) OMe CH₂S (O) Et
CH₂C (O) OMe CH₂S (O)₂Et
CH₂C (O) OMe CH₂SPr-n
CH₂C (O) OMe CH₂S (O) Pr-n
CH₂C (O) OMe CH₂S (O)₂Pr-n
CH₂C (O) OMe CH₂SPr-i
CH₂C (O) OMe CH₂S (O) Pr-i
CH₂C (O) OMe CH₂S (O)₂Pr-i
CH₂C (O) OMe CH₂SPr-c
CH₂C (O) OMe CH₂S (O) Pr-c
CH₂C (O) OMe CH₂S (O)₂Pr-c
CH₂C (O) OMe CH₂SCH₂CH = CH₂
CH₂C (O) OMe CH₂S (O) CH₂CH = CH₂
CH₂C (O) OMe CH₂S (O)₂CH₂CH = CH₂
CH₂C (O) OMe CH₂SCH₂C≡CH
CH₂C (O) OMe CH₂S (O) CH₂C≡CH
CH₂C (O) OMe CH₂S (O)₂CH₂C≡CH
CH₂C (O) OMe CH₂SCH₂CF_Three
CH₂C (O) OMe CH₂S (O) CH₂CF_Three
CH₂C (O) OMe CH₂S (O)₂CH₂CF_Three
CH₂C (O) OMe CH₂SCH₂CH (OMe)₂
CH₂C (O) OMe CH₂SCH₂CH (= NOMe)
CH₂C (O) OMe CH (Me) SMe
CH₂C (O) OMe CH (Me) S (O) Me
CH₂C (O) OMe CH (Me) S (O)₂Me
CH₂C (O) OMe CH (Me) SEt
CH₂C (O) OMe CH (Me) S (O) Et
CH₂C (O) OMe CH (Me) S (O)₂Et
CH₂C (O) OMe CH (Me) S (= NCN) Et
CH₂C (O) OMe CH (Me) S (O) (= NCN) Et
CH₂C (O) OMe CH (Me) SPr-n
CH₂C (O) OMe CH (Me) S (O) Pr-n
CH₂C (O) OMe CH (Me) S (O)₂Pr-n
CH₂C (O) OMe CH (Me) SPr-i
CH₂C (O) OMe CH (Me) S (O) Pr-i
CH₂C (O) OMe CH (Me) S (O)₂Pr-i
CH₂C (O) OMe CH (Me) SBu-t
CH₂C (O) OMe CH (Me) S (O) Bu-t
CH₂C (O) OMe CH (Me) S (O)₂Bu-t
CH₂C (O) OMe CH (Me) SCH₂Pr-c
CH₂C (O) OMe CH (Me) S (O) CH₂Pr-c
CH₂C (O) OMe CH (Me) S (O)₂CH₂Pr-c
CH₂C (O) OMe CH (Me) SCH₂OMe
CH₂C (O) OMe CH (Me) SCH₂SMe
CH₂C (O) OMe CH (Me) S (O) CH₂SMe
CH₂C (O) OMe CH (Me) S (O)₂CH₂SMe
CH₂C (O) OMe CH (Me) SCH₂C = CH₂
CH₂C (O) OMe CH (Me) S (O) CH₂C = CH₂
CH₂C (O) OMe CH (Me) S (O)₂CH₂C = CH₂
CH₂C (O) OMe CH (Me) SCH₂C≡CH
CH₂C (O) OMe CH (Me) S (O) CH₂C≡CH
CH₂C (O) OMe CH (Me) S (O)₂CH₂C≡CH
CH₂C (O) OMe CH (Me) SCH₂C (O) NHMe
CH₂C (O) OMe CH (Me) S (O) CH₂C (O) NHMe
CH₂C (O) OMe CH (Me) S (O)₂CH₂C (O) NHMe
CH₂C (O) OMe CH (Me) SCH₂C (O) OMe
CH₂C (O) OMe CH (Me) S (O) CH₂C (O) OMe
CH₂C (O) OMe CH (Me) S (O)₂CH₂C (O) OMe
CH₂C (O) OMe CH (Me) SCH₂CH₂CH₂Cl
CH₂C (O) OMe CH (Me) S (O) CH₂CH₂CH₂Cl
CH₂C (O) OMe CH (Me) S (O)₂CH₂CH₂CH₂Cl
CH₂C (O) OMe CH (Me) SCH₂CF_Three
CH₂C (O) OMe CH (Me) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Me) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Me) SCH₂Ph
CH₂C (O) OMe CH (Me) S (O) CH₂Ph
CH₂C (O) OMe CH (Me) S (O)₂CH₂Ph
CH₂C (O) OMe CH (Me) SCH₂(D2-34a)
CH₂C (O) OMe H (Me) S (O) CH₂(D2-34a)
CH₂C (O) OMe H (Me) S (O)₂CH₂(D2-34a)
CH₂C (O) OMe CH (CH_Three) SCH₂Si (CH_Three)_Three
CH₂C (O) OMe CH (Me) SCN
CH₂C (O) OMe CH (Me) SCH₂CN
CH₂C (O) OMe CH (Me) SC (O) Me
CH₂C (O) OMe CH (Me) S (D2-12a)
CH₂C (O) OMe CH (Me) S (D2-32a)
CH₂C (O) OMe CH (Me) S {D2-32b (3-NO₂)}
CH₂C (O) OMe CH (Me) S {D2-32b (3-CF_Three)}
CH₂C (O) OMe CH (Me) S (D2-37a)
CH₂C (O) OMe CH (Me) S (D2-51a)
CH₂C (O) OMe CH (Et) SMe
CH₂C (O) OMe CH (Et) S (O) Me
CH₂C (O) OMe CH (Et) S (O)₂Me
CH₂C (O) OMe CH (Et) SEt
CH₂C (O) OMe CH (Et) S (O) Et
CH₂C (O) OMe CH (Et) S (O)₂Et
CH₂C (O) OMe CH (Et) SCH₂CF_Three
CH₂C (O) OMe CH (Et) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Et) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Pr-n) SMe
CH₂C (O) OMe CH (Pr-n) S (O) Me
CH₂C (O) OMe CH (Pr-n) S (O)₂Me
CH₂C (O) OMe CH (Pr-n) SEt
CH₂C (O) OMe CH (Pr-n) S (O) Et
CH₂C (O) OMe CH (Pr-n) S (O)₂Et
CH₂C (O) OMe CH (Pr-n) S (= NCN) Et
CH₂C (O) OMe CH (Pr-n) S (O) (= NCN) Et
CH₂C (O) OMe CH (Pr-n) SPr-n
CH₂C (O) OMe CH (Pr-n) S (O) Pr-n
CH₂C (O) OMe CH (Pr-n) S (O)₂Pr-n
CH₂C (O) OMe CH (Pr-n) SPr-i
CH₂C (O) OMe CH (Pr-n) S (O) Pr-i
CH₂C (O) OMe CH (Pr-n) S (O)₂Pr-i
CH₂C (O) OMe CH (Pr-n) SPr-c
CH₂C (O) OMe CH (Pr-n) S (O) Pr-c
CH₂C (O) OMe CH (Pr-n) S (O)₂Pr-c
CH₂C (O) OMe CH (Pr-n) SCH₂CF_Three
CH₂C (O) OMe CH (Pr-n) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Pr-n) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Pr-i) SMe
CH₂C (O) OMe CH (Pr-i) S (O) Me
CH₂C (O) OMe CH (Pr-i) S (O)₂Me
CH₂C (O) OMe CH (Pr-i) SEt
CH₂C (O) OMe CH (Pr-i) S (O) Et
CH₂C (O) OMe CH (Pr-i) S (O)₂Et
CH₂C (O) OMe CH (Pr-i) S (= NCN) Et
CH₂C (O) OMe CH (Pr-i) S (O) (= NCN) Et
CH₂C (O) OMe CH (Pr-i) SPr-n
CH₂C (O) OMe CH (Pr-i) S (O) Pr-n
CH₂C (O) OMe CH (Pr-i) S (O)₂Pr-n
CH₂C (O) OMe CH (Pr-i) SPr-i
CH₂C (O) OMe CH (Pr-i) S (O) Pr-i
CH₂C (O) OMe CH (Pr-i) S (O)₂Pr-i
CH₂C (O) OMe CH (Pr-i) SPr-c
CH₂C (O) OMe CH (Pr-i) S (O) Pr-c
CH₂C (O) OMe CH (Pr-i) S (O)₂Pr-c
CH₂C (O) OMe CH (Pr-i) SCH₂CF_Three
CH₂C (O) OMe CH (Pr-i) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Pr-i) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Pr-c) SMe
CH₂C (O) OMe CH (Pr-c) S (O) Me
CH₂C (O) OMe CH (Pr-c) S (O)₂Me
CH₂C (O) OMe CH (Pr-c) SEt
CH₂C (O) OMe CH (Pr-c) S (O) Et
CH₂C (O) OMe CH (Pr-c) S (O)₂Et
CH₂C (O) OMe CH (Pr-c) S (= NCN) Et
CH₂C (O) OMe CH (Pr-c) S (O) (= NCN) Et
CH₂C (O) OMe CH (Pr-c) SPr-n
CH₂C (O) OMe CH (Pr-c) S (O) Pr-n
CH₂C (O) OMe CH (Pr-c) S (O)₂Pr-n
CH₂C (O) OMe CH (Pr-c) SPr-i
CH₂C (O) OMe CH (Pr-c) S (O) Pr-i
CH₂C (O) OMe CH (Pr-c) S (O)₂Pr-i
CH₂C (O) OMe CH (Pr-c) SPr-c
CH₂C (O) OMe CH (Pr-c) S (O) Pr-c
CH₂C (O) OMe CH (Pr-c) S (O)₂Pr-c
CH₂C (O) OMe CH (Pr-c) SCH₂CF_Three
CH₂C (O) OMe CH (Pr-c) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Pr-c) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Bu-n) SMe
CH₂C (O) OMe CH (Bu-n) S (O) Me
CH₂C (O) OMe CH (Bu-n) S (O)₂Me
CH₂C (O) OMe CH (Bu-n) SEt
CH₂C (O) OMe CH (Bu-n) S (O) Et
CH₂C (O) OMe CH (Bu-n) S (O)₂Et
CH₂C (O) OMe CH (Bu-n) S (= NCN) Et
CH₂C (O) OMe CH (Bu-n) S (O) (= NCN) Et
CH₂C (O) OMe CH (Bu-n) SPr-n
CH₂C (O) OMe CH (Bu-n) S (O) Pr-n
CH₂C (O) OMe CH (Bu-n) S (O)₂Pr-n
CH₂C (O) OMe CH (Bu-n) SPr-i
CH₂C (O) OMe CH (Bu-n) S (O) Pr-i
CH₂C (O) OMe CH (Bu-n) S (O)₂Pr-i
CH₂C (O) OMe CH (Bu-n) SPr-c
CH₂C (O) OMe CH (Bu-n) S (O) Pr-c
CH₂C (O) OMe CH (Bu-n) S (O)₂Pr-c
CH₂C (O) OMe CH (Bu-n) SCH₂CF_Three
CH₂C (O) OMe CH (Bu-n) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Bu-n) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (F) SMe
CH₂C (O) OMe CH (F) S (O) Me
CH₂C (O) OMe CH (F) S (O)₂Me
CH₂C (O) OMe CH (F) SEt
CH₂C (O) OMe CH (F) S (O) Et
CH₂C (O) OMe CH (F) S (O)₂Et
CH₂C (O) OMe CH (F) S (= NCN) Et
CH₂C (O) OMe CH (F) S (O) (= NCN) Et
CH₂C (O) OMe CH (F) SCH₂CF_Three
CH₂C (O) OMe CH (F) S (O) CH₂CF_Three
CH₂C (O) OMe CH (F) S (O)₂CH₂CF_Three
CH₂C (O) OMe C (F)₂SMe
CH₂C (O) OMe C (F)₂S (O) Me
CH₂C (O) OMe C (F)₂S (O)₂Me
CH₂C (O) OMe C (F)₂SEt
CH₂C (O) OMe C (F)₂S (O) Et
CH₂C (O) OMe C (F)₂S (O)₂Et
CH₂C (O) OMe C (F)₂S (= NCN) Et
CH₂C (O) OMe C (F)₂S (O) (= NCN) Et
CH₂C (O) OMe C (F)₂SCH₂CF_Three
CH₂C (O) OMe C (F)₂S (O) CH₂CF_Three
CH₂C (O) OMe C (F)₂S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Cl) SMe
CH₂C (O) OMe CH (Cl) S (O) Me
CH₂C (O) OMe CH (Cl) S (O)₂Me
CH₂C (O) OMe CH (Cl) SEt
CH₂C (O) OMe CH (Cl) S (O) Et
CH₂C (O) OMe CH (Cl) S (O)₂Et
CH₂C (O) OMe CH (Cl) S (= NCN) Et
CH₂C (O) OMe CH (Cl) S (O) (= NCN) Et
CH₂C (O) OMe CH (Cl) SCH₂CF_Three
CH₂C (O) OMe CH (Cl) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Cl) S (O)₂CH₂CF_Three
CH₂C (O) OMe C (Cl)₂SMe
CH₂C (O) OMe C (Cl)₂S (O) Me
CH₂C (O) OMe C (Cl)₂S (O)₂Me
CH₂C (O) OMe C (Cl)₂SEt
CH₂C (O) OMe C (Cl)₂S (O) Et
CH₂C (O) OMe C (Cl)₂S (O)₂Et
CH₂C (O) OMe C (Cl)₂S (= NCN) Et
CH₂C (O) OMe C (Cl)₂S (O) (= NCN) Et
CH₂C (O) OMe C (Cl)₂SCH₂CF_Three
CH₂C (O) OMe C (Cl)₂S (O) CH₂CF_Three
CH₂C (O) OMe C (Cl)₂S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (Br) SMe
CH₂C (O) OMe CH (Br) S (O) Me
CH₂C (O) OMe CH (Br) S (O)₂Me
CH₂C (O) OMe CH (Br) SEt
CH₂C (O) OMe CH (Br) S (O) Et
CH₂C (O) OMe CH (Br) S (O)₂Et
CH₂C (O) OMe CH (Br) S (= NCN) Et
CH₂C (O) OMe CH (Br) S (O) (= NCN) Et
CH₂C (O) OMe CH (Br) SCH₂CF_Three
CH₂C (O) OMe CH (Br) S (O) CH₂CF_Three
CH₂C (O) OMe CH (Br) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH (I) SMe
CH₂C (O) OMe CH (I) S (O) Me
CH₂C (O) OMe CH (I) S (O)₂Me
CH₂C (O) OMe CH (I) SEt
CH₂C (O) OMe CH (I) S (O) Et
CH₂C (O) OMe CH (I) S (O)₂Et
CH₂C (O) OMe CH (I) S (= NCN) Et
CH₂C (O) OMe CH (I) S (O) (= NCN) Et
CH₂C (O) OMe CH (I) SCH₂CF_Three
CH₂C (O) OMe CH (I) S (O) CH₂CF_Three
CH₂C (O) OMe CH (I) S (O)₂CH₂CF_Three
CH₂C (O) OMe CH {OC (O) Me} SMe
CH₂C (O) OMe CH {OC (O) Me} S (O) Me
CH₂C (O) OMe CH {OC (O) Me} S (O)₂Me
CH₂C (O) OMe CH {OC (O) OMe} SEt
CH₂C (O) OMe CH {OC (O) OMe} S (O) Et
CH₂C (O) OMe CH {OC (O) OMe} S (O)₂Et
CH₂C (O) OMe CH {OC (O) OMe} S (= NCN) Et
CH₂C (O) OMe CH {OC (O) OMe} S (O) (= NCN) Et
CH₂C (O) OMe CH {OC (O) OEt} SMe
CH₂C (O) OMe CH {OC (O) OEt} S (O) Me
CH₂C (O) OMe CH {OC (O) OEt} S (O)₂Me
CH₂C (O) OMe CH {OC (O) OEt} SEt
CH₂C (O) OMe CH {OC (O) OEt} S (O) Et
CH₂C (O) OMe CH {OC (O) OEt} S (O)₂Et
CH₂C (O) OMe CH {OC (O) OEt} S (= NCN) Et
CH₂C (O) OMe CH {OC (O) OEt} S (O) (= NCN) Et
CH₂C (O) OMe CH (OMe) SMe
CH₂C (O) OMe CH (OMe) S (O) Me
CH₂C (O) OMe CH (OMe) S (O)₂Me
CH₂C (O) OMe CH (OMe) SEt
CH₂C (O) OMe CH (OMe) S (O) Et
CH₂C (O) OMe CH (OMe) S (O)₂Et
CH₂C (O) OMe CH (OMe) S (= NCN) Et
CH₂C (O) OMe CH (OMe) S (O) (= NCN) Et
CH₂C (O) OMe CH (OEt) SMe
CH₂C (O) OMe CH (OEt) S (O) Me
CH₂C (O) OMe CH (OEt) S (O)₂Me
CH₂C (O) OMe CH (OEt) SEt
CH₂C (O) OMe CH (OEt) S (O) Et
CH₂C (O) OMe CH (OEt) S (O)₂Et
CH₂C (O) OMe CH (OEt) S (= NCN) Et
CH₂C (O) OMe CH (OEt) S (O) (= CN) Et
CH₂C (O) OMe CH (SMe)₂
CH₂C (O) OMe CH (SMe) S (O) Me
CH₂C (O) OMe CH (SMe) S (O)₂Me
CH₂C (O) OMe CH (SMe) SEt
CH₂C (O) OMe CH (SMe) S (O) Et
CH₂C (O) OMe CH (SMe) S (O)₂Et
CH₂C (O) OMe CH (SMe) S (= NCN) Et
CH₂C (O) OMe CH (SMe) S (O) (= NCN) Et
CH₂C (O) OMe CH (SEt) SMe
CH₂C (O) OMe CH (SEt) S (O) Me
CH₂C (O) OMe CH (SEt) S (O)₂Me
CH₂C (O) OMe CH (SEt) SEt
CH₂C (O) OMe CH (SEt) S (O) Et
CH₂C (O) OMe CH (SEt) S (O)₂Et
CH₂C (O) OMe CH (SEt) S (= NCN) Et
CH₂C (O) OMe CH (SEt) S (O) (= NCN) Et
CH₂C (O) OMe CH (CN) SMe
CH₂C (O) OMe CH (CN) S (O) Me
CH₂C (O) OMe CH (CN) S (O)₂Me
CH₂C (O) OMe CH (CN) SEt
CH₂C (O) OMe CH (CN) S (O) Et
CH₂C (O) OMe CH (CN) S (O)₂Et
CH₂C (O) OMe CH (CN) S (= NCN) Et
CH₂C (O) OMe CH (CN) S (O) (= NCN) Et
CH₂C (O) OMe CH {C (O) OMe} SMe
CH₂C (O) OMe CH {C (O) OMe} S (O) Me
CH₂C (O) OMe CH {C (O) OMe} S (O)₂Me
CH₂C (O) OMe CH {C (O) OMe} SMe
CH₂C (O) OMe CH {C (O) OMe} S (O) Me
CH₂C (O) OMe CH {C (O) OMe} S (O)₂Me
CH₂C (O) OMe CH {C (O) OMe} SEt
CH₂C (O) OMe CH {C (O) OMe} S (O) Et
CH₂C (O) OMe CH {C (O) OMe} S (O)₂Et
CH₂C (O) OMe CH {C (O) OMe} S (= NCN) Et
CH₂C (O) OMe CH {C (O) OMe} S (O) (= NCN) Et
CH₂C (O) OMe CH {C (O) OEt} SMe
CH₂C (O) OMe CH {C (O) OEt} S (O) Me
CH₂C (O) OMe CH {C (O) OEt} S (O)₂Me
CH₂C (O) OMe CH {C (O) OEt} SEt
CH₂C (O) OMe CH {C (O) OEt} S (O) Et
CH₂C (O) OMe CH {C (O) OEt} S (O)₂Et
CH₂C (O) OMe CH {C (O) OEt} S (= NCN) Et
CH₂C (O) OMe CH {C (O) OEt} S (O) (= NCN) Et
CH₂C (O) OMe C (Me)₂SMe
CH₂C (O) OMe C (Me)₂S (O) Me
CH₂C (O) OMe C (Me)₂S (O)₂Me
CH₂C (O) OMe CH₂CH₂SMe
CH₂C (O) OMe CH₂CH₂S (O) Me
CH₂C (O) OMe CH₂CH₂S (O)₂Me
CH₂C (O) OMe CH (Me) CH₂SMe
CH₂C (O) OMe CH (Me) CH₂S (O) Me
CH₂C (O) OMe CH (Me) CH₂S (O)₂Me
CH₂C (O) OMe NHPh
CH₂C (O) OMe NH (D2-1a)
CH₂C (O) OMe NH (D2-2a)
CH₂C (O) OMe NH (D2-2b)
CH₂C (O) OMe NH (D2-5a)
CH₂C (O) OMe NH (D2-5b)
CH₂C (O) OMe NH (D2-5c)
CH₂C (O) OMe NH (D2-6a)
CH₂C (O) OMe NH (D2-6b)
CH₂C (O) OMe NH (D2-6c)
CH₂C (O) OMe NH (D2-7a)
CH₂C (O) OMe NH (D2-8a)
CH₂C (O) OMe NH (D2-8b)
CH₂C (O) OMe NH (D2-8c)
CH₂C (O) OMe NH (D2-9a)
CH₂C (O) OMe NH (D2-9b)
CH₂C (O) OMe NH (D2-9c)
CH₂C (O) OMe NH (D2-10a)
CH₂C (O) OMe NH (D2-10b)
CH₂C (O) OMe NH (D2-10c)
CH₂C (O) OMe NH (D2-11a)
CH₂C (O) OMe NH (D2-12a)
CH₂C (O) OMe NH (D2-12b)
CH₂C (O) OMe NH (D2-12c)
CH₂C (O) OMe NH (D2-13a)
CH₂C (O) OMe NH (D2-13b)
CH₂C (O) OMe NH (D2-14a)
CH₂C (O) OMe NH (D2-14b)
CH₂C (O) OMe NH (D2-15a)
CH₂C (O) OMe NH (D2-15b)
CH₂C (O) OMe NH (D2-16a)
CH₂C (O) OMe NH (D2-17a)
CH₂C (O) OMe NH (D2-18a)
CH₂C (O) OMe NH (D2-19a)
CH₂C (O) OMe NH (D2-20a)
CH₂C (O) OMe NH (D2-21a)
CH₂C (O) OMe NH (D2-21b)
CH₂C (O) OMe NH (D2-22a)
CH₂C (O) OMe NH (D2-23a)
CH₂C (O) OMe NH (D2-23b)
CH₂C (O) OMe NH (D2-24a)
CH₂C (O) OMe NH (D2-25a)
CH₂C (O) OMe NH (D2-26a)
CH₂C (O) OMe NH (D2-27a)
CH₂C (O) OMe NH (D2-28a)
CH₂C (O) OMe NH (D2-29a)
CH₂C (O) OMe NH (D2-30a)
CH₂C (O) OMe NH (D2-31a)
CH₂C (O) OMe NH (D2-32a)
CH₂C (O) OMe NH (D2-33a)
CH₂C (O) OMe NH (D2-34a)
CH₂C (O) OMe NH (D2-35a)
CH₂C (O) OMe NH (D2-35b)
CH₂C (O) OMe NH (D2-36a)
CH₂C (O) OMe NH (D2-37a)
CH₂C (O) OMe NH (D2-38a)
CH₂C (O) OMe NH (D2-39a)
CH₂C (O) OMe NH (D2-40a)
CH₂C (O) OMe NH (D2-40b)
CH₂C (O) OMe NH (D2-40c)
CH₂C (O) OMe NH (D2-41a)
CH₂C (O) OMe NH (D2-42a)
CH₂C (O) OMe NH (D2-43a)
CH₂C (O) OMe NH (D2-45a)
CH₂C (O) OMe NH (D2-49a)
CH₂C (O) OMe NH (D2-51a)
CH₂C (O) OMe NH (D2-59a)
CH₂C (O) OMe NH (D2-61a)
CH₂C (O) OMe NH (D2-79a)
CH₂C (O) OMe NH (D2-80a)
CH₂C (O) OMe NH {D2-108b (2-Cl)}
CH₂C (O) OMe NH {D2-108b (3-Cl)}
CH₂C (O) OMe NH {D2-108b (4-Cl)}
CH₂C (O) OMe NH {D2-108b (2-Me)}
CH₂C (O) OMe NH {D2-108b (3-Me)}
CH₂C (O) OMe NH {D2-108b (4-Me)}
CH₂C (O) OMe N (Me) Ph
CH₂C (O) OMe N (Me) (D2-1a)
CH₂C (O) OMe N (Me) (D2-2a)
CH₂C (O) OMe N (Me) (D2-2b)
CH₂C (O) OMe N (Me) (D2-4a)
CH₂C (O) OMe N (Me) (D2-5a)
CH₂C (O) OMe N (Me) (D2-5b)
CH₂C (O) OMe N (Me) (D2-5c)
CH₂C (O) OMe N (Me) (D2-6a)
CH₂C (O) OMe N (Me) (D2-6b)
CH₂C (O) OMe N (Me) (D2-6c)
CH₂C (O) OMe N (Me) (D2-7a)
CH₂C (O) OMe N (Me) (D2-8a)
CH₂C (O) OMe N (Me) (D2-8b)
CH₂C (O) OMe N (Me) (D2-8c)
CH₂C (O) OMe N (Me) (D2-9a)
CH₂C (O) OMe N (Me) (D2-9b)
CH₂C (O) OMe N (Me) (D2-9c)
CH₂C (O) OMe N (Me) (D2-10a)
CH₂C (O) OMe N (Me) (D2-10b)
CH₂C (O) OMe N (Me) (D2-10c)
CH₂C (O) OMe N (Me) (D2-11a)
CH₂C (O) OMe N (Me) (D2-12a)
CH₂C (O) OMe N (Me) (D2-12b)
CH₂C (O) OMe N (Me) (D2-12c)
CH₂C (O) OMe N (Me) (D2-13a)
CH₂C (O) OMe N (Me) (D2-13b)
CH₂C (O) OMe N (Me) (D2-14a)
CH₂C (O) OMe N (Me) (D2-14b)
CH₂C (O) OMe N (Me) (D2-15a)
CH₂C (O) OMe N (Me) (D2-15b)
CH₂C (O) OMe N (Me) (D2-16a)
CH₂C (O) OMe N (Me) (D2-17a)
CH₂C (O) OMe N (Me) (D2-18a)
CH₂C (O) OMe N (Me) (D2-19a)
CH₂C (O) OMe N (Me) (D2-20a)
CH₂C (O) OMe N (Me) (D2-21a)
CH₂C (O) OMe N (Me) (D2-21b)
CH₂C (O) OMe N (Me) (D2-22a)
CH₂C (O) OMe N (Me) (D2-23a)
CH₂C (O) OMe N (Me) (D2-23b)
CH₂C (O) OMe N (Me) (D2-24a)
CH₂C (O) OMe N (Me) (D2-25a)
CH₂C (O) OMe N (Me) (D2-26a)
CH₂C (O) OMe N (Me) (D2-27a)
CH₂C (O) OMe N (Me) (D2-28a)
CH₂C (O) OMe N (Me) (D2-29a)
CH₂C (O) OMe N (Me) (D2-30a)
CH₂C (O) OMe N (Me) (D2-31a)
CH₂C (O) OMe N (Me) (D2-32a)
CH₂C (O) OMe N (Me) (D2-34a)
CH₂C (O) OMe N (Me) (D2-35a)
CH₂C (O) OMe N (Me) (D2-35b)
CH₂C (O) OMe N (Me) (D2-36a)
CH₂C (O) OMe N (Me) (D2-37a)
CH₂C (O) OMe N (Me) (D2-38a)
CH₂C (O) OMe N (Me) (D2-39a)
CH₂C (O) OMe N (Me) (D2-40a)
CH₂C (O) OMe N (Me) (D2-40b)
CH₂C (O) OMe N (Me) (D2-40c)
CH₂C (O) OMe N (Me) (D2-41a)
CH₂C (O) OMe N (Me) (D2-42a)
CH₂C (O) OMe N (Me) (D2-43a)
CH₂C (O) OMe N (Me) (D2-45a)
CH₂C (O) OMe N (Me) (D2-49a)
CH₂C (O) OMe N (Me) (D2-51a)
CH₂C (O) OMe N (Me) (D2-59a)
CH₂C (O) OMe N (Me) (D2-61a)
CH₂C (O) OMe N (Me) (D2-79a)
CH₂C (O) OMe N (Me) (D2-80a)
CH₂C (O) OMe N (Me) {D2-108b (2-Cl)}
CH₂C (O) OMe N (Me) {D2-108b (3-Cl)}
CH₂C (O) OMe N (Me) {D2-108b (4-Cl)}
CH₂C (O) OMe N (Me) {D2-108b (2-Me)}
CH₂C (O) OMe N (Me) {D2-108b (3-Me)}
CH₂C (O) OMe N (Me) {D2-108b (4-Me)}
CH₂C (O) OEt CH₂SMe
CH₂C (O) OEt CH₂S (O) Me
CH₂C (O) OEt CH₂S (O)₂Me
CH₂C (O) OEt CH₂SEt
CH₂C (O) OEt CH₂S (O) Et
CH₂C (O) OEt CH₂S (O)₂Et
CH₂C (O) OEt CH₂SPr-n
CH₂C (O) OEt CH₂S (O) Pr-n
CH₂C (O) OEt CH₂S (O)₂Pr-n
CH₂C (O) OEt CH₂SPr-i
CH₂C (O) OEt CH₂S (O) Pr-i
CH₂C (O) OEt CH₂S (O)₂Pr-i
CH₂C (O) OEt CH₂SPr-c
CH₂C (O) OEt CH₂S (O) Pr-c
CH₂C (O) OEt CH₂S (O)₂Pr-c
CH₂C (O) OEt CH₂SCH₂CH = CH₂
CH₂C (O) OEt CH₂S (O) CH₂CH = CH₂
CH₂C (O) OEt CH₂S (O)₂CH₂CH = CH₂
CH₂C (O) OEt CH₂SCH₂C≡CH
CH₂C (O) OEt CH₂S (O) CH₂C≡CH
CH₂C (O) OEt CH₂S (O)₂CH₂C≡CH
CH₂C (O) OEt CH₂SCH₂CF_Three
CH₂C (O) OEt CH₂S (O) CH₂CF_Three
CH₂C (O) OEt CH₂S (O)₂CH₂CF_Three
CH₂C (O) OEt CH₂SCH₂CH (OMe)₂
CH₂C (O) OEt CH₂SCH₂CH (= NOMe)
CH₂C (O) OEt CH (Me) SMe
CH₂C (O) OEt CH (Me) S (O) Me
CH₂C (O) OEt CH (Me) S (O)₂Me
CH₂C (O) OEt CH (Me) SEt
CH₂C (O) OEt CH (Me) S (O) Et
CH₂C (O) OEt CH (Me) S (O)₂Et
CH₂C (O) OEt CH (Me) S (= NCN) Et
CH₂C (O) OEt CH (Me) S (O) (= NCN) Et
CH₂C (O) OEt CH (Me) SPr-n
CH₂C (O) OEt CH (Me) S (O) Pr-n
CH₂C (O) OEt CH (Me) S (O)₂Pr-n
CH₂C (O) OEt CH (Me) SPr-i
CH₂C (O) OEt CH (Me) S (O) Pr-i
CH₂C (O) OEt CH (Me) S (O)₂Pr-i
CH₂C (O) OEt CH (Me) SBu-t
CH₂C (O) OEt CH (Me) S (O) Bu-t
CH₂C (O) OEt CH (Me) S (O)₂Bu-t
CH₂C (O) OEt CH (Me) SCH₂Pr-c
CH₂C (O) OEt CH (Me) S (O) CH₂Pr-c
CH₂C (O) OEt CH (Me) S (O)₂CH₂Pr-c
CH₂C (O) OEt CH (Me) SCH₂OMe
CH₂C (O) OEt CH (Me) SCH₂SMe
CH₂C (O) OEt CH (Me) S (O) CH₂SMe
CH₂C (O) OEt CH (Me) S (O)₂CH₂SMe
CH₂C (O) OEt CH (Me) SCH₂C = CH₂
CH₂C (O) OEt CH (Me) S (O) CH₂C = CH₂
CH₂C (O) OEt CH (Me) S (O)₂CH₂C = CH₂
CH₂C (O) OEt CH (Me) SCH₂C≡CH
CH₂C (O) OEt CH (Me) S (O) CH₂C≡CH
CH₂C (O) OEt CH (Me) S (O)₂CH₂C≡CH
CH₂C (O) OEt CH (Me) SCH₂C (O) NHMe
CH₂C (O) OEt CH (Me) S (O) CH₂C (O) NHMe
CH₂C (O) OEt CH (Me) S (O)₂CH₂C (O) NHMe
CH₂C (O) OEt CH (Me) SCH₂C (O) OMe
CH₂C (O) OEt CH (Me) S (O) CH₂C (O) OMe
CH₂C (O) OEt CH (Me) S (O)₂CH₂C (O) OMe
CH₂C (O) OEt CH (Me) SCH₂CH₂CH₂Cl
CH₂C (O) OEt CH (Me) S (O) CH₂CH₂CH₂Cl
CH₂C (O) OEt CH (Me) S (O)₂CH₂CH₂CH₂Cl
CH₂C (O) OEt CH (Me) SCH₂CF_Three
CH₂C (O) OEt CH (Me) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Me) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Me) SCH₂Ph
CH₂C (O) OEt CH (Me) S (O) CH₂Ph
CH₂C (O) OEt CH (Me) S (O)₂CH₂Ph
CH₂C (O) OEt CH (Me) SCH₂(D2-34a)
CH₂C (O) OEt CH (Me) S (O) CH₂(D2-34a)
CH₂C (O) OEt CH (Me) S (O)₂CH₂(D2-34a)
CH₂C (O) OEt CH (CH_Three) SCH₂Si (CH_Three)_Three
CH₂C (O) OEt CH (Me) SCN
CH₂C (O) OEt CH (Me) SCH₂CN
CH₂C (O) OEt CH (Me) SC (O) Me
CH₂C (O) OEt CH (Me) S (D2-12a)
CH₂C (O) OEt CH (Me) S (D2-32a)
CH₂C (O) OEt CH (Me) S {D2-32b (3-NO₂)}
CH₂C (O) OEt CH (Me) S {D2-32b (3-CF_Three)}
CH₂C (O) OEt CH (Me) S (D2-37a)
CH₂C (O) OEt CH (Me) S (D2-51a)
CH₂C (O) OEt CH (Et) SMe
CH₂C (O) OEt CH (Et) S (O) Me
CH₂C (O) OEt CH (Et) S (O)₂Me
CH₂C (O) OEt CH (Et) SEt
CH₂C (O) OEt CH (Et) S (O) Et
CH₂C (O) OEt CH (Et) S (O)₂Et
CH₂C (O) OEt CH (Et) SCH₂CF_Three
CH₂C (O) OEt CH (Et) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Et) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Pr-n) SMe
CH₂C (O) OEt CH (Pr-n) S (O) Me
CH₂C (O) OEt CH (Pr-n) S (O)₂Me
CH₂C (O) OEt CH (Pr-n) SEt
CH₂C (O) OEt CH (Pr-n) S (O) Et
CH₂C (O) OEt CH (Pr-n) S (O)₂Et
CH₂C (O) OEt CH (Pr-n) S (= NCN) Et
CH₂C (O) OEt CH (Pr-n) S (O) (= NCN) Et
CH₂C (O) OEt CH (Pr-n) SPr-n
CH₂C (O) OEt CH (Pr-n) S (O) Pr-n
CH₂C (O) OEt CH (Pr-n) S (O)₂Pr-n
CH₂C (O) OEt CH (Pr-n) SPr-i
CH₂C (O) OEt CH (Pr-n) S (O) Pr-i
CH₂C (O) OEt CH (Pr-n) S (O)₂Pr-i
CH₂C (O) OEt CH (Pr-n) SPr-c
CH₂C (O) OEt CH (Pr-n) S (O) Pr-c
CH₂C (O) OEt CH (Pr-n) S (O)₂Pr-c
CH₂C (O) OEt CH (Pr-n) SCH₂CF_Three
CH₂C (O) OEt CH (Pr-n) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Pr-n) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Pr-i) SMe
CH₂C (O) OEt CH (Pr-i) S (O) Me
CH₂C (O) OEt CH (Pr-i) S (O)₂Me
CH₂C (O) OEt CH (Pr-i) SEt
CH₂C (O) OEt CH (Pr-i) S (O) Et
CH₂C (O) OEt CH (Pr-i) S (O)₂Et
CH₂C (O) OEt CH (Pr-i) S (= NCN) Et
CH₂C (O) OEt CH (Pr-i) S (O) (= NCN) Et
CH₂C (O) OEt CH (Pr-i) SPr-n
CH₂C (O) OEt CH (Pr-i) S (O) Pr-n
CH₂C (O) OEt CH (Pr-i) S (O)₂Pr-n
CH₂C (O) OEt CH (Pr-i) SPr-i
CH₂C (O) OEt CH (Pr-i) S (O) Pr-i
CH₂C (O) OEt CH (Pr-i) S (O)₂Pr-i
CH₂C (O) OEt CH (Pr-i) SPr-c
CH₂C (O) OEt CH (Pr-i) S (O) Pr-c
CH₂C (O) OEt CH (Pr-i) S (O)₂Pr-c
CH₂C (O) OEt CH (Pr-i) SCH₂CF_Three
CH₂C (O) OEt CH (Pr-i) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Pr-i) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Pr-c) SMe
CH₂C (O) OEt CH (Pr-c) S (O) Me
CH₂C (O) OEt CH (Pr-c) S (O)₂Me
CH₂C (O) OEt CH (Pr-c) SEt
CH₂C (O) OEt CH (Pr-c) S (O) Et
CH₂C (O) OEt CH (Pr-c) S (O)₂Et
CH₂C (O) OEt CH (Pr-c) S (= NCN) Et
CH₂C (O) OEt CH (Pr-c) S (O) (= NCN) Et
CH₂C (O) OEt CH (Pr-c) SPr-n
CH₂C (O) OEt CH (Pr-c) S (O) Pr-n
CH₂C (O) OEt CH (Pr-c) S (O)₂Pr-n
CH₂C (O) OEt CH (Pr-c) SPr-i
CH₂C (O) OEt CH (Pr-c) S (O) Pr-i
CH₂C (O) OEt CH (Pr-c) S (O)₂Pr-i
CH₂C (O) OEt CH (Pr-c) SPr-c
CH₂C (O) OEt CH (Pr-c) S (O) Pr-c
CH₂C (O) OEt CH (Pr-c) S (O)₂Pr-c
CH₂C (O) OEt CH (Pr-c) SCH₂CF_Three
CH₂C (O) OEt CH (Pr-c) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Pr-c) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Bu-n) SMe
CH₂C (O) OEt CH (Bu-n) S (O) Me
CH₂C (O) OEt CH (Bu-n) S (O)₂Me
CH₂C (O) OEt CH (Bu-n) SEt
CH₂C (O) OEt CH (Bu-n) S (O) Et
CH₂C (O) OEt CH (Bu-n) S (O)₂Et
CH₂C (O) OEt CH (Bu-n) S (= NCN) Et
CH₂C (O) OEt CH (Bu-n) S (O) (= NCN) Et
CH₂C (O) OEt CH (Bu-n) SPr-n
CH₂C (O) OEt CH (Bu-n) S (O) Pr-n
CH₂C (O) OEt CH (Bu-n) S (O)₂Pr-n
CH₂C (O) OEt CH (Bu-n) SPr-i
CH₂C (O) OEt CH (Bu-n) S (O) Pr-i
CH₂C (O) OEt CH (Bu-n) S (O)₂Pr-i
CH₂C (O) OEt CH (Bu-n) SPr-c
CH₂C (O) OEt CH (Bu-n) S (O) Pr-c
CH₂C (O) OEt CH (Bu-n) S (O)₂Pr-c
CH₂C (O) OEt CH (Bu-n) SCH₂CF_Three
CH₂C (O) OEt CH (Bu-n) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Bu-n) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (F) SMe
CH₂C (O) OEt CH (F) S (O) Me
CH₂C (O) OEt CH (F) S (O)₂Me
CH₂C (O) OEt CH (F) SEt
CH₂C (O) OEt CH (F) S (O) Et
CH₂C (O) OEt CH (F) S (O)₂Et
CH₂C (O) OEt CH (F) S (= NCN) Et
CH₂C (O) OEt CH (F) S (O) (= NCN) Et
CH₂C (O) OEt CH (F) SCH₂CF_Three
CH₂C (O) OEt CH (F) S (O) CH₂CF_Three
CH₂C (O) OEt CH (F) S (O)₂CH₂CF_Three
CH₂C (O) OEt C (F)₂SMe
CH₂C (O) OEt C (F)₂S (O) Me
CH₂C (O) OEt C (F)₂S (O)₂Me
CH₂C (O) OEt C (F)₂SEt
CH₂C (O) OEt C (F)₂S (O) Et
CH₂C (O) OEt C (F)₂S (O)₂Et
CH₂C (O) OEt C (F)₂S (= NCN) Et
CH₂C (O) OEt C (F)₂S (O) (= NCN) Et
CH₂C (O) OEt C (F)₂SCH₂CF_Three
CH₂C (O) OEt C (F)₂S (O) CH₂CF_Three
CH₂C (O) OEt C (F)₂S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Cl) SMe
CH₂C (O) OEt CH (Cl) S (O) Me
CH₂C (O) OEt CH (Cl) S (O)₂Me
CH₂C (O) OEt CH (Cl) SEt
CH₂C (O) OEt CH (Cl) S (O) Et
CH₂C (O) OEt CH (Cl) S (O)₂Et
CH₂C (O) OEt CH (Cl) S (= NCN) Et
CH₂C (O) OEt CH (Cl) S (O) (= NCN) Et
CH₂C (O) OEt CH (Cl) SCH₂CF_Three
CH₂C (O) OEt CH (Cl) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Cl) S (O)₂CH₂CF_Three
CH₂C (O) OEt C (Cl)₂SMe
CH₂C (O) OEt C (Cl)₂S (O) Me
CH₂C (O) OEt C (Cl)₂S (O)₂Me
CH₂C (O) OEt C (Cl)₂SEt
CH₂C (O) OEt C (Cl)₂S (O) Et
CH₂C (O) OEt C (Cl)₂S (O)₂Et
CH₂C (O) OEt C (Cl)₂S (= NCN) Et
CH₂C (O) OEt C (Cl)₂S (O) (= NCN) Et
CH₂C (O) OEt C (Cl)₂SCH₂CF_Three
CH₂C (O) OEt C (Cl)₂S (O) CH₂CF_Three
CH₂C (O) OEt C (Cl)₂S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (Br) SMe
CH₂C (O) OEt CH (Br) S (O) Me
CH₂C (O) OEt CH (Br) S (O)₂Me
CH₂C (O) OEt CH (Br) SEt
CH₂C (O) OEt CH (Br) S (O) Et
CH₂C (O) OEt CH (Br) S (O)₂Et
CH₂C (O) OEt CH (Br) S (= NCN) Et
CH₂C (O) OEt CH (Br) S (O) (= NCN) Et
CH₂C (O) OEt CH (Br) SCH₂CF_Three
CH₂C (O) OEt CH (Br) S (O) CH₂CF_Three
CH₂C (O) OEt CH (Br) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH (I) SMe
CH₂C (O) OEt CH (I) S (O) Me
CH₂C (O) OEt CH (I) S (O)₂Me
CH₂C (O) OEt CH (I) SEt
CH₂C (O) OEt CH (I) S (O) Et
CH₂C (O) OEt CH (I) S (O)₂Et
CH₂C (O) OEt CH (I) S (= NCN) Et
CH₂C (O) OEt CH (I) S (O) (= NCN) Et
CH₂C (O) OEt CH (I) SCH₂CF_Three
CH₂C (O) OEt CH (I) S (O) CH₂CF_Three
CH₂C (O) OEt CH (I) S (O)₂CH₂CF_Three
CH₂C (O) OEt CH {OC (O) Me} SMe
CH₂C (O) OEt CH {OC (O) Me} S (O) Me
CH₂C (O) OEt CH {OC (O) Me} S (O)₂Me
CH₂C (O) OEt CH {OC (O) OMe} SEt
CH₂C (O) OEt CH {OC (O) OMe} S (O) Et
CH₂C (O) OEt CH {OC (O) OMe} S (O)₂Et
CH₂C (O) OEt CH {OC (O) OMe} S (= NCN) Et
CH₂C (O) OEt CH {OC (O) OMe} S (O) (= NCN) Et
CH₂C (O) OEt CH {OC (O) OEt} SMe
CH₂C (O) OEt CH {OC (O) OEt} S (O) Me
CH₂C (O) OEt CH {OC (O) OEt} S (O)₂Me
CH₂C (O) OEt CH {OC (O) OEt} SEt
CH₂C (O) OEt CH {OC (O) OEt} S (O) Et
CH₂C (O) OEt CH {OC (O) OEt} S (O)₂Et
CH₂C (O) OEt CH {OC (O) OEt} S (= NCN) Et
CH₂C (O) OEt CH {OC (O) OEt} S (O) (= NCN) Et
CH₂C (O) OEt CH (OMe) SMe
CH₂C (O) OEt CH (OMe) S (O) Me
CH₂C (O) OEt CH (OMe) S (O)₂Me
CH₂C (O) OEt CH (OMe) SEt
CH₂C (O) OEt CH (OMe) S (O) Et
CH₂C (O) OEt CH (OMe) S (O)₂Et
CH₂C (O) OEt CH (OMe) S (= NCN) Et
CH₂C (O) OEt CH (OMe) S (O) (= NCN) Et
CH₂C (O) OEt CH (OEt) SMe
CH₂C (O) OEt CH (OEt) S (O) Me
CH₂C (O) OEt CH (OEt) S (O)₂Me
CH₂C (O) OEt CH (OEt) SEt
CH₂C (O) OEt CH (OEt) S (O) Et
CH₂C (O) OEt CH (OEt) S (O)₂Et
CH₂C (O) OEt CH (OEt) S (= NCN) Et
CH₂C (O) OEt CH (OEt) S (O) (= NCN) Et
CH₂C (O) OEt CH (SMe)₂
CH₂C (O) OEt CH (SMe) S (O) Me
CH₂C (O) OEt CH (SMe) S (O)₂Me
CH₂C (O) OEt CH (SMe) SEt
CH₂C (O) OEt CH (SMe) S (O) Et
CH₂C (O) OEt CH (SMe) S (O)₂Et
CH₂C (O) OEt CH (SMe) S (= NCN) Et
CH₂C (O) OEt CH (SMe) S (O) (= NCN) Et
CH₂C (O) OEt CH (SEt) SMe
CH₂C (O) OEt CH (SEt) S (O) Me
CH₂C (O) OEt CH (SEt) S (O)₂Me
CH₂C (O) OEt CH (SEt) SEt
CH₂C (O) OEt CH (SEt) S (O) Et
CH₂C (O) OEt CH (SEt) S (O)₂Et
CH₂C (O) OEt CH (SEt) S (= NCN) Et
CH₂C (O) OEt CH (SEt) S (O) (= NCN) Et
CH₂C (O) OEt CH (CN) SMe
CH₂C (O) OEt CH (CN) S (O) Me
CH₂C (O) OEt CH (CN) S (O)₂Me
CH₂C (O) OEt CH (CN) SEt
CH₂C (O) OEt CH (CN) S (O) Et
CH₂C (O) OEt CH (CN) S (O)₂Et
CH₂C (O) OEt CH (CN) S (= NCN) Et
CH₂C (O) OEt CH (CN) S (O) (= NCN) Et
CH₂C (O) OEt CH {C (O) OMe} SMe
CH₂C (O) OEt CH {C (O) OMe} S (O) Me
CH₂C (O) OEt CH {C (O) OMe} S (O)₂Me
CH₂C (O) OEt CH {C (O) OMe} SMe
CH₂C (O) OEt CH {C (O) OMe} S (O) Me
CH₂C (O) OEt CH {C (O) OMe} S (O)₂Me
CH₂C (O) OEt CH {C (O) OMe} SEt
CH₂C (O) OEt CH {C (O) OMe} S (O) Et
CH₂C (O) OEt CH {C (O) OMe} S (O)₂Et
CH₂C (O) OEt CH {C (O) OMe} S (= NCN) Et
CH₂C (O) OEt CH {C (O) OMe} S (O) (= NCN) Et
CH₂C (O) OEt CH {C (O) OEt} SMe
CH₂C (O) OEt CH {C (O) OEt} S (O) Me
CH₂C (O) OEt CH {C (O) OEt} S (O)₂Me
CH₂C (O) OEt CH {C (O) OEt} SEt
CH₂C (O) OEt CH {C (O) OEt} S (O) Et
CH₂C (O) OEt CH {C (O) OEt} S (O)₂Et
CH₂C (O) OEt CH {C (O) OEt} S (= NCN) Et
CH₂C (O) OEt CH {C (O) OEt} S (O) (= NCN) Et
CH₂C (O) OEt C (Me)₂SMe
CH₂C (O) OEt C (Me)₂S (O) Me
CH₂C (O) OEt C (Me)₂S (O)₂Me
CH₂C (O) OEt CH₂CH₂SMe
CH₂C (O) OEt CH₂CH₂S (O) Me
CH₂C (O) OEt CH₂CH₂S (O)₂Me
CH₂C (O) OEt CH (Me) CH₂SMe
CH₂C (O) OEt CH (Me) CH₂S (O) Me
CH₂C (O) OEt CH (Me) CH₂S (O)₂Me
C (O) OMe CH₂SMe
C (O) OMe CH₂S (O) Me
C (O) OMe CH₂S (O)₂Me
C (O) OMe CH₂SEt
C (O) OMe CH₂S (O) Et
C (O) OMe CH₂S (O)₂Et
C (O) OMe CH₂SPr-n
C (O) OMe CH₂S (O) Pr-n
C (O) OMe CH₂S (O)₂Pr-n
C (O) OMe CH₂SPr-i
C (O) OMe CH₂S (O) Pr-i
C (O) OMe CH₂S (O)₂Pr-i
C (O) OMe CH₂SPr-c
C (O) OMe CH₂S (O) Pr-c
C (O) OMe CH₂S (O)₂Pr-c
C (O) OMe CH₂SCH₂CH = CH₂
C (O) OMe CH₂S (O) CH₂CH = CH₂
C (O) OMe CH₂S (O)₂CH₂CH = CH₂
C (O) OMe CH₂SCH₂C≡CH
C (O) OMe CH₂S (O) CH₂C≡CH
C (O) OMe CH₂S (O)₂CH₂C≡CH
C (O) OMe CH₂SCH₂CF_Three
C (O) OMe CH₂S (O) CH₂CF_Three
C (O) OMe CH₂S (O)₂CH₂CF_Three
C (O) OMe CH₂SCH₂CH (OMe)₂
C (O) OMe CH₂SCH₂CH (= NOMe)
C (O) OMe CH (Me) SMe
C (O) OMe CH (Me) S (O) Me
C (O) OMe CH (Me) S (O)₂Me
C (O) OMe CH (Me) SEt
C (O) OMe CH (Me) S (O) Et
C (O) OMe CH (Me) S (O)₂Et
C (O) OMe CH (Me) S (= NCN) Et
C (O) OMe CH (Me) S (O) (= NCN) Et
C (O) OMe CH (Me) SPr-n
C (O) OMe CH (Me) S (O) Pr-n
C (O) OMe CH (Me) S (O)₂Pr-n
C (O) OMe CH (Me) SPr-i
C (O) OMe CH (Me) S (O) Pr-i
C (O) OMe CH (Me) S (O)₂Pr-i
C (O) OMe CH (Me) SBu-t
C (O) OMe CH (Me) S (O) Bu-t
C (O) OMe CH (Me) S (O)₂Bu-t
C (O) OMe CH (Me) SCH₂Pr-c
C (O) OMe CH (Me) S (O) CH₂Pr-c
C (O) OMe CH (Me) S (O)₂CH₂Pr-c
C (O) OMe CH (Me) SCH₂OMe
C (O) OMe CH (Me) SCH₂SMe
C (O) OMe CH (Me) S (O) CH₂SMe
C (O) OMe CH (Me) S (O)₂CH₂SMe
C (O) OMe CH (Me) SCH₂C = CH₂
C (O) OMe CH (Me) S (O) CH₂C = CH₂
C (O) OMe CH (Me) S (O)₂CH₂C = CH₂
C (O) OMe CH (Me) SCH₂C≡CH
C (O) OMe CH (Me) S (O) CH₂C≡CH
C (O) OMe CH (Me) S (O)₂CH₂C≡CH
C (O) OMe CH (Me) SCH₂C (O) NHMe
C (O) OMe CH (Me) S (O) CH₂C (O) NHMe
C (O) OMe CH (Me) S (O)₂CH₂C (O) NHMe
C (O) OMe CH (Me) SCH₂C (O) OMe
C (O) OMe CH (Me) S (O) CH₂C (O) OMe
C (O) OMe CH (Me) S (O)₂CH₂C (O) OMe
C (O) OMe CH (Me) SCH₂CH₂CH₂Cl
C (O) OMe CH (Me) S (O) CH₂CH₂CH₂Cl
C (O) OMe CH (Me) S (O)₂CH₂CH₂CH₂Cl
C (O) OMe CH (Me) SCH₂CF_Three
C (O) OMe CH (Me) S (O) CH₂CF_Three
C (O) OMe CH (Me) S (O)₂CH₂CF_Three
C (O) OMe CH (Me) SCH₂Ph
C (O) OMe CH (Me) S (O) CH₂Ph
C (O) OMe CH (Me) S (O)₂CH₂Ph
C (O) OMe CH (Me) SCH₂(D2-34a)
C (O) OMe CH (Me) S (O) CH₂(D2-34a)
C (O) OMe CH (Me) S (O)₂CH₂(D2-34a)
C (O) OMe CH (CH_Three) SCH₂Si (CH_Three)_Three
C (O) OMe CH (Me) SCN
C (O) OMe CH (Me) SCH₂CN
C (O) OMe CH (Me) SC (O) Me
C (O) OMe CH (Me) S (D2-12a)
C (O) OMe CH (Me) S (D2-32a)
C (O) OMe CH (Me) S {D2-32b (3-NO₂)}
C (O) OMe CH (Me) S {D2-32b (3-CF_Three)}
C (O) OMe CH (Me) S (D2-37a)
C (O) OMe CH (Me) S (D2-51a)
C (O) OMe CH (Et) SMe
C (O) OMe CH (Et) S (O) Me
C (O) OMe CH (Et) S (O)₂Me
C (O) OMe CH (Et) SEt
C (O) OMe CH (Et) S (O) Et
C (O) OMe CH (Et) S (O)₂Et
C (O) OMe CH (Et) SCH₂CF_Three
C (O) OMe CH (Et) S (O) CH₂CF_Three
C (O) OMe CH (Et) S (O)₂CH₂CF_Three
C (O) OMe CH (Pr-n) SMe
C (O) OMe CH (Pr-n) S (O) Me
C (O) OMe CH (Pr-n) S (O)₂Me
C (O) OMe CH (Pr-n) SEt
C (O) OMe CH (Pr-n) S (O) Et
C (O) OMe CH (Pr-n) S (O)₂Et
C (O) OMe CH (Pr-n) S (= NCN) Et
C (O) OMe CH (Pr-n) S (O) (= NCN) Et
C (O) OMe CH (Pr-n) SPr-n
C (O) OMe CH (Pr-n) S (O) Pr-n
C (O) OMe CH (Pr-n) S (O)₂Pr-n
C (O) OMe CH (Pr-n) SPr-i
C (O) OMe CH (Pr-n) S (O) Pr-i
C (O) OMe CH (Pr-n) S (O)₂Pr-i
C (O) OMe CH (Pr-n) SPr-c
C (O) OMe CH (Pr-n) S (O) Pr-c
C (O) OMe CH (Pr-n) S (O)₂Pr-c
C (O) OMe CH (Pr-n) SCH₂CF_Three
C (O) OMe CH (Pr-n) S (O) CH₂CF_Three
C (O) OMe CH (Pr-n) S (O)₂CH₂CF_Three
C (O) OMe CH (Pr-i) SMe
C (O) OMe CH (Pr-i) S (O) Me
C (O) OMe CH (Pr-i) S (O)₂Me
C (O) OMe CH (Pr-i) SEt
C (O) OMe CH (Pr-i) S (O) Et
C (O) OMe CH (Pr-i) S (O)₂Et
C (O) OMe CH (Pr-i) S (= NCN) Et
C (O) OMe CH (Pr-i) S (O) (= NCN) Et
C (O) OMe CH (Pr-i) SPr-n
C (O) OMe CH (Pr-i) S (O) Pr-n
C (O) OMe CH (Pr-i) S (O)₂Pr-n
C (O) OMe CH (Pr-i) SPr-i
C (O) OMe CH (Pr-i) S (O) Pr-i
C (O) OMe CH (Pr-i) S (O)₂Pr-i
C (O) OMe CH (Pr-i) SPr-c
C (O) OMe CH (Pr-i) S (O) Pr-c
C (O) OMe CH (Pr-i) S (O)₂Pr-c
C (O) OMe CH (Pr-i) SCH₂CF_Three
C (O) OMe CH (Pr-i) S (O) CH₂CF_Three
C (O) OMe CH (Pr-i) S (O)₂CH₂CF_Three
C (O) OMe CH (Pr-c) SMe
C (O) OMe CH (Pr-c) S (O) Me
C (O) OMe CH (Pr-c) S (O)₂Me
C (O) OMe CH (Pr-c) SEt
C (O) OMe CH (Pr-c) S (O) Et
C (O) OMe CH (Pr-c) S (O)₂Et
C (O) OMe CH (Pr-c) S (= NCN) Et
C (O) OMe CH (Pr-c) S (O) (= NCN) Et
C (O) OMe CH (Pr-c) SPr-n
C (O) OMe CH (Pr-c) S (O) Pr-n
C (O) OMe CH (Pr-c) S (O)₂Pr-n
C (O) OMe CH (Pr-c) SPr-i
C (O) OMe CH (Pr-c) S (O) Pr-i
C (O) OMe CH (Pr-c) S (O)₂Pr-i
C (O) OMe CH (Pr-c) SPr-c
C (O) OMe CH (Pr-c) S (O) Pr-c
C (O) OMe CH (Pr-c) S (O)₂Pr-c
C (O) OMe CH (Pr-c) SCH₂CF_Three
C (O) OMe CH (Pr-c) S (O) CH₂CF_Three
C (O) OMe CH (Pr-c) S (O)₂CH₂CF_Three
C (O) OMe CH (Bu-n) SMe
C (O) OMe CH (Bu-n) S (O) Me
C (O) OMe CH (Bu-n) S (O)₂Me
C (O) OMe CH (Bu-n) SEt
C (O) OMe CH (Bu-n) S (O) Et
C (O) OMe CH (Bu-n) S (O)₂Et
C (O) OMe CH (Bu-n) S (= NCN) Et
C (O) OMe CH (Bu-n) S (O) (= NCN) Et
C (O) OMe CH (Bu-n) SPr-n
C (O) OMe CH (Bu-n) S (O) Pr-n
C (O) OMe CH (Bu-n) S (O)₂Pr-n
C (O) OMe CH (Bu-n) SPr-i
C (O) OMe CH (Bu-n) S (O) Pr-i
C (O) OMe CH (Bu-n) S (O)₂Pr-i
C (O) OMe CH (Bu-n) SPr-c
C (O) OMe CH (Bu-n) S (O) Pr-c
C (O) OMe CH (Bu-n) S (O)₂Pr-c
C (O) OMe CH (Bu-n) SCH₂CF_Three
C (O) OMe CH (Bu-n) S (O) CH₂CF_Three
C (O) OMe CH (Bu-n) S (O)₂CH₂CF_Three
C (O) OMe CH (F) SMe
C (O) OMe CH (F) S (O) Me
C (O) OMe CH (F) S (O)₂Me
C (O) OMe CH (F) SEt
C (O) OMe CH (F) S (O) Et
C (O) OMe CH (F) S (O)₂Et
C (O) OMe CH (F) S (= NCN) Et
C (O) OMe CH (F) S (O) (= NCN) Et
C (O) OMe CH (F) SCH₂CF_Three
C (O) OMe CH (F) S (O) CH₂CF_Three
C (O) OMe CH (F) S (O)₂CH₂CF_Three
C (O) OMe C (F)₂SMe
C (O) OMe C (F)₂S (O) Me
C (O) OMe C (F)₂S (O)₂Me
C (O) OMe C (F)₂SEt
C (O) OMe C (F)₂S (O) Et
C (O) OMe C (F)₂S (O)₂Et
C (O) OMe C (F)₂S (= NCN) Et
C (O) OMe C (F)₂S (O) (= NCN) Et
C (O) OMe C (F)₂SCH₂CF_Three
C (O) OMe C (F)₂S (O) CH₂CF_Three
C (O) OMe C (F)₂S (O)₂CH₂CF_Three
C (O) OMe CH (Cl) SMe
C (O) OMe CH (Cl) S (O) Me
C (O) OMe CH (Cl) S (O)₂Me
C (O) OMe CH (Cl) SEt
C (O) OMe CH (Cl) S (O) Et
C (O) OMe CH (Cl) S (O)₂Et
C (O) OMe CH (Cl) S (= NCN) Et
C (O) OMe CH (Cl) S (O) (= NCN) Et
C (O) OMe CH (Cl) SCH₂CF_Three
C (O) OMe CH (Cl) S (O) CH₂CF_Three
C (O) OMe CH (Cl) S (O)₂CH₂CF_Three
C (O) OMe C (Cl)₂SMe
C (O) OMe C (Cl)₂S (O) Me
C (O) OMe C (Cl)₂S (O)₂Me
C (O) OMe C (Cl)₂SEt
C (O) OMe C (Cl)₂S (O) Et
C (O) OMe C (Cl)₂S (O)₂Et
C (O) OMe C (Cl)₂S (= NCN) Et
C (O) OMe C (Cl)₂S (O) (= NCN) Et
C (O) OMe C (Cl)₂SCH₂CF_Three
C (O) OMe C (Cl)₂S (O) CH₂CF_Three
C (O) OMe C (Cl)₂S (O)₂CH₂CF_Three
C (O) OMe CH (Br) SMe
C (O) OMe CH (Br) S (O) Me
C (O) OMe CH (Br) S (O)₂Me
C (O) OMe CH (Br) SEt
C (O) OMe CH (Br) S (O) Et
C (O) OMe CH (Br) S (O)₂Et
C (O) OMe CH (Br) S (= NCN) Et
C (O) OMe CH (Br) S (O) (= NCN) Et
C (O) OMe CH (Br) SCH₂CF_Three
C (O) OMe CH (Br) S (O) CH₂CF_Three
C (O) OMe CH (Br) S (O)₂CH₂CF_Three
C (O) OMe CH (I) SMe
C (O) OMe CH (I) S (O) Me
C (O) OMe CH (I) S (O)₂Me
C (O) OMe CH (I) SEt
C (O) OMe CH (I) S (O) Et
C (O) OMe CH (I) S (O)₂Et
C (O) OMe CH (I) S (= NCN) Et
C (O) OMe CH (I) S (O) (= NCN) Et
C (O) OMe CH (I) SCH₂CF_Three
C (O) OMe CH (I) S (O) CH₂CF_Three
C (O) OMe CH (I) S (O)₂CH₂CF_Three
C (O) OMe CH {OC (O) Me} SMe
C (O) OMe CH {OC (O) Me} S (O) Me
C (O) OMe CH {OC (O) Me} S (O)₂Me
C (O) OMe CH {OC (O) OMe} SEt
C (O) OMe CH {OC (O) OMe} S (O) Et
C (O) OMe CH {OC (O) OMe} S (O)₂Et
C (O) OMe CH {OC (O) OMe} S (= NCN) Et
C (O) OMe CH {OC (O) OMe} S (O) (= NCN) Et
C (O) OMe CH {OC (O) OEt} SMe
C (O) OMe CH {OC (O) OEt} S (O) Me
C (O) OMe CH {OC (O) OEt} S (O)₂Me
C (O) OMe CH {OC (O) OEt} SEt
C (O) OMe CH {OC (O) OEt} S (O) Et
C (O) OMe CH {OC (O) OEt} S (O)₂Et
C (O) OMe CH {OC (O) OEt} S (= NCN) Et
C (O) OMe CH {OC (O) OEt} S (O) (= NCN) Et
C (O) OMe CH (OMe) SMe
C (O) OMe CH (OMe) S (O) Me
C (O) OMe CH (OMe) S (O)₂Me
C (O) OMe CH (OMe) SEt
C (O) OMe CH (OMe) S (O) Et
C (O) OMe CH (OMe) S (O)₂Et
C (O) OMe CH (OMe) S (= NCN) Et
C (O) OMe CH (OMe) S (O) (= NCN) Et
C (O) OMe CH (OEt) SMe
C (O) OMe CH (OEt) S (O) Me
C (O) OMe CH (OEt) S (O)₂Me
C (O) OMe CH (OEt) SEt
C (O) OMe CH (OEt) S (O) Et
C (O) OMe CH (OEt) S (O)₂Et
C (O) OMe CH (OEt) S (= NCN) Et
C (O) OMe CH (OEt) S (O) (= NCN) Et
C (O) OMe CH (SMe)₂
C (O) OMe CH (SMe) S (O) Me
C (O) OMe CH (SMe) S (O)₂Me
C (O) OMe CH (SMe) SEt
C (O) OMe CH (SMe) S (O) Et
C (O) OMe CH (SMe) S (O)₂Et
C (O) OMe CH (SMe) S (= NCN) Et
C (O) OMe CH (SMe) S (O) (= NCN) Et
C (O) OMe CH (SEt) SMe
C (O) OMe CH (SEt) S (O) Me
C (O) OMe CH (SEt) S (O)₂Me
C (O) OMe CH (SEt) SEt
C (O) OMe CH (SEt) S (O) Et
C (O) OMe CH (SEt) S (O)₂Et
C (O) OMe CH (SEt) S (= NCN) Et
C (O) OMe CH (SEt) S (O) (= NCN) Et
C (O) OMe CH (CN) SMe
C (O) OMe CH (CN) S (O) Me
C (O) OMe CH (CN) S (O)₂Me
C (O) OMe CH (CN) SEt
C (O) OMe CH (CN) S (O) Et
C (O) OMe CH (CN) S (O)₂Et
C (O) OMe CH (CN) S (= NCN) Et
C (O) OMe CH (CN) S (O) (= NCN) Et
C (O) OMe CH {C (O) OMe} SMe
C (O) OMe CH {C (O) OMe} S (O) Me
C (O) OMe CH {C (O) OMe} S (O)₂Me
C (O) OMe CH {C (O) OMe} SMe
C (O) OMe CH {C (O) OMe} S (O) Me
C (O) OMe CH {C (O) OMe} S (O)₂Me
C (O) OMe CH {C (O) OMe} SEt
C (O) OMe CH {C (O) OMe} S (O) Et
C (O) OMe CH {C (O) OMe} S (O)₂Et
C (O) OMe CH {C (O) OMe} S (= NCN) Et
C (O) OMe CH {C (O) OMe} S (O) (= NCN) Et
C (O) OMe CH {C (O) OEt} SMe
C (O) OMe CH {C (O) OEt} S (O) Me
C (O) OMe CH {C (O) OEt} S (O)₂Me
C (O) OMe CH {C (O) OEt} SEt
C (O) OMe CH {C (O) OEt} S (O) Et
C (O) OMe CH {C (O) OEt} S (O)₂Et
C (O) OMe CH {C (O) OEt} S (= NCN) Et
C (O) OMe CH {C (O) OEt} S (O) (= NCN) Et
C (O) OMe C (Me)₂SMe
C (O) OMe C (Me)₂S (O) Me
C (O) OMe C (Me)₂S (O)₂Me
C (O) OMe CH₂CH₂SMe
C (O) OMe CH₂CH₂S (O) Me
C (O) OMe CH₂CH₂S (O)₂Me
C (O) OMe CH (Me) CH₂SMe
C (O) OMe CH (Me) CH₂S (O) Me
C (O) OMe CH (Me) CH₂S (O)₂Me
C (O) OEt CH₂SMe
C (O) OEt CH₂S (O) Me
C (O) OEt CH₂S (O)₂Me
C (O) OEt CH₂SEt
C (O) OEt CH₂S (O) Et
C (O) OEt CH₂S (O)₂Et
C (O) OEt CH₂SPr-n
C (O) OEt CH₂S (O) Pr-n
C (O) OEt CH₂S (O)₂Pr-n
C (O) OEt CH₂SPr-i
C (O) OEt CH₂S (O) Pr-i
C (O) OEt CH₂S (O)₂Pr-i
C (O) OEt CH₂SPr-c
C (O) OEt CH₂S (O) Pr-c
C (O) OEt CH₂S (O)₂Pr-c
C (O) OEt CH₂SCH₂CH = CH₂
C (O) OEt CH₂S (O) CH₂CH = CH₂
C (O) OEt CH₂S (O)₂CH₂CH = CH₂
C (O) OEt CH₂SCH₂C≡CH
C (O) OEt CH₂S (O) CH₂C≡CH
C (O) OEt CH₂S (O)₂CH₂C≡CH
C (O) OEt CH₂SCH₂CF_Three
C (O) OEt CH₂S (O) CH₂CF_Three
C (O) OEt CH₂S (O)₂CH₂CF_Three
C (O) OEt CH₂SCH₂CH (OMe)₂
C (O) OEt CH₂SCH₂CH (= NOMe)
C (O) OEt CH (Me) SMe
C (O) OEt CH (Me) S (O) Me
C (O) OEt CH (Me) S (O)₂Me
C (O) OEt CH (Me) SEt
C (O) OEt CH (Me) S (O) Et
C (O) OEt CH (Me) S (O)₂Et
C (O) OEt CH (Me) S (= NCN) Et
C (O) OEt CH (Me) S (O) (= NCN) Et
C (O) OEt CH (Me) SPr-n
C (O) OEt CH (Me) S (O) Pr-n
C (O) OEt CH (Me) S (O)₂Pr-n
C (O) OEt CH (Me) SPr-i
C (O) OEt CH (Me) S (O) Pr-i
C (O) OEt CH (Me) S (O)₂Pr-i
C (O) OEt CH (Me) SBu-t
C (O) OEt CH (Me) S (O) Bu-t
C (O) OEt CH (Me) S (O)₂Bu-t
C (O) OEt CH (Me) SCH₂Pr-c
C (O) OEt CH (Me) S (O) CH₂Pr-c
C (O) OEt CH (Me) S (O)₂CH₂Pr-c
C (O) OEt CH (Me) SCH₂OMe
C (O) OEt CH (Me) SCH₂SMe
C (O) OEt CH (Me) S (O) CH₂SMe
C (O) OEt CH (Me) S (O)₂CH₂SMe
C (O) OEt CH (Me) SCH₂C = CH₂
C (O) OEt CH (Me) S (O) CH₂C = CH₂
C (O) OEt CH (Me) S (O)₂CH₂C = CH₂
C (O) OEt CH (Me) SCH₂C≡CH
C (O) OEt CH (Me) S (O) CH₂C≡CH
C (O) OEt CH (Me) S (O)₂CH₂C≡CH
C (O) OEt CH (Me) SCH₂C (O) NHMe
C (O) OEt CH (Me) S (O) CH₂C (O) NHMe
C (O) OEt CH (Me) S (O)₂CH₂C (O) NHMe
C (O) OEt CH (Me) SCH₂C (O) OMe
C (O) OEt CH (Me) S (O) CH₂C (O) OMe
C (O) OEt CH (Me) S (O)₂CH₂C (O) OMe
C (O) OEt CH (Me) SCH₂CH₂CH₂Cl
C (O) OEt CH (Me) S (O) CH₂CH₂CH₂Cl
C (O) OEt CH (Me) S (O)₂CH₂CH₂CH₂Cl
C (O) OEt CH (Me) SCH₂CF_Three
C (O) OEt CH (Me) S (O) CH₂CF_Three
C (O) OEt CH (Me) S (O)₂CH₂CF_Three
C (O) OEt CH (Me) SCH₂Ph
C (O) OEt CH (Me) S (O) CH₂Ph
C (O) OEt CH (Me) S (O)₂CH₂Ph
C (O) OEt CH (Me) SCH₂(D2-34a)
C (O) OEt CH (Me) S (O) CH₂(D2-34a)
C (O) OEt CH (Me) S (O)₂CH₂(D2-34a)
C (O) OEt CH (CH_Three) SCH₂Si (CH_Three)_Three
C (O) OEt CH (Me) SCN
C (O) OEt CH (Me) SCH₂CN
C (O) OEt CH (Me) SC (O) Me
C (O) OEt CH (Me) S (D2-12a)
C (O) OEt CH (Me) S (D2-32a)
C (O) OEt CH (Me) S {D2-32b (3-NO₂)}
C (O) OEt CH (Me) S {D2-32b (3-CF_Three)}
C (O) OEt CH (Me) S (D2-37a)
C (O) OEt CH (Me) S (D2-51a)
C (O) OEt CH (Et) SMe
C (O) OEt CH (Et) S (O) Me
C (O) OEt CH (Et) S (O)₂Me
C (O) OEt CH (Et) SEt
C (O) OEt CH (Et) S (O) Et
C (O) OEt CH (Et) S (O)₂Et
C (O) OEt CH (Et) SCH₂CF_Three
C (O) OEt CH (Et) S (O) CH₂CF_Three
C (O) OEt CH (Et) S (O)₂CH₂CF_Three
C (O) OEt CH (Pr-n) SMe
C (O) OEt CH (Pr-n) S (O) Me
C (O) OEt CH (Pr-n) S (O)₂Me
C (O) OEt CH (Pr-n) SEt
C (O) OEt CH (Pr-n) S (O) Et
C (O) OEt CH (Pr-n) S (O)₂Et
C (O) OEt CH (Pr-n) S (= NCN) Et
C (O) OEt CH (Pr-n) S (O) (= NCN) Et
C (O) OEt CH (Pr-n) SPr-n
C (O) OEt CH (Pr-n) S (O) Pr-n
C (O) OEt CH (Pr-n) S (O)₂Pr-n
C (O) OEt CH (Pr-n) SPr-i
C (O) OEt CH (Pr-n) S (O) Pr-i
C (O) OEt CH (Pr-n) S (O)₂Pr-i
C (O) OEt CH (Pr-n) SPr-c
C (O) OEt CH (Pr-n) S (O) Pr-c
C (O) OEt CH (Pr-n) S (O)₂Pr-c
C (O) OEt CH (Pr-n) SCH₂CF_Three
C (O) OEt CH (Pr-n) S (O) CH₂CF_Three
C (O) OEt CH (Pr-n) S (O)₂CH₂CF_Three
C (O) OEt CH (Pr-i) SMe
C (O) OEt CH (Pr-i) S (O) Me
C (O) OEt CH (Pr-i) S (O)₂Me
C (O) OEt CH (Pr-i) SEt
C (O) OEt CH (Pr-i) S (O) Et
C (O) OEt CH (Pr-i) S (O)₂Et
C (O) OEt CH (Pr-i) S (= NCN) Et
C (O) OEt CH (Pr-i) S (O) (= NCN) Et
C (O) OEt CH (Pr-i) SPr-n
C (O) OEt CH (Pr-i) S (O) Pr-n
C (O) OEt CH (Pr-i) S (O)₂Pr-n
C (O) OEt CH (Pr-i) SPr-i
C (O) OEt CH (Pr-i) S (O) Pr-i
C (O) OEt CH (Pr-i) S (O)₂Pr-i
C (O) OEt CH (Pr-i) SPr-c
C (O) OEt CH (Pr-i) S (O) Pr-c
C (O) OEt CH (Pr-i) S (O)₂Pr-c
C (O) OEt CH (Pr-i) SCH₂CF_Three
C (O) OEt CH (Pr-i) S (O) CH₂CF_Three
C (O) OEt CH (Pr-i) S (O)₂CH₂CF_Three
C (O) OEt CH (Pr-c) SMe
C (O) OEt CH (Pr-c) S (O) Me
C (O) OEt CH (Pr-c) S (O)₂Me
C (O) OEt CH (Pr-c) SEt
C (O) OEt CH (Pr-c) S (O) Et
C (O) OEt CH (Pr-c) S (O)₂Et
C (O) OEt CH (Pr-c) S (= NCN) Et
C (O) OEt CH (Pr-c) S (O) (= NCN) Et
C (O) OEt CH (Pr-c) SPr-n
C (O) OEt CH (Pr-c) S (O) Pr-n
C (O) OEt CH (Pr-c) S (O)₂Pr-n
C (O) OEt CH (Pr-c) SPr-i
C (O) OEt CH (Pr-c) S (O) Pr-i
C (O) OEt CH (Pr-c) S (O)₂Pr-i
C (O) OEt CH (Pr-c) SPr-c
C (O) OEt CH (Pr-c) S (O) Pr-c
C (O) OEt CH (Pr-c) S (O)₂Pr-c
C (O) OEt CH (Pr-c) SCH₂CF_Three
C (O) OEt CH (Pr-c) S (O) CH₂CF_Three
C (O) OEt CH (Pr-c) S (O)₂CH₂CF_Three
C (O) OEt CH (Bu-n) SMe
C (O) OEt CH (Bu-n) S (O) Me
C (O) OEt CH (Bu-n) S (O)₂Me
C (O) OEt CH (Bu-n) SEt
C (O) OEt CH (Bu-n) S (O) Et
C (O) OEt CH (Bu-n) S (O)₂Et
C (O) OEt CH (Bu-n) S (= NCN) Et
C (O) OEt CH (Bu-n) S (O) (= NCN) Et
C (O) OEt CH (Bu-n) SPr-n
C (O) OEt CH (Bu-n) S (O) Pr-n
C (O) OEt CH (Bu-n) S (O)₂Pr-n
C (O) OEt CH (Bu-n) SPr-i
C (O) OEt CH (Bu-n) S (O) Pr-i
C (O) OEt CH (Bu-n) S (O)₂Pr-i
C (O) OEt CH (Bu-n) SPr-c
C (O) OEt CH (Bu-n) S (O) Pr-c
C (O) OEt CH (Bu-n) S (O)₂Pr-c
C (O) OEt CH (Bu-n) SCH₂CF_Three
C (O) OEt CH (Bu-n) S (O) CH₂CF_Three
C (O) OEt CH (Bu-n) S (O)₂CH₂CF_Three
C (O) OEt CH (F) SMe
C (O) OEt CH (F) S (O) Me
C (O) OEt CH (F) S (O)₂Me
C (O) OEt CH (F) SEt
C (O) OEt CH (F) S (O) Et
C (O) OEt CH (F) S (O)₂Et
C (O) OEt CH (F) S (= NCN) Et
C (O) OEt CH (F) S (O) (= NCN) Et
C (O) OEt CH (F) SCH₂CF_Three
C (O) OEt CH (F) S (O) CH₂CF_Three
C (O) OEt CH (F) S (O)₂CH₂CF_Three
C (O) OEt C (F)₂SMe
C (O) OEt C (F)₂S (O) Me
C (O) OEt C (F)₂S (O)₂Me
C (O) OEt C (F)₂SEt
C (O) OEt C (F)₂S (O) Et
C (O) OEt C (F)₂S (O)₂Et
C (O) OEt C (F)₂S (= NCN) Et
C (O) OEt C (F)₂S (O) (= NCN) Et
C (O) OEt C (F)₂SCH₂CF_Three
C (O) OEt C (F)₂S (O) CH₂CF_Three
C (O) OEt C (F)₂S (O)₂CH₂CF_Three
C (O) OEt CH (Cl) SMe
C (O) OEt CH (Cl) S (O) Me
C (O) OEt CH (Cl) S (O)₂Me
C (O) OEt CH (Cl) SEt
C (O) OEt CH (Cl) S (O) Et
C (O) OEt CH (Cl) S (O)₂Et
C (O) OEt CH (Cl) S (= NCN) Et
C (O) OEt CH (Cl) S (O) (= NCN) Et
C (O) OEt CH (Cl) SCH₂CF_Three
C (O) OEt CH (Cl) S (O) CH₂CF_Three
C (O) OEt CH (Cl) S (O)₂CH₂CF_Three
C (O) OEt C (Cl)₂SMe
C (O) OEt C (Cl)₂S (O) Me
C (O) OEt C (Cl)₂S (O)₂Me
C (O) OEt C (Cl)₂SEt
C (O) OEt C (Cl)₂S (O) Et
C (O) OEt C (Cl)₂S (O)₂Et
C (O) OEt C (Cl)₂S (= NCN) Et
C (O) OEt C (Cl)₂S (O) (= NCN) Et
C (O) OEt C (Cl)₂SCH₂CF_Three
C (O) OEt C (Cl)₂S (O) CH₂CF_Three
C (O) OEt C (Cl)₂S (O)₂CH₂CF_Three
C (O) OEt CH (Br) SMe
C (O) OEt CH (Br) S (O) Me
C (O) OEt CH (Br) S (O)₂Me
C (O) OEt CH (Br) SEt
C (O) OEt CH (Br) S (O) Et
C (O) OEt CH (Br) S (O)₂Et
C (O) OEt CH (Br) S (= NCN) Et
C (O) OEt CH (Br) S (O) (= NCN) Et
C (O) OEt CH (Br) SCH₂CF_Three
C (O) OEt CH (Br) S (O) CH₂CF_Three
C (O) OEt CH (Br) S (O)₂CH₂CF_Three
C (O) OEt CH (I) SMe
C (O) OEt CH (I) S (O) Me
C (O) OEt CH (I) S (O)₂Me
C (O) OEt CH (I) SEt
C (O) OEt CH (I) S (O) Et
C (O) OEt CH (I) S (O)₂Et
C (O) OEt CH (I) S (= NCN) Et
C (O) OEt CH (I) S (O) (= NCN) Et
C (O) OEt CH (I) SCH₂CF_Three
C (O) OEt CH (I) S (O) CH₂CF_Three
C (O) OEt CH (I) S (O)₂CH₂CF_Three
C (O) OEt CH {OC (O) Me} SMe
C (O) OEt CH {OC (O) Me} S (O) Me
C (O) OEt CH {OC (O) Me} S (O)₂Me
C (O) OEt CH {OC (O) OMe} SEt
C (O) OEt CH {OC (O) OMe} S (O) Et
C (O) OEt CH {OC (O) OMe} S (O)₂Et
C (O) OEt CH {OC (O) OMe} S (= NCN) Et
C (O) OEt CH {OC (O) OMe} S (O) (= NCN) Et
C (O) OEt CH {OC (O) OEt} SMe
C (O) OEt CH {OC (O) OEt} S (O) Me
C (O) OEt CH {OC (O) OEt} S (O)₂Me
C (O) OEt CH {OC (O) OEt} SEt
C (O) OEt CH {OC (O) OEt} S (O) Et
C (O) OEt CH {OC (O) OEt} S (O)₂Et
C (O) OEt CH {OC (O) OEt} S (= NCN) Et
C (O) OEt CH {OC (O) OEt} S (O) (= NCN) Et
C (O) OEt CH (OMe) SMe
C (O) OEt CH (OMe) S (O) Me
C (O) OEt CH (OMe) S (O)₂Me
C (O) OEt CH (OMe) SEt
C (O) OEt CH (OMe) S (O) Et
C (O) OEt CH (OMe) S (O)₂Et
C (O) OEt CH (OMe) S (= NCN) Et
C (O) OEt CH (OMe) S (O) (= NCN) Et
C (O) OEt CH (OEt) SMe
C (O) OEt CH (OEt) S (O) Me
C (O) OEt CH (OEt) S (O)₂Me
C (O) OEt CH (OEt) SEt
C (O) OEt CH (OEt) S (O) Et
C (O) OEt CH (OEt) S (O)₂Et
C (O) OEt CH (OEt) S (= NCN) Et
C (O) OEt CH (OEt) S (O) (= NCN) Et
C (O) OEt CH (SMe)₂
C (O) OEt CH (SMe) S (O) Me
C (O) OEt CH (SMe) S (O)₂Me
C (O) OEt CH (SMe) SEt
C (O) OEt CH (SMe) S (O) Et
C (O) OEt CH (SMe) S (O)₂Et
C (O) OEt CH (SMe) S (= NCN) Et
C (O) OEt CH (SMe) S (O) (= NCN) Et
C (O) OEt CH (SEt) SMe
C (O) OEt CH (SEt) S (O) Me
C (O) OEt CH (SEt) S (O)₂Me
C (O) OEt CH (SEt) SEt
C (O) OEt CH (SEt) S (O) Et
C (O) OEt CH (SEt) S (O)₂Et
C (O) OEt CH (SEt) S (= NCN) Et
C (O) OEt CH (SEt) S (O) (= NCN) Et
C (O) OEt CH (CN) SMe
C (O) OEt CH (CN) S (O) Me
C (O) OEt CH (CN) S (O)₂Me
C (O) OEt CH (CN) SEt
C (O) OEt CH (CN) S (O) Et
C (O) OEt CH (CN) S (O)₂Et
C (O) OEt CH (CN) S (= NCN) Et
C (O) OEt CH (CN) S (O) (= NCN) Et
C (O) OEt CH {C (O) OMe} SMe
C (O) OEt CH {C (O) OMe} S (O) Me
C (O) OEt CH {C (O) OMe} S (O)₂Me
C (O) OEt CH {C (O) OMe} SMe
C (O) OEt CH {C (O) OMe} S (O) Me
C (O) OEt CH {C (O) OMe} S (O)₂Me
C (O) OEt CH {C (O) OMe} SEt
C (O) OEt CH {C (O) OMe} S (O) Et
C (O) OEt CH {C (O) OMe} S (O)₂Et
C (O) OEt CH {C (O) OMe} S (= NCN) Et
C (O) OEt CH {C (O) OMe} S (O) (= NCN) Et
C (O) OEt CH {C (O) OEt} SMe
C (O) OEt CH {C (O) OEt} S (O) Me
C (O) OEt CH {C (O) OEt} S (O)₂Me
C (O) OEt CH {C (O) OEt} SEt
C (O) OEt CH {C (O) OEt} S (O) Et
C (O) OEt CH {C (O) OEt} S (O)₂Et
C (O) OEt CH {C (O) OEt} S (= NCN) Et
C (O) OEt CH {C (O) OEt} S (O) (= NCN) Et
C (O) OEt C (Me)₂SMe
C (O) OEt C (Me)₂S (O) Me
C (O) OEt C (Me)₂S (O)₂Me
C (O) OEt CH₂CH₂SMe
C (O) OEt CH₂CH₂S (O) Me
C (O) OEt CH₂CH₂S (O)₂Me
C (O) OEt CH (Me) CH₂SMe
C (O) OEt CH (Me) CH₂S (O) Me
C (O) OEt CH (Me) CH₂S (O)₂Me
CH₂CF_Three                    CH₂SMe
CH₂CF_Three                    CH₂S (O) Me
CH₂CF_Three                    CH₂S (O)₂Me
CH₂CF_Three                    CH₂SEt
CH₂CF_Three                    CH₂S (O) Et
CH₂CF_Three                    CH₂S (O)₂Et
CH₂CF_Three                    CH₂SPr-n
CH₂CF_Three                    CH₂S (O) Pr-n
CH₂CF_Three                    CH₂S (O)₂Pr-n
CH₂CF_Three                    CH₂SPr-i
CH₂CF_Three                    CH₂S (O) Pr-i
CH₂CF_Three                    CH₂S (O)₂Pr-i
CH₂CF_Three                    CH₂SPr-c
CH₂CF_Three                    CH₂S (O) Pr-c
CH₂CF_Three                    CH₂S (O)₂Pr-c
CH₂CF_Three                    CH₂SCH₂CH = CH₂
CH₂CF_Three                  CH₂S (O) CH₂CH = CH₂
CH₂CF_Three                 CH₂S (O)₂CH₂CH = CH₂
CH₂CF_Three                    CH₂SCH₂C≡CH
CH₂CF_Three                  CH₂S (O) CH₂C≡CH
CH₂CF_Three                  CH₂S (O)₂CH₂C≡CH
CH₂CF_Three                    CH₂SCH₂CF_Three
CH₂CF_Three                    CH₂S (O) CH₂CF_Three
CH₂CF_Three                    CH₂S (O)₂CH₂CF_Three
CH₂CF_Three                   CH₂SCH₂CH (OMe)₂
CH₂CF_Three                 CH₂SCH₂CH (= NOMe)
CH₂CF_Three                    CH (Me) SMe
CH₂CF_Three                    CH (Me) S (O) Me
CH₂CF_Three                    CH (Me) S (O)₂Me
CH₂CF_Three                    CH (Me) SEt
CH₂CF_Three                    CH (Me) S (O) Et
CH₂CF_Three                    CH (Me) S (O)₂Et
CH₂CF_Three                 CH (Me) S (= NCN) Et
CH₂CF_Three              CH (Me) S (O) (= NCN) Et
CH₂CF_Three                    CH (Me) SPr-n
CH₂CF_Three                  CH (Me) S (O) Pr-n
CH₂CF_Three                  CH (Me) S (O)₂Pr-n
CH₂CF_Three                    CH (Me) SPr-i
CH₂CF_Three                  CH (Me) S (O) Pr-i
CH₂CF_Three                  CH (Me) S (O)₂Pr-i
CH₂CF_Three                    CH (Me) SBu-t
CH₂CF_Three                  CH (Me) S (O) Bu-t
CH₂CF_Three                  CH (Me) S (O)₂Bu-t
CH₂CF_Three                   CH (Me) SCH₂Pr-c
CH₂CF_Three                CH (Me) S (O) CH₂Pr-c
CH₂CF_Three               CH (Me) S (O)₂CH₂Pr-c
CH₂CF_Three                    CH (Me) SCH₂OMe
CH₂CF_Three                    CH (Me) SCH₂SMe
CH₂CF_Three                 CH (Me) S (O) CH₂SMe
CH₂CF_Three                CH (Me) S (O)₂CH₂SMe
CH₂CF_Three                  CH (Me) SCH₂C = CH₂
CH₂CF_Three               CH (Me) S (O) CH₂C = CH₂
CH₂CF_Three               CH (Me) S (O)₂CH₂C = CH₂
CH₂CF_Three                  CH (Me) SCH₂C≡CH
CH₂CF_Three               CH (Me) S (O) CH₂C≡CH
CH₂CF_Three              CH (Me) S (O)₂CH₂C≡CH
CH₂CF_Three               CH (Me) SCH₂C (O) NHMe
CH₂CF_Three            CH (Me) S (O) CH₂C (O) NHMe
CH₂CF_Three           CH (Me) S (O)₂CH₂C (O) NHMe
CH₂CF_Three                CH (Me) SCH₂C (O) OMe
CH₂CF_Three             CH (Me) S (O) CH₂C (O) OMe
CH₂CF_Three            CH (Me) S (O)₂CH₂C (O) OMe
CH₂CF_Three                CH (Me) SCH₂CH₂CH₂Cl
CH₂CF_Three             CH (Me) S (O) CH₂CH₂CH₂Cl
CH₂CF_Three            CH (Me) S (O)₂CH₂CH₂CH₂Cl
CH₂CF_Three                    CH (Me) SCH₂CF_Three
CH₂CF_Three                 CH (Me) S (O) CH₂CF_Three
CH₂CF_Three                 CH (Me) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Me) SCH₂Ph
CH₂CF_Three                  CH (Me) S (O) CH₂Ph
CH₂CF_Three                 CH (Me) S (O)₂CH₂Ph
CH₂CF_Three               CH (Me) SCH₂(D2-34a)
CH₂CF_Three            CH (Me) S (O) CH₂(D2-34a)
CH₂CF_Three           CH (Me) S (O)₂CH₂(D2-34a)
CH₂CF_Three               CH (CH_Three) SCH₂Si (CH_Three)_Three
CH₂CF_Three                    CH (Me) SCN
CH₂CF_Three                    CH (Me) SCH₂CN
CH₂CF_Three                   CH (Me) SC (O) Me
CH₂CF_Three          CH (Me) S (D2-12a)
CH₂CF_Three                 CH (Me) S (D2-32a)
CH₂CF_Three           CH (Me) S {D2-32b (3-NO₂)}
CH₂CF_Three           CH (Me) S {D2-32b (3-CF_Three)}
CH₂CF_Three                 CH (Me) S (D2-37a)
CH₂CF_Three                 CH (Me) S (D2-51a)
CH₂CF_Three                    CH (Et) SMe
CH₂CF_Three                    CH (Et) S (O) Me
CH₂CF_Three                    CH (Et) S (O)₂Me
CH₂CF_Three                    CH (Et) SEt
CH₂CF_Three                    CH (Et) S (O) Et
CH₂CF_Three                    CH (Et) S (O)₂Et
CH₂CF_Three                    CH (Et) SCH₂CF_Three
CH₂CF_Three                 CH (Et) S (O) CH₂CF_Three
CH₂CF_Three                 CH (Et) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Pr-n) SMe
CH₂CF_Three                  CH (Pr-n) S (O) Me
CH₂CF_Three                  CH (Pr-n) S (O)₂Me
CH₂CF_Three                    CH (Pr-n) SEt
CH₂CF_Three                  CH (Pr-n) S (O) Et
CH₂CF_Three                  CH (Pr-n) S (O)₂Et
CH₂CF_Three               CH (Pr-n) S (= NCN) Et
CH₂CF_Three            CH (Pr-n) S (O) (= NCN) Et
CH₂CF_Three                   CH (Pr-n) SPr-n
CH₂CF_Three                CH (Pr-n) S (O) Pr-n
CH₂CF_Three                CH (Pr-n) S (O)₂Pr-n
CH₂CF_Three                   CH (Pr-n) SPr-i
CH₂CF_Three                CH (Pr-n) S (O) Pr-i
CH₂CF_Three                CH (Pr-n) S (O)₂Pr-i
CH₂CF_Three                   CH (Pr-n) SPr-c
CH₂CF_Three                CH (Pr-n) S (O) Pr-c
CH₂CF_Three                CH (Pr-n) S (O)₂Pr-c
CH₂CF_Three                  CH (Pr-n) SCH₂CF_Three
CH₂CF_Three               CH (Pr-n) S (O) CH₂CF_Three
CH₂CF_Three               CH (Pr-n) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Pr-i) SMe
CH₂CF_Three                  CH (Pr-i) S (O) Me
CH₂CF_Three                  CH (Pr-i) S (O)₂Me
CH₂CF_Three                    CH (Pr-i) SEt
CH₂CF_Three                  CH (Pr-i) S (O) Et
CH₂CF_Three                  CH (Pr-i) S (O)₂Et
CH₂CF_Three               CH (Pr-i) S (= NCN) Et
CH₂CF_Three            CH (Pr-i) S (O) (= NCN) Et
CH₂CF_Three                   CH (Pr-i) SPr-n
CH₂CF_Three                CH (Pr-i) S (O) Pr-n
CH₂CF_Three                CH (Pr-i) S (O)₂Pr-n
CH₂CF_Three                   CH (Pr-i) SPr-i
CH₂CF_Three                CH (Pr-i) S (O) Pr-i
CH₂CF_Three                CH (Pr-i) S (O)₂Pr-i
CH₂CF_Three                   CH (Pr-i) SPr-c
CH₂CF_Three                CH (Pr-i) S (O) Pr-c
CH₂CF_Three                CH (Pr-i) S (O)₂Pr-c
CH₂CF_Three                  CH (Pr-i) SCH₂CF_Three
CH₂CF_Three               CH (Pr-i) S (O) CH₂CF_Three
CH₂CF_Three               CH (Pr-i) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Pr-c) SMe
CH₂CF_Three                  CH (Pr-c) S (O) Me
CH₂CF_Three                  CH (Pr-c) S (O)₂Me
CH₂CF_Three                    CH (Pr-c) SEt
CH₂CF_Three                  CH (Pr-c) S (O) Et
CH₂CF_Three                  CH (Pr-c) S (O)₂Et
CH₂CF_Three               CH (Pr-c) S (= NCN) Et
CH₂CF_Three            CH (Pr-c) S (O) (= NCN) Et
CH₂CF_Three                   CH (Pr-c) SPr-n
CH₂CF_Three                CH (Pr-c) S (O) Pr-n
CH₂CF_Three                CH (Pr-c) S (O)₂Pr-n
CH₂CF_Three                   CH (Pr-c) SPr-i
CH₂CF_Three                CH (Pr-c) S (O) Pr-i
CH₂CF_Three                CH (Pr-c) S (O)₂Pr-i
CH₂CF_Three                   CH (Pr-c) SPr-c
CH₂CF_Three                CH (Pr-c) S (O) Pr-c
CH₂CF_Three                CH (Pr-c) S (O)₂Pr-c
CH₂CF_Three                  CH (Pr-c) SCH₂CF_Three
CH₂CF_Three               CH (Pr-c) S (O) CH₂CF_Three
CH₂CF_Three               CH (Pr-c) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Bu-n) SMe
CH₂CF_Three                  CH (Bu-n) S (O) Me
CH₂CF_Three                  CH (Bu-n) S (O)₂Me
CH₂CF_Three                    CH (Bu-n) SEt
CH₂CF_Three                  CH (Bu-n) S (O) Et
CH₂CF_Three                  CH (Bu-n) S (O)₂Et
CH₂CF_Three               CH (Bu-n) S (= NCN) Et
CH₂CF_Three            CH (Bu-n) S (O) (= NCN) Et
CH₂CF_Three                   CH (Bu-n) SPr-n
CH₂CF_Three                CH (Bu-n) S (O) Pr-n
CH₂CF_Three                CH (Bu-n) S (O)₂Pr-n
CH₂CF_Three                   CH (Bu-n) SPr-i
CH₂CF_Three                CH (Bu-n) S (O) Pr-i
CH₂CF_Three                CH (Bu-n) S (O)₂Pr-i
CH₂CF_Three                   CH (Bu-n) SPr-c
CH₂CF_Three                CH (Bu-n) S (O) Pr-c
CH₂CF_Three                CH (Bu-n) S (O)₂Pr-c
CH₂CF_Three                  CH (Bu-n) SCH₂CF_Three
CH₂CF_Three               CH (Bu-n) S (O) CH₂CF_Three
CH₂CF_Three               CH (Bu-n) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (F) SMe
CH₂CF_Three                    CH (F) S (O) Me
CH₂CF_Three                    CH (F) S (O)₂Me
CH₂CF_Three                    CH (F) SEt
CH₂CF_Three                    CH (F) S (O) Et
CH₂CF_Three                    CH (F) S (O)₂Et
CH₂CF_Three                  CH (F) S (= NCN) Et
CH₂CF_Three               CH (F) S (O) (= NCN) Et
CH₂CF_Three                    CH (F) SCH₂CF_Three
CH₂CF_Three                  CH (F) S (O) CH₂CF_Three
CH₂CF_Three                  CH (F) S (O)₂CH₂CF_Three
CH₂CF_Three                    C (F)₂SMe
CH₂CF_Three                    C (F)₂S (O) Me
CH₂CF_Three                    C (F)₂S (O)₂Me
CH₂CF_Three                    C (F)₂SEt
CH₂CF_Three                    C (F)₂S (O) Et
CH₂CF_Three                    C (F)₂S (O)₂Et
CH₂CF_Three                   C (F)₂S (= NCN) Et
CH₂CF_Three                C (F)₂S (O) (= NCN) Et
CH₂CF_Three                    C (F)₂SCH₂CF_Three
CH₂CF_Three                   C (F)₂S (O) CH₂CF_Three
CH₂CF_Three                  C (F)₂S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Cl) SMe
CH₂CF_Three                    CH (Cl) S (O) Me
CH₂CF_Three                    CH (Cl) S (O)₂Me
CH₂CF_Three                    CH (Cl) SEt
CH₂CF_Three                    CH (Cl) S (O) Et
CH₂CF_Three                    CH (Cl) S (O)₂Et
CH₂CF_Three                 CH (Cl) S (= NCN) Et
CH₂CF_Three              CH (Cl) S (O) (= NCN) Et
CH₂CF_Three                    CH (Cl) SCH₂CF_Three
CH₂CF_Three                 CH (Cl) S (O) CH₂CF_Three
CH₂CF_Three                 CH (Cl) S (O)₂CH₂CF_Three
CH₂CF_Three                    C (Cl)₂SMe
CH₂CF_Three                    C (Cl)₂S (O) Me
CH₂CF_Three                    C (Cl)₂S (O)₂Me
CH₂CF_Three                    C (Cl)₂SEt
CH₂CF_Three                    C (Cl)₂S (O) Et
CH₂CF_Three                    C (Cl)₂S (O)₂Et
CH₂CF_Three                  C (Cl)₂S (= NCN) Et
CH₂CF_Three               C (Cl)₂S (O) (= NCN) Et
CH₂CF_Three                    C (Cl)₂SCH₂CF_Three
CH₂CF_Three                  C (Cl)₂S (O) CH₂CF_Three
CH₂CF_Three                 C (Cl)₂S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (Br) SMe
CH₂CF_Three                    CH (Br) S (O) Me
CH₂CF_Three                    CH (Br) S (O)₂Me
CH₂CF_Three                    CH (Br) SEt
CH₂CF_Three                    CH (Br) S (O) Et
CH₂CF_Three                    CH (Br) S (O)₂Et
CH₂CF_Three                 CH (Br) S (= NCN) Et
CH₂CF_Three              CH (Br) S (O) (= NCN) Et
CH₂CF_Three                    CH (Br) SCH₂CF_Three
CH₂CF_Three                 CH (Br) S (O) CH₂CF_Three
CH₂CF_Three                 CH (Br) S (O)₂CH₂CF_Three
CH₂CF_Three                    CH (I) SMe
CH₂CF_Three                    CH (I) S (O) Me
CH₂CF_Three                    CH (I) S (O)₂Me
CH₂CF_Three                    CH (I) SEt
CH₂CF_Three                    CH (I) S (O) Et
CH₂CF_Three                    CH (I) S (O)₂Et
CH₂CF_Three                  CH (I) S (= NCN) Et
CH₂CF_Three               CH (I) S (O) (= NCN) Et
CH₂CF_Three                    CH (I) SCH₂CF_Three
CH₂CF_Three                  CH (I) S (O) CH₂CF_Three
CH₂CF_Three                  CH (I) S (O)₂CH₂CF_Three
CH₂CF_Three                  CH {OC (O) Me} SMe
CH₂CF_Three               CH {OC (O) Me} S (O) Me
CH₂CF_Three               CH {OC (O) Me} S (O)₂Me
CH₂CF_Three                 CH {OC (O) OMe} SEt
CH₂CF_Three              CH {OC (O) OMe} S (O) Et
CH₂CF_Three              CH {OC (O) OMe} S (O)₂Et
CH₂CF_Three           CH {OC (O) OMe} S (= NCN) Et
CH₂CF_Three        CH {OC (O) OMe} S (O) (= NCN) Et
CH₂CF_Three                 CH {OC (O) OEt} SMe
CH₂CF_Three              CH {OC (O) OEt} S (O) Me
CH₂CF_Three              CH {OC (O) OEt} S (O)₂Me
CH₂CF_Three                 CH {OC (O) OEt} SEt
CH₂CF_Three              CH {OC (O) OEt} S (O) Et
CH₂CF_Three              CH {OC (O) OEt} S (O)₂Et
CH₂CF_Three           CH {OC (O) OEt} S (= NCN) Et
CH₂CF_Three        CH {OC (O) OEt} S (O) (= NCN) Et
CH₂CF_Three                    CH (OMe) SMe
CH₂CF_Three                   CH (OMe) S (O) Me
CH₂CF_Three                   CH (OMe) S (O)₂Me
CH₂CF_Three                    CH (OMe) SEt
CH₂CF_Three                   CH (OMe) S (O) Et
CH₂CF_Three                   CH (OMe) S (O)₂Et
CH₂CF_Three                CH (OMe) S (= NCN) Et
CH₂CF_Three             CH (OMe) S (O) (= NCN) Et
CH₂CF_Three                    CH (OEt) SMe
CH₂CF_Three                   CH (OEt) S (O) Me
CH₂CF_Three                   CH (OEt) S (O)₂Me
CH₂CF_Three                    CH (OEt) SEt
CH₂CF_Three                   CH (OEt) S (O) Et
CH₂CF_Three                   CH (OEt) S (O)₂Et
CH₂CF_Three                CH (OEt) S (= NCN) Et
CH₂CF_Three             CH (OEt) S (O) (= NCN) Et
CH₂CF_Three                    CH (SMe)₂
CH₂CF_Three                   CH (SMe) S (O) Me
CH₂CF_Three                   CH (SMe) S (O)₂Me
CH₂CF_Three                    CH (SMe) SEt
CH₂CF_Three                   CH (SMe) S (O) Et
CH₂CF_Three                   CH (SMe) S (O)₂Et
CH₂CF_Three                CH (SMe) S (= NCN) Et
CH₂CF_Three             CH (SMe) S (O) (= NCN) Et
CH₂CF_Three                    CH (SEt) SMe
CH₂CF_Three                   CH (SEt) S (O) Me
CH₂CF_Three                   CH (SEt) S (O)₂Me
CH₂CF_Three                    CH (SEt) SEt
CH₂CF_Three                   CH (SEt) S (O) Et
CH₂CF_Three                   CH (SEt) S (O)₂Et
CH₂CF_Three                CH (SEt) S (= NCN) Et
CH₂CF_Three             CH (SEt) S (O) (= NCN) Et
CH₂CF_Three                    CH (CN) SMe
CH₂CF_Three                    CH (CN) S (O) Me
CH₂CF_Three                    CH (CN) S (O)₂Me
CH₂CF_Three                    CH (CN) SEt
CH₂CF_Three                    CH (CN) S (O) Et
CH₂CF_Three                    CH (CN) S (O)₂Et
CH₂CF_Three                 CH (CN) S (= NCN) Et
CH₂CF_Three              CH (CN) S (O) (= NCN) Et
CH₂CF_Three                  CH {C (O) OMe} SMe
CH₂CF_Three               CH {C (O) OMe} S (O) Me
CH₂CF_Three               CH {C (O) OMe} S (O)₂Me
CH₂CF_Three                  CH {C (O) OMe} SMe
CH₂CF_Three               CH {C (O) OMe} S (O) Me
CH₂CF_Three               CH {C (O) OMe} S (O)₂Me
CH₂CF_Three                  CH {C (O) OMe} SEt
CH₂CF_Three               CH {C (O) OMe} S (O) Et
CH₂CF_Three               CH {C (O) OMe} S (O)₂Et
CH₂CF_Three            CH {C (O) OMe} S (= NCN) Et
CH₂CF_Three         CH {C (O) OMe} S (O) (= NCN) Et
CH₂CF_Three                  CH {C (O) OEt} SMe
CH₂CF_Three               CH {C (O) OEt} S (O) Me
CH₂CF_Three               CH {C (O) OEt} S (O)₂Me
CH₂CF_Three                  CH {C (O) OEt} SEt
CH₂CF_Three               CH {C (O) OEt} S (O) Et
CH₂CF_Three               CH {C (O) OEt} S (O)₂Et
CH₂CF_Three            CH {C (O) OEt} S (= NCN) Et
CH₂CF_Three         CH {C (O) OEt} S (O) (= NCN) Et
CH₂CF_Three                    C (Me)₂SMe
CH₂CF_Three                    C (Me)₂S (O) Me
CH₂CF_Three                    C (Me)₂S (O)₂Me
CH₂CF_Three                    OBu-t
S (O)₂Me CH₂SMe
S (O)₂Me CH₂S (O) Me
S (O)₂Me CH₂S (O)₂Me
S (O)₂Me CH₂SEt
S (O)₂Me CH₂S (O) Et
S (O)₂Me CH₂S (O)₂Et
S (O)₂Me CH₂SPr-n
S (O)₂Me CH₂S (O) Pr-n
S (O)₂Me CH₂S (O)₂Pr-n
S (O)₂Me CH₂SPr-i
S (O)₂Me CH₂S (O) Pr-i
S (O)₂Me CH₂S (O)₂Pr-i
S (O)₂Me CH₂SPr-c
S (O)₂Me CH₂S (O) Pr-c
S (O)₂Me CH₂S (O)₂Pr-c
S (O)₂Me CH₂SCH₂CH = CH₂
S (O)₂Me CH₂S (O) CH₂CH = CH₂
S (O)₂Me CH₂S (O)₂CH₂CH = CH₂
S (O)₂Me CH₂SCH₂C≡CH
S (O)₂Me CH₂S (O) CH₂C≡CH
S (O)₂Me CH₂S (O)₂CH₂C≡CH
S (O)₂Me CH₂SCH₂CF_Three
S (O)₂Me CH₂S (O) CH₂CF_Three
S (O)₂Me CH₂S (O)₂CH₂CF_Three
S (O)₂Me CH₂SCH₂CH (OMe)₂
S (O)₂Me CH₂SCH₂CH (= NOMe)
S (O)₂Me CH (Me) SMe
S (O)₂Me CH (Me) S (O) Me
S (O)₂Me CH (Me) S (O)₂Me
S (O)₂Me CH (Me) SEt
S (O)₂Me CH (Me) S (O) Et
S (O)₂Me CH (Me) S (O)₂Et
S (O)₂Me CH (Me) S (= NCN) Et
S (O)₂Me CH (Me) S (O) (= NCN) Et
S (O)₂Me CH (Me) SPr-n
S (O)₂Me CH (Me) S (O) Pr-n
S (O)₂Me CH (Me) S (O)₂Pr-n
S (O)₂Me CH (Me) SPr-i
S (O)₂Me CH (Me) S (O) Pr-i
S (O)₂Me CH (Me) S (O)₂Pr-i
S (O)₂Me CH (Me) SBu-t
S (O)₂Me CH (Me) S (O) Bu-t
S (O)₂Me CH (Me) S (O)₂Bu-t
S (O)₂Me CH (Me) SCH₂Pr-c
S (O)₂Me CH (Me) S (O) CH₂Pr-c
S (O)₂Me CH (Me) S (O)₂CH₂Pr-c
S (O)₂Me CH (Me) SCH₂OMe
S (O)₂Me CH (Me) SCH₂SMe
S (O)₂Me CH (Me) S (O) CH₂SMe
S (O)₂Me CH (Me) S (O)₂CH₂SMe
S (O)₂Me CH (Me) SCH₂C = CH₂
S (O)₂Me CH (Me) S (O) CH₂C = CH₂
S (O)₂Me CH (Me) S (O)₂CH₂C = CH₂
S (O)₂Me CH (Me) SCH₂C≡CH
S (O)₂Me CH (Me) S (O) CH₂C≡CH
S (O)₂Me CH (Me) S (O)₂CH₂C≡CH
S (O)₂Me CH (Me) SCH₂C (O) NHMe
S (O)₂Me CH (Me) S (O) CH₂C (O) NHMe
S (O)₂Me CH (Me) S (O)₂CH₂C (O) NHMe
S (O)₂Me CH (Me) SCH₂C (O) OMe
S (O)₂Me CH (Me) S (O) CH₂C (O) OMe
S (O)₂Me CH (Me) S (O)₂CH₂C (O) OMe
S (O)₂Me CH (Me) SCH₂CH₂CH₂Cl
S (O)₂Me CH (Me) S (O) CH₂CH₂CH₂Cl
S (O)₂Me CH (Me) S (O)₂CH₂CH₂CH₂Cl
S (O)₂Me CH (Me) SCH₂CF_Three
S (O)₂Me CH (Me) S (O) CH₂CF_Three
S (O)₂Me CH (Me) S (O)₂CH₂CF_Three
S (O)₂Me CH (Me) SCH₂Ph
S (O)₂Me CH (Me) S (O) CH₂Ph
S (O)₂Me CH (Me) S (O)₂CH₂Ph
S (O)₂Me CH (Me) SCH₂(D2-34a)
S (O)₂Me CH (Me) S (O) CH₂(D2-34a)
S (O)₂Me CH (Me) S (O)₂CH₂(D2-34a)
S (O)₂Me CH (CH_Three) SCH₂Si (CH_Three)_Three
S (O)₂Me CH (Me) SCN
S (O)₂Me CH (Me) SCH₂CN
S (O)₂Me CH (Me) SC (O) Me
S (O)₂Me CH (Me) S (D2-12a)
S (O)₂Me CH (Me) S (D2-32a)
S (O)₂Me CH (Me) S {D2-32b (3-NO₂)}
S (O)₂Me CH (Me) S {D2-32b (3-CF_Three)}
S (O)₂Me CH (Me) S (D2-37a)
S (O)₂Me CH (Me) S (D2-51a)
S (O)₂Me CH (Et) SMe
S (O)₂Me CH (Et) S (O) Me
S (O)₂Me CH (Et) S (O)₂Me
S (O)₂Me CH (Et) SEt
S (O)₂Me CH (Et) S (O) Et
S (O)₂Me CH (Et) S (O)₂Et
S (O)₂Me CH (Et) SCH₂CF_Three
S (O)₂Me CH (Et) S (O) CH₂CF_Three
S (O)₂Me CH (Et) S (O)₂CH₂CF_Three
S (O)₂Me CH (Pr-n) SMe
S (O)₂Me CH (Pr-n) S (O) Me
S (O)₂Me CH (Pr-n) S (O)₂Me
S (O)₂Me CH (Pr-n) SEt
S (O)₂Me CH (Pr-n) S (O) Et
S (O)₂Me CH (Pr-n) S (O)₂Et
S (O)₂Me CH (Pr-n) S (= NCN) Et
S (O)₂Me CH (Pr-n) S (O) (= NCN) Et
S (O)₂Me CH (Pr-n) SPr-n
S (O)₂Me CH (Pr-n) S (O) Pr-n
S (O)₂Me CH (Pr-n) S (O)₂Pr-n
S (O)₂Me CH (Pr-n) SPr-i
S (O)₂Me CH (Pr-n) S (O) Pr-i
S (O)₂Me CH (Pr-n) S (O)₂Pr-i
S (O)₂Me CH (Pr-n) SPr-c
S (O)₂Me CH (Pr-n) S (O) Pr-c
S (O)₂Me CH (Pr-n) S (O)₂Pr-c
S (O)₂Me CH (Pr-n) SCH₂CF_Three
S (O)₂Me CH (Pr-n) S (O) CH₂CF_Three
S (O)₂Me CH (Pr-n) S (O)₂CH₂CF_Three
S (O)₂Me CH (Pr-i) SMe
S (O)₂Me CH (Pr-i) S (O) Me
S (O)₂Me CH (Pr-i) S (O)₂Me
S (O)₂Me CH (Pr-i) SEt
S (O)₂Me CH (Pr-i) S (O) Et
S (O)₂Me CH (Pr-i) S (O)₂Et
S (O)₂Me CH (Pr-i) S (= NCN) Et
S (O)₂Me CH (Pr-i) S (O) (= NCN) Et
S (O)₂Me CH (Pr-i) SPr-n
S (O)₂Me CH (Pr-i) S (O) Pr-n
S (O)₂Me CH (Pr-i) S (O)₂Pr-n
S (O)₂Me CH (Pr-i) SPr-i
S (O)₂Me CH (Pr-i) S (O) Pr-i
S (O)₂Me CH (Pr-i) S (O)₂Pr-i
S (O)₂Me CH (Pr-i) SPr-c
S (O)₂Me CH (Pr-i) S (O) Pr-c
S (O)₂Me CH (Pr-i) S (O)₂Pr-c
S (O)₂Me CH (Pr-i) SCH₂CF_Three
S (O)₂Me CH (Pr-i) S (O) CH₂CF_Three
S (O)₂Me CH (Pr-i) S (O)₂CH₂CF_Three
S (O)₂Me CH (Pr-c) SMe
S (O)₂Me CH (Pr-c) S (O) Me
S (O)₂Me CH (Pr-c) S (O)₂Me
S (O)₂Me CH (Pr-c) SEt
S (O)₂Me CH (Pr-c) S (O) Et
S (O)₂Me CH (Pr-c) S (O)₂Et
S (O)₂Me CH (Pr-c) S (= NCN) Et
S (O)₂Me CH (Pr-c) S (O) (= NCN) Et
S (O)₂Me CH (Pr-c) SPr-n
S (O)₂Me CH (Pr-c) S (O) Pr-n
S (O)₂Me CH (Pr-c) S (O)₂Pr-n
S (O)₂Me CH (Pr-c) SPr-i
S (O)₂Me CH (Pr-c) S (O) Pr-i
S (O)₂Me CH (Pr-c) S (O)₂Pr-i
S (O)₂Me CH (Pr-c) SPr-c
S (O)₂Me CH (Pr-c) S (O) Pr-c
S (O)₂Me CH (Pr-c) S (O)₂Pr-c
S (O)₂Me CH (Pr-c) SCH₂CF_Three
S (O)₂Me CH (Pr-c) S (O) CH₂CF_Three
S (O)₂Me CH (Pr-c) S (O)₂CH₂CF_Three
S (O)₂Me CH (Bu-n) SMe
S (O)₂Me CH (Bu-n) S (O) Me
S (O)₂Me CH (Bu-n) S (O)₂Me
S (O)₂Me CH (Bu-n) SEt
S (O)₂Me CH (Bu-n) S (O) Et
S (O)₂Me CH (Bu-n) S (O)₂Et
S (O)₂Me CH (Bu-n) S (= NCN) Et
S (O)₂Me CH (Bu-n) S (O) (= NCN) Et
S (O)₂Me CH (Bu-n) SPr-n
S (O)₂Me CH (Bu-n) S (O) Pr-n
S (O)₂Me CH (Bu-n) S (O)₂Pr-n
S (O)₂Me CH (Bu-n) SPr-i
S (O)₂Me CH (Bu-n) S (O) Pr-i
S (O)₂Me CH (Bu-n) S (O)₂Pr-i
S (O)₂Me CH (Bu-n) SPr-c
S (O)₂Me CH (Bu-n) S (O) Pr-c
S (O)₂Me CH (Bu-n) S (O)₂Pr-c
S (O)₂Me CH (Bu-n) SCH₂CF_Three
S (O)₂Me CH (Bu-n) S (O) CH₂CF_Three
S (O)₂Me CH (Bu-n) S (O)₂CH₂CF_Three
S (O)₂Me CH (F) SMe
S (O)₂Me CH (F) S (O) Me
S (O)₂Me CH (F) S (O)₂Me
S (O)₂Me CH (F) SEt
S (O)₂Me CH (F) S (O) Et
S (O)₂Me CH (F) S (O)₂Et
S (O)₂Me CH (F) S (= NCN) Et
S (O)₂Me CH (F) S (O) (= NCN) Et
S (O)₂Me CH (F) SCH₂CF_Three
S (O)₂Me CH (F) S (O) CH₂CF_Three
S (O)₂Me CH (F) S (O)₂CH₂CF_Three
S (O)₂Me C (F)₂SMe
S (O)₂Me C (F)₂S (O) Me
S (O)₂Me C (F)₂S (O)₂Me
S (O)₂Me C (F)₂SEt
S (O)₂Me C (F)₂S (O) Et
S (O)₂Me C (F)₂S (O)₂Et
S (O)₂Me C (F)₂S (= NCN) Et
S (O)₂Me C (F)₂S (O) (= NCN) Et
S (O)₂Me C (F)₂SCH₂CF_Three
S (O)₂Me C (F)₂S (O) CH₂CF_Three
S (O)₂Me C (F)₂S (O)₂CH₂CF_Three
S (O)₂Me CH (Cl) SMe
S (O)₂Me CH (Cl) S (O) Me
S (O)₂Me CH (Cl) S (O)₂Me
S (O)₂Me CH (Cl) SEt
S (O)₂Me CH (Cl) S (O) Et
S (O)₂Me CH (Cl) S (O)₂Et
S (O)₂Me CH (Cl) S (= NCN) Et
S (O)₂Me CH (Cl) S (O) (= NCN) Et
S (O)₂Me CH (Cl) SCH₂CF_Three
S (O)₂Me CH (Cl) S (O) CH₂CF_Three
S (O)₂Me CH (Cl) S (O)₂CH₂CF_Three
S (O)₂Me C (Cl)₂SMe
S (O)₂Me C (Cl)₂S (O) Me
S (O)₂Me C (Cl)₂S (O)₂Me
S (O)₂Me C (Cl)₂SEt
S (O)₂Me C (Cl)₂S (O) Et
S (O)₂Me C (Cl)₂S (O)₂Et
S (O)₂Me C (Cl)₂S (= NCN) Et
S (O)₂Me C (Cl)₂S (O) (= NCN) Et
S (O)₂Me C (Cl)₂SCH₂CF_Three
S (O)₂Me C (Cl)₂S (O) CH₂CF_Three
S (O)₂Me C (Cl)₂S (O)₂CH₂CF_Three
S (O)₂Me CH (Br) SMe
S (O)₂Me CH (Br) S (O) Me
S (O)₂Me CH (Br) S (O)₂Me
S (O)₂Me CH (Br) SEt
S (O)₂Me CH (Br) S (O) Et
S (O)₂Me CH (Br) S (O)₂Et
S (O)₂Me CH (Br) S (= NCN) Et
S (O)₂Me CH (Br) S (O) (= NCN) Et
S (O)₂Me CH (Br) SCH₂CF_Three
S (O)₂Me CH (Br) S (O) CH₂CF_Three
S (O)₂Me CH (Br) S (O)₂CH₂CF_Three
S (O)₂Me CH (I) SMe
S (O)₂Me CH (I) S (O) Me
S (O)₂Me CH (I) S (O)₂Me
S (O)₂Me CH (I) SEt
S (O)₂Me CH (I) S (O) Et
S (O)₂Me CH (I) S (O)₂Et
S (O)₂Me CH (I) S (= NCN) Et
S (O)₂Me CH (I) S (O) (= NCN) Et
S (O)₂Me CH (I) SCH₂CF_Three
S (O)₂Me CH (I) S (O) CH₂CF_Three
S (O)₂Me CH (I) S (O)₂CH₂CF_Three
S (O)₂Me CH {OC (O) Me} SMe
S (O)₂Me CH {OC (O) Me} S (O) Me
S (O)₂Me CH {OC (O) Me} S (O)₂Me
S (O)₂Me CH {OC (O) OMe} SEt
S (O)₂Me CH {OC (O) OMe} S (O) Et
S (O)₂Me CH {OC (O) OMe} S (O)₂Et
S (O)₂Me CH {OC (O) OMe} S (= NCN) Et
S (O)₂Me CH {OC (O) OMe} S (O) (= NCN) Et
S (O)₂Me CH {OC (O) OEt} SMe
S (O)₂Me CH {OC (O) OEt} S (O) Me
S (O)₂Me CH {OC (O) OEt} S (O)₂Me
S (O)₂Me CH {OC (O) OEt} SEt
S (O)₂Me CH {OC (O) OEt} S (O) Et
S (O)₂Me CH {OC (O) OEt} S (O)₂Et
S (O)₂Me CH {OC (O) OEt} S (= NCN) Et
S (O)₂Me CH {OC (O) OEt} S (O) (= NCN) Et
S (O)₂Me CH (OMe) SMe
S (O)₂Me CH (OMe) S (O) Me
S (O)₂Me CH (OMe) S (O)₂Me
S (O)₂Me CH (OMe) SEt
S (O)₂Me CH (OMe) S (O) Et
S (O)₂Me CH (OMe) S (O)₂Et
S (O)₂Me CH (OMe) S (= NCN) Et
S (O)₂Me CH (OMe) S (O) (= NCN) Et
S (O)₂Me CH (OEt) SMe
S (O)₂Me CH (OEt) S (O) Me
S (O)₂Me CH (OEt) S (O)₂Me
S (O)₂Me CH (OEt) SEt
S (O)₂Me CH (OEt) S (O) Et
S (O)₂Me CH (OEt) S (O)₂Et
S (O)₂Me CH (OEt) S (= NCN) Et
S (O)₂Me CH (OEt) S (O) (= NCN) Et
S (O)₂Me CH (SMe)₂
S (O)₂Me CH (SMe) S (O) Me
S (O)₂Me CH (SMe) S (O)₂Me
S (O)₂Me CH (SMe) SEt
S (O)₂Me CH (SMe) S (O) Et
S (O)₂Me CH (SMe) S (O)₂Et
S (O)₂Me CH (SMe) S (= NCN) Et
S (O)₂Me CH (SMe) S (O) (= NCN) Et
S (O)₂Me CH (SEt) SMe
S (O)₂Me CH (SEt) S (O) Me
S (O)₂Me CH (SEt) S (O)₂Me
S (O)₂Me CH (SEt) SEt
S (O)₂Me CH (SEt) S (O) Et
S (O)₂Me CH (SEt) S (O)₂Et
S (O)₂Me CH (SEt) S (= NCN) Et
S (O)₂Me CH (SEt) S (O) (= NCN) Et
S (O)₂Me CH (CN) SMe
S (O)₂Me CH (CN) S (O) Me
S (O)₂Me CH (CN) S (O)₂Me
S (O)₂Me CH (CN) SEt
S (O)₂Me CH (CN) S (O) Et
S (O)₂Me CH (CN) S (O)₂Et
S (O)₂Me CH (CN) S (= NCN) Et
S (O)₂Me CH (CN) S (O) (= NCN) Et
S (O)₂Me CH {C (O) OMe} SMe
S (O)₂Me CH {C (O) OMe} S (O) Me
S (O)₂Me CH {C (O) OMe} S (O)₂Me
S (O)₂Me CH {C (O) OMe} SMe
S (O)₂Me CH {C (O) OMe} S (O
S (O)₂Me CH {C (O) OMe} S (O)₂Me
S (O)₂Me CH {C (O) OMe} SEt
S (O)₂Me CH {C (O) OMe} S (O) Et
S (O)₂Me CH {C (O) OMe} S (O)₂Et
S (O)₂Me CH {C (O) OMe} S (= NCN) Et
S (O)₂Me CH {C (O) OMe} S (O) (= NCN) Et
S (O)₂Me CH {C (O) OEt} SMe
S (O)₂Me CH {C (O) OEt} S (O) Me
S (O)₂Me CH {C (O) OEt} S (O)₂Me
S (O)₂Me CH {C (O) OEt} SEt
S (O)₂Me CH {C (O) OEt} S (O) Et
S (O)₂Me CH {C (O) OEt} S (O)₂Et
S (O)₂Me CH {C (O) OEt} S (= NCN) Et
S (O)₂Me CH {C (O) OEt} S (O) (= NCN) Et
S (O)₂Me C (Me)₂SMe
S (O)₂Me C (Me)₂S (O) Me
S (O)₂Me C (Me)₂S (O)₂Me
SC (Cl)_Three                  CH (Me) SMe
SC (Cl)_Three                  CH (Me) S (O) Me
SC (Cl)_Three                  CH (Me) S (O)₂Me
SC (Cl)_Three                  CH (Me) SEt
SC (Cl)_Three                  CH (Me) S (O) Et
SC (Cl)_Three                  CH (Me) S (O)₂Et
SC (Cl)_Three                  CH (Me) CH₂SMe
CH₂CH₂CH₂SMe Me
CH₂CH₂SMe Me
NH₂                       OBu-t
NHC (O) CH₂SMe OBu-t
N (Me) C (O) CH₂SMe OBu-t
NHC (O) CH (Me) SMe OBu-t
N (Me) C (O) CH (Me) SMe OBu-t
NHC (O) CH₂CH₂SMe OBu-t
N {C (O) OBu-t}₂             OBu-t
NHC (O) OBu-t OBu-t
―――――――――――――――――――
[Table 6]

第６表
―――――――――――――――――――
R^f2 R^f3
―――――――――――――――――――
H CH₂CF₃
H CH₂CN
H CH₂SMe
H CH₂S(O)Me
H CH₂S(O)₂Me
H CH₂CH₂SMe
H CH₂CH₂S(O)Me
H CH₂CH₂S(O)₂Me
H CH(Me)CH₂SMe
H CH(Me)CH₂S(O)Me
H CH(Me)CH₂S(O)₂Me
H CH₂CH(OMe)₂
H CH₂CH(OEt)₂
H NHC(O)OMe
H NHC(O)OEt
H NHC(O)OPr-n
H NHC(O)OPr-i
H NHC(O)OBu-n
H NHC(O)OBu-i
H NHC(O)OBu-s
H NHC(O)OBu-t
H D2-32a
H D2-33a
H D2-34a
H D2-37a
H CH₂(D2-32a)
H CH₂(D2-33a)
H CH₂(D2-34a)
H CH₂(D2-37a)
Me CH₂CF₃
Me CH₂CH₂SMe
Me CH₂CH₂S(O)Me
Me CH₂CH₂S(O)₂Me
Me CH(Me)CH₂SMe
Me CH(Me)CH₂S(O)Me
Me CH(Me)CH₂S(O)₂Me
Me CH₂CH(OMe)₂
Me CH₂CH(OEt)₂
Me NHC(O)OMe
Me NHC(O)OEt
Me NHC(O)OPr-n
Me NHC(O)OPr-i
Me NHC(O)OBu-n
Me NHC(O)OBu-i
Me NHC(O)OBu-s
Me NHC(O)OBu-t
Me D2-32a
Me D2-33a
Me D2-34a
Me D2-37a
Me CH₂(D2-32a)
Me CH₂(D2-33a)
Me CH₂(D2-34a)
Me CH₂(D2-37a)
H H
H Me
H Et
H n-Pr
H i-Pr
H c-Pr
H n-Bu
H i-Bu
H s-Bu
H t-Bu
H c-Bu
H n-Pen
H c-Pen
H n-Hex
H c-Hex
H Hep
H Oct
H CH₂Pr-c
H CH₂Bu-i
H CH₂Bu-s
H CH₂Bu-t
H CH₂Bu-c
H CH₂Pen-c
H CH₂Hex-c
H CH(CH₃)Pr-n
H CH(CH₃)Pr-i
H CH(CH₃)Pr-n
H CH(CH₃)Bu-i
H CH(Et)₂
H C(CH₃)₂Et
H C(CH₃)₂Pr-n
H CH₂CH₂F
H CH₂CH₂Cl
H CH₂CH₂Br
H CH₂CHF₂
H CH₂CHFCl
H CH₂CHCl₂
H CH₂CHFBr
H CH₂CF₂Cl
H CH₂CFCl₂
H CH₂CCl₃
H CH₂CF₂Br
H CH₂CFClBr
H CH₂CCl₂Br
H CH(CH₃)CH₂F
H CH(CH₃)CH₂Cl
H CH(CH₃)CH₂Br
H CH₂CHFCH₃
H CH₂CHClCH₃
H CH₂CHBrCH₃
H CH₂CFClCH₃
H CH₂CHClCH₂Cl
H CH₂CHBrCH₂F
H CH₂CHClCH₂Br
H CH₂CHBrCH₂Cl
H CH₂CHBrCHCl₂
H CH₂CClBrCH₃
H CH₂CHBrCH₂Br
H CH₂CH₂CF₃
H CH₂CH₂CF₂Br
H CH₂CClBrCH₂Cl
H CH₂CF₂CF₂H
H CH₂CHClCF₃
H CH₂CF₂CF₃
H CH₂CF(CH₃)₂
H CH₂CHFCH₂CH₃
H CH₂CHClCH₂CH₃
H CH₂CF₂CHFCF₃
H CH₂CF₂CF₂CHF₂
H CH₂CF₂CF₂CF₃
H C(CH₃)₂CH₂Cl
H C(CH₃)₂CH₂Br
H C(CH₃)₂CHBrCH₂Br
H CH₂CF₃
Me CH₂CF₃
Et CH₂CF₃
n-Pr CH₂CF₃
i-Pr CH₂CF₃
CH₂OCH₃ CH₂CF₃
CH₂CH₂OEt CH₂CF₃
CH₂SCH₃ CH₂CF₃
CH₂CN CH₂CF₃
CH₂CO₂Me CH₂CF₃
CH₂CO₂Et CH₂CF₃
CH₂CH=CH₂ CH₂CF₃
CH₂CH≡CH CH₂CF₃
C(O)CH₃ CH₂CF₃
C(O)Et CH₂CF₃
C(O)Pr-n CH₂CF₃
C(O)Pr-c CH₂CF₃
C(O)Bu-t CH₂CF₃
C(O)CH₂OCH₃ CH₂CF₃
C(O)CH₂SCH₃ CH₂CF₃
C(O)OMe CH₂CF₃
C(O)OEt CH₂CF₃
C(O)CH₂CH₂Cl CH₂CF₃
C(O)CH₂CH₂OMe CH₂CF₃
C(O)OCH₂CH=CH₂ CH₂CF₃
C(O)SCH₃ CH₂CF₃
C(S)OCH₃ CH₂CF₃
C(S)SCH₃ CH₂CF₃
SMe CH₂CF₃
SPh CH₂CF₃
SNEt₂ CH₂CF₃
SO₂Me CH₂CF₃
SO₂Et CH₂CF₃
SO₂Ph CH₂CF₃
SO₂NMe₂ CH₂CF₃
NH₂ CH₂CF₃
NHMe CH₂CF₃
NHCHO CH₂CF₃
NHC(O)CH₃ CH₂CF₃
NHC(O)OCH₃ CH₂CF₃
N=C(CH₃)₂ CH₂CF₃
N=CHPh CH₂CF₃
H CH(CF₃)Me
H CH(CF₃)Et
H CH(CF₃)OH
H CH(CF₃)OMe
H CH₂CH(OMe)₂
H CH₂CH(OEt)₂
H CH₂CN
H CH(Me)CN
H C(Me)₂CN
H CH(OMe)CN
H CH₂CH₂CN
H CH₂C(O)Me
H CH₂C(O)OMe
H CH₂C(O)OEt
H CH₂C(O)OCH₂CF₃
H CH(Me)C(O)OMe
H CH(Me)C(O)OEt
H CH(Me)C(O)OCH₂CF₃
H CH(OMe)C(O)OMe
H CH(OMe)C(O)OEt
H CH(OMe)C(O)OCH₂CF₃
H CH(Ph)C(O)OMe
H CH(Ph)C(O)OEt
H CH(Ph)C(O)OCH₂CF₃
H CH(CF₃)C(O)OMe
H CH(CF₃)C(O)OEt
H CH(CF₃)C(O)OCH₂CF₃
H CH₂CH₂C(O)OMe
H CH₂CH₂C(O)OEt
H CH₂CH₂C(O)OCH₂CF₃
H CH₂CH(Me)C(O)OMe
H CH₂CH(Me)C(O)OEt
H CH(Me)CH₂C(O)OMe
H CH(Me)CH₂C(O)OEt
H CH₂C(O)NH₂
H CH₂C(O)NHMe
H CH₂C(O)NHEt
H CH₂C(O)NHPr-n
H CH₂C(O)NHPr-i
H CH₂C(O)NHPr-c
H CH₂C(O)NHBu-n
H CH₂C(O)NHBu-i
H CH₂C(O)NHBu-s
H CH₂C(O)NHBu-t
H CH₂C(O)NHBu-c
H CH₂C(O)NHHex-n
H CH₂C(O)NHHex-c
H CH₂C(O)N(Me)₂
H CH₂C(O)N(Et)₂
H CH₂C(O)N(n-Pr)₂
H CH₂C(O)N(Me)Et
H CH₂C(O)N(Me)Pr-n
H CH₂C(O)N(Me)Pr-i
H CH₂C(O)NHCH₂CH₂F
H CH₂C(O)NHCH₂CH₂Cl
H CH₂C(O)NHCH₂CH₂Br
H CH₂C(O)N(Me)CH₂CH₂F
H CH₂C(O)N(Me)CH₂CH₂Cl
H CH₂C(O)N(Me)CH₂CH₂Br
H CH₂C(O)NHCH₂CF₃
CH₂OCH₃ CH₂C(O)NHCH₂CF₃
CH₂CN CH₂C(O)NHCH₂CF₃
CH₂CO₂Me CH₂C(O)NHCH₂CF₃
CH₂CO₂Et CH₂C(O)NHCH₂CF₃
CH₂CH=CH₂ CH₂C(O)NHCH₂CF₃
CH₂CH≡CH CH₂C(O)NHCH₂CF₃
C(O)Me CH₂C(O)NHCH₂CF₃
C(O)OMe CH₂C(O)NHCH₂CF₃
H CH₂C(O)N(Me)CH₂CF₃
H CH₂C(O)NHCH₂CF₂Cl
H CH₂C(O)NHCH₂CN
H CH₂C(O)NHCH₂CH=CH₂
H CH₂C(O)NHCH₂CH≡CH
H CH₂C(O)NHCH₂CH₂CH₂Cl
H CH₂C(O)NHCH₂CH₂OCH₃
H CH₂C(O)NHCH₂CH₂SCH₃
H CH₂C(O)NHCH₂CH₂SO₂CH₃
H CH(Me)C(O)NH₂
H CH(Me)C(O)NHMe
H CH(Me)C(O)NHEt
H CH(Me)C(O)NHPr-n
H CH(Me)C(O)NHPr-i
H CH(Me)C(O)NHPr-c
H CH(Me)C(O)NHBu-n
H CH(Me)C(O)NHBu-i
H CH(Me)C(O)NHBu-s
H CH(Me)C(O)NHBu-t
H CH(Me)C(O)NHBu-c
H CH(Me)C(O)NHHex-n
H CH(Me)C(O)NHHex-c
H CH(Me)C(O)N(Me)₂
H CH(Me)C(O)N(Et)₂
H CH(Me)C(O)N(n-Pr)₂
H CH(Me)C(O)N(Me)Et
H CH(Me)C(O)N(Me)Pr-n
H CH(Me)C(O)N(Me)Pr-i
H CH(Me)C(O)NHCH₂CH₂F
H CH(Me)C(O)NHCH₂CH₂Cl
H CH(Me)C(O)NHCH₂CH₂Br
H CH(Me)C(O)NHCH₂CF₃
H CH(Et)C(O)NHCH₂CF₃
H CH(i-Pr)C(O)NHCH₂CF₃
H CH(CH₂OCH₃)C(O)NHCH₂CF₃
H CH(CH₂SCH₃)C(O)NHCH₂CF₃
H CH(Ph)C(O)NHCH₂CF₃
H CH(CH₂Ph)C(O)NHCH₂CF₃
H CH(CF₃)C(O)NHMe
H CH(CF₃)C(O)NHEt
H CH(CF₃)C(O)NHPr-n
H CH(CF₃)C(O)NHPr-i
H CH(CF₃)C(O)NHPr-c
H CH(CF₃)C(O)NHBu-n
H CH(CF₃)C(O)NHBu-i
H CH(CF₃)C(O)NHBu-s
H CH(CF₃)C(O)NHBu-t
H CH(CF₃)C(O)NHBu-c
H CH(CF₃)C(O)NHHex-n
H CH(CF₃)C(O)NHHex-c
H CH(CF₃)C(O)N(Me)₂
H CH(CF₃)C(O)N(Et)₂
H CH(CF₃)C(O)N(n-Pr)₂
H CH(CF₃)C(O)N(Me)Et
H CH(CF₃)C(O)N(Me)Pr-n
H CH(CF₃)C(O)N(Me)Pr-i
H CH(CF₃)C(O)NHCH₂CH₂F
H CH(CF₃)C(O)NHCH₂CH₂Cl
H CH(CF₃)C(O)NHCH₂CH₂Br
H CH(CF₃)C(O)NHCH₂CF₃
H CH₂CH₂C(O)NHCH₂CF₃
H CH₂C(O)N(Me)₂
H CH₂C(O)N(Et)₂
H CH₂C(O)N(n-Pr)₂
H CH₂CH=CH₂
H CH₂C(Me)=CH₂
H CH₂C(Et)=CH₂
H CH(Me)CH=CH₂
H CH₂CH=C(Me)₂
H CH₂C(Me)=CHCH₃
H CH(Me)CH=CHCH₃
H CH₂C(F)=CH₂
H CH₂CH=CHCl
H CH₂C(Cl)=CH₂
H CH₂CH=CCl₂
H CH₂CH=CHBr
H CH₂C(Br)=CH₂
H CH₂C(Br)=CHBr
H CH₂C(Me)=CHBr
H CH₂CH=C(Cl)CH₃
H CH₂CH=C(Br)CH₃
H CH₂C(OMe)=CH₂
H CH₂C(Br)=CHOMe
H CH₂C(Br)=CHOEt
H CH₂C(Br)=CHPh
H CH₂C≡CH
H CH₂C≡CCl
H CH₂C≡CBr
H CH₂C≡CI
H CH₂C≡CPh
H CH₂OMe
H CH₂CH₂OH
H CH₂CH₂OMe
H CH₂CH₂OEt
H CH₂CH₂OPr-n
H CH₂CH₂OPr-i
H CH₂CH₂OBu-i
H CH₂CH₂OCH₂CH₂Cl
H CH₂CH₂OCH₂CF3
H CH₂CH₂OCH₂CH₂OCH₃
H CH₂CH₂OCH₂CH₂SCH₃
H CH₂CH₂OC(O)CH₃
H CH₂CH(Me)OH
H CH₂CH(Me)OMe
H CH₂CH(Me)OCH₂CF₃
H CH(Me)CH₂OH
H CH(Me)CH₂OMe
H CH(Me)CH₂OCH₂CF₃
H CH(Ph)CH₂OH
H CH(Ph)CH₂OMe
H CH(Ph)CH₂OCH₂CF₃
H C(Me)₂CH₂OH
H C(Me)₂CH₂OMe
H C(Me)₂CH₂OCH₂CF₃
H CH₂CH₂CH₂OH
H CH₂CH₂CH₂OMe
H CH₂CH₂CH₂OCH₂CF₃
H CH₂CH₂CH₂CH₂OH
H CH₂CH₂CH₂CH₂OMe
H CH₂CH₂CH₂CH₂OCH₂CF₃
H CH₂SMe
H CH(CF₃)SMe
H CH(CF₃)SEt
H CH₂CH₂SMe
H CH₂CH₂S(O)Me
H CH₂CH₂S(O)₂Me
H CH₂CH₂SEt
H CH₂CH₂S(O)Et
H CH₂CH₂S(O)₂Et
H CH₂CH₂SPr-n
H CH₂CH₂S(O)Pr-n
H CH₂CH₂S(O)₂Pr-n
H CH₂CH₂SPr-i
H CH₂CH₂S(O)Pr-i
H CH₂CH₂S(O)₂Pr-i
H CH₂CH₂SCH₂CF₃
H CH₂CH₂S(O)CH₂CF₃
H CH₂CH₂S(O)₂CH₂CF₃
H CH₂CH₂SCH₂CH₂OH
H CH₂CH₂S(O)CH₂CH₂OH
H CH₂CH₂S(O)₂CH₂CH₂OH
H CH₂CH₂SCH₂CH₂OMe
H CH₂CH₂S(O)CH₂CH₂OMe
H CH₂CH₂S(O)₂CH₂CH₂OMe
H CH₂CH₂SCH₂C(O)OMe
H CH₂CH₂S(O)CH₂C(O)OMe
H CH₂CH₂S(O)₂CH₂C(O)OMe
H CH₂CH₂SCH₂C(O)NHMe
H CH₂CH₂S(O)CH₂C(O)NHMe
H CH₂CH₂S(O)₂CH₂C(O)NHMe
H CH₂CH₂SCH₂C(O)NMe
H CH₂CH₂S(O)CH₂C(O)NMe
H CH₂CH₂S(O)₂CH₂C(O)N(Me)₂
H CH₂CH₂SCH₂CH=CH₂
H CH₂CH₂SCH₂CH≡CH
H CH₂CH₂S(O)₂NHMe
H CH₂CH₂S(O)₂N(Me)₂
H CH₂CH₂S(O)₂NHEt
H CH₂CH₂S(O)₂N(Et)₂
H CH₂CH₂S(O)₂NHPr-n
H CH₂CH₂S(O)₂N(Pr-n)₂
H CH₂CH₂S(O)₂NHPr-i
H CH₂CH₂S(O)₂N(Pr-i)₂
H CH₂CH₂S(O)₂NHPr-c
H CH₂CH₂S(O)₂NHBu-t
H CH₂CH₂S(O)₂NHCH₂CF₃
H CH₂CH₂S(O)₂NHCH₂CH₂OMe
H CH₂CH₂S(O)₂NHCH₂CH₂SMe
H CH₂CH₂S(O)₂NHCH₂CH=CH₂
H CH₂CH₂S(O)₂NHCH₂CH≡CH
H CH₂CH₂S(O)(=NCN)Me
H CH₂CH(Me)SMe
H CH₂CH(Me)S(O)Me
H CH₂CH(Me)S(O)₂Me
H CH₂CH(Me)SEt
H CH₂CH(Me)S(O)Et
H CH₂CH(Me)S(O)₂Et
H CH₂CH(Et)SMe
H CH₂CH(Et)S(O)Me
H CH₂CH(Et)S(O)₂Me
H CH₂CH(n-Pr)SMe
H CH₂CH(n-Pr)S(O)Me
H CH₂CH(n-Pr)S(O)₂Me
H CH₂CH(i-Pr)SMe
H CH₂CH(i-Pr)S(O)Me
H CH₂CH(i-Pr)S(O)₂Me
H CH₂CH(Ph)SMe
H CH₂CH(Ph)S(O)Me
H CH₂CH(Ph)S(O)₂Me
H CH(Me)CH₂SMe
H CH(Me)CH₂S(O)Me
H CH(Me)CH₂S(O)₂Me
H CH(Me)CH₂SEt
H CH(Me)CH₂S(O)Et
H CH(Me)CH₂S(O)₂Et
H CH(Me)CH₂SPr-n
H CH(Me)CH₂S(O)Pr-n
H CH(Me)CH₂S(O)₂Pr-n
H CH(Me)CH₂SPr-i
H CH(Me)CH₂S(O)Pr-i
H CH(Me)CH₂S(O)₂Pr-i
H CH(Me)CH₂SPh
H CH(Me)CH₂S(O)Ph
H CH(Me)CH₂S(O)₂Ph
H CH(Ph)CH₂SMe
H CH(Ph)CH₂S(O)Me
H CH(Ph)CH₂S(O)₂Me
H CH(Me)CH(Me)SMe
H CH(Me)CH(Me)S(O)Me
H CH(Me)CH(Me)S(O)₂Me
H C(Me)₂CH₂SMe
H C(Me)₂CH₂S(O)Me
H C(Me)₂CH₂S(O)₂Me
H CH₂CH₂CH₂SMe
H CH₂CH₂CH₂S(O)Me
H CH₂CH₂CH₂S(O)₂Me
H CH₂CH₂CH(Me)SMe
H CH₂CH₂CH(Me)S(O)Me
H CH₂CH₂CH(Me)S(O)₂Me
H CH₂CH(Me)CH₂SMe
H CH₂CH(Me)CH₂S(O)Me
H CH₂CH(Me)CH₂S(O)₂Me
H CH(Me)CH₂CH₂SMe
H CH(Me)CH₂CH₂S(O)Me
H CH(Me)CH₂CH₂S(O)₂Me
H C(Me)₂CH₂CH₂SMe
H C(Me)₂CH₂CH₂S(O)Me
H C(Me)₂CH₂CH₂S(O)₂Me
H CH(Me)(CH₂)₃SMe
H CH(Me)(CH₂)₃S(O)Me
H CH(Me)(CH₂)₃S(O)₂Me
H CH(Me)(CH₂)₄SMe
H CH(Me)(CH₂)₄S(O)Me
H CH(Me)(CH₂)₄S(O)₂Me
H CH₂NHC(O)Me
H CH₂NHC(O)Et
H CH₂NHC(O)Pr-n
H CH₂CH₂NHC(O)Me
H CH₂CH₂NHC(O)Et
H CH₂CH₂NHC(O)Pr-n
H CH₂CH₂NHC(O)Pr-i
H CH₂CH₂NHC(O)Pr-c
H CH₂CH₂NHC(O)Bu-n
H CH₂CH₂NHC(O)Bu-i
H CH₂CH₂NHC(O)Bu-s
H CH₂CH₂NHC(O)Bu-t
H CH₂CH₂NHC(O)CF₃
H CH₂CH₂NHC(O)CF₂Cl
H CH₂CH₂NHC(O)Ph
H CH₂CH₂NHC(O)CH₂CF₃
H CH₂CH₂NHC(O)CH₂SMe
H CH₂CH₂NHC(O)CH₂S(O)Me
H CH₂CH₂NHC(O)CH₂S(O)₂Me
H CH₂CH₂N(Me)C(O)Me
H CH₂CH₂N(Me)C(O)Et
H CH₂CH₂N(Me)C(O)CF₃
H CH₂CH₂N(Me)C(O)CH₂CF₃
H CH₂CH₂N(Me)C(O)CH₂SMe
H CH₂CH₂N(Me)C(O)CH₂S(O)Me
H CH₂CH₂N(Me)C(O)CH₂S(O)₂Me
H CH₂CH₂NHC(O)OMe
H CH₂CH₂NHC(O)OEt
H CH₂CH₂NHC(O)OPr-n
H CH₂CH₂NHC(O)OBu-t
H CH₂CH₂NHC(O)NHEt
H CH₂CH₂NHC(O)NHPr-n
H CH₂CH₂NHC(O)NHPr-i
H CH₂CH₂NHC(O)NHBu-t
H CH₂CH₂NHC(O)N(Me)₂
H CH₂CH₂NHSO₂Me
H CH₂CH₂NHSO₂Et
H CH₂CH₂NHSO₂CF₃
H CH₂CH₂NHSO₂Ph
H CH₂CH₂NHSO₂N(Me)₂
H CH₂CH₂NHP(S)(OMe)₂
H CH₂CH₂NHP(S)(OEt)₂
H CH₂CH₂N(Me)SO₂Me
H CH₂CH₂N(Me)SO₂CF₃
H CH₂CH₂N(Me)OMe
H CH₂CH(Me)NHC(O)Me
H CH₂CH(Me)NHC(O)CF₃
H CH₂CH(Me)NHC(O)CH₂CF₃
H CH₂CH(Me)NHC(O)CH₂SMe
H CH₂CH(Me)NHC(O)CH₂S(O)Me
H CH₂CH(Me)NHC(O)CH₂S(O)₂Me
H CH₂CH(Me)NHC(O)OMe
H CH(Me)CH₂NHC(O)Me
H CH(Me)CH₂NHC(O)CF₃
H CH(Me)CH₂NHC(O)CH₂CF₃
H CH(Me)CH₂NHC(O)CH₂SMe
H CH(Me)CH₂NHC(O)CH₂S(O)Me
H CH(Me)CH₂NHC(O)CH₂S(O)₂Me
H CH(Me)CH₂NHC(O)OMe
H CH₂CH₂CH₂NHC(O)Me
H CH₂CH₂CH₂NHC(O)OMe
H OMe
H OPr-i
H OCH₂CF₃
H OCH₂CH=CH₂
H OCH₂CH=CHCl
H N(Me)₂
H N(Et)₂
H N(n-Pr)₂
H NHCH₂CF₃
H N(Me)CH₂CF₃
H N(CH₂CF₃)C(O)Me
H N(CH₂CF₃)C(O)OMe
H N(CH₂CF₃)C(O)OEt
H NHCHO
H NHC(O)Me
H NHC(O)Et
H NHC(O)Pr-n
H NHC(O)Pr-i
H NHC(O)Pr-c
H NHC(O)Bu-n
H NHC(O)Bu-i
H NHC(O)Bu-s
H NHC(O)Bu-t
H NHC(O)Hex-n
H NHC(O)Hex-c
H NHC(O)CH₂CF₃
H NHC(O)CH₂SMe
H NHC(O)CH₂S(O)Me
H NHC(O)CH₂S(O)₂Me
H NHC(O)OMe
H NHC(O)OEt
H NHC(O)OBu-t
H NHC(O)SMe
H NHC(S)OMe
H NHC(S)SMe
H N(Me)CHO
H N(Me)C(O)Me
H N(Me)C(O)Et
H N(Me)C(O)Pr-n
H N(Me)C(O)Pr-i
H N(Me)C(O)Pr-c
H N(Me)C(O)Bu-n
H N(Me)C(O)Bu-i
H N(Me)C(O)Bu-s
H N(Me)C(O)Bu-t
H N(Me)C(O)Hex-n
H N(Me)C(O)Hex-c
H N(Me)C(O)CH₂CF₃
H N(Me)C(O)CH₂SMe
H N(Me)C(O)CH₂S(O)Me
H N(Me)C(O)CH₂S(O)₂Me
H N(Me)C(O)OMe
H N(Me)C(O)OEt
H N(Me)C(O)OBu-t
H N(Et)CHO
H N(Et)C(O)Me
H N(Et)C(O)Et
H N(Et)C(O)Pr-n
H N(Et)C(O)Pr-i
H N(Et)C(O)Pr-c
H N(Et)C(O)Bu-n
H N(Et)C(O)Bu-i
H N(Et)C(O)Bu-s
H N(Et)C(O)Bu-t
H N(Et)C(O)Hex-n
H N(Et)C(O)Hex-c
H N(Et)C(O)CH₂CF₃
H N(Et)C(O)CH₂SMe
H N(Et)C(O)CH₂S(O)Me
H N(Et)C(O)CH₂S(O)₂Me
H N(Et)C(O)OMe
H N(Et)C(O)OEt
H N(Et)C(O)OBu-t
H NHC(O)NHMe
H NHC(O)NHCH₂CF₃
H NHC(S)NHMe
H NHC(S)NHCH₂CF₃
H C(O)NHMe
H C(O)NHEt
H C(O)NHPr-n
H C(O)NHPr-i
H C(O)NHPr-c
H C(O)NHBu-n
H C(O)NHBu-i
H C(O)NHBu-s
H C(O)NHBu-t
H C(O)NHCH₂CH₂F
H C(O)NHCH₂CH₂Cl
H C(O)NHCH₂CH₂Br
H C(O)NHCH₂CF₃
H C(O)NHCH₂CF₂Cl
H C(O)NHCH₂CF₂CF₃
H C(O)NHCH₂CF₂CF₂H
H C(O)NHCH₂CH₂OMe
H C(O)NHCH₂CH₂SMe
H C(O)NHCH₂CH₂S(O)Me
H C(O)NHCH₂CH₂S(O)₂Me
H C(O)NHCH₂CN
H C(O)NHCH₂CH=CH₂
H C(O)NHCH₂CH≡CH
H C(O)N(Me)₂
H C(O)N(Me)Et
H C(O)N(Me)Pr-n
H C(O)N(Me)Pr-i
H C(O)N(Me)Pr-c
H C(O)N(Me)Bu-n
H C(O)N(Me)Bu-i
H C(O)N(Me)Bu-s
H C(O)N(Me)Bu-t
H C(O)N(Me)CH₂CH₂F
H C(O)N(Me)CH₂CH₂Cl
H C(O)N(Me)CH₂CH₂Br
H C(O)N(Me)CH₂CF₃
H C(O)N(Me)CH₂CF₂Cl
H C(O)N(Me)CH₂CF₂CF₃
H C(O)N(Me)CH₂CF₂CF₂H
H C(O)N(Me)CH₂CH₂OMe
H C(O)N(Me)CH₂CH₂SMe
H C(O)N(Me)CH₂CH₂S(O)Me
H C(O)N(Me)CH₂CH₂S(O)₂Me
H C(O)N(Me)CH₂CN
H C(O)N(Me)CH₂CH=CH₂
H C(O)N(Me)CH₂CH≡CH
H C(S)NHMe
H C(S)NHEt
H C(S)NHPr-n
H C(S)NHPr-i
H C(S)NHPr-c
H C(S)NHBu-n
H C(S)NHBu-i
H C(S)NHBu-s
H C(S)NHBu-t
H C(S)NHCH₂CH₂F
H C(S)NHCH₂CH₂Cl
H C(S)NHCH₂CH₂Br
H C(S)NHCH₂CF₃
H C(S)NHCH₂CF₂Cl
H C(S)NHCH₂CF₂CF₃
H C(S)NHCH₂CF₂CF₂H
H C(S)NHCH₂CH₂OMe
H C(S)NHCH₂CH₂SMe
H C(S)NHCH₂CH₂S(O)Me
H C(S)NHCH₂CH₂S(O)₂Me
H C(S)NHCH₂CN
H C(S)NHCH₂CH=CH₂
H C(S)NHCH₂CH≡CH
H C(S)N(Me)₂
H C(S)N(Me)Et
H C(S)N(Me)Pr-n
H C(S)N(Me)Pr-i
H C(S)N(Me)Pr-c
H C(S)N(Me)Bu-n
H C(S)N(Me)Bu-i
H C(S)N(Me)Bu-s
H C(S)N(Me)Bu-t
H C(S)N(Me)CH₂CH₂F
H C(S)N(Me)CH₂CH₂Cl
H C(S)N(Me)CH₂CH₂Br
H C(S)N(Me)CH₂CF₃
H C(S)N(Me)CH₂CF₂Cl
H C(S)N(Me)CH₂CF₂CF₃
H C(S)N(Me)CH₂CF₂CF₂H
H C(S)N(Me)CH₂CH₂OMe
H C(S)N(Me)CH₂CH₂SMe
H C(S)N(Me)CH₂CH₂S(O)Me
H C(S)N(Me)CH₂CH₂S(O)₂Me
H C(S)N(Me)CH₂CN
H C(S)N(Me)CH₂CH=CH₂
H C(S)N(Me)CH₂CH≡CH
H C(O)CH₂CF3
H C(O)CH₂SMe
H C(O)CH₂S(O)Me
H C(O)CH₂S(O)₂Me
H D2-1a
H D2-1b
H D2-2a
H D2-2b
H D2-5a
H D2-5b
H D2-5c
H D2-6a
H D2-6b
H D2-6c
H D2-7a
H D2-8a
H D2-8b
H D2-8c
H D2-9a
H D2-9b
H D2-9c
H D2-10a
H D2-10b
H D2-10c
H D2-11a
H D2-12a
H D2-12b
H D2-12c
H D2-13a
H D2-13b
H D2-14a
H D2-14b
H D2-15a
H D2-15b
H D2-16a
H D2-17a
H D2-18a
H D2-19a
H D2-21a
H D2-21b
H D2-22a
H D2-23a
H D2-23b
H D2-24a
H D2-25a
H D2-27a
H D2-30a
H D2-31a
H D2-32a
H D2-34a
H D2-36a
H D2-37a
H D2-41a
H D2-43a
H D2-45a
H D2-46a
H D2-49a
H D2-51a
H D2-53a
H D2-59a
H D2-61a
H D2-63a
H D2-68a
H D2-75a
H D2-76a
H D2-76b
H D2-77a
H D2-77b
H D2-78a
H D2-78b
H D2-79a
H D2-81a
H D2-82a
H D2-84a
H D2-85a
H D2-87a
H D2-90a
H D2-100a
H D2-100b
H D2-100c
H D2-100d
H D2-100e
H D2-101a
H D2-101b
H D2-101c
H D2-101d
H D2-102a
H D2-102b
H D2-102c
H D2-102d
H D2-102e
H D2-102f
H D2-103a
H CH₂(D2-1a)
H CH₂(D2-1b)
H CH₂(D2-2a)
H CH₂(D2-2b)
H CH₂(D2-4a)
H CH₂(D2-4b)
H CH₂(D2-5a)
H CH₂(D2-5b)
H CH₂(D2-5c)
H CH₂(D2-6a)
H CH₂(D2-6b)
H CH₂(D2-6c)
H CH₂(D2-7a)
H CH₂(D2-8a)
H CH₂(D2-8b)
H CH₂(D2-8c)
H CH₂(D2-9a)
H CH₂(D2-9b)
H CH₂(D2-9c)
H CH₂(D2-10a)
H CH₂(D2-10b)
H CH₂(D2-10c)
H CH₂(D2-12a)
H CH₂(D2-12b)
H CH₂(D2-12c)
H CH₂(D2-13a)
H CH₂(D2-13b)
H CH₂(D2-14a)
H CH₂(D2-14b)
H CH₂(D2-15a)
H CH₂(D2-15b)
H CH₂(D2-16a)
H CH₂(D2-17a)
H CH₂(D2-18a)
H CH₂(D2-19a)
H CH₂(D2-20a)
H CH₂(D2-21a)
H CH₂(D2-21b)
H CH₂(D2-23a)
H CH₂(D2-23b)
H CH₂(D2-25a)
H CH₂(D2-27a)
H CH₂(D2-30a)
H CH₂(D2-31a)
H CH₂(D2-32a)
Me CH₂(D2-32a)
Et CH₂(D2-32a)
n-Pr CH₂(D2-32a)
i-Pr CH₂(D2-32a)
CH₂OCH₃ CH₂(D2-32a)
CH₂CH₂OEt CH₂(D2-32a)
CH₂SCH₃ CH₂(D2-32a)
CH₂CN CH₂(D2-32a)
CH₂CO₂Me CH₂(D2-32a)
CH₂CO₂Et CH₂(D2-32a)
CH₂CH=CH₂ CH₂(D2-32a)
CH₂CH≡CH CH₂(D2-32a)
C(O)CH₃ CH₂(D2-32a)
C(O)Et CH₂(D2-32a)
C(O)Pr-n CH₂(D2-32a)
C(O)Pr-c CH₂(D2-32a)
C(O)Bu-t CH₂(D2-32a)
C(O)CH₂OCH₃ CH₂(D2-32a)
C(O)CH₂SCH₃ CH₂(D2-32a)
C(O)OMe CH₂(D2-32a)
C(O)OEt CH₂(D2-32a)
C(O)CH₂CH₂ CH₂(D2-32a)
C(O)CH₂CH₂ CH₂(D2-32a)
C(O)OCH₂CH=CH₂ CH₂(D2-32a)
C(O)SCH₃ CH₂(D2-32a)
C(S)OCH₃ CH₂(D2-32a)
C(S)SCH₃ CH₂(D2-32a)
SMe CH₂(D2-32a)
SPh CH₂(D2-32a)
SNEt₂ CH₂(D2-32a)
SO₂Me CH₂(D2-32a)
SO₂Et CH₂(D2-32a)
SO₂Ph CH₂(D2-32a)
SO₂NMe₂ CH₂(D2-32a)
NH₂ CH₂(D2-32a)
NHMe CH₂(D2-32a)
NHCHO CH₂(D2-32a)
NHC(O)CH₃ CH₂(D2-32a)
NHC(O)OCH₃ CH₂(D2-32a)
N=C(CH₃)₂ CH₂(D2-32a)
N=CHPh CH₂(D2-32a)
H CH₂(D2-33a)
H CH₂(D2-34a)
H CH₂(D2-35a)
H CH₂(D2-35b)
H CH₂(D2-36a)
H CH₂(D2-37a)
Me CH₂(D2-37a)
Et CH₂(D2-37a)
n-Pr CH₂(D2-37a)
i-Pr CH₂(D2-37a)
CH₂OCH₃ CH₂(D2-37a)
CH₂CH₂OEt CH₂(D2-37a)
CH₂SCH₃ CH₂(D2-37a)
CH₂CN CH₂(D2-37a)
CH₂CO₂Me CH₂(D2-37a)
CH₂CO₂Et CH₂(D2-37a)
CH₂CH=CH₂ CH₂(D2-37a)
CH₂CH≡CH CH₂(D2-37a)
C(O)CH₃ CH₂(D2-37a)
C(O)Et CH₂(D2-37a)
C(O)Pr-n CH₂(D2-37a)
C(O)Pr-c CH₂(D2-37a)
C(O)Bu-t CH₂(D2-37a)
C(O)CH₂OCH₃ CH₂(D2-37a)
C(O)CH₂SCH₃ CH₂(D2-37a)
C(O)OMe CH₂(D2-37a)
C(O)OEt CH₂(D2-37a)
C(O)CH₂CH₂ CH₂(D2-37a)
C(O)CH₂CH₂ CH₂(D2-37a)
C(O)OCH₂CH=CH₂ CH₂(D2-37a)
C(O)SCH₃ CH₂(D2-37a)
C(S)OCH₃ CH₂(D2-37a)
C(S)SCH₃ CH₂(D2-37a)
SMe CH₂(D2-37a)
SPh CH₂(D2-37a)
SNEt₂ CH₂(D2-37a)
SO₂Me CH₂(D2-37a)
SO₂Et CH₂(D2-37a)
SO₂Ph CH₂(D2-37a)
SO₂NMe₂ CH₂(D2-37a)
NH₂ CH₂(D2-37a)
NHMe CH₂(D2-37a)
NHCHO CH₂(D2-37a)
NHC(O)CH₃ CH₂(D2-37a)
NHC(O)OCH₃ CH₂(D2-37a)
N=C(CH₃)₂ CH₂(D2-37a)
N=CHPh CH₂(D2-37a)
H CH₂(D2-38a)
H CH₂(D2-39a)
H CH₂(D2-40a)
H CH₂(D2-41a)
H CH₂(D2-42a)
H CH₂(D2-43a)
H CH₂(D2-45a)
H CH₂(D2-46a)
H CH₂(D2-49a)
H CH₂(D2-51a)
H CH₂(D2-53a)
H CH₂(D2-59a)
H CH₂(D2-61a)
H CH₂(D2-63a)
H CH₂(D2-68a)
H CH₂(D2-75a)
H CH₂(D2-76a)
H CH₂(D2-76b)
H CH₂(D2-77a)
H CH₂(D2-77b)
H CH₂(D2-78a)
H CH₂(D2-78b)
H CH₂(D2-79a)
H CH₂(D2-81a)
H CH₂(D2-82a)
H CH₂(D2-84a)
H CH₂(D2-85a)
H CH₂(D2-87a)
H CH₂(D2-90a)
H CH₂(D2-100a)
H CH₂(D2-100b)
H CH₂(D2-100c)
H CH₂(D2-100d)
H CH₂(D2-100e)
H CH₂(D2-101a)
H CH₂(D2-101b)
H CH₂(D2-101c)
H CH₂(D2-101d)
H CH₂(D2-102a)
H CH₂(D2-102b)
H CH₂(D2-102c)
H CH₂(D2-102d)
H CH₂(D2-102e)
H CH₂(D2-102f)
H CH₂(D2-103a)
H CH₂(D2-108a)
H CH(Me)(D2-1a)
H CH(Me)(D2-2a)
H CH(Me)(D2-5a)
H CH(Me)(D2-5c)
H CH(Me)(D2-6c)
H CH(Me)(D2-8c)
H CH(Me)(D2-9b)
H CH(Me)(D2-9c)
H CH(Me)(D2-10b)
H CH(Me)(D2-10c)
H CH(Me)(D2-12b)
H CH(Me)(D2-12c)
H CH(Me)(D2-13b)
H CH(Me)(D2-14a)
H CH(Me)(D2-14b)
H CH(Me)(D2-15a)
H CH(Me)(D2-15b)
H CH(Me)(D2-16a)
H CH(Me)(D2-17a)
H CH(Me)(D2-18a)
H CH(Me)(D2-23b)
H CH(Me)(D2-27a)
H CH(Me)(D2-31a)
H CH(Me)(D2-32a)
H CH(Me)(D2-35a)
H CH(Me)(D2-36a)
H CH(Me)(D2-37a)
H CH(Me)(D2-39a)
H CH(Me)(D2-41a)
H CH₂C(O)NH(D2-1a)
H CH₂C(O)NH(D2-2a)
H CH₂C(O)NH(D2-5a)
H CH₂C(O)NH(D2-5c)
H CH₂C(O)NH(D2-6c)
H CH₂C(O)NH(D2-8c)
H CH₂C(O)NH(D2-9b)
H CH₂C(O)NH(D2-9c)
H CH₂C(O)NH(D2-10b)
H CH₂C(O)NH(D2-10c)
H CH₂C(O)NH(D2-12b)
H CH₂C(O)NH(D2-12c)
H CH₂C(O)NH(D2-13b)
H CH₂C(O)NH(D2-14a)
H CH₂C(O)NH(D2-14b)
H CH₂C(O)NH(D2-15a)
H CH₂C(O)NH(D2-15b)
H CH₂C(O)NH(D2-16a)
H CH₂C(O)NH(D2-17a)
H CH₂C(O)NH(D2-18a)
H CH₂C(O)NH(D2-23b)
H CH₂C(O)NH(D2-27a)
H CH₂C(O)NH(D2-31a)
H CH₂C(O)NH(D2-32a)
H CH₂C(O)NH(D2-35a)
H CH₂C(O)NH(D2-36a)
H CH₂C(O)NH(D2-37a)
H CH₂C(O)NH(D2-39a)
H CH₂C(O)NH(D2-41a)
H CH₂C(O)NH(D2-45a)
H CH₂C(O)NH(D2-46a)
H CH₂C(O)NH(D2-49a)
H CH₂C(O)NH(D2-51a)
H CH₂C(O)NH(D2-53a)
H CH₂C(O)NH(D2-59a)
H CH₂C(O)NH(D2-61a)
H CH₂C(O)NH(D2-63a)
H CH₂C(O)NH(D2-68a)
H CH₂C(O)NH(D2-75a)
H CH₂C(O)NH(D2-76a)
H CH₂C(O)NH(D2-76b)
H CH₂C(O)NH(D2-77a)
H CH₂C(O)NH(D2-77b)
H CH₂C(O)NH(D2-78a)
H CH₂C(O)NH(D2-78b)
H CH₂C(O)NH(D2-79a)
H CH₂C(O)NH(D2-82a)
H CH₂C(O)NH(D2-84a)
H CH₂C(O)NH(D2-85a)
H CH₂C(O)NH(D2-87a)
H CH₂C(O)NH(D2-90a)
H CH₂C(O)NH(D2-100a)
H CH₂C(O)NH(D2-100b)
H CH₂C(O)NH(D2-100c)
H CH₂C(O)NH(D2-100d)
H CH₂C(O)NH(D2-100e)
H CH₂C(O)NH(D2-101a)
H CH₂C(O)NH(D2-101b)
H CH₂C(O)NH(D2-101c)
H CH₂C(O)NH(D2-101d)
H CH₂C(O)NH(D2-108a)
H CH₂C(O)NHCH₂(D2-1a)
H CH₂C(O)NHCH₂(D2-2a)
H CH₂C(O)NHCH₂(D2-5a)
H CH₂C(O)NHCH₂(D2-5c)
H CH₂C(O)NHCH₂(D2-6c)
H CH₂C(O)NHCH₂(D2-8c)
H CH₂C(O)NHCH₂(D2-9b)
H CH₂C(O)NHCH₂(D2-9c)
H CH₂C(O)NHCH₂(D2-10b)
H CH₂C(O)NHCH₂(D2-10c)
H CH₂C(O)NHCH₂(D2-12b)
H CH₂C(O)NHCH₂(D2-12c)
H CH₂C(O)NHCH₂(D2-13b)
H CH₂C(O)NHCH₂(D2-14a)
H CH₂C(O)NHCH₂(D2-14b)
H CH₂C(O)NHCH₂(D2-15a)
H CH₂C(O)NHCH₂(D2-15b)
H CH₂C(O)NHCH₂(D2-16a)
H CH₂C(O)NHCH₂(D2-17a)
H CH₂C(O)NHCH₂(D2-18a)
H CH₂C(O)NHCH₂(D2-23b)
H CH₂C(O)NHCH₂(D2-27a)
H CH₂C(O)NHCH₂(D2-31a)
H CH₂C(O)NHCH₂(D2-32a)
H CH₂C(O)NHCH₂(D2-35a)
H CH₂C(O)NHCH₂(D2-36a)
H CH₂C(O)NHCH₂(D2-37a)
H CH₂C(O)NHCH₂(D2-39a)
H CH₂C(O)NHCH₂(D2-41a)
H CH₂C(O)NHCH₂(D2-45a)
H CH₂C(O)NHCH₂(D2-46a)
H CH₂C(O)NHCH₂(D2-49a)
H CH₂C(O)NHCH₂(D2-51a)
H CH₂C(O)NHCH₂(D2-53a)
H CH₂C(O)NHCH₂(D2-59a)
H CH₂C(O)NHCH₂(D2-61a)
H CH₂C(O)NHCH₂(D2-63a)
H CH₂C(O)NHCH₂(D2-68a)
H CH₂C(O)NHCH₂(D2-75a)
H CH₂C(O)NHCH₂(D2-76a)
H CH₂C(O)NHCH₂(D2-76b)
H CH₂C(O)NHCH₂(D2-77a)
H CH₂C(O)NHCH₂(D2-77b)
H CH₂C(O)NHCH₂(D2-78a)
H CH₂C(O)NHCH₂(D2-78b)
H CH₂C(O)NHCH₂(D2-79a)
H CH₂C(O)NHCH₂(D2-82a)
H CH₂C(O)NHCH₂(D2-84a)
H CH₂C(O)NHCH₂(D2-85a)
H CH₂C(O)NHCH₂(D2-87a)
H CH₂C(O)NHCH₂(D2-90a)
H CH₂C(O)NHCH₂(D2-102a)
H CH₂C(O)NHCH₂(D2-102b)
H CH₂C(O)NHCH₂(D2-102c)
H CH₂C(O)NHCH₂(D2-102d)
H CH₂C(O)NHCH₂(D2-102e)
H CH₂C(O)NHCH₂(D2-102f)
H CH₂C(O)NHCH₂(D2-103a)
H CH₂C(O)NHCH₂(D2-108a)
H NH(D2-7a)
H NH(D2-10c)
H NH(D2-22a)
H NH(D2-24a)
H NH(D2-32a)
H NC(O)Me(D2-32a)
H NC(O)OMe(D2-32a)
H NC(O)Et(D2-32a)
H NC(O)OEt(D2-32a)
H NC(O)CH₂CF₃(D2-32a)
H NSO₂Me(D2-32a)
H NSO₂CF₃(D2-32a)
H NSO₂Ph(D2-32a)
H NH(D2-35a)
H NH(D2-36a)
H NH(D2-37a)
H NH(D2-39a)
H NH(D2-43a)
H NH(D2-45a)
H NH(D2-49a)
H NH(D2-51a)
H NH(D2-53a)
H NH(D2-59a)
H NH(D2-61a)
H NH(D2-63a)
H NH(D2-108a)
H NH{D2-32b(3-Cl)}
H NH{D2-32b(4-Cl)}
H NH{D2-32b(5-Cl)}
H NH{D2-32b(6-Cl)}
H NH{D2-32b(4-CF₃)}
H NH{D2-108b(2-Cl)}
H NH{D2-108b(3-Cl)}
H NH{D2-108b(4-Cl)}
H NH{D2-108b(2-Me)}
H NH{D2-108b(3-Me)}
H NH{D2-108b(4-Me)}
H CH₂CH₂(D2-1a)
H CH₂CH₂(D2-1b)
H CH₂CH₂(D2-2a)
H CH₂CH₂(D2-2b)
H CH₂CH₂(D2-5c)
H CH₂CH₂(D2-6c)
H CH₂CH₂(D2-7a)
H CH₂CH₂(D2-8c)
H CH₂CH₂(D2-9b)
H CH₂CH₂(D2-10b)
H CH₂CH₂(D2-10c)
H CH₂CH₂(D2-11a)
H CH₂CH₂(D2-20a)
H CH₂CH₂(D2-22a)
H CH₂CH₂(D2-24a)
H CH₂CH₂(D2-26a)
H CH₂CH₂(D2-28a)
H CH₂CH₂(D2-29a)
H CH₂CH₂(D2-32a)
H CH₂CH₂(D2-36a)
H CH₂CH₂(D2-37a)
H CH₂CH₂OCH₂(D2-1a)
H CH₂CH₂OCH₂(D2-1b)
H CH₂CH₂OCH₂(D2-2a)
H CH₂CH₂OCH₂(D2-2b)
H CH₂CH₂OCH₂(D2-4a)
H CH₂CH₂OCH₂(D2-4b)
H CH₂CH₂OCH₂(D2-5a)
H CH₂CH₂OCH₂(D2-5b)
H CH₂CH₂OCH₂(D2-5c)
H CH₂CH₂OCH₂(D2-6a)
H CH₂CH₂OCH₂(D2-6b)
H CH₂CH₂OCH₂(D2-6c)
H CH₂CH₂OCH₂(D2-7a)
H CH₂CH₂OCH₂(D2-8a)
H CH₂CH₂OCH₂(D2-8b)
H CH₂CH₂OCH₂(D2-8c)
H CH₂CH₂OCH₂(D2-9a)
H CH₂CH₂OCH₂(D2-9b)
H CH₂CH₂OCH₂(D2-9c)
H CH₂CH₂OCH₂(D2-10a)
H CH₂CH₂OCH₂(D2-10b)
H CH₂CH₂OCH₂(D2-10c)
H CH₂CH₂OCH₂(D2-12a)
H CH₂CH₂OCH₂(D2-12b)
H CH₂CH₂OCH₂(D2-12c)
H CH₂CH₂OCH₂(D2-13a)
H CH₂CH₂OCH₂(D2-13b)
H CH₂CH₂OCH₂(D2-14a)
H CH₂CH₂OCH₂(D2-14b)
H CH₂CH₂OCH₂(D2-15a)
H CH₂CH₂OCH₂(D2-15b)
H CH₂CH₂OCH₂(D2-16a)
H CH₂CH₂OCH₂(D2-17a)
H CH₂CH₂OCH₂(D2-18a)
H CH₂CH₂OCH₂(D2-19a)
H CH₂CH₂OCH₂(D2-20a)
H CH₂CH₂OCH₂(D2-21a)
H CH₂CH₂OCH₂(D2-21b)
H CH₂CH₂OCH₂(D2-23a)
H CH₂CH₂OCH₂(D2-23b)
H CH₂CH₂OCH₂(D2-25a)
H CH₂CH₂OCH₂(D2-27a)
H CH₂CH₂OCH₂(D2-30a)
H CH₂CH₂OCH₂(D2-31a)
H CH₂CH₂OCH₂(D2-32a)
H CH₂CH₂OCH₂(D2-33a)
H CH₂CH₂OCH₂(D2-34a)
H CH₂CH₂OCH₂(D2-35a)
H CH₂CH₂OCH₂(D2-35b)
H CH₂CH₂OCH₂(D2-36a)
H CH₂CH₂OCH₂(D2-37a)
H CH₂CH₂OCH₂(D2-38a)
H CH₂CH₂OCH₂(D2-39a)
H CH₂CH₂OCH₂(D2-40a)
H CH₂CH₂OCH₂(D2-41a)
H CH₂CH₂OCH₂(D2-42a)
H CH₂CH₂OCH₂(D2-43a)
H CH₂CH₂OCH₂(D2-45a)
H CH₂CH₂OCH₂(D2-46a)
H CH₂CH₂OCH₂(D2-49a)
H CH₂CH₂OCH₂(D2-51a)
H CH₂CH₂OCH₂(D2-53a)
H CH₂CH₂OCH₂(D2-59a)
H CH₂CH₂OCH₂(D2-61a)
H CH₂CH₂OCH₂(D2-63a)
H CH₂CH₂OCH₂(D2-68a)
H CH₂CH₂OCH₂(D2-75a)
H CH₂CH₂OCH₂(D2-76a)
H CH₂CH₂OCH₂(D2-76b)
H CH₂CH₂OCH₂(D2-77a)
H CH₂CH₂OCH₂(D2-77b)
H CH₂CH₂OCH₂(D2-78a)
H CH₂CH₂OCH₂(D2-78b)
H CH₂CH₂OCH₂(D2-79a)
H CH₂CH₂OCH₂(D2-81a)
H CH₂CH₂OCH₂(D2-82a)
H CH₂CH₂OCH₂(D2-84a)
H CH₂CH₂OCH₂(D2-85a)
H CH₂CH₂OCH₂(D2-87a)
H CH₂CH₂OCH₂(D2-90a)
H CH₂CH₂OCH₂(D2-100a)
H CH₂CH₂OCH₂(D2-100b)
H CH₂CH₂OCH₂(D2-100c)
H CH₂CH₂OCH₂(D2-100d)
H CH₂CH₂OCH₂(D2-100e)
H CH₂CH₂OCH₂(D2-101a)
H CH₂CH₂OCH₂(D2-101b)
H CH₂CH₂OCH₂(D2-101c)
H CH₂CH₂OCH₂(D2-101d)
H CH₂CH₂OCH₂(D2-102a)
H CH₂CH₂OCH₂(D2-102b)
H CH₂CH₂OCH₂(D2-102c)
H CH₂CH₂OCH₂(D2-102d)
H CH₂CH₂OCH₂(D2-102e)
H CH₂CH₂OCH₂(D2-102f)
H CH₂CH₂OCH₂(D2-103a)
H CH₂CH₂OCH₂(D2-108a)
H CH₂CH₂SCH₂(D2-1a)
H CH₂CH₂SCH₂(D2-1b)
H CH₂CH₂SCH₂(D2-2a)
H CH₂CH₂SCH₂(D2-2b)
H CH₂CH₂SCH₂(D2-4a)
H CH₂CH₂SCH₂(D2-4b)
H CH₂CH₂SCH₂(D2-5a)
H CH₂CH₂SCH₂(D2-5b)
H CH₂CH₂SCH₂(D2-5c)
H CH₂CH₂SCH₂(D2-6a)
H CH₂CH₂SCH₂(D2-6b)
H CH₂CH₂SCH₂(D2-6c)
H CH₂CH₂SCH₂(D2-7a)
H CH₂CH₂SCH₂(D2-8a)
H CH₂CH₂SCH₂(D2-8b)
H CH₂CH₂SCH₂(D2-8c)
H CH₂CH₂SCH₂(D2-9a)
H CH₂CH₂SCH₂(D2-9b)
H CH₂CH₂SCH₂(D2-9c)
H CH₂CH₂SCH₂(D2-10a)
H CH₂CH₂SCH₂(D2-10b)
H CH₂CH₂SCH₂(D2-10c)
H CH₂CH₂SCH₂(D2-12a)
H CH₂CH₂SCH₂(D2-12b)
H CH₂CH₂SCH₂(D2-12c)
H CH₂CH₂SCH₂(D2-13a)
H CH₂CH₂SCH₂(D2-13b)
H CH₂CH₂OCH₂(D2-14a)
H CH₂CH₂SCH₂(D2-14b)
H CH₂CH₂SCH₂(D2-15a)
H CH₂CH₂SCH₂(D2-15b)
H CH₂CH₂SCH₂(D2-16a)
H CH₂CH₂SCH₂(D2-17a)
H CH₂CH₂SCH₂(D2-18a)
H CH₂CH₂SCH₂(D2-19a)
H CH₂CH₂SCH₂(D2-20a)
H CH₂CH₂SCH₂(D2-21a)
H CH₂CH₂SCH₂(D2-21b)
H CH₂CH₂SCH₂(D2-23a)
H CH₂CH₂SCH₂(D2-23b)
H CH₂CH₂SCH₂(D2-25a)
H CH₂CH₂SCH₂(D2-27a)
H CH₂CH₂SCH₂(D2-30a)
H CH₂CH₂SCH₂(D2-31a)
H CH₂CH₂SCH₂(D2-32a)
H CH₂CH₂SCH₂(D2-33a)
H CH₂CH₂SCH₂(D2-34a)
H CH₂CH₂SCH₂(D2-35a)
H CH₂CH₂SCH₂(D2-35b)
H CH₂CH₂SCH₂(D2-36a)
H CH₂CH₂SCH₂(D2-37a)
H CH₂CH₂SCH₂(D2-38a)
H CH₂CH₂SCH₂(D2-39a)
H CH₂CH₂SCH₂(D2-40a)
H CH₂CH₂SCH₂(D2-41a)
H CH₂CH₂SCH₂(D2-42a)
H CH₂CH₂SCH₂(D2-43a)
H CH₂CH₂SCH₂(D2-45a)
H CH₂CH₂SCH₂(D2-46a)
H CH₂CH₂SCH₂(D2-49a)
H CH₂CH₂SCH₂(D2-51a)
H CH₂CH₂SCH₂(D2-53a)
H CH₂CH₂SCH₂(D2-59a)
H CH₂CH₂SCH₂(D2-61a)
H CH₂CH₂SCH₂(D2-63a)
H CH₂CH₂SCH₂(D2-68a)
H CH₂CH₂SCH₂(D2-75a)
H CH₂CH₂SCH₂(D2-76a)
H CH₂CH₂SCH₂(D2-76b)
H CH₂CH₂SCH₂(D2-77a)
H CH₂CH₂SCH₂(D2-77b)
H CH₂CH₂SCH₂(D2-78a)
H CH₂CH₂SCH₂(D2-78b)
H CH₂CH₂SCH₂(D2-79a)
H CH₂CH₂SCH₂(D2-81a)
H CH₂CH₂SCH₂(D2-82a)
H CH₂CH₂SCH₂(D2-84a)
H CH₂CH₂SCH₂(D2-85a)
H CH₂CH₂SCH₂(D2-87a)
H CH₂CH₂SCH₂(D2-90a)
H CH₂CH₂SCH₂(D2-100a)
H CH₂CH₂SCH₂(D2-100b)
H CH₂CH₂SCH₂(D2-100c)
H CH₂CH₂SCH₂(D2-100d)
H CH₂CH₂SCH₂(D2-100e)
H CH₂CH₂SCH₂(D2-101a)
H CH₂CH₂SCH₂(D2-101b)
H CH₂CH₂SCH₂(D2-101c)
H CH₂CH₂SCH₂(D2-101d)
H CH₂CH₂SCH₂(D2-102a)
H CH₂CH₂SCH₂(D2-102b)
H CH₂CH₂SCH₂(D2-102c)
H CH₂CH₂SCH₂(D2-102d)
H CH₂CH₂SCH₂(D2-102e)
H CH₂CH₂SCH₂(D2-102f)
H CH₂CH₂SCH₂(D2-103a)
H CH₂CH₂SCH₂(D2-108a)
H CH₂{D2-1c(3-Me)}
H CH₂{D2-1d(5-Cl)}
H CH₂{D2-2c(5-Br)}
H CH₂{D2-2d(5-Cl)}
H CH₂{D2-4c(5-Cl)}
H CH₂{D2-4d(5-Cl)}
H CH₂{D2-5d(3-Me)}
H CH₂{D2-5e(3-Me)}
H CH₂{D2-5f(5-Me)}
H CH₂{D2-6d(3-Cl)}
H CH₂{D2-6e(3-Me)}
H CH₂{D2-6f(5-Me)}
H CH₂{D2-7a(3-Me)}
H CH₂{D2-8d(3-Cl)}
H CH₂{D2-8e(3-CF₃)}
H CH₂{D2-8f(5-Me)}
H CH₂{D2-9d(2-Me)}
H CH₂{D2-9e(2-Me)}
H CH₂{D2-9f(4-Me)}
H CH₂{D2-10e(2-Me)}
H CH₂{D2-10f(2-Cl)}
H CH₂{D2-10e(2-Br)}
H CH₂{D2-12d(4-Me)}
H CH₂{D2-12e(5-Me)}
H CH₂{D2-12f(5-Cl)}
H CH₂{D2-13c(Me)}
H CH₂{D2-13d(Cl)}
H CH₂{D2-14c(Me)}
H CH₂{D2-14d(Me)}
H CH₂{D2-15c(Cl)}
H CH₂{D2-15d(Me)}
H CH₂{D2-16b(Ph)}
H CH₂{D2-17b(Ph)}
H CH₂{D2-18b(Me)}
H CH₂{D2-19b(Cl)}
H CH₂{D2-20b(Me)}
H CH₂{D2-21c(Me)}
H CH₂{D2-21d(Me)}
H CH₂{D2-23c(t-Bu)}
H CH₂{D2-23d(Ph)}
H CH₂{D2-25b(Me)}
H CH₂{D2-27a(Me)}
H CH₂{D2-32b(3-Cl)}
H CH₂{D2-32b(4-Cl)}
H CH₂{D2-32b(5-Cl)}
H CH₂{D2-32b(6-Cl)}
H CH₂{D2-32b(3-Me)}
H CH₂{D2-32b(4-Me)}
H CH₂{D2-32b(5-Me)}
H CH₂{D2-32b(6-Me)}
H CH₂{D2-32b(5-CF₃)}
H CH₂{D2-33b(4-CF₃)}
H CH₂{D2-34b(3-Cl)}
H CH₂{D2-35c(3-Cl)}
H CH₂{D2-35d(3-Cl)}
H CH₂{D2-36b(2-Me)}
H CH₂{D2-37b(4-Me)}
H CH₂{D2-38b(2-Me)}
H CH₂{D2-39b(5-Me)}
H CH₂{D2-108b(2-Cl)}
H CH₂{D2-108b(3-Cl)}
H CH₂{D2-108b(4-Cl)}
H CH₂{D2-108b(2-Me)}
H CH₂{D2-108b(3-Me)}
H CH₂{D2-108b(4-Me)}
H CH₂{D2-108b(2-CF₃)}
H CH₂{D2-108b(3-CF₃)}
H CH₂{D2-108b(4-CF₃)}
H CH₂{D2-108b(2-OMe)}
H CH₂{D2-108b(3-OMe)}
H CH₂{D2-108b(4-OMe)}
H CH₂CH₂{D2-7b(4-Cl)}
H CH₂CH₂{D2-10e(2-Cl)}
H CH₂CH₂{D2-11b(2-Me)}
H CH₂CH₂{D2-20b(4-Me)}
H CH₂CH₂{D2-22b(3-SMe)}
H CH₂CH₂{D2-24b(3-Me)}
H CH₂CH₂{D2-26b(4-CO₂Me)}
H CH₂CH₂{D2-28b(Me)}
H CH₂CH₂{D2-29a(Ph)}
H CH₂CH₂{D2-32b(3-Cl)}
H CH₂CH₂{D2-36b(2-Me)}
H CH₂CH₂{D2-37b(4-Me)
―――――――――――――――――――
本発明化合物は、農園芸作物及び樹木などを加害する所謂農業害虫、家畜・家禽類に寄生する所謂家畜害虫、家屋等の人間の生活環境で様々な悪影響を与える所謂衛生害虫、倉庫に貯蔵された穀物等を加害する所謂貯穀害虫等としての昆虫類、及び同様の場面で発生、加害するダニ類、甲殻類、軟体動物、線虫類の何れの有害生物も低濃度で有効に防除できる。 Table 6 ――――――――――――――――――――
R ^f2 R ^f3
―――――――――――――――――――
H CH ₂ CF ₃
H CH ₂ CN
H CH ₂ SMe
H CH ₂ S (O) Me
H CH ₂ S (O) ₂ Me
H CH ₂ CH ₂ SMe
H CH ₂ CH ₂ S (O) Me
H CH ₂ CH ₂ S (O) ₂ Me
H CH (Me) CH ₂ SMe
H CH (Me) CH ₂ S (O) Me
H CH (Me) CH ₂ S (O) ₂ Me
H CH ₂ CH (OMe) ₂
H CH ₂ CH (OEt) ₂
H NHC (O) OMe
H NHC (O) OEt
H NHC (O) OPr-n
H NHC (O) OPr-i
H NHC (O) OBu-n
H NHC (O) OBu-i
H NHC (O) OBu-s
H NHC (O) OBu-t
H D2-32a
H D2-33a
H D2-34a
H D2-37a
H CH ₂ (D2-32a)
H CH ₂ (D2-33a)
H CH ₂ (D2-34a)
H CH ₂ (D2-37a)
Me CH ₂ CF ₃
Me CH ₂ CH ₂ SMe
Me CH ₂ CH ₂ S (O) Me
Me CH ₂ CH ₂ S (O) ₂ Me
Me CH (Me) CH ₂ SMe
Me CH (Me) CH ₂ S (O) Me
Me CH (Me) CH ₂ S (O) ₂ Me
Me CH ₂ CH (OMe) ₂
Me CH ₂ CH (OEt) ₂
Me NHC (O) OMe
Me NHC (O) OEt
Me NHC (O) OPr-n
Me NHC (O) OPr-i
Me NHC (O) OBu-n
Me NHC (O) OBu-i
Me NHC (O) OBu-s
Me NHC (O) OBu-t
Me D2-32a
Me D2-33a
Me D2-34a
Me D2-37a
Me CH ₂ (D2-32a)
Me CH ₂ (D2-33a)
Me CH ₂ (D2-34a)
Me CH ₂ (D2-37a)
HH
H Me
H Et
H n-Pr
H i-Pr
H c-Pr
H n-Bu
H i-Bu
H s-Bu
H t-Bu
H c-Bu
H n-Pen
H c-Pen
H n-Hex
H c-Hex
H Hep
H Oct
H CH ₂ Pr-c
H CH ₂ Bu-i
H CH ₂ Bu-s
H CH ₂ Bu-t
H CH ₂ Bu-c
H CH ₂ Pen-c
H CH ₂ Hex-c
H CH (CH ₃ ) Pr-n
H CH (CH ₃ ) Pr-i
H CH (CH ₃ ) Pr-n
H CH (CH ₃ ) Bu-i
H CH (Et) ₂
HC (CH ₃ ) ₂ Et
HC (CH ₃ ) ₂ Pr-n
H CH ₂ CH ₂ F
H CH ₂ CH ₂ Cl
H CH ₂ CH ₂ Br
H CH ₂ CHF ₂
H CH ₂ CHFCl
H CH ₂ CHCl ₂
H CH ₂ CHFBr
H CH ₂ CF ₂ Cl
H CH ₂ CFCl ₂
H CH ₂ CCl ₃
H CH ₂ CF ₂ Br
H CH ₂ CFClBr
H CH ₂ CCl ₂ Br
H CH (CH ₃ ) CH ₂ F
H CH (CH ₃ ) CH ₂ Cl
H CH (CH ₃ ) CH ₂ Br
H CH ₂ CHFCH ₃
H CH ₂ CHClCH ₃
H CH ₂ CHBrCH ₃
H CH ₂ CFClCH ₃
H CH ₂ CHClCH ₂ Cl
H CH ₂ CHBrCH ₂ F
H CH ₂ CHClCH ₂ Br
H CH ₂ CHBrCH ₂ Cl
H CH ₂ CHBrCHCl ₂
H CH ₂ CClBrCH ₃
H CH ₂ CHBrCH ₂ Br
H CH ₂ CH ₂ CF ₃
H CH ₂ CH ₂ CF ₂ Br
H CH ₂ CClBrCH ₂ Cl
H CH ₂ CF ₂ CF ₂ H
H CH ₂ CHClCF ₃
H CH ₂ CF ₂ CF ₃
H CH ₂ CF (CH ₃ ) ₂
H CH ₂ CHFCH ₂ CH ₃
H CH ₂ CHClCH ₂ CH ₃
H CH ₂ CF ₂ CHFCF ₃
H CH ₂ CF ₂ CF ₂ CHF ₂
H CH ₂ CF ₂ CF ₂ CF ₃
HC (CH ₃ ) ₂ CH ₂ Cl
HC (CH ₃ ) ₂ CH ₂ Br
HC (CH ₃ ) ₂ CHBrCH ₂ Br
H CH ₂ CF ₃
Me CH ₂ CF ₃
Et CH ₂ CF ₃
n-Pr CH ₂ CF ₃
i-Pr CH ₂ CF ₃
CH ₂ OCH ₃ CH ₂ CF ₃
CH ₂ CH ₂ OEt CH ₂ CF ₃
CH ₂ SCH ₃ CH ₂ CF ₃
CH ₂ CN CH ₂ CF ₃
CH ₂ CO ₂ Me CH ₂ CF ₃
CH ₂ CO ₂ Et CH ₂ CF ₃
CH ₂ CH = CH ₂ CH ₂ CF ₃
CH ₂ CH≡CH CH ₂ CF ₃
C (O) CH ₃ CH ₂ CF ₃
C (O) Et CH ₂ CF ₃
C (O) Pr-n CH ₂ CF ₃
C (O) Pr-c CH ₂ CF ₃
C (O) Bu-t CH ₂ CF ₃
C (O) CH ₂ OCH ₃ CH ₂ CF ₃
C (O) CH ₂ SCH ₃ CH ₂ CF ₃
C (O) OMe CH ₂ CF ₃
C (O) OEt CH ₂ CF ₃
C (O) CH ₂ CH ₂ Cl CH ₂ CF ₃
C (O) CH ₂ CH ₂ OMe CH ₂ CF ₃
C (O) OCH ₂ CH = CH ₂ CH ₂ CF ₃
C (O) SCH ₃ CH ₂ CF ₃
C (S) OCH ₃ CH ₂ CF ₃
C (S) SCH ₃ CH ₂ CF ₃
SMe CH ₂ CF ₃
SPh CH ₂ CF ₃
SNEt ₂ CH ₂ CF ₃
SO ₂ Me CH ₂ CF ₃
SO ₂ Et CH ₂ CF ₃
SO ₂ Ph CH ₂ CF ₃
SO ₂ NMe ₂ CH ₂ CF ₃
NH ₂ CH ₂ CF ₃
NHMe CH ₂ CF ₃
NHCHO CH ₂ CF ₃
NHC (O) CH ₃ CH ₂ CF ₃
NHC (O) OCH ₃ CH ₂ CF ₃
N = C (CH ₃ ) ₂ CH ₂ CF ₃
N = CHPh CH ₂ CF ₃
H CH (CF ₃ ) Me
H CH (CF ₃ ) Et
H CH (CF ₃ ) OH
H CH (CF ₃ ) OMe
H CH ₂ CH (OMe) ₂
H CH ₂ CH (OEt) ₂
H CH ₂ CN
H CH (Me) CN
HC (Me) ₂ CN
H CH (OMe) CN
H CH ₂ CH ₂ CN
H CH ₂ C (O) Me
H CH ₂ C (O) OMe
H CH ₂ C (O) OEt
H CH ₂ C (O) OCH ₂ CF ₃
H CH (Me) C (O) OMe
H CH (Me) C (O) OEt
H CH (Me) C (O) OCH ₂ CF ₃
H CH (OMe) C (O) OMe
H CH (OMe) C (O) OEt
H CH (OMe) C (O) OCH ₂ CF ₃
H CH (Ph) C (O) OMe
H CH (Ph) C (O) OEt
H CH (Ph) C (O) OCH ₂ CF ₃
H CH (CF ₃ ) C (O) OMe
H CH (CF ₃ ) C (O) OEt
H CH (CF ₃ ) C (O) OCH ₂ CF ₃
H CH ₂ CH ₂ C (O) OMe
H CH ₂ CH ₂ C (O) OEt
H CH ₂ CH ₂ C (O) OCH ₂ CF ₃
H CH ₂ CH (Me) C (O) OMe
H CH ₂ CH (Me) C (O) OEt
H CH (Me) CH ₂ C (O) OMe
H CH (Me) CH ₂ C (O) OEt
H CH ₂ C (O) NH ₂
H CH ₂ C (O) NHMe
H CH ₂ C (O) NHEt
H CH ₂ C (O) NHPr-n
H CH ₂ C (O) NHPr-i
H CH ₂ C (O) NHPr-c
H CH ₂ C (O) NHBu-n
H CH ₂ C (O) NHBu-i
H CH ₂ C (O) NHBu-s
H CH ₂ C (O) NHBu-t
H CH ₂ C (O) NHBu-c
H CH ₂ C (O) NHHex-n
H CH ₂ C (O) NHHex-c
H CH ₂ C (O) N (Me) ₂
H CH ₂ C (O) N (Et) ₂
H CH ₂ C (O) N (n-Pr) ₂
H CH ₂ C (O) N (Me) Et
H CH ₂ C (O) N (Me) Pr-n
H CH ₂ C (O) N (Me) Pr-i
H CH ₂ C (O) NHCH ₂ CH ₂ F
H CH ₂ C (O) NHCH ₂ CH ₂ Cl
H CH ₂ C (O) NHCH ₂ CH ₂ Br
H CH ₂ C (O) N (Me) CH ₂ CH ₂ F
H CH ₂ C (O) N (Me) CH ₂ CH ₂ Cl
H CH ₂ C (O) N (Me) CH ₂ CH ₂ Br
H CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ OCH ₃ CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ CN CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ CO ₂ Me CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ CO ₂ Et CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ CH = CH ₂ CH ₂ C (O) NHCH ₂ CF ₃
CH ₂ CH≡CH CH ₂ C (O) NHCH ₂ CF ₃
C (O) Me CH ₂ C (O) NHCH ₂ CF ₃
C (O) OMe CH ₂ C (O) NHCH ₂ CF ₃
H CH ₂ C (O) N (Me) CH ₂ CF ₃
H CH ₂ C (O) NHCH ₂ CF ₂ Cl
H CH ₂ C (O) NHCH ₂ CN
H CH ₂ C (O) NHCH ₂ CH = CH ₂
H CH ₂ C (O) NHCH ₂ CH≡CH
H CH ₂ C (O) NHCH ₂ CH ₂ CH ₂ Cl
H CH ₂ C (O) NHCH ₂ CH ₂ OCH ₃
H CH ₂ C (O) NHCH ₂ CH ₂ SCH ₃
H CH ₂ C (O) NHCH ₂ CH ₂ SO ₂ CH ₃
H CH (Me) C (O) NH ₂
H CH (Me) C (O) NHMe
H CH (Me) C (O) NHEt
H CH (Me) C (O) NHPr-n
H CH (Me) C (O) NHPr-i
H CH (Me) C (O) NHPr-c
H CH (Me) C (O) NHBu-n
H CH (Me) C (O) NHBu-i
H CH (Me) C (O) NHBu-s
H CH (Me) C (O) NHBu-t
H CH (Me) C (O) NHBu-c
H CH (Me) C (O) NHHex-n
H CH (Me) C (O) NHHex-c
H CH (Me) C (O) N (Me) ₂
H CH (Me) C (O) N (Et) ₂
H CH (Me) C (O) N (n-Pr) ₂
H CH (Me) C (O) N (Me) Et
H CH (Me) C (O) N (Me) Pr-n
H CH (Me) C (O) N (Me) Pr-i
H CH (Me) C (O) NHCH ₂ CH ₂ F
H CH (Me) C (O) NHCH ₂ CH ₂ Cl
H CH (Me) C (O) NHCH ₂ CH ₂ Br
H CH (Me) C (O) NHCH ₂ CF ₃
H CH (Et) C (O) NHCH ₂ CF ₃
H CH (i-Pr) C (O) NHCH ₂ CF ₃
H CH (CH ₂ OCH ₃ ) C (O) NHCH ₂ CF ₃
H CH (CH ₂ SCH ₃ ) C (O) NHCH ₂ CF ₃
H CH (Ph) C (O) NHCH ₂ CF ₃
H CH (CH ₂ Ph) C (O) NHCH ₂ CF ₃
H CH (CF ₃ ) C (O) NHMe
H CH (CF ₃ ) C (O) NHEt
H CH (CF ₃ ) C (O) NHPr-n
H CH (CF ₃ ) C (O) NHPr-i
H CH (CF ₃ ) C (O) NHPr-c
H CH (CF ₃ ) C (O) NHBu-n
H CH (CF ₃ ) C (O) NHBu-i
H CH (CF ₃ ) C (O) NHBu-s
H CH (CF ₃ ) C (O) NHBu-t
H CH (CF ₃ ) C (O) NHBu-c
H CH (CF ₃ ) C (O) NHHex-n
H CH (CF ₃ ) C (O) NHHex-c
H CH (CF ₃ ) C (O) N (Me) ₂
H CH (CF ₃ ) C (O) N (Et) ₂
H CH (CF ₃ ) C (O) N (n-Pr) ₂
H CH (CF ₃ ) C (O) N (Me) Et
H CH (CF ₃ ) C (O) N (Me) Pr-n
H CH (CF ₃ ) C (O) N (Me) Pr-i
H CH (CF ₃ ) C (O) NHCH ₂ CH ₂ F
H CH (CF ₃ ) C (O) NHCH ₂ CH ₂ Cl
H CH (CF ₃ ) C (O) NHCH ₂ CH ₂ Br
H CH (CF ₃ ) C (O) NHCH ₂ CF ₃
H CH ₂ CH ₂ C (O) NHCH ₂ CF ₃
H CH ₂ C (O) N (Me) ₂
H CH ₂ C (O) N (Et) ₂
H CH ₂ C (O) N (n-Pr) ₂
H CH ₂ CH = CH ₂
H CH ₂ C (Me) = CH ₂
H CH ₂ C (Et) = CH ₂
H CH (Me) CH = CH ₂
H CH ₂ CH = C (Me) ₂
H CH ₂ C (Me) = CHCH ₃
H CH (Me) CH = CHCH ₃
H CH ₂ C (F) = CH ₂
H CH ₂ CH = CHCl
H CH ₂ C (Cl) = CH ₂
H CH ₂ CH = CCl ₂
H CH ₂ CH = CHBr
H CH ₂ C (Br) = CH ₂
H CH ₂ C (Br) = CHBr
H CH ₂ C (Me) = CHBr
H CH ₂ CH = C (Cl) CH ₃
H CH ₂ CH = C (Br) CH ₃
H CH ₂ C (OMe) = CH ₂
H CH ₂ C (Br) = CHOMe
H CH ₂ C (Br) = CHOEt
H CH ₂ C (Br) = CHPh
H CH ₂ C≡CH
H CH ₂ C≡CCl
H CH ₂ C≡CBr
H CH ₂ C≡CI
H CH ₂ C≡CPh
H CH ₂ OMe
H CH ₂ CH ₂ OH
H CH ₂ CH ₂ OMe
H CH ₂ CH ₂ OEt
H CH ₂ CH ₂ OPr-n
H CH ₂ CH ₂ OPr-i
H CH ₂ CH ₂ OBu-i
H CH ₂ CH ₂ OCH ₂ CH ₂ Cl
H CH ₂ CH ₂ OCH ₂ CF3
H CH ₂ CH ₂ OCH ₂ CH ₂ OCH ₃
H CH ₂ CH ₂ OCH ₂ CH ₂ SCH ₃
H CH ₂ CH ₂ OC (O) CH ₃
H CH ₂ CH (Me) OH
H CH ₂ CH (Me) OMe
H CH ₂ CH (Me) OCH ₂ CF ₃
H CH (Me) CH ₂ OH
H CH (Me) CH ₂ OMe
H CH (Me) CH ₂ OCH ₂ CF ₃
H CH (Ph) CH ₂ OH
H CH (Ph) CH ₂ OMe
H CH (Ph) CH ₂ OCH ₂ CF ₃
HC (Me) ₂ CH ₂ OH
HC (Me) ₂ CH ₂ OMe
HC (Me) ₂ CH ₂ OCH ₂ CF ₃
H CH ₂ CH ₂ CH ₂ OH
H CH ₂ CH ₂ CH ₂ OMe
H CH ₂ CH ₂ CH ₂ OCH ₂ CF ₃
H CH ₂ CH ₂ CH ₂ CH ₂ OH
H CH ₂ CH ₂ CH ₂ CH ₂ OMe
H CH ₂ CH ₂ CH ₂ CH ₂ OCH ₂ CF ₃
H CH ₂ SMe
H CH (CF ₃ ) SMe
H CH (CF ₃ ) SEt
H CH ₂ CH ₂ SMe
H CH ₂ CH ₂ S (O) Me
H CH ₂ CH ₂ S (O) ₂ Me
H CH ₂ CH ₂ SEt
H CH ₂ CH ₂ S (O) Et
H CH ₂ CH ₂ S (O) ₂ Et
H CH ₂ CH ₂ SPr-n
H CH ₂ CH ₂ S (O) Pr-n
H CH ₂ CH ₂ S (O) ₂ Pr-n
H CH ₂ CH ₂ SPr-i
H CH ₂ CH ₂ S (O) Pr-i
H CH ₂ CH ₂ S (O) ₂ Pr-i
H CH ₂ CH ₂ SCH ₂ CF ₃
H CH ₂ CH ₂ S (O) CH ₂ CF ₃
H CH ₂ CH ₂ S (O) ₂ CH ₂ CF ₃
H CH ₂ CH ₂ SCH ₂ CH ₂ OH
H CH ₂ CH ₂ S (O) CH ₂ CH ₂ OH
H CH ₂ CH ₂ S (O) ₂ CH ₂ CH ₂ OH
H CH ₂ CH ₂ SCH ₂ CH ₂ OMe
H CH ₂ CH ₂ S (O) CH ₂ CH ₂ OMe
H CH ₂ CH ₂ S (O) ₂ CH ₂ CH ₂ OMe
H CH ₂ CH ₂ SCH ₂ C (O) OMe
H CH ₂ CH ₂ S (O) CH ₂ C (O) OMe
H CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) OMe
H CH ₂ CH ₂ SCH ₂ C (O) NHMe
H CH ₂ CH ₂ S (O) CH ₂ C (O) NHMe
H CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) NHMe
H CH ₂ CH ₂ SCH ₂ C (O) NMe
H CH ₂ CH ₂ S (O) CH ₂ C (O) NMe
H CH ₂ CH ₂ S (O) ₂ CH ₂ C (O) N (Me) ₂
H CH ₂ CH ₂ SCH ₂ CH = CH ₂
H CH ₂ CH ₂ SCH ₂ CH≡CH
H CH ₂ CH ₂ S (O) ₂ NHMe
H CH ₂ CH ₂ S (O) ₂ N (Me) ₂
H CH ₂ CH ₂ S (O) ₂ NHEt
H CH ₂ CH ₂ S (O) ₂ N (Et) ₂
H CH ₂ CH ₂ S (O) ₂ NHPr-n
H CH ₂ CH ₂ S (O) ₂ N (Pr-n) ₂
H CH ₂ CH ₂ S (O) ₂ NHPr-i
H CH ₂ CH ₂ S (O) ₂ N (Pr-i) ₂
H CH ₂ CH ₂ S (O) ₂ NHPr-c
H CH ₂ CH ₂ S (O) ₂ NHBu-t
H CH ₂ CH ₂ S (O) ₂ NHCH ₂ CF ₃
H CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH ₂ OMe
H CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH ₂ SMe
H CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH = CH ₂
H CH ₂ CH ₂ S (O) ₂ NHCH ₂ CH≡CH
H CH ₂ CH ₂ S (O) (= NCN) Me
H CH ₂ CH (Me) SMe
H CH ₂ CH (Me) S (O) Me
H CH ₂ CH (Me) S (O) ₂ Me
H CH ₂ CH (Me) SEt
H CH ₂ CH (Me) S (O) Et
H CH ₂ CH (Me) S (O) ₂ Et
H CH ₂ CH (Et) SMe
H CH ₂ CH (Et) S (O) Me
H CH ₂ CH (Et) S (O) ₂ Me
H CH ₂ CH (n-Pr) SMe
H CH ₂ CH (n-Pr) S (O) Me
H CH ₂ CH (n-Pr) S (O) ₂ Me
H CH ₂ CH (i-Pr) SMe
H CH ₂ CH (i-Pr) S (O) Me
H CH ₂ CH (i-Pr) S (O) ₂ Me
H CH ₂ CH (Ph) SMe
H CH ₂ CH (Ph) S (O) Me
H CH ₂ CH (Ph) S (O) ₂ Me
H CH (Me) CH ₂ SMe
H CH (Me) CH ₂ S (O) Me
H CH (Me) CH ₂ S (O) ₂ Me
H CH (Me) CH ₂ SEt
H CH (Me) CH ₂ S (O) Et
H CH (Me) CH ₂ S (O) ₂ Et
H CH (Me) CH ₂ SPr-n
H CH (Me) CH ₂ S (O) Pr-n
H CH (Me) CH ₂ S (O) ₂ Pr-n
H CH (Me) CH ₂ SPr-i
H CH (Me) CH ₂ S (O) Pr-i
H CH (Me) CH ₂ S (O) ₂ Pr-i
H CH (Me) CH ₂ SPh
H CH (Me) CH ₂ S (O) Ph
H CH (Me) CH ₂ S (O) ₂ Ph
H CH (Ph) CH ₂ SMe
H CH (Ph) CH ₂ S (O) Me
H CH (Ph) CH ₂ S (O) ₂ Me
H CH (Me) CH (Me) SMe
H CH (Me) CH (Me) S (O) Me
H CH (Me) CH (Me) S (O) ₂ Me
HC (Me) ₂ CH ₂ SMe
HC (Me) ₂ CH ₂ S (O) Me
HC (Me) ₂ CH ₂ S (O) ₂ Me
H CH ₂ CH ₂ CH ₂ SMe
H CH ₂ CH ₂ CH ₂ S (O) Me
H CH ₂ CH ₂ CH ₂ S (O) ₂ Me
H CH ₂ CH ₂ CH (Me) SMe
H CH ₂ CH ₂ CH (Me) S (O) Me
H CH ₂ CH ₂ CH (Me) S (O) ₂ Me
H CH ₂ CH (Me) CH ₂ SMe
H CH ₂ CH (Me) CH ₂ S (O) Me
H CH ₂ CH (Me) CH ₂ S (O) ₂ Me
H CH (Me) CH ₂ CH ₂ SMe
H CH (Me) CH ₂ CH ₂ S (O) Me
H CH (Me) CH ₂ CH ₂ S (O) ₂ Me
HC (Me) ₂ CH ₂ CH ₂ SMe
HC (Me) ₂ CH ₂ CH ₂ S (O) Me
HC (Me) ₂ CH ₂ CH ₂ S (O) ₂ Me
H CH (Me) (CH ₂ ) ₃ SMe
H CH (Me) (CH ₂ ) ₃ S (O) Me
H CH (Me) (CH ₂ ) ₃ S (O) ₂ Me
H CH (Me) (CH ₂ ) ₄ SMe
H CH (Me) (CH ₂ ) ₄ S (O) Me
H CH (Me) (CH ₂ ) ₄ S (O) ₂ Me
H CH ₂ NHC (O) Me
H CH ₂ NHC (O) Et
H CH ₂ NHC (O) Pr-n
H CH ₂ CH ₂ NHC (O) Me
H CH ₂ CH ₂ NHC (O) Et
H CH ₂ CH ₂ NHC (O) Pr-n
H CH ₂ CH ₂ NHC (O) Pr-i
H CH ₂ CH ₂ NHC (O) Pr-c
H CH ₂ CH ₂ NHC (O) Bu-n
H CH ₂ CH ₂ NHC (O) Bu-i
H CH ₂ CH ₂ NHC (O) Bu-s
H CH ₂ CH ₂ NHC (O) Bu-t
H CH ₂ CH ₂ NHC (O) CF ₃
H CH ₂ CH ₂ NHC (O) CF ₂ Cl
H CH ₂ CH ₂ NHC (O) Ph
H CH ₂ CH ₂ NHC (O) CH ₂ CF ₃
H CH ₂ CH ₂ NHC (O) CH ₂ SMe
H CH ₂ CH ₂ NHC (O) CH ₂ S (O) Me
H CH ₂ CH ₂ NHC (O) CH ₂ S (O) ₂ Me
H CH ₂ CH ₂ N (Me) C (O) Me
H CH ₂ CH ₂ N (Me) C (O) Et
H CH ₂ CH ₂ N (Me) C (O) CF ₃
H CH ₂ CH ₂ N (Me) C (O) CH ₂ CF ₃
H CH ₂ CH ₂ N (Me) C (O) CH ₂ SMe
H CH ₂ CH ₂ N (Me) C (O) CH ₂ S (O) Me
H CH ₂ CH ₂ N (Me) C (O) CH ₂ S (O) ₂ Me
H CH ₂ CH ₂ NHC (O) OMe
H CH ₂ CH ₂ NHC (O) OEt
H CH ₂ CH ₂ NHC (O) OPr-n
H CH ₂ CH ₂ NHC (O) OBu-t
H CH ₂ CH ₂ NHC (O) NHEt
H CH ₂ CH ₂ NHC (O) NHPr-n
H CH ₂ CH ₂ NHC (O) NHPr-i
H CH ₂ CH ₂ NHC (O) NHBu-t
H CH ₂ CH ₂ NHC (O) N (Me) ₂
H CH ₂ CH ₂ NHSO ₂ Me
H CH ₂ CH ₂ NHSO ₂ Et
H CH ₂ CH ₂ NHSO ₂ CF ₃
H CH ₂ CH ₂ NHSO ₂ Ph
H CH ₂ CH ₂ NHSO ₂ N (Me) ₂
H CH ₂ CH ₂ NHP (S) (OMe) ₂
H CH ₂ CH ₂ NHP (S) (OEt) ₂
H CH ₂ CH ₂ N (Me) SO ₂ Me
H CH ₂ CH ₂ N (Me) SO ₂ CF ₃
H CH ₂ CH ₂ N (Me) OMe
H CH ₂ CH (Me) NHC (O) Me
H CH ₂ CH (Me) NHC (O) CF ₃
H CH ₂ CH (Me) NHC (O) CH ₂ CF ₃
H CH ₂ CH (Me) NHC (O) CH ₂ SMe
H CH ₂ CH (Me) NHC (O) CH ₂ S (O) Me
H CH ₂ CH (Me) NHC (O) CH ₂ S (O) ₂ Me
H CH ₂ CH (Me) NHC (O) OMe
H CH (Me) CH ₂ NHC (O) Me
H CH (Me) CH ₂ NHC (O) CF ₃
H CH (Me) CH ₂ NHC (O) CH ₂ CF ₃
H CH (Me) CH ₂ NHC (O) CH ₂ SMe
H CH (Me) CH ₂ NHC (O) CH ₂ S (O) Me
H CH (Me) CH ₂ NHC (O) CH ₂ S (O) ₂ Me
H CH (Me) CH ₂ NHC (O) OMe
H CH ₂ CH ₂ CH ₂ NHC (O) Me
H CH ₂ CH ₂ CH ₂ NHC (O) OMe
H OMe
H OPr-i
H OCH ₂ CF ₃
H OCH ₂ CH = CH ₂
H OCH ₂ CH = CHCl
HN (Me) ₂
HN (Et) ₂
HN (n-Pr) ₂
H NHCH ₂ CF ₃
HN (Me) CH ₂ CF ₃
HN (CH ₂ CF ₃ ) C (O) Me
HN (CH ₂ CF ₃ ) C (O) OMe
HN (CH ₂ CF ₃ ) C (O) OEt
H NHCHO
H NHC (O) Me
H NHC (O) Et
H NHC (O) Pr-n
H NHC (O) Pr-i
H NHC (O) Pr-c
H NHC (O) Bu-n
H NHC (O) Bu-i
H NHC (O) Bu-s
H NHC (O) Bu-t
H NHC (O) Hex-n
H NHC (O) Hex-c
H NHC (O) CH ₂ CF ₃
H NHC (O) CH ₂ SMe
H NHC (O) CH ₂ S (O) Me
H NHC (O) CH ₂ S (O) ₂ Me
H NHC (O) OMe
H NHC (O) OEt
H NHC (O) OBu-t
H NHC (O) SMe
H NHC (S) OMe
H NHC (S) SMe
HN (Me) CHO
HN (Me) C (O) Me
HN (Me) C (O) Et
HN (Me) C (O) Pr-n
HN (Me) C (O) Pr-i
HN (Me) C (O) Pr-c
HN (Me) C (O) Bu-n
HN (Me) C (O) Bu-i
HN (Me) C (O) Bu-s
HN (Me) C (O) Bu-t
HN (Me) C (O) Hex-n
HN (Me) C (O) Hex-c
HN (Me) C (O) CH ₂ CF ₃
HN (Me) C (O) CH ₂ SMe
HN (Me) C (O) CH ₂ S (O) Me
HN (Me) C (O) CH ₂ S (O) ₂ Me
HN (Me) C (O) OMe
HN (Me) C (O) OEt
HN (Me) C (O) OBu-t
HN (Et) CHO
HN (Et) C (O) Me
HN (Et) C (O) Et
HN (Et) C (O) Pr-n
HN (Et) C (O) Pr-i
HN (Et) C (O) Pr-c
HN (Et) C (O) Bu-n
HN (Et) C (O) Bu-i
HN (Et) C (O) Bu-s
HN (Et) C (O) Bu-t
HN (Et) C (O) Hex-n
HN (Et) C (O) Hex-c
HN (Et) C (O) CH ₂ CF ₃
HN (Et) C (O) CH ₂ SMe
HN (Et) C (O) CH ₂ S (O) Me
HN (Et) C (O) CH ₂ S (O) ₂ Me
HN (Et) C (O) OMe
HN (Et) C (O) OEt
HN (Et) C (O) OBu-t
H NHC (O) NHMe
H NHC (O) NHCH ₂ CF ₃
H NHC (S) NHMe
H NHC (S) NHCH ₂ CF ₃
HC (O) NHMe
HC (O) NHEt
HC (O) NHPr-n
HC (O) NHPr-i
HC (O) NHPr-c
HC (O) NHBu-n
HC (O) NHBu-i
HC (O) NHBu-s
HC (O) NHBu-t
HC (O) NHCH ₂ CH ₂ F
HC (O) NHCH ₂ CH ₂ Cl
HC (O) NHCH ₂ CH ₂ Br
HC (O) NHCH ₂ CF ₃
HC (O) NHCH ₂ CF ₂ Cl
HC (O) NHCH ₂ CF ₂ CF ₃
HC (O) NHCH ₂ CF ₂ CF ₂ H
HC (O) NHCH ₂ CH ₂ OMe
HC (O) NHCH ₂ CH ₂ SMe
HC (O) NHCH ₂ CH ₂ S (O) Me
HC (O) NHCH ₂ CH ₂ S (O) ₂ Me
HC (O) NHCH ₂ CN
HC (O) NHCH ₂ CH = CH ₂
HC (O) NHCH ₂ CH≡CH
HC (O) N (Me) ₂
HC (O) N (Me) Et
HC (O) N (Me) Pr-n
HC (O) N (Me) Pr-i
HC (O) N (Me) Pr-c
HC (O) N (Me) Bu-n
HC (O) N (Me) Bu-i
HC (O) N (Me) Bu-s
HC (O) N (Me) Bu-t
HC (O) N (Me) CH ₂ CH ₂ F
HC (O) N (Me) CH ₂ CH ₂ Cl
HC (O) N (Me) CH ₂ CH ₂ Br
HC (O) N (Me) CH ₂ CF ₃
HC (O) N (Me) CH ₂ CF ₂ Cl
HC (O) N (Me) CH ₂ CF ₂ CF ₃
HC (O) N (Me) CH ₂ CF ₂ CF ₂ H
HC (O) N (Me) CH ₂ CH ₂ OMe
HC (O) N (Me) CH ₂ CH ₂ SMe
HC (O) N (Me) CH ₂ CH ₂ S (O) Me
HC (O) N (Me) CH ₂ CH ₂ S (O) ₂ Me
HC (O) N (Me) CH ₂ CN
HC (O) N (Me) CH ₂ CH = CH ₂
HC (O) N (Me) CH ₂ CH≡CH
HC (S) NHMe
HC (S) NHEt
HC (S) NHPr-n
HC (S) NHPr-i
HC (S) NHPr-c
HC (S) NHBu-n
HC (S) NHBu-i
HC (S) NHBu-s
HC (S) NHBu-t
HC (S) NHCH ₂ CH ₂ F
HC (S) NHCH ₂ CH ₂ Cl
HC (S) NHCH ₂ CH ₂ Br
HC (S) NHCH ₂ CF ₃
HC (S) NHCH ₂ CF ₂ Cl
HC (S) NHCH ₂ CF ₂ CF ₃
HC (S) NHCH ₂ CF ₂ CF ₂ H
HC (S) NHCH ₂ CH ₂ OMe
HC (S) NHCH ₂ CH ₂ SMe
HC (S) NHCH ₂ CH ₂ S (O) Me
HC (S) NHCH ₂ CH ₂ S (O) ₂ Me
HC (S) NHCH ₂ CN
HC (S) NHCH ₂ CH = CH ₂
HC (S) NHCH ₂ CH≡CH
HC (S) N (Me) ₂
HC (S) N (Me) Et
HC (S) N (Me) Pr-n
HC (S) N (Me) Pr-i
HC (S) N (Me) Pr-c
HC (S) N (Me) Bu-n
HC (S) N (Me) Bu-i
HC (S) N (Me) Bu-s
HC (S) N (Me) Bu-t
HC (S) N (Me) CH ₂ CH ₂ F
HC (S) N (Me) CH ₂ CH ₂ Cl
HC (S) N (Me) CH ₂ CH ₂ Br
HC (S) N (Me) CH ₂ CF ₃
HC (S) N (Me) CH ₂ CF ₂ Cl
HC (S) N (Me) CH ₂ CF ₂ CF ₃
HC (S) N (Me) CH ₂ CF ₂ CF ₂ H
HC (S) N (Me) CH ₂ CH ₂ OMe
HC (S) N (Me) CH ₂ CH ₂ SMe
HC (S) N (Me) CH ₂ CH ₂ S (O) Me
HC (S) N (Me) CH ₂ CH ₂ S (O) ₂ Me
HC (S) N (Me) CH ₂ CN
HC (S) N (Me) CH ₂ CH = CH ₂
HC (S) N (Me) CH ₂ CH≡CH
HC (O) CH ₂ CF3
HC (O) CH ₂ SMe
HC (O) CH ₂ S (O) Me
HC (O) CH ₂ S (O) ₂ Me
H D2-1a
H D2-1b
H D2-2a
H D2-2b
H D2-5a
H D2-5b
H D2-5c
H D2-6a
H D2-6b
H D2-6c
H D2-7a
H D2-8a
H D2-8b
H D2-8c
H D2-9a
H D2-9b
H D2-9c
H D2-10a
H D2-10b
H D2-10c
H D2-11a
H D2-12a
H D2-12b
H D2-12c
H D2-13a
H D2-13b
H D2-14a
H D2-14b
H D2-15a
H D2-15b
H D2-16a
H D2-17a
H D2-18a
H D2-19a
H D2-21a
H D2-21b
H D2-22a
H D2-23a
H D2-23b
H D2-24a
H D2-25a
H D2-27a
H D2-30a
H D2-31a
H D2-32a
H D2-34a
H D2-36a
H D2-37a
H D2-41a
H D2-43a
H D2-45a
H D2-46a
H D2-49a
H D2-51a
H D2-53a
H D2-59a
H D2-61a
H D2-63a
H D2-68a
H D2-75a
H D2-76a
H D2-76b
H D2-77a
H D2-77b
H D2-78a
H D2-78b
H D2-79a
H D2-81a
H D2-82a
H D2-84a
H D2-85a
H D2-87a
H D2-90a
H D2-100a
H D2-100b
H D2-100c
H D2-100d
H D2-100e
H D2-101a
H D2-101b
H D2-101c
H D2-101d
H D2-102a
H D2-102b
H D2-102c
H D2-102d
H D2-102e
H D2-102f
H D2-103a
H CH ₂ (D2-1a)
H CH ₂ (D2-1b)
H CH ₂ (D2-2a)
H CH ₂ (D2-2b)
H CH ₂ (D2-4a)
H CH ₂ (D2-4b)
H CH ₂ (D2-5a)
H CH ₂ (D2-5b)
H CH ₂ (D2-5c)
H CH ₂ (D2-6a)
H CH ₂ (D2-6b)
H CH ₂ (D2-6c)
H CH ₂ (D2-7a)
H CH ₂ (D2-8a)
H CH ₂ (D2-8b)
H CH ₂ (D2-8c)
H CH ₂ (D2-9a)
H CH ₂ (D2-9b)
H CH ₂ (D2-9c)
H CH ₂ (D2-10a)
H CH ₂ (D2-10b)
H CH ₂ (D2-10c)
H CH ₂ (D2-12a)
H CH ₂ (D2-12b)
H CH ₂ (D2-12c)
H CH ₂ (D2-13a)
H CH ₂ (D2-13b)
H CH ₂ (D2-14a)
H CH ₂ (D2-14b)
H CH ₂ (D2-15a)
H CH ₂ (D2-15b)
H CH ₂ (D2-16a)
H CH ₂ (D2-17a)
H CH ₂ (D2-18a)
H CH ₂ (D2-19a)
H CH ₂ (D2-20a)
H CH ₂ (D2-21a)
H CH ₂ (D2-21b)
H CH ₂ (D2-23a)
H CH ₂ (D2-23b)
H CH ₂ (D2-25a)
H CH ₂ (D2-27a)
H CH ₂ (D2-30a)
H CH ₂ (D2-31a)
H CH ₂ (D2-32a)
Me CH ₂ (D2-32a)
Et CH ₂ (D2-32a)
n-Pr CH ₂ (D2-32a)
i-Pr CH ₂ (D2-32a)
CH ₂ OCH ₃ CH ₂ (D2-32a)
CH ₂ CH ₂ OEt CH ₂ (D2-32a)
CH ₂ SCH ₃ CH ₂ (D2-32a)
CH ₂ CN CH ₂ (D2-32a)
CH ₂ CO ₂ Me CH ₂ (D2-32a)
CH ₂ CO ₂ Et CH ₂ (D2-32a)
CH ₂ CH = CH ₂ CH ₂ (D2-32a)
CH ₂ CH≡CH CH ₂ (D2-32a)
C (O) CH ₃ CH ₂ (D2-32a)
C (O) Et CH ₂ (D2-32a)
C (O) Pr-n CH ₂ (D2-32a)
C (O) Pr-c CH ₂ (D2-32a)
C (O) Bu-t CH ₂ (D2-32a)
C (O) CH ₂ OCH ₃ CH ₂ (D2-32a)
C (O) CH ₂ SCH ₃ CH ₂ (D2-32a)
C (O) OMe CH ₂ (D2-32a)
C (O) OEt CH ₂ (D2-32a)
C (O) CH ₂ CH ₂ CH ₂ (D2-32a)
C (O) CH ₂ CH ₂ CH ₂ (D2-32a)
C (O) OCH ₂ CH = CH ₂ CH ₂ (D2-32a)
C (O) SCH ₃ CH ₂ (D2-32a)
C (S) OCH ₃ CH ₂ (D2-32a)
C (S) SCH ₃ CH ₂ (D2-32a)
SMe CH ₂ (D2-32a)
SPh CH ₂ (D2-32a)
SNEt ₂ CH ₂ (D2-32a)
SO ₂ Me CH ₂ (D2-32a)
SO ₂ Et CH ₂ (D2-32a)
SO ₂ Ph CH ₂ (D2-32a)
SO ₂ NMe ₂ CH ₂ (D2-32a)
NH ₂ CH ₂ (D2-32a)
NHMe CH ₂ (D2-32a)
NHCHO CH ₂ (D2-32a)
NHC (O) CH ₃ CH ₂ (D2-32a)
NHC (O) OCH ₃ CH ₂ (D2-32a)
N = C (CH ₃ ) ₂ CH ₂ (D2-32a)
N = CHPh CH ₂ (D2-32a)
H CH ₂ (D2-33a)
H CH ₂ (D2-34a)
H CH ₂ (D2-35a)
H CH ₂ (D2-35b)
H CH ₂ (D2-36a)
H CH ₂ (D2-37a)
Me CH ₂ (D2-37a)
Et CH ₂ (D2-37a)
n-Pr CH ₂ (D2-37a)
i-Pr CH ₂ (D2-37a)
CH ₂ OCH ₃ CH ₂ (D2-37a)
CH ₂ CH ₂ OEt CH ₂ (D2-37a)
CH ₂ SCH ₃ CH ₂ (D2-37a)
CH ₂ CN CH ₂ (D2-37a)
CH ₂ CO ₂ Me CH ₂ (D2-37a)
CH ₂ CO ₂ Et CH ₂ (D2-37a)
CH ₂ CH = CH ₂ CH ₂ (D2-37a)
CH ₂ CH≡CH CH ₂ (D2-37a)
C (O) CH ₃ CH ₂ (D2-37a)
C (O) Et CH ₂ (D2-37a)
C (O) Pr-n CH ₂ (D2-37a)
C (O) Pr-c CH ₂ (D2-37a)
C (O) Bu-t CH ₂ (D2-37a)
C (O) CH ₂ OCH ₃ CH ₂ (D2-37a)
C (O) CH ₂ SCH ₃ CH ₂ (D2-37a)
C (O) OMe CH ₂ (D2-37a)
C (O) OEt CH ₂ (D2-37a)
C (O) CH ₂ CH ₂ CH ₂ (D2-37a)
C (O) CH ₂ CH ₂ CH ₂ (D2-37a)
C (O) OCH ₂ CH = CH ₂ CH ₂ (D2-37a)
C (O) SCH ₃ CH ₂ (D2-37a)
C (S) OCH ₃ CH ₂ (D2-37a)
C (S) SCH ₃ CH ₂ (D2-37a)
SMe CH ₂ (D2-37a)
SPh CH ₂ (D2-37a)
SNEt ₂ CH ₂ (D2-37a)
SO ₂ Me CH ₂ (D2-37a)
SO ₂ Et CH ₂ (D2-37a)
SO ₂ Ph CH ₂ (D2-37a)
SO ₂ NMe ₂ CH ₂ (D2-37a)
NH ₂ CH ₂ (D2-37a)
NHMe CH ₂ (D2-37a)
NHCHO CH ₂ (D2-37a)
NHC (O) CH ₃ CH ₂ (D2-37a)
NHC (O) OCH ₃ CH ₂ (D2-37a)
N = C (CH ₃ ) ₂ CH ₂ (D2-37a)
N = CHPh CH ₂ (D2-37a)
H CH ₂ (D2-38a)
H CH ₂ (D2-39a)
H CH ₂ (D2-40a)
H CH ₂ (D2-41a)
H CH ₂ (D2-42a)
H CH ₂ (D2-43a)
H CH ₂ (D2-45a)
H CH ₂ (D2-46a)
H CH ₂ (D2-49a)
H CH ₂ (D2-51a)
H CH ₂ (D2-53a)
H CH ₂ (D2-59a)
H CH ₂ (D2-61a)
H CH ₂ (D2-63a)
H CH ₂ (D2-68a)
H CH ₂ (D2-75a)
H CH ₂ (D2-76a)
H CH ₂ (D2-76b)
H CH ₂ (D2-77a)
H CH ₂ (D2-77b)
H CH ₂ (D2-78a)
H CH ₂ (D2-78b)
H CH ₂ (D2-79a)
H CH ₂ (D2-81a)
H CH ₂ (D2-82a)
H CH ₂ (D2-84a)
H CH ₂ (D2-85a)
H CH ₂ (D2-87a)
H CH ₂ (D2-90a)
H CH ₂ (D2-100a)
H CH ₂ (D2-100b)
H CH ₂ (D2-100c)
H CH ₂ (D2-100d)
H CH ₂ (D2-100e)
H CH ₂ (D2-101a)
H CH ₂ (D2-101b)
H CH ₂ (D2-101c)
H CH ₂ (D2-101d)
H CH ₂ (D2-102a)
H CH ₂ (D2-102b)
H CH ₂ (D2-102c)
H CH ₂ (D2-102d)
H CH ₂ (D2-102e)
H CH ₂ (D2-102f)
H CH ₂ (D2-103a)
H CH ₂ (D2-108a)
H CH (Me) (D2-1a)
H CH (Me) (D2-2a)
H CH (Me) (D2-5a)
H CH (Me) (D2-5c)
H CH (Me) (D2-6c)
H CH (Me) (D2-8c)
H CH (Me) (D2-9b)
H CH (Me) (D2-9c)
H CH (Me) (D2-10b)
H CH (Me) (D2-10c)
H CH (Me) (D2-12b)
H CH (Me) (D2-12c)
H CH (Me) (D2-13b)
H CH (Me) (D2-14a)
H CH (Me) (D2-14b)
H CH (Me) (D2-15a)
H CH (Me) (D2-15b)
H CH (Me) (D2-16a)
H CH (Me) (D2-17a)
H CH (Me) (D2-18a)
H CH (Me) (D2-23b)
H CH (Me) (D2-27a)
H CH (Me) (D2-31a)
H CH (Me) (D2-32a)
H CH (Me) (D2-35a)
H CH (Me) (D2-36a)
H CH (Me) (D2-37a)
H CH (Me) (D2-39a)
H CH (Me) (D2-41a)
H CH ₂ C (O) NH (D2-1a)
H CH ₂ C (O) NH (D2-2a)
H CH ₂ C (O) NH (D2-5a)
H CH ₂ C (O) NH (D2-5c)
H CH ₂ C (O) NH (D2-6c)
H CH ₂ C (O) NH (D2-8c)
H CH ₂ C (O) NH (D2-9b)
H CH ₂ C (O) NH (D2-9c)
H CH ₂ C (O) NH (D2-10b)
H CH ₂ C (O) NH (D2-10c)
H CH ₂ C (O) NH (D2-12b)
H CH ₂ C (O) NH (D2-12c)
H CH ₂ C (O) NH (D2-13b)
H CH ₂ C (O) NH (D2-14a)
H CH ₂ C (O) NH (D2-14b)
H CH ₂ C (O) NH (D2-15a)
H CH ₂ C (O) NH (D2-15b)
H CH ₂ C (O) NH (D2-16a)
H CH ₂ C (O) NH (D2-17a)
H CH ₂ C (O) NH (D2-18a)
H CH ₂ C (O) NH (D2-23b)
H CH ₂ C (O) NH (D2-27a)
H CH ₂ C (O) NH (D2-31a)
H CH ₂ C (O) NH (D2-32a)
H CH ₂ C (O) NH (D2-35a)
H CH ₂ C (O) NH (D2-36a)
H CH ₂ C (O) NH (D2-37a)
H CH ₂ C (O) NH (D2-39a)
H CH ₂ C (O) NH (D2-41a)
H CH ₂ C (O) NH (D2-45a)
H CH ₂ C (O) NH (D2-46a)
H CH ₂ C (O) NH (D2-49a)
H CH ₂ C (O) NH (D2-51a)
H CH ₂ C (O) NH (D2-53a)
H CH ₂ C (O) NH (D2-59a)
H CH ₂ C (O) NH (D2-61a)
H CH ₂ C (O) NH (D2-63a)
H CH ₂ C (O) NH (D2-68a)
H CH ₂ C (O) NH (D2-75a)
H CH ₂ C (O) NH (D2-76a)
H CH ₂ C (O) NH (D2-76b)
H CH ₂ C (O) NH (D2-77a)
H CH ₂ C (O) NH (D2-77b)
H CH ₂ C (O) NH (D2-78a)
H CH ₂ C (O) NH (D2-78b)
H CH ₂ C (O) NH (D2-79a)
H CH ₂ C (O) NH (D2-82a)
H CH ₂ C (O) NH (D2-84a)
H CH ₂ C (O) NH (D2-85a)
H CH ₂ C (O) NH (D2-87a)
H CH ₂ C (O) NH (D2-90a)
H CH ₂ C (O) NH (D2-100a)
H CH ₂ C (O) NH (D2-100b)
H CH ₂ C (O) NH (D2-100c)
H CH ₂ C (O) NH (D2-100d)
H CH ₂ C (O) NH (D2-100e)
H CH ₂ C (O) NH (D2-101a)
H CH ₂ C (O) NH (D2-101b)
H CH ₂ C (O) NH (D2-101c)
H CH ₂ C (O) NH (D2-101d)
H CH ₂ C (O) NH (D2-108a)
H CH ₂ C (O) NHCH ₂ (D2-1a)
H CH ₂ C (O) NHCH ₂ (D2-2a)
H CH ₂ C (O) NHCH ₂ (D2-5a)
H CH ₂ C (O) NHCH ₂ (D2-5c)
H CH ₂ C (O) NHCH ₂ (D2-6c)
H CH ₂ C (O) NHCH ₂ (D2-8c)
H CH ₂ C (O) NHCH ₂ (D2-9b)
H CH ₂ C (O) NHCH ₂ (D2-9c)
H CH ₂ C (O) NHCH ₂ (D2-10b)
H CH ₂ C (O) NHCH ₂ (D2-10c)
H CH ₂ C (O) NHCH ₂ (D2-12b)
H CH ₂ C (O) NHCH ₂ (D2-12c)
H CH ₂ C (O) NHCH ₂ (D2-13b)
H CH ₂ C (O) NHCH ₂ (D2-14a)
H CH ₂ C (O) NHCH ₂ (D2-14b)
H CH ₂ C (O) NHCH ₂ (D2-15a)
H CH ₂ C (O) NHCH ₂ (D2-15b)
H CH ₂ C (O) NHCH ₂ (D2-16a)
H CH ₂ C (O) NHCH ₂ (D2-17a)
H CH ₂ C (O) NHCH ₂ (D2-18a)
H CH ₂ C (O) NHCH ₂ (D2-23b)
H CH ₂ C (O) NHCH ₂ (D2-27a)
H CH ₂ C (O) NHCH ₂ (D2-31a)
H CH ₂ C (O) NHCH ₂ (D2-32a)
H CH ₂ C (O) NHCH ₂ (D2-35a)
H CH ₂ C (O) NHCH ₂ (D2-36a)
H CH ₂ C (O) NHCH ₂ (D2-37a)
H CH ₂ C (O) NHCH ₂ (D2-39a)
H CH ₂ C (O) NHCH ₂ (D2-41a)
H CH ₂ C (O) NHCH ₂ (D2-45a)
H CH ₂ C (O) NHCH ₂ (D2-46a)
H CH ₂ C (O) NHCH ₂ (D2-49a)
H CH ₂ C (O) NHCH ₂ (D2-51a)
H CH ₂ C (O) NHCH ₂ (D2-53a)
H CH ₂ C (O) NHCH ₂ (D2-59a)
H CH ₂ C (O) NHCH ₂ (D2-61a)
H CH ₂ C (O) NHCH ₂ (D2-63a)
H CH ₂ C (O) NHCH ₂ (D2-68a)
H CH ₂ C (O) NHCH ₂ (D2-75a)
H CH ₂ C (O) NHCH ₂ (D2-76a)
H CH ₂ C (O) NHCH ₂ (D2-76b)
H CH ₂ C (O) NHCH ₂ (D2-77a)
H CH ₂ C (O) NHCH ₂ (D2-77b)
H CH ₂ C (O) NHCH ₂ (D2-78a)
H CH ₂ C (O) NHCH ₂ (D2-78b)
H CH ₂ C (O) NHCH ₂ (D2-79a)
H CH ₂ C (O) NHCH ₂ (D2-82a)
H CH ₂ C (O) NHCH ₂ (D2-84a)
H CH ₂ C (O) NHCH ₂ (D2-85a)
H CH ₂ C (O) NHCH ₂ (D2-87a)
H CH ₂ C (O) NHCH ₂ (D2-90a)
H CH ₂ C (O) NHCH ₂ (D2-102a)
H CH ₂ C (O) NHCH ₂ (D2-102b)
H CH ₂ C (O) NHCH ₂ (D2-102c)
H CH ₂ C (O) NHCH ₂ (D2-102d)
H CH ₂ C (O) NHCH ₂ (D2-102e)
H CH ₂ C (O) NHCH ₂ (D2-102f)
H CH ₂ C (O) NHCH ₂ (D2-103a)
H CH ₂ C (O) NHCH ₂ (D2-108a)
H NH (D2-7a)
H NH (D2-10c)
H NH (D2-22a)
H NH (D2-24a)
H NH (D2-32a)
H NC (O) Me (D2-32a)
H NC (O) OMe (D2-32a)
H NC (O) Et (D2-32a)
H NC (O) OEt (D2-32a)
H NC (O) CH ₂ CF ₃ (D2-32a)
H NSO ₂ Me (D2-32a)
H NSO ₂ CF ₃ (D2-32a)
H NSO ₂ Ph (D2-32a)
H NH (D2-35a)
H NH (D2-36a)
H NH (D2-37a)
H NH (D2-39a)
H NH (D2-43a)
H NH (D2-45a)
H NH (D2-49a)
H NH (D2-51a)
H NH (D2-53a)
H NH (D2-59a)
H NH (D2-61a)
H NH (D2-63a)
H NH (D2-108a)
H NH {D2-32b (3-Cl)}
H NH {D2-32b (4-Cl)}
H NH {D2-32b (5-Cl)}
H NH {D2-32b (6-Cl)}
H NH {D2-32b (4-CF ₃ )}
H NH {D2-108b (2-Cl)}
H NH {D2-108b (3-Cl)}
H NH {D2-108b (4-Cl)}
H NH {D2-108b (2-Me)}
H NH {D2-108b (3-Me)}
H NH {D2-108b (4-Me)}
H CH ₂ CH ₂ (D2-1a)
H CH ₂ CH ₂ (D2-1b)
H CH ₂ CH ₂ (D2-2a)
H CH ₂ CH ₂ (D2-2b)
H CH ₂ CH ₂ (D2-5c)
H CH ₂ CH ₂ (D2-6c)
H CH ₂ CH ₂ (D2-7a)
H CH ₂ CH ₂ (D2-8c)
H CH ₂ CH ₂ (D2-9b)
H CH ₂ CH ₂ (D2-10b)
H CH ₂ CH ₂ (D2-10c)
H CH ₂ CH ₂ (D2-11a)
H CH ₂ CH ₂ (D2-20a)
H CH ₂ CH ₂ (D2-22a)
H CH ₂ CH ₂ (D2-24a)
H CH ₂ CH ₂ (D2-26a)
H CH ₂ CH ₂ (D2-28a)
H CH ₂ CH ₂ (D2-29a)
H CH ₂ CH ₂ (D2-32a)
H CH ₂ CH ₂ (D2-36a)
H CH ₂ CH ₂ (D2-37a)
H CH ₂ CH ₂ OCH ₂ (D2-1a)
H CH ₂ CH ₂ OCH ₂ (D2-1b)
H CH ₂ CH ₂ OCH ₂ (D2-2a)
H CH ₂ CH ₂ OCH ₂ (D2-2b)
H CH ₂ CH ₂ OCH ₂ (D2-4a)
H CH ₂ CH ₂ OCH ₂ (D2-4b)
H CH ₂ CH ₂ OCH ₂ (D2-5a)
H CH ₂ CH ₂ OCH ₂ (D2-5b)
H CH ₂ CH ₂ OCH ₂ (D2-5c)
H CH ₂ CH ₂ OCH ₂ (D2-6a)
H CH ₂ CH ₂ OCH ₂ (D2-6b)
H CH ₂ CH ₂ OCH ₂ (D2-6c)
H CH ₂ CH ₂ OCH ₂ (D2-7a)
H CH ₂ CH ₂ OCH ₂ (D2-8a)
H CH ₂ CH ₂ OCH ₂ (D2-8b)
H CH ₂ CH ₂ OCH ₂ (D2-8c)
H CH ₂ CH ₂ OCH ₂ (D2-9a)
H CH ₂ CH ₂ OCH ₂ (D2-9b)
H CH ₂ CH ₂ OCH ₂ (D2-9c)
H CH ₂ CH ₂ OCH ₂ (D2-10a)
H CH ₂ CH ₂ OCH ₂ (D2-10b)
H CH ₂ CH ₂ OCH ₂ (D2-10c)
H CH ₂ CH ₂ OCH ₂ (D2-12a)
H CH ₂ CH ₂ OCH ₂ (D2-12b)
H CH ₂ CH ₂ OCH ₂ (D2-12c)
H CH ₂ CH ₂ OCH ₂ (D2-13a)
H CH ₂ CH ₂ OCH ₂ (D2-13b)
H CH ₂ CH ₂ OCH ₂ (D2-14a)
H CH ₂ CH ₂ OCH ₂ (D2-14b)
H CH ₂ CH ₂ OCH ₂ (D2-15a)
H CH ₂ CH ₂ OCH ₂ (D2-15b)
H CH ₂ CH ₂ OCH ₂ (D2-16a)
H CH ₂ CH ₂ OCH ₂ (D2-17a)
H CH ₂ CH ₂ OCH ₂ (D2-18a)
H CH ₂ CH ₂ OCH ₂ (D2-19a)
H CH ₂ CH ₂ OCH ₂ (D2-20a)
H CH ₂ CH ₂ OCH ₂ (D2-21a)
H CH ₂ CH ₂ OCH ₂ (D2-21b)
H CH ₂ CH ₂ OCH ₂ (D2-23a)
H CH ₂ CH ₂ OCH ₂ (D2-23b)
H CH ₂ CH ₂ OCH ₂ (D2-25a)
H CH ₂ CH ₂ OCH ₂ (D2-27a)
H CH ₂ CH ₂ OCH ₂ (D2-30a)
H CH ₂ CH ₂ OCH ₂ (D2-31a)
H CH ₂ CH ₂ OCH ₂ (D2-32a)
H CH ₂ CH ₂ OCH ₂ (D2-33a)
H CH ₂ CH ₂ OCH ₂ (D2-34a)
H CH ₂ CH ₂ OCH ₂ (D2-35a)
H CH ₂ CH ₂ OCH ₂ (D2-35b)
H CH ₂ CH ₂ OCH ₂ (D2-36a)
H CH ₂ CH ₂ OCH ₂ (D2-37a)
H CH ₂ CH ₂ OCH ₂ (D2-38a)
H CH ₂ CH ₂ OCH ₂ (D2-39a)
H CH ₂ CH ₂ OCH ₂ (D2-40a)
H CH ₂ CH ₂ OCH ₂ (D2-41a)
H CH ₂ CH ₂ OCH ₂ (D2-42a)
H CH ₂ CH ₂ OCH ₂ (D2-43a)
H CH ₂ CH ₂ OCH ₂ (D2-45a)
H CH ₂ CH ₂ OCH ₂ (D2-46a)
H CH ₂ CH ₂ OCH ₂ (D2-49a)
H CH ₂ CH ₂ OCH ₂ (D2-51a)
H CH ₂ CH ₂ OCH ₂ (D2-53a)
H CH ₂ CH ₂ OCH ₂ (D2-59a)
H CH ₂ CH ₂ OCH ₂ (D2-61a)
H CH ₂ CH ₂ OCH ₂ (D2-63a)
H CH ₂ CH ₂ OCH ₂ (D2-68a)
H CH ₂ CH ₂ OCH ₂ (D2-75a)
H CH ₂ CH ₂ OCH ₂ (D2-76a)
H CH ₂ CH ₂ OCH ₂ (D2-76b)
H CH ₂ CH ₂ OCH ₂ (D2-77a)
H CH ₂ CH ₂ OCH ₂ (D2-77b)
H CH ₂ CH ₂ OCH ₂ (D2-78a)
H CH ₂ CH ₂ OCH ₂ (D2-78b)
H CH ₂ CH ₂ OCH ₂ (D2-79a)
H CH ₂ CH ₂ OCH ₂ (D2-81a)
H CH ₂ CH ₂ OCH ₂ (D2-82a)
H CH ₂ CH ₂ OCH ₂ (D2-84a)
H CH ₂ CH ₂ OCH ₂ (D2-85a)
H CH ₂ CH ₂ OCH ₂ (D2-87a)
H CH ₂ CH ₂ OCH ₂ (D2-90a)
H CH ₂ CH ₂ OCH ₂ (D2-100a)
H CH ₂ CH ₂ OCH ₂ (D2-100b)
H CH ₂ CH ₂ OCH ₂ (D2-100c)
H CH ₂ CH ₂ OCH ₂ (D2-100d)
H CH ₂ CH ₂ OCH ₂ (D2-100e)
H CH ₂ CH ₂ OCH ₂ (D2-101a)
H CH ₂ CH ₂ OCH ₂ (D2-101b)
H CH ₂ CH ₂ OCH ₂ (D2-101c)
H CH ₂ CH ₂ OCH ₂ (D2-101d)
H CH ₂ CH ₂ OCH ₂ (D2-102a)
H CH ₂ CH ₂ OCH ₂ (D2-102b)
H CH ₂ CH ₂ OCH ₂ (D2-102c)
H CH ₂ CH ₂ OCH ₂ (D2-102d)
H CH ₂ CH ₂ OCH ₂ (D2-102e)
H CH ₂ CH ₂ OCH ₂ (D2-102f)
H CH ₂ CH ₂ OCH ₂ (D2-103a)
H CH ₂ CH ₂ OCH ₂ (D2-108a)
H CH ₂ CH ₂ SCH ₂ (D2-1a)
H CH ₂ CH ₂ SCH ₂ (D2-1b)
H CH ₂ CH ₂ SCH ₂ (D2-2a)
H CH ₂ CH ₂ SCH ₂ (D2-2b)
H CH ₂ CH ₂ SCH ₂ (D2-4a)
H CH ₂ CH ₂ SCH ₂ (D2-4b)
H CH ₂ CH ₂ SCH ₂ (D2-5a)
H CH ₂ CH ₂ SCH ₂ (D2-5b)
H CH ₂ CH ₂ SCH ₂ (D2-5c)
H CH ₂ CH ₂ SCH ₂ (D2-6a)
H CH ₂ CH ₂ SCH ₂ (D2-6b)
H CH ₂ CH ₂ SCH ₂ (D2-6c)
H CH ₂ CH ₂ SCH ₂ (D2-7a)
H CH ₂ CH ₂ SCH ₂ (D2-8a)
H CH ₂ CH ₂ SCH ₂ (D2-8b)
H CH ₂ CH ₂ SCH ₂ (D2-8c)
H CH ₂ CH ₂ SCH ₂ (D2-9a)
H CH ₂ CH ₂ SCH ₂ (D2-9b)
H CH ₂ CH ₂ SCH ₂ (D2-9c)
H CH ₂ CH ₂ SCH ₂ (D2-10a)
H CH ₂ CH ₂ SCH ₂ (D2-10b)
H CH ₂ CH ₂ SCH ₂ (D2-10c)
H CH ₂ CH ₂ SCH ₂ (D2-12a)
H CH ₂ CH ₂ SCH ₂ (D2-12b)
H CH ₂ CH ₂ SCH ₂ (D2-12c)
H CH ₂ CH ₂ SCH ₂ (D2-13a)
H CH ₂ CH ₂ SCH ₂ (D2-13b)
H CH ₂ CH ₂ OCH ₂ (D2-14a)
H CH ₂ CH ₂ SCH ₂ (D2-14b)
H CH ₂ CH ₂ SCH ₂ (D2-15a)
H CH ₂ CH ₂ SCH ₂ (D2-15b)
H CH ₂ CH ₂ SCH ₂ (D2-16a)
H CH ₂ CH ₂ SCH ₂ (D2-17a)
H CH ₂ CH ₂ SCH ₂ (D2-18a)
H CH ₂ CH ₂ SCH ₂ (D2-19a)
H CH ₂ CH ₂ SCH ₂ (D2-20a)
H CH ₂ CH ₂ SCH ₂ (D2-21a)
H CH ₂ CH ₂ SCH ₂ (D2-21b)
H CH ₂ CH ₂ SCH ₂ (D2-23a)
H CH ₂ CH ₂ SCH ₂ (D2-23b)
H CH ₂ CH ₂ SCH ₂ (D2-25a)
H CH ₂ CH ₂ SCH ₂ (D2-27a)
H CH ₂ CH ₂ SCH ₂ (D2-30a)
H CH ₂ CH ₂ SCH ₂ (D2-31a)
H CH ₂ CH ₂ SCH ₂ (D2-32a)
H CH ₂ CH ₂ SCH ₂ (D2-33a)
H CH ₂ CH ₂ SCH ₂ (D2-34a)
H CH ₂ CH ₂ SCH ₂ (D2-35a)
H CH ₂ CH ₂ SCH ₂ (D2-35b)
H CH ₂ CH ₂ SCH ₂ (D2-36a)
H CH ₂ CH ₂ SCH ₂ (D2-37a)
H CH ₂ CH ₂ SCH ₂ (D2-38a)
H CH ₂ CH ₂ SCH ₂ (D2-39a)
H CH ₂ CH ₂ SCH ₂ (D2-40a)
H CH ₂ CH ₂ SCH ₂ (D2-41a)
H CH ₂ CH ₂ SCH ₂ (D2-42a)
H CH ₂ CH ₂ SCH ₂ (D2-43a)
H CH ₂ CH ₂ SCH ₂ (D2-45a)
H CH ₂ CH ₂ SCH ₂ (D2-46a)
H CH ₂ CH ₂ SCH ₂ (D2-49a)
H CH ₂ CH ₂ SCH ₂ (D2-51a)
H CH ₂ CH ₂ SCH ₂ (D2-53a)
H CH ₂ CH ₂ SCH ₂ (D2-59a)
H CH ₂ CH ₂ SCH ₂ (D2-61a)
H CH ₂ CH ₂ SCH ₂ (D2-63a)
H CH ₂ CH ₂ SCH ₂ (D2-68a)
H CH ₂ CH ₂ SCH ₂ (D2-75a)
H CH ₂ CH ₂ SCH ₂ (D2-76a)
H CH ₂ CH ₂ SCH ₂ (D2-76b)
H CH ₂ CH ₂ SCH ₂ (D2-77a)
H CH ₂ CH ₂ SCH ₂ (D2-77b)
H CH ₂ CH ₂ SCH ₂ (D2-78a)
H CH ₂ CH ₂ SCH ₂ (D2-78b)
H CH ₂ CH ₂ SCH ₂ (D2-79a)
H CH ₂ CH ₂ SCH ₂ (D2-81a)
H CH ₂ CH ₂ SCH ₂ (D2-82a)
H CH ₂ CH ₂ SCH ₂ (D2-84a)
H CH ₂ CH ₂ SCH ₂ (D2-85a)
H CH ₂ CH ₂ SCH ₂ (D2-87a)
H CH ₂ CH ₂ SCH ₂ (D2-90a)
H CH ₂ CH ₂ SCH ₂ (D2-100a)
H CH ₂ CH ₂ SCH ₂ (D2-100b)
H CH ₂ CH ₂ SCH ₂ (D2-100c)
H CH ₂ CH ₂ SCH ₂ (D2-100d)
H CH ₂ CH ₂ SCH ₂ (D2-100e)
H CH ₂ CH ₂ SCH ₂ (D2-101a)
H CH ₂ CH ₂ SCH ₂ (D2-101b)
H CH ₂ CH ₂ SCH ₂ (D2-101c)
H CH ₂ CH ₂ SCH ₂ (D2-101d)
H CH ₂ CH ₂ SCH ₂ (D2-102a)
H CH ₂ CH ₂ SCH ₂ (D2-102b)
H CH ₂ CH ₂ SCH ₂ (D2-102c)
H CH ₂ CH ₂ SCH ₂ (D2-102d)
H CH ₂ CH ₂ SCH ₂ (D2-102e)
H CH ₂ CH ₂ SCH ₂ (D2-102f)
H CH ₂ CH ₂ SCH ₂ (D2-103a)
H CH ₂ CH ₂ SCH ₂ (D2-108a)
H CH ₂ {D2-1c (3-Me)}
H CH ₂ {D2-1d (5-Cl)}
H CH ₂ {D2-2c (5-Br)}
H CH ₂ {D2-2d (5-Cl)}
H CH ₂ {D2-4c (5-Cl)}
H CH ₂ {D2-4d (5-Cl)}
H CH ₂ {D2-5d (3-Me)}
H CH ₂ {D2-5e (3-Me)}
H CH ₂ {D2-5f (5-Me)}
H CH ₂ {D2-6d (3-Cl)}
H CH ₂ {D2-6e (3-Me)}
H CH ₂ {D2-6f (5-Me)}
H CH ₂ {D2-7a (3-Me)}
H CH ₂ {D2-8d (3-Cl)}
H CH ₂ {D2-8e (3-CF ₃ )}
H CH ₂ {D2-8f (5-Me)}
H CH ₂ {D2-9d (2-Me)}
H CH ₂ {D2-9e (2-Me)}
H CH ₂ {D2-9f (4-Me)}
H CH ₂ {D2-10e (2-Me)}
H CH ₂ {D2-10f (2-Cl)}
H CH ₂ {D2-10e (2-Br)}
H CH ₂ {D2-12d (4-Me)}
H CH ₂ {D2-12e (5-Me)}
H CH ₂ {D2-12f (5-Cl)}
H CH ₂ {D2-13c (Me)}
H CH ₂ {D2-13d (Cl)}
H CH ₂ {D2-14c (Me)}
H CH ₂ {D2-14d (Me)}
H CH ₂ {D2-15c (Cl)}
H CH ₂ {D2-15d (Me)}
H CH ₂ {D2-16b (Ph)}
H CH ₂ {D2-17b (Ph)}
H CH ₂ {D2-18b (Me)}
H CH ₂ {D2-19b (Cl)}
H CH ₂ {D2-20b (Me)}
H CH ₂ {D2-21c (Me)}
H CH ₂ {D2-21d (Me)}
H CH ₂ {D2-23c (t-Bu)}
H CH ₂ {D2-23d (Ph)}
H CH ₂ {D2-25b (Me)}
H CH ₂ {D2-27a (Me)}
H CH ₂ {D2-32b (3-Cl)}
H CH ₂ {D2-32b (4-Cl)}
H CH ₂ {D2-32b (5-Cl)}
H CH ₂ {D2-32b (6-Cl)}
H CH ₂ {D2-32b (3-Me)}
H CH ₂ {D2-32b (4-Me)}
H CH ₂ {D2-32b (5-Me)}
H CH ₂ {D2-32b (6-Me)}
H CH ₂ {D2-32b (5-CF ₃ )}
H CH ₂ {D2-33b (4-CF ₃ )}
H CH ₂ {D2-34b (3-Cl)}
H CH ₂ {D2-35c (3-Cl)}
H CH ₂ {D2-35d (3-Cl)}
H CH ₂ {D2-36b (2-Me)}
H CH ₂ {D2-37b (4-Me)}
H CH ₂ {D2-38b (2-Me)}
H CH ₂ {D2-39b (5-Me)}
H CH ₂ {D2-108b (2-Cl)}
H CH ₂ {D2-108b (3-Cl)}
H CH ₂ {D2-108b (4-Cl)}
H CH ₂ {D2-108b (2-Me)}
H CH ₂ {D2-108b (3-Me)}
H CH ₂ {D2-108b (4-Me)}
H CH ₂ {D2-108b (2-CF ₃ )}
H CH ₂ {D2-108b (3-CF ₃ )}
H CH ₂ {D2-108b (4-CF ₃ )}
H CH ₂ {D2-108b (2-OMe)}
H CH ₂ {D2-108b (3-OMe)}
H CH ₂ {D2-108b (4-OMe)}
H CH ₂ CH ₂ {D2-7b (4-Cl)}
H CH ₂ CH ₂ {D2-10e (2-Cl)}
H CH ₂ CH ₂ {D2-11b (2-Me)}
H CH ₂ CH ₂ {D2-20b (4-Me)}
H CH ₂ CH ₂ {D2-22b (3-SMe)}
H CH ₂ CH ₂ {D2-24b (3-Me)}
H CH ₂ CH ₂ {D2-26b (4-CO ₂ Me)}
H CH ₂ CH ₂ {D2-28b (Me)}
H CH ₂ CH ₂ {D2-29a (Ph)}
H CH ₂ CH ₂ {D2-32b (3-Cl)}
H CH ₂ CH ₂ {D2-36b (2-Me)}
H CH ₂ CH ₂ (D2-37b (4-Me)
―――――――――――――――――――
The compounds of the present invention are stored in warehouses, so-called agricultural pests that harm agricultural and horticultural crops and trees, so-called livestock pests that parasitize livestock and poultry, so-called sanitary pests that cause various adverse effects in the human living environment such as houses. It is possible to effectively control insects such as so-called stored grain pests that harm cereals and the like, and pests such as mites, crustaceans, molluscs, and nematodes that occur and harm in similar situations at low concentrations.

本発明化合物を用いて防除しうる昆虫類、ダニ類、甲殻類、軟体動物及び線虫類には具体的に、例えば、
クリタマバチChestnut gall wasp（Dryocosmus kuriphilus）、アルゼンチンアリArgentine ant（Linepithema humile）、グンタイアリArmy ant（Eciton burchelli, E. schmitti）、クロオオアリJapanese carpenter ant（Camponotus japonicus）、イエヒメアリPharaoh ant（Monomorium pharaonis）、ブルドックアント類Bulldog ant（Myrmecia spp.）、ファイヤーアント類Fire ant（Solenopsis spp.）、オオスズメバチAsian giant hornet（Vespa mandarina）、キイロスズメバチJapanese yellow hornet（Vespa simillima）、チュウレンジハバチLarge rose sawfly（Arge pagana）、マツノキハバチEuropean pine sawfly（Neodiprion sertifer）、クリハバチChestnut sawfly（Apethymus kuri）、セグロカブラハバチCabbage sawfly（Athalia infumata）、カブラハバチTurnip sawfly（Athalia rosae）等の膜翅目（Hymenoptera）昆虫、
ナシチビガPear leaf miner（Bucculatrix pyrivorella）、チャノホソガTea leafroller（Caloptilia theivora）、キンモンホソガApple leafminer（Phyllonorycter ringoniella）、ミカンハモグリガCitrus leafminer（Phyllocnistis citrella）、イモキバガSweetpotato leaffolder（Helcystogramma triannulella）、ワタアカミムシPink bollworm（Pectinophora gossypiella）、カキノヘタムシガPersimmon fruit moth（Stathmopoda masinissa）、モモシンクイガPeach fruit moth（Carposina sasakii）、ネギコガAllium leafminer（Acrolepiopsis sapporensis）、ヤマノイモコガYam leafminer（Acrolepiopsis suzukiella）、モモハモグリガPeach leafminer（Lyonetia clerkella）、ギンモンハモグリガ（Lyonetia prunifoliella malinella）、コナガDiamondback moth（Plutella xylostella）、ニカメイガRice stem borer（Chilo suppressalis）、シバツトガBluegrass webworm（Parapediasia teterrella）、ハイマダラノメイガCabbage webworm（Hellula undalis）、コブノメイガRice leafroller（Cnaphalocrocis medinalis）、モモノゴマダラノメイガYellow peach moth（Conogethes punctiferalis）、ワタヘリクロノメイガCucumber moth（Diaphania indica）、クワノメイガMulberry pyralid（Glyphodes pyloalis）、アワノメイガAsian corn borer（Ostrinia furnacalis）、ヨーロッパアワノメイガEuropean corn borer（Ostrinia nubilalis）、アズキノメイガAdzuki bean borer（Ostrinia scapulalis）、モロコシマダラメイガLesser corn stalk borer（Elasmopalpus lignosellus）、シロイチモジマダラメイガLimabean pod borer（Etiella zinckenella）、ピーチツリーボーラーPeach tree borer（Synanthedon exitiosa）、コスカシバCherry tree borer（Synanthedon hector）、クビアカスカシバ（Toleria romanovi）、イラガOriental moth（Monema flavescens）、アオイラガ（Parasa consocia）、ヒロヘリアオイラガ（Parasa lepida）、クロシタアオイラガ（Parasa siniea）、タケノホソクロバ（Artona martini）、リンゴハマキクロバ（Illiberis pruni）、ウメスカシクロバ（Illiberis rotundata）、ヒメボクトウCarpenter moth（Cossus insularis）、コドリンガCodling moth（Cydia pomonella）、スモモヒメシンクイPlum fruit moth（Grapholita dimorpha）、ナシヒメシンクイOriental fruit moth（Grapholita molesta）、マメシンクイガSoybean pod borer（Leguminivora glycinivorella）、マメヒメサヤムシガSoybean podworm（Matsumuraeses phaseoli）、グレープベリーモスGrape berry moth（Endopiza viteana）、チャノコカクモンハマキSmaller tea tortrix（Adoxophyes honmai）、リンゴコカクモンハマキSummer fruit tortrix（Adoxophyes orana fasciata）、リンゴモンハマキAsiatic leafroller（Archips breviplicanus）、ミダレカクモンハマキApple tortrix（Archips fuscocupreanus）、チャハマキOriental tea tortrix（Homona magnanima）、トビハマキDark fruit-tree tortrix（Pandemis heparana）、マツカレハPine moth（Dendrolimus spectabilis）、ツガカレハJananese hemlock caterpillar（Dendrolimus superans）、タケカレハJapanese bamboo lappet moth（Euthrix albomaculata）、ヨシカレハDrinker moth（Euthrix potatoria）、カレハガOriental lappet（Gastropacha orientalis）、クヌギカレハ（Kunugia undans）、ヤマダカレハ（Kunugia yamadai）、トマトホーンワームTomato hornworm（Manduca quinquemaculata）、タバコスズメガTobacco hornworm（Manduca sexta）、アメリカシロヒトリFall webworm moth（Hyphantria cunea）、クワゴマダラヒトリMulberry tiger moth（Lemyra imparilis）、ヤネホソバ（Eilema fuscodorsalis）、ツマキホソバ（Eilema laevis）、ドクガOriental tussock moth（Artaxa subflava）、キドクガ（Euproctis piperita）、チャドクガTea tussock moth（Euproctis pseudoconspersa）、モンシロドクガSwan moth（Sphrageidus similis）、マイマイガGypsy moth（Lymantria dispar）、ヒメシロモンドクガWhite-spotted tussock moth（Orgyia thyellina）、フタオビコヤガRice green caterpillar（Naranga aenescens）、アケビコノハ（Adris tyrannus）、ナカジロシタバSweet potato leaf worm（Aedia leucomelas）、ヨトウガCabbage armyworm（Mamestra brassicae）、アワヨトウOriental armyworm（Pseudaletia separata）、スジキリヨトウLawn grass cutworm（Spodoptera depravata）、サザンアーミーワームSouthern armyworm（Spodoptera eridania）、シロイチモジヨトウBeet armyworm（Spodoptera exigua）、フォールアーミーワームFall armyworm（Spodoptera frugiperda）、コットンリーフワームCotton leafworm（Spodoptera littoralis）、ハスモンヨトウCommon cutworm（Spodoptera litura）、オオタバコガCotton bollworm（Helicoverpa armigera）、タバコガOriental tobacco budworm（Helicoverpa assulta）、タバコバッドワームTobacco budworm（Heliothis virescens）、アメリカタバコガCorn earworm（Helicoverpa zea）、タマナヤガBlack cutworm（Agrotis ipsilon）、カブラヤガTurnip moth（Agrotis segetum）、タマナギンウワバAsiatic common looper（Autographa nigrisigna）、ミツモンキンウワバThreespotted plusia（Ctenoplusia agnata）、ソイビーンルーパーSoybean looper（Pseudoplusia includens）、イラクサギンウワバCabbage looper（Trichoplusia ni）、ヨモギエダシャクJapanese giant looper（Ascotis selenaria）、オオモンシロチョウLarge white（Pieris brassicae）、モンシロチョウCabbage white butterfly（Pieris rapae crucivora）、イチモンジセセリStraight swift（Parnara guttata）、コットンリーフワームcotton leafworm (Alabama argillacea)、サトウキビメイガsugarcane borer（Diatraea sacharalis）等の鱗翅目（Lepidoptera）昆虫、
ウリミバエMelon fly（Bactrocera cucurbitae）、ミカンコミバエOriental fruit fly（Bactrocera dorsalis）、クイーンズランドミバエQueensland fruit fly（Bactrocera tryoni）、ミカンバエJapanese orange fly（Bactrocera tsuneonis）、チチュウカイミバエMediterranean fruit fly（Ceratitis capitata）、メキシコミバエMexican fruit fly（Anastrepha ludens）、リンゴミバエApple maggot（Rhagoletis pomonella）、イネハモグリバエRice leaf miner（Agromyza oryzae）、ナモグリバエPea leaf miner（Chromatomyia horticola）、アブラナハモグリバエCabbage leafminer（Liriomyza brassicae）、ナスハモグリバエTomato leaf miner（Liriomyza bryoniae）、ネギハモグリバエStone leek leafminer（Liriomyza chinensis）、アシグロハモグリバエPea leafminer（Liriomyza huidobrensis）、トマトハモグリバエTomato leafminer（Liriomyza sativae）、マメハモグリバエSerpentine leafminer（Liriomyza trifolii）、オウトウショウジョウバエJapanese fruit fly（Drosophila suzukii）、イネヒメハモグリバエSmaller rice leaf miner（Hydrellia griseola）、ツェツェバエTsetse fly（Glossina morsitans, G. palpalis）、ウマシラミバエForest fly（Hippobosca equina）、ヒツジシラミバエSheep ked（Melophagus ovinus）、タマネギバエOnion fly（Delia antiqua）、タネバエSeed corn maggot（Delia platura）、テンサイモグリハナバエBeet leaf miner（Pegomya cunicularia）、ヒメイエバエLesser house fly（Fannia canicularis）、シープヘッドフライSheep headfly（Hydrotaea irritans）、スウィートフライSweat fly（Morellia simplex）、フェイスフライFace fly（Musca autumnalis）、イエバエHousefly（Musca domestica）、オーストラリアブッシュフライAustralian bush fly（Musca vetustissima）、ノサシバエHorn fly（Haematobia irritans）、サシバエStable fly（Stomoxys calcitrans）、オオクロバエ（Calliphora lata）、ホホアカクロバエBottle fly（Calliphora vicina）、旧世界ラセンウジバエOld World screw-worm fly（Chrysomya bezziana）、ブロウフライBlow fly（Chrysomya chloropyga）、オビキンバエOriental latrine fly（Chrysomya megacephala）、アメリカオビキンバエNew World screw-worm fly（Cochliomyia hominivorax）、クロキンバエBlack blow fly（Phormia regina）、ルリキンバエNorthern blowfly（Protophormia terraenovae）、ヒツジキンバエAustralian sheep blowfly（Lucilia cuprina）、ミドリキンバエGreen bottle fly（Lucilia illustris）、ヒロズキンバエCommon green bottle fly（Lucilia sericata）、ボットフライBot flies（Cuterebra spp.）、ヒトヒフバエHuman botfly（Dermatobia hominis）、アトアカウマバエHorse nose bot fly（Gasterophilus haemorrhoidalis）、ウマバエHorse bot fly（Gasterophilus intestinalis）、アカウマバエThroat bot fly（Gasterophilus nasalis）、ウシヒフバエWarble fly（Hypoderma bovis）、キスジウシバエCommon cattle grub（Hypoderma lineatum）、ヒツジバエSheep nasal bot fly（Oestrus ovis）、フレッシュフライFlesh fly（Sarcophaga carnaria）、センチニクバエFlesh fly（Sarcophaga peregrina）、スプレイドディアーフライSplayed deerfly（Chrysops caecutiens）、メクラアブDeer fly（Chrysops suavis）、コモンホースフライCommon horse fly（Haematopota pluvialis）、グリーンヘッドホースフライGreenhead horse fly（Tabanus nigrovittatus）、ウシアブHorse fly（Tabanus trigonus）、ダイズサヤタマバエSoybean pod gall midge（Asphondylia yushimai）、ヘシアンバエHessian fly（Mayetiola destructor）、ムギアカタマバエOrange wheat blossom midge（Sitodiplosis mosellana）、ニワトリヌカカBiting midge（Culicoides arakawae）、トクナガクロヌカカBlack gnat（Leptoconops nipponensis）、キアシオオブユ（Prosimulium yezoensis）、ブラックフライBlack fly（Simulium ochraceum）、ガンビエハマダラカAfrican malaria mosquito（Anopheles gambiae）、シナハマダラカ（Anopheles hyrcanus sinesis）、オオツルハマダラカ（Anopheles lesteri）、ネッタイシマカYellow fever mosquito（Aedes aegypti）、ヒトスジシマカAsian tiger mosquito（Aedes albopictus）、チカイエカHouse mosquito（Culex pipiens molestus）、アカイエカHouse mosquito（Culex pipiens pallens）、コガタアカイエカ（Culex tritaeniorhynchus）、サシチョウバエSandfly（Phlebotomus spp.）、オオチョウバエMoth fly（Telmatoscopus albipunctatus）等の双翅目（Diptera）昆虫、
ニワトリノミHen flea（Ceratophyllus gallinae)、スナノミChigoe flea（Tunga penetrans)、イヌノミDog flea（Ctenocephalides canis)、ネコノミCat flea（Ctenocephalides felis）、ニワトリフトノミSticktight flea（Echidnophaga gallinacea)、ヒトノミHuman flea（Pulex irritans）、ケオプスネズミノミOriental rat flea（Xenopsylla cheopis）等の隠翅目（Siphonaptera）昆虫、
タバコシバンムシTobacco beetle（Lasioderma serricorne）、インゲンマメゾウムシCommon bean weevil（Acanthoscelides obtectus）、アズキゾウムシAdzuki bean beetle（Callosobruchus chinensis）、ブドウトラカミキリGrape borer（Xylotrechus pyrrhoderus）、ツヤハダゴマダラカミキリAsian long-horn beetle（Anoplophora glabripennis）、ゴマダラカミキリWhite-spotted longicorn beetle（Anoplophora malasiaca）、マツノマダラカミキリJapanese pine sawyer（Monochamus alternatus）、キボシカミキリYellow-spotted longicorn beetle（Psacothea hilaris）、コロラドハムシColorado potato beetle（Leptinotarsa decemlineata）、マスタードリーフビートルMustard leaf beetle（Phaedon cochleariae）、イネドロオイムシRice leaf beetle（Oulema oryzae）、マダラカサハラハムシReaf beetle（Demotina fasciculata）、ウリハムシCucurbit leaf beetle（Aulacophora femoralis）、テンサイトビハムシBeet flea beetle（Chaetocnema concinna）、ノーザンコーンルートワームNorthern corn rootworm（Diabrotica barberi）、ジュウイチホシウリハムシSouthern corn rootworm（Diabrotica undecimpunctata）、ウエスタンコーンルートワームWestern corn rootworm（Diabrotica virgifera）、キスジノミハムシStriped flea beetle（Phyllotreta striolata）、ナスナガスネトビハムシSolanum flea beetle（Psylliodes angusticollis）、インゲンテントウMexican been beetle（Epilachna varivestis）、オオニジュウヤホシテントウLarge twenty-eight-spotted ladybird（Epilachna vigintioctomaculata）、ニジュウヤホシテントウTwentyeight-spotted ladybird（Epilachna vigintioctopunctata）、ヒメヒラタケシキスイ（Epuraea domina）、ポーレンビートルPollen beetle（Meligethes aeneus）、モモチョッキリゾウムシPeach curculio（Rhynchites heros）、アリモドキゾウムシSweetpotato weevil（Cylas formicarius）、イモゾウムシWest Indian sweet potato weevil（Euscepes postfasciatus）、ワタミゾウムシBoll weevil（Anthonomus grandis）、シロヘリクチブトゾウムシWhite-fringed beetle（Graphognatus leucoloma）、キンケクチブトゾウムシBlack vine weevil（Otiorhynchus sulcatus）、アルファルファタコゾウムシAlfalfa weevil（Hypera postica）、グラナリアコクゾウGranary weevil（Sitophilus granarius）、コクゾウムシMaize weevil（Sitophilus zeamais）、シバオサゾウムシHunting billbug（Sphenophorus venatus vestitus）、イネゾウムシRice plant weevil（Echinocnemus squameus）、イネミズゾウムシRice water weevil（Lissohoptrus oryzophilus）、チャイロコメノゴミムシダマシYellow mealworm（Tenebrio molitor）、コクヌストモドキRed flour beetle（Tribolium castaneum）、マルクビクシコメツキSweetpotato wireworm（Melanotus fortnumi）、カンシャクシコメツキSugarcane wireworm（Melanotus tamsuyensis）、コアオハナムグリCitrus flower chafer（Gametis jucunda）、ナガチャコガネYellowish elongate chafer（Heptophylla picea）、ドウガネブイブイCupreous chafer（Anomala cuprea）、ヒメコガネSoybean beetle（Anomala rufocuprea）、マメコガネJapanese beetle（Popillia japonica）、アオバアリガタハネカクシRove beetle（Paederus fuscipes）等の鞘翅目（Coleoptera）昆虫、
ミカンキジラミAsian citrus psyllid（Diaphorina citri）、ナシキジラミPear sucker（Psylla pyrisuga）、チャトゲコナジラミCamellia spiny whitefly（Aleurocanthus camelliae）、ミカントゲコナジラミOrange spiny whitefly（Aleurocanthus spiniferus）、シルバーリーフコナジラミSilverleaf whitefly（Bemisia argentifolii）、タバココナジラミSweetpotato whitefly（Bemisia tabaci）、ミカンコナジラミCitrus whitefly（Dialeurodes citri）、オンシツコナジラミGreenhouse whitefly（Trialeurodes vaporariorum）、エンドウヒゲナガアブラムシPea aphid（Acyrthosiphon pisum）、マメアブラムシCowpea aphid（Aphis craccivora）、マメクロアブラムシBlack bean aphid（Aphis fabae）、ダイズアブラムシSoybean aphid（Aphis glycines）、ワタアブラムシCotton aphid（Aphis gossypii）、リンゴアブラムシGreen apple aphid（Aphis pomi）、ユキヤナギアブラムシSpiraea aphid（Aphis spiraecola）、ジャガイモヒゲナガアブラムシFoxglove aphid（Aulacorthum solani）、ムギワラギクオマルアブラムシLeafcurl plum aphid（Brachycaudus helichrysi）、ダイコンアブラムシCabbage aphid（Brevicoryne brassicae）、ウォールナットアフィッドWalnut aphid（Chromaphis juglandicola）、ロシアンウィートアフィッドRussian wheat aphid（Diuraphis noxia）、オオバコアブラムシRosy apple aphid（Dysaphis plantaginea）、モモコフキアブラムシMealy plum aphid（Hyalopterus pruni）、ニセダイコンアブラムシTurnip aphid（Lipaphis erysimi）、チューリップヒゲナガアブラムシPotato aphid（Macrosiphum euphorbiae）、ブラックマージンドアフィッドBlackmargined aphid（Monellia caryella）、モモアカアブラムシGreen peach aphid（Myzus persicae）、レタスヒゲナガアブラムシLettuce aphid（Nasonovia ribisnigri）、ネギアブラムシOnion aphid（Neotoxoptera formosana）、ムギクビレアブラムシBird cherry-oat aphid（Rhopalosiphum padi）、オカボノアカアブラムシRice root aphid（Rhopalosiphum rufiabdominalis）、ムギヒゲナガアブラムシCorn leaf aphid（Sitobion akebiae）、イングリッシュグレインアフィッドEnglish grain aphid（Sitobion avenae）、ムギミドリアブラムシGreenbug（Schizaphis graminum）、コミカンアブラムシBlack citrus aphid（Toxoptera aurantii）、ミカンクロアブラムシBrown citrus aphid（Toxoptera citricida）、リンゴワタムシWooly apple aphid（Eriosoma lanigerum）、ブドウネアブラムシGrape phylloxera（Viteus vitifolii）、ツノロウムシIndian wax scale（Ceroplastes ceriferus）、ルビーロウムシRed wax scale（Ceroplastes rubens）、カンキツカタカイガラムシCitricola scale（Coccus pseudomagnoliarum）、アカマルカイガラムシCalifornia red scale（Aonidiella aurantii）、ナシマルカイガラムシSan jose scale（Comstockaspis perniciosa）、チャコノハカイガラムシTea scale（Fiorinia theae）、チャノマルカイガラムシPeony scale（Pseudaonidia paeoniae）、クワシロカイガラムシMulberry scale（Pseudaulacaspis pentagona）、ウメシロカイガラムシWhite peach scale（Pseudaulacaspis prunicola）、ニセヤノネカイガラムシCitrus snow scale（Unaspis citri）、マサキナガカイガラムシEuonymus scale（Unaspis euonymi）、ヤノネカイガラムシArrowhead scale（Unaspis yanonensis）、オオワラジカイガラムシGiant margarodid scale（Drosicha corpulenta）、イセリアカイガラムシCottony cushion scale（Icerya purchasi）、ナスコナカイガラムシCotton mealy bug（Phenacoccus solani）、ミカンコナカイガラムシCitrus mealybug（Planococcus citri）、フジコナカイガラムシJapanese mealybug（Planococcus kuraunhiae）、クワコナカイガラムシComstock mealybug（Pseudococcus comstocki）、グレープミールバグGrape mealybug（Pseudococcus maritimus）、ヒメトビウンカSmall brown planthopper（Laodelphax striatella）、トビイロウンカBrown rice planthopper（Nilaparvata lugens）、セジロウンカWhite-backed rice planthopper（Sogatella furcifera）、フタテンオオヨコバイGrape Leafhopper（Epiacanthus stramineus）、インディアンコットンリーフホッパーIndian cotton leafhopper（Amrasca devastans）、ミドリナガヨコバイBeardsley leafhopper（Balclutha saltuella）、フタテンヨコバイAster leafhopper（Macrosteles fascifrons）、ヒメフタテンヨコバイ（Macrosteles striifrons）、ツマグロヨコバイGreen rice leafhopper（Nephotettix cincticeps）、フタテンヒメヨコバイGrape Leafhopper（Arboridia apicalis）、ポテトリーフホッパーPotato Leafhopper（Empoasca fabae）、カキノヒメヨコバイ（Empoasca nipponica）、チャノミドリヒメヨコバイTea green leafhopper（Empoasca onukii）、マメノミドリヒメヨコバイBean's smaller green leafhopper（Empoasca sakaii）、ブチヒゲカメムシSloe bug（Dolycoris baccarum）、ナガメCabbage bug（Eurydema rugosa）、トゲシラホシカメムシWhitespotted spined bug（Eysarcoris aeneus）、オオトゲシラホシカメムシ（Eysarcoris lewisi）、シラホシカメムシWhite-spotted stink bug（Eysarcoris ventralis）、ツヤアオカメムシSheild bug（Glaucias subpunctatus）、クサギカメムシBrown marmorated stink bug（Halyomorpha halys）、アオクサカメムシEastern green stink bug（Nezara antennata）、ミナミアオカメムシSouthern green stink bug（Nezara viridula）、レッドバンディドスティンクバグRedbanded stink bug（Piezodorus guildinii）、イチモンジカメムシRedbanded shield bug（Piezodorus hybneri）、チャバネアオカメムシBrown-winged green bug（Plautia crossota）、イネクロカメムシJapanese black rice bug（Scotinophora lurida）、ホソヘリカメムシBean bug（Riptortus clavatus）、クモヘリカメムシRice bug（Leptocorisa chinensis）、ホソハリカメムシRice stink bug（Cletus punctiger）、ミナミトゲヘリカメムシSquash bug（Paradasynus spinosus）、アカヒメヘリカメムシRhopalid bug（Rhopalus maculatus）、アメリカコバネナガカメムシTrue chinch bug（Blissus leucopterus）、カンシャコバネナガカメムシOriental chinch bug（Cavelerius saccharivorus）、コバネヒョウタンナガカメムシSeed bug（Togo hemipterus）、アカホシカメムシRed cotton bug（Dysdercus cingulatus）、ベネズエラサシガメBlood-sucking bug（Rhodnius prolixus）、メキシコサシガメKissing bug（Triatoma dimidiata）、ブラジルサシガメKissing bug（Triatoma infestans）、グリーンスティンクバッグgreen stink bug (Acrosternum hilare)、ブロウンスティンクバッグbrown stink bug (Euschistus servus)、サウザングリーンスティンクバッグsouthern green stink bug (Nezara viridula)、ターニッシュプラントバッグTarnished plant bug (Lygus lineolaris)、スティンクバッグ（Dichelops furcatus）、シュガーカンスピットルバッグsugarcane spittlebug (Mahanarva fimbriolata)、ツツジグンバイAzalea lace bug（Stephanitis pyrioides）、トコジラミBed bug（Cimex lectularius）、ツマグロアオカスミカメPale greenplant bug（Apolygus spinolae）、ウェスタンターニッシュドプラントバグWestern tarnished plant bug（Lygus hesperus）、サビイロカスミカメTarnished plant bug（Lygus lineolaris）、ナガムギカスミカメRice stink bug（Stenodema sibiricum）、アカスジカスミカメSorghum plant bug（Stenotus rubrovittatus）、イネホソミドリカスミカメRice leaf bug（Trigonotylus caelestialium）、クロトビカスミカメIsland fleahopper（Halticus insularis）、ワタノミハムシCotton fleahopper（Pseudatomoscelis seriatus）等の半翅目（Hemiptera）昆虫
ヒラズハナアザミウマFlower thrips（Frankliniella intonsa）、ミカンキイロアザミウマWestern flower thrips（Frankliniella occidentalis）、クロトンアザミウマGreenhouse thrips（Heliothrips haemorrhoidalis）、チャノキイロアザミウマYellow tea thrips（Scirtothrips dorsalis）、ミナミキイロアザミウマMelon thrips（Thrips palmi）、ネギアザミウマOnion thrips（Thrips tabaci）、カキクダアザミウマJapanese gall-forming thrips（Ponticulothrips diospyrosi）等の総翅目（Thysanoptera）昆虫、
ニワトリツノハジラミBody louse（Menacanthus cornutus）、ウスイロニワトリハジラミSmall body louse（Menacanthus pallidulus）、ニワトリオオハジラミChicken body louse（Menacanthus stramineus）、ニワトリハジラミChicken shaft louse（Menopon gallinae）、ハバビロナガハジラミChicken head louse（Cuclotogaster heterographa）、カクアゴハジラミBrown chicken louse（Goniodes dissmilis）、ヒメニワトリハジラミFluff louse（Goniodes gallinae）、マルハジラミLarge hen louse（Goniodes gigas）、ニワトリナガハジラミWing louse（Lipeurus caponis）、ウシハジラミCattle chewing louse（Damalinia bovis）、ネコハジラミCat louse（Felicola subrostrata）、イヌハジラミDog biting louse（Trichodectes canis）、ウシジラミShort-nosed cattle louse（Haematopinus eurysternus）、ウシジラミTail switch louse（Haematopinus quadripertusus）、ブタジラミLarge pig louse（Haematopinus suis）、スイギュウジラミBuffalo louse（Haematopinus tuberculatus）、イヌジラミDog sucking louse（Linognathus setosus）、ウシホソジラミLong-nosed cattle louse（Linognathus vituri）、ラビットロウズRabbit louse（Haemodipsus ventricosus）、ケブカウシジラミLittle blue cattle louse（Solenopotes capillatus）、ヒトジラミHead louse（Pediculus humanus）、ハツカネズミジラミMouse louse（Polyplax serratus）、ケジラミCrab louse（Pthirus pubis）等の咀顎目（Psocodea）昆虫、
サバクトビバッタDesert locust（Schistocerca gregaria）、オーストラリアトビバッタAustralian plague locust（Chortoicetes terminifera）、トノサマバッタMigratory locust（Locusta migratoria）、ハネナガイナゴLesser paddy grasshopper（Oxya japonica）、コバネイナゴRice grasshopper（Oxya yezoensis）、エンマコオロギEmma field cricket（Teleogryllus emma）、ケラOriental mole cricket（Gryllotalpa orientalis）等の直翅目（Orthoptera）昆虫、
チャバネゴキブリGerman cockroach（Blattella germanica）、ワモンゴキブリAmerican cockroach（Periplaneta americana）、クロゴキブリSmoky-brown cockroach（Periplaneta fuliginosa）、ヤマトゴキブリJapanese cockroach（Periplaneta japonica）、ダイコクシロアリDaikoku dry-wood termite（Cryptotermes domesticus）、アメリカカンザイシロアリWestern dry-wood termite（Incisitermes minor）、イエシロアリFormosan subterranean termite（Coptotermes formosanus）、ヤマトシロアリJapanese subterranean termite（Reticulitermes speratus）、タイワンシロアリBlack-winged subterranean termite（Odontotermes formosanus）等の網翅目（Dictyoptera）昆虫、
トゲナシシロトビムシRootfeeding springtail（Onychiurus folsomi）、シベリアシロトビムシ（Onychiurus sibiricus）、キボシマルトビムシGarden springtail（Bourletiella hortensis）等の粘管目（Collembola）六脚類、
オカダンゴムシPill bug（Armadillidium vulgare）、ワラジムシCommon rough woodlouse（Porcellio scaber）等の等脚目（Isopoda）甲殻類、
チョウモドキ（Argulus coregoni）、チョウJapanese fishlouse（Argulus japonicus）、ウミチョウ（Argulus scutiformis）等のチョウ目（Arguloida）甲殻類、
ウオジラミSea louse（Caligus curtus, C. elongatus）、サーモンローズSalmon louse（Lepeophtheirus salmonis）等のシフォノストム目（Siphonostomatoida）甲殻類、
サヤアシニクダニStorage mite（Glycyphagus destructor）、イエニクダニHouse itch mite（Glycyphagus domesticus）、ムギコナダニBrown-legged grain mite（Aleuroglyphus ovatus）、ケナガコナダニCheese mite（Tyrophagus putrescentiae）、ホウレンソウケナガコナダニ（Tyrophagus similis）、ロビンネダニBulb mite（Rhizoglyphus robini）、ヒシガタウモウダニFeather mite（Pterolichus obtusus）、ニワトリウモウダニFeather mite（Megninia cubitalis）、コナヒョウヒダニAmerican house dust mite（Dermatophagoides farinae）、ヤケヒョウヒダニHouse dust mite（Dermatophagoides pteronyssinus）、ウシショクヒヒゼンダニChorioptic mange mite（Chorioptes bovis）、イヌミミヒゼンダニDog ear mite（Otodectes cynotis）、ウシキュウセンヒゼンダニPsoroptic mite（Psoroptes communis）、ウサギキュウセンヒゼンダニRabbit ear mite（Psoroptes cuniculi）、ヒツジキュウセンヒゼンダニSheep scab mite（Psoroptes ovis）、センコウヒゼンダニItch mite（Sarcoptes scabiei）、ネコショウセンコウヒゼンダニCat mange mite（Notoedres cati）等のコナダニ亜目（Astigmata）ダニ類、
イエササラダニ（Haplochthonius simplex）等のササラダニ亜目（Oribatida）ダニ類、
ミナミツメダニ（Chelacaropsis moorei）、ネコツメダニ（Cheyletiella blakei）、ウサギツメダニRabbit fur mite（Cheyletiella parasitovorax）、イヌツメダニ（Cheyletiella yasguri）、ホソツメダニ（Cheyletus eruditus）、クワガタツメダニ（Cheyletus malaccensis）、イヌニキビダニDog follicle mite（Demodex canis）、ネコニキビダニCat follicle mite（Demodex cati）、ニキビダニFace mite（Demodex folliculorum）、チューリップサビダニWheat curl mite（Aceria tulipae）、ニセナシサビダニPear rust mite（Eriophyes chibaensis）、ピーチバドマイトPeach bud mite（Eriophyes insidiosus）、ペアリーフブリスターマイトPearleaf blister mite（Eriophyes pyri）、チャノナガサビダニTea rust mite（Acaphylla theavagrans）、トマトサビダニTomato russet mite（Aculops lycopersici）、ミカンサビダニPink citrus rust mite（Aculops pelekassi）、リンゴサビダニApple rust mite（Aculus schlechtendali）、シトラスラストマイトCitrus rust mite（Phyllocoptruta oleivora）、チャノホコリダニBroad mite（Polyphagotarsonemus latus）、シクラメンホコリダニCyclamen mite（Phytonemus pallidus）、スジブトホコリダニTarsonemid mite（Tarsonemus bilobatus）、イネハダニ（Oligonychus shinkajii）、ミカンハダニCitrus red mite（Panonychus citri）、クワオオハダニSpider mite（Panonychus mori）、リンゴハダニEuropean red mite（Panonychus ulmi）、カンザワハダニKanzawa spider mite（Tetranychus kanzawai）、ナミハダニTwo-spotted spider mite（Tetranychus urticae）、ハクサイダニ（Penthaleus erythrocephalus）、ムギダニWinter grain mite（Penthaleus major）、ナンヨウツツガムシ（Eutrombicula wichmanni）、ミヤガワタマツツガムシTrombiculid mite（Helenicula miyagawai）、アカツツガムシ（Leptotrombidium akamushi）、フトゲツツガムシ（Leptotrombidium pallida）、タテツツガムシTsutsugamushi mite（Leptotrombidium scutellare）等のケダニ亜目（Prostigmata）ダニ類、
イングリッシュファウルティックEnglish fowl tick（Argas persicus）、カズキダニSoft tick（Ornithodoros moubata）、回帰熱ティックRelapsing fever tick（Ornithodoros turicata）、スピノウズイヤーティックSpinose ear tick（Otobius megnini）、ローン・スターマダニLone star tick（Amblyomma americanum）、メキシコ湾岸マダニGulf coast tick（Amblyomma maculatum）、ツリガネチマダニ（Haemaphysalis campanulata）、キチマダニ（Haemaphysalis flava）、フタトゲチマダニBush tick（Haemaphysalis longicornis）、オオトゲチマダニ（Haemaphysalis megaspinosa）、トルトイスティックTortoise tick（Hyalomma aegyptium）、メディトレニアンティックMediterranean tick（Hyalomma marginatum）、オウシマダニTropical cattle tick（Boophilus microplus）、タネガタマダニ（Ixodes nipponensis）、ヤマトマダニ（Ixodes ovatus）、西部クロアシダニWestern black-legged tick（Ixodes pacifcus）、シュルツェマダニTaiga tick（Ixodes persulcatus）、ヒツジダニCastor bean tick（Ixodes ricinus）、クロアシダニBlack-legged tick（Ixodes scapularis）、トロピカルホースティックTropical horse tick（Anocentor nitens）、ロッキー山脈森林マダニRocky Mountain wood tick（Dermacentor andersoni）、西海岸マダニPacific Coast tick（Dermacentor occidentalis）、アミメカクマダニOrnate cow tick（Dermacentor reticulatus）、アメリカンドッグティックAmerican dog tick（Dermacentor variabilis）、リピセントール属（Rhipicentor spp.）、アメリカンキャトルティックAmerican cattle tick（Rhipicephalus annulatus）、クリイロコイタマダニBrown dog tick（Rhipicephalus sanguineus）等のマダニ亜目（Metastigmata）ダニ類、
ワクモRed mite（Dermanyssus gallinae）、イエダニTropical rat mite（Ornithonyssus bacoti）、トリサシダニNorthern fowl mite（Ornithonyssus sylviarum）、ハニービーマイトHoneybee mite（Varroa destructor）、ミツバチヘギイタダニVarroa mite（Varroa jacobsoni）等のトゲダニ亜目（Mesostigmata）ダニ類、
スクミリンゴガイApple snail（Pomacea canaliculata）等の盤足目（Architaenioglossa）腹足類、
アフリカマイマイGiant African snail（Achatina fulica）、チャコウラナメクジTerrestrial slug（Limax marginatus）、ナメクジSlug（Meghimatium bilineatum）、ウスカワマイマイKorean round snail（Acusta despecta sieboldiana）、ミスジマイマイLand snail（Euhadra peliomphala）等のマイマイ目（Stylommatophora）腹足類、
腎虫Giant kidney worm（Dioctophyma renale）、有環毛細線虫Thread worms（Capillaria annulata）、捻転毛細線虫Cropworm（Capillaria contorta）、肝毛細線虫Capillary liver worm（Capillaria hepatica）、穿通毛細線虫（Capillaria perforans）、フィリピン毛細線虫（Capillaria philippinensis）、豚毛細線虫（Capillaria suis）、牛鞭虫Whipworm（Trichuris discolor）、羊鞭虫Whipworm（Trichuris ovis）、豚鞭虫Pig whipworm（Trichuris suis）、ヒト鞭虫Human whipworm（Trichuris trichiura）、犬鞭虫Dog whipworm（Trichuris vulpis）、旋毛虫Pork worm（Trichinella spiralis）等のエノプルス目（Enoplida）線虫、
乳頭糞線虫Intestinal threadworm（Strongyloides papillosus）、猫糞線虫（Strongyloides planiceps）、豚糞線虫Pig threadworm（Strongyloides ransomi）、ヒト糞線虫Threadworm（Strongyloides stercoralis）、ミクロネマ属（Micronema spp.）等の桿線虫目（Rhabditida）線虫、
ブラジル鉤虫Hookworm（Ancylostoma braziliense）、犬鉤虫Dog hookworm（Ancylostoma caninum）、ズビニ鉤虫Old World hookworm（Ancylostoma duodenale）、猫鉤虫Cat hookworm（Ancylostoma tubaeforme）、狭頭鉤虫The Northern hookworm of dogs（Uncinaria stenocephala）、牛鉤虫Cattle hookworm（Bunostomum phlebotomum）、羊鉤虫Small ruminant hookworm（Bunostomum trigonocephalum）、アメリカ鉤虫New World hookworm（Necator americanus）、シアトストーマム属（Cyathostomum spp.）、シリコシクラス属（Cylicocyclus spp.）、シリコドントフォラス属（Cylicodontophorus spp.）、シリコステファナス属（Cylicostephanus spp.）、ロバ円虫（Strongylus asini）、無歯円虫（Strongylus edentatus）、馬円虫Blood worm（Strongylus equinus）、普通円虫Blood worm（Strongylus vulgaris）、羊縮小線虫Large-mouthed bowel worm（Chabertia ovina）、インド腸結節虫Nodular worm（Oesophagostomum brevicaudatum）、コロンビア腸結節虫Nodule worm（Oesophagostomum columbianum）、豚腸結節虫Nodule worm（Oesophagostomum dentatum）、アメリカ腸結節虫Nodular worm（Oesophagostomum georgianum）、腸結節虫Nodular worm（Oesophagostomum maplestonei）、豚盲結虫Nodular worm（Oesophagostomum quadrispinulatum）、牛腸結節虫Nodular worm（Oesophagostomum radiatum）、山羊腸結節虫Nodular worm（Oesophagostomum venulosum）、スクリジャビン開嘴虫（Syngamus skrjabinomorpha）、鶏開嘴虫Gapeworm（Syngamus trachea）、豚腎虫Swine kidney worm（Stephanurus dentatus）、クーペリアCattle bankrupt worm（Cooperia oncophora）、紅色毛様線虫Red stomach worm（Hyostrongylus rubidus）、皺胃毛様線虫Stomach hair worm（Trichostrongylus axei）、蛇状毛様線虫（Trichostrongylus colubriformis）、東洋毛様線虫Oriental trichostrongylus（Trichostrongylus orientalis）、捻転胃虫Red stomach worm（Haemonchus contortus）、牛捻転胃虫Cattle stomach worm（Mecistocirrus digitatus）、オステルターグ胃虫Brown stomach worm（Ostertagia ostertagi）、糸状肺虫Common lungworm（Dictyocaulus filaria）、牛肺虫Bovine lungworm（Dictyocaulus viviparus）、細頸毛円虫Thin-necked intestinal worm（Nematodirus filicollis）、豚肺虫Swine lungworm（Metastrongylus elongatus）、犬肺虫Lungworm（Filaroides hirthi）、肺毛細線虫Lungworm（Crenosoma aerophila）、キツネ肺虫Fox lungworm（Crenosoma vulpis）、広東住血線虫Rat lung worm（Angiostrongylus cantonensis）、住血線虫French heartworm（Angiostrongylus vasorum）、プロトストロンギラス属（Protostrongylus spp.）等の円虫目（Strongylida）線虫、
イネシンガレセンチュウRice white tip nematode（Aphelenchoides besseyi）、マツノザイセンチュウPine wood nematode（Bursaphelenchus xylophilus）等の葉線虫目（Aphelenchida）線虫、
ジャガイモシストセンチュウPotato cyst nematode（Globodera rostochiensis）、ムギシストセンチュウCereal cyst nematode（Heterodera avenae）、ダイズシストセンチュウSoybean cyst nematode（Heterodera glycines）、アレナリアネコブセンチュウPeanut root-knot nematode（Meloidogyne arenaria）、キタネコブセンチュウNorthern root-knot nematode（Meloidogyne hapla）、サツマイモネコブセンチュウSouthern root-knot nematode（Meloidogyne incognita）、ジャワネコブセンチュウJavanese root-knot nematode（Meloidogyne javanica）、ミナミネグサレセンチュウCoffee root-lesion nematode（Pratylenchus coffeae）、チャネグサレセンチュウTea root-lesion nematode（Pratylenchus loosi）、キタネグサレセンチュウCobb's root-lesion nematode（Pratylenchus penetrans）、クルミネグサレセンチュウWalnut root-lesion nematode（Pratylenchus vulnus）等のハリセンチュウ目（Tylenchida）線虫、
ヒト蟯虫Pinworm（Enterobius vermicularis）、馬蟯虫Equine pinworm（Oxyuris equi）、ウサギ蟯虫Rabbit pinworm（Passalurus ambiguus）等の蟯虫目（Oxyurida）線虫、
豚回虫Pig roundworm（Ascaris suum）、馬回虫Horse roundworm（Parascaris equorum）、犬小回虫Dog roundworm（Toxascaris leonina）、犬回虫Dog intestinal roundworm（Toxocara canis）、猫回虫Feline roundworm（Toxocara cati）、牛回虫Large cattle roundworm（Toxocara vitulorum）、アニサキス属（Anisakis spp.）、シュードテラノーバ属（Pseudoterranova spp.）、鶏盲腸虫Caecal worm（Heterakis gallinarum）、鶏回虫Chicken roundworm（Ascaridia galli）等の回虫目（Ascaridida）線虫、
メジナ虫Guinea worm（Dracunculus medinensis）、ドロレス顎口虫（Gnathostoma doloresi）、剛棘顎口虫（Gnathostoma hispidum）、日本顎口虫（Gnathostoma nipponicum）、有棘顎口虫Reddish‐coloured worm（Gnathostoma spinigerum）、犬胃虫Dog stomach worm（Physaloptera canis）、猫胃虫Cat stomach worm（Physaloptera felidis, P. praeputialis）、ラーラ胃虫Feline/canine stomach worm（Physaloptera rara）、東洋眼虫Eye worm（Thelazia callipaeda）、ロデシア眼虫Bovine eyeworm（Thelazia rhodesi）、大口馬胃虫Large mouth stomach worm（Draschia megastoma）、小口胃虫Equine stomach worm（Habronema microstoma）、ハエ胃虫Stomach worm（Habronema muscae）、美麗食道虫Gullet worm（Gongylonema pulchrum）、類円豚胃虫Thick stomach worm（Ascarops strongylina）、牛パラフィラリアParafilaria（Parafilaria bovicola）、多乳頭糸状虫（Parafilaria multipapillosa）、沖縄糸状虫（Stephanofilaria okinawaensis）、バンクロフト糸状虫Bancroft filaria（Wuchereria bancrofti）、マレー糸状虫（Brugia malayi）、頸部糸状虫Neck threadworm（Onchocerca cervicalis）、ギブソン糸状虫（Onchocerca gibsoni）、咽頭糸状虫Cattle filarial worm（Onchocerca gutturosa）、回旋糸状虫（Onchocerca volvulus）、指状糸状虫Bovine filarial worm（Setaria digitata）、馬糸状虫Peritoneal worm（Setaria equina）、唇乳頭糸状虫（Setaria labiatopapillosa）、マーシャル糸状虫（Setaria marshalli）、犬糸状虫Dog heartworm（Dirofilaria immitis）、ロア糸状虫African eye worm（Loa loa）等の旋尾線虫目（Spirurida）線虫、
鎖状鉤頭虫（Moniliformis moniliformis）、大鉤頭虫Giant thorny-headed worm（Macracanthorhynchus hirudinaceus）等の鉤頭虫類、
広節裂頭条虫Fish tapeworm（Diphyllobothrium latum）、日本海裂頭条虫（Diphyllobothrium nihonkaiense）、マンソン裂頭条虫Manson tapeworm（Spirometra erinaceieuropaei）、大複殖門条虫（Diplogonoporus grandis）等の擬葉目（Pseudophyllidea）条虫、
有線条虫（Mesocestoides lineatus）、有輪条虫Chicken tapeworm（Raillietina cesticillus）、棘溝条虫Fowl tapeworm（Raillietina echinobothrida）、方形条虫Chicken tapeworm（Raillietina tetragona）、胞状条虫Canine tapeworm（Taenia hydatigena）、多頭条虫Canine tapeworm（Taenia multiceps）、羊条虫Sheep measles（Taenia ovis）、豆状条虫Dog tapeworm（Taenia pisiformis）、無鉤条虫Beef tapeworm（Taenia saginata）、連節条虫Tapeworm（Taenia serialis）、有鉤条虫Pork tapeworm（Taenia solium）、猫条虫Feline tapeworm（Taenia taeniaeformis）、単包条虫Hydatid tapeworm（Echinococcus granulosus）、多包条虫Small fox tapeworm（Echinococcus multilocularis）、ヤマネコ包条虫（Echinococcus oligarthrus）、フォーゲル包条虫（Echinococcus vogeli）、縮小条虫Rat tapeworm（Hymenolepis diminuta）、小型条虫Dwarf tapeworm（Hymenolepis nana）、瓜実条虫Double-pored dog tapeworm（Dipylidium caninum）、楔状条虫（Amoebotaenia sphenoides）、漏斗状条虫（Choanotaenia infundibulum）、ウズラ条虫（Metroliasthes coturnix）、大条虫Equine tapeworm（Anoplocephala magna）、葉状条虫Cecal tapeworm（Anoplocephala perfoliata）、乳頭条虫Dwarf equine tapeworm（Paranoplocephala mamillana）、ベネデン条虫Common tapeworm（Moniezia benedeni）、拡張条虫Sheep tapeworm（Moniezia expansa）、スティレシア属（Stilesia spp.）等の円葉目（Cyclophyllidea）条虫、
壷型吸虫（Pharyngostomum cordatum）、ビルハルツ住血吸虫Blood fluke（Schistosoma haematobium）、日本住血吸虫Blood fluke（Schistosoma japonicum）、マンソン住血吸虫Blood fluke（Schistosoma mansoni）等の有壁吸虫目（Strigeidida）吸虫、
移睾棘口吸虫（Echinostoma cinetorchis）、浅田棘口吸虫（Echinostoma hortense）、巨大肝蛭Giant liver fluke（Fasciola gigantica）、肝蛭Common liver fluke（Fasciola hepatica）、肥大吸虫（Fasciolopsis buski）、平腹双口吸虫（Homalogaster paloniae）等の棘口吸虫目（Echinostomida）吸虫、
大陸槍型吸虫（Dicrocoelium chinensis）、槍型吸虫Lancet liver fluke（Dicrocoelium dendriticum）、アフリカ槍型吸虫African lancet fluke（Dicrocoelium hospes）、小型膵蛭（Eurytrema coelomaticum）、膵蛭Pancreatic fluke（Eurytrema pancreaticum）、宮崎肺吸虫（Paragonimus miyazakii）、大平肺吸虫（Paragonimus ohirai）、ウエステルマン肺吸虫Lung fluke（Paragonimus westermani）等の斜睾吸虫目（Plagiorchiida）吸虫、
アンフィメルス属（Amphimerus spp.）、肝吸虫Chinese liver fluke（Clonorchis sinensis）、猫肝吸虫Cat liver fluke（Opisthorchis felineus）、タイ肝吸虫Southeast Aasian liver fluke（Opisthorchis viverrini）、シュードアンフィストーマム属（Pseudamphistomum spp.）、メトロキス属（Metorchis spp.）、パラメトロキス属（Parametorchis spp.）、異形吸虫Intestinal fluke（Heterophyes heterophyes）、横川吸虫（Metagonimus yokokawai）、前腸異形吸虫（Pygidiopsis summa）等の後睾吸虫目（Opisthorchiida）吸虫、
赤痢アメーバ（Entamoeba histolytica, E. invadens）等のアメーバ類、
フタゴバベシア（Babesia bigemina）、牛バベシア（Babesia bovis）、大形馬バベシア（Babesia caballi）、犬バベシア（Babesia canis）、猫バベシア（Babesia felis）、ギブソン犬バベシア（Babesia gibsoni）、大型ピロプラズマ（Babesia ovata）、サイタウクスゾーン・フェリス（Cytauxzoon felis）、熱帯ピロプラズマ病タイレリア（Theileria annulata）、仮性沿岸熱タイレリア（Theileria mutans）、小型ピロプラズマ（Theileria orientalis）、東沿岸熱タイレリア（Theileria parva）等のピロプラズマ目（Piroplasmida）胞子虫類、
ヘモプロテウス・マンソニ（Haemoproteus mansoni）、鶏ロイコチトゾーン（Leucocytozoon caulleryi）、熱帯熱マラリア原虫（Plasmodium falciparum）、四日熱マラリア原虫（Plasmodium malariae）、卵形マラリア原虫（Plasmodium ovale）、三日熱マラリア原虫（Plasmodium vivax）等の住血胞子虫目（Haemosporida）胞子虫類、
カリオスポラ属（Caryospora spp.）、エイメリア・アセルブリナ（Eimeria acervulina）、エイメリア・ボビス（Eimeria bovis）、エイメリア・ブルネッチ（Eimeria brunetti）、エイメリア・マクシマ（Eimeria maxima）、エイメリア・ネカトリクス（Eimeria necatrix）、エイメリア・オビノイダリス（Eimeria ovinoidalis）、ウサギ肝コクシジウム（Eimeria stiedae）、鶏盲腸コクシジウム（Eimeria tenella）、犬イソスポーラ（Isospora canis）、猫イソスポーラ（Isospora felis）、豚イソスポーラ（Isospora suis）、ティゼリア・アレニ（Tyzzeria alleni）、ティゼリア・アンセリス（Tyzzeria anseris）、ティゼリア・パーニシオサ（Tyzzeria perniciosa）、ウェニョネラ・アナティス（Wenyonella anatis）、ウェニョネラ・ガガリ（Wenyonella gagari）、犬クリプトスポリジウム（Cryptosporidium canis）、猫クリプトスポリジウム（Cryptosporidium felis）、ヒトクリプトスポリジウム（Cryptosporidium hominis）、シチメンチョウクリプトスポリジウム（Cryptosporidium meleagridis）、ネズミクリプトスポリジウム（Cryptosporidium muris）、小形クリプトスポリジウム（Cryptosporidium parvum）、サルコシスチス・カニス（Sarcocystis canis）、クルーズ肉胞子虫（Sarcocystis cruzi）、サルコシスチス・フェリス（Sarcocystis felis）、ヒト肉胞子虫（Sarcocystis hominis）、サルコシスチス・ミーシェリアナ（Sarcocystis miescheriana）、サルコシスチス・ニューロナ（Sarcocystis neurona）、サルコシスチス・テネラ（Sarcocystis tenella）、サルコシスチス・オバリス（Sarcocystis ovalis）、トキソプラズマ（Toxoplasma gondii）、犬ヘパトゾーン（Hepatozoon canis）、猫ヘパトゾーン（Hepatozoon felis）等の真コクシジウム目（Eucoccidiorida）胞子虫類、
大腸バランチジウム（Balantidium coli）等の前庭目（Vestibuliferida）繊毛虫類、
ヒストモナス（Histomanas meleagridis）、腸トリコモナス（Pentatrichomonas hominis）、口腔トリコモナス（Trichomonas tenax）等のトリコモナス目（Trichomonadida）鞭毛虫類、
ランブル鞭毛虫（Giardia intestinalis）、ジアルディア・ムリス（Giardia muris）、シチメンチョウヘキサミタ（Hexamita meleagridis）、ヘキサミタ・パルバ（Hexamita parva）等のディプロモナス目（Diplomonadida）鞭毛虫類、
ドノバンリーシュマニア（Leishmania donovani）、幼児リーシュマニア（Leishmania infantum）、大形リーシュマニア（Leishmania major）、熱帯リーシュマニア（Leishmania tropica）、ガンビアトリパノソーマ（Trypanosoma brucei gambiense）、ローデシアトリパノソーマ（Trypanosoma brucei rhodesiense）、クルーズトリパノソーマ（Trypanosoma cruzi）、媾疫トリパノソーマ（Trypanosoma equiperdum）、エバンストリパノソーマ（Trypanosoma evansi）等のキネトプラスト目（Kinetoplastida）鞭毛虫類、
等が挙げられるが、本発明化合物を用いて防除しうる農園芸分野の有害生物及び家畜、家禽、愛玩動物等の外部又は内部寄生虫はこれらのみに限定されるものではない。 Specific examples of insects, mites, crustaceans, molluscs and nematodes that can be controlled using the compounds of the present invention include:
Chestnut gall wasp (Dryocosmus kuriphilus), Argentine ant Argentine ant (Linepithema humile), Gantai ant Army ant (Eciton burchelli, E. schmitti), Japanese carpenter ant (Camponotus japonicus), Yhihara ant Mona Pharaohant Bulldog ant (Myrmecia spp.), Fire Ant (Solenopsis spp.), Asian giant hornet (Vespa mandarina), Japanese yellow hornet (Vespa simillima), Large-ranged bee Large rose sawfly (Arge pagana) Hymenoptera insects such as pine sawfly (Neodiprion sertifer), chestnut wasp Chestnut sawfly (Apethymus kuri), sedge bee wasp Cabbage sawfly (Athalia infumata), bee turnip sawfly (Athalia rosae),
Pear leaf miner (Bucculatrix pyrivorella), tea leaf roller (Caloptilia theivora), golden leaf soy Apple leafminer (Phyllonorycter ringoniella), citrus leafminer (Phyllocnistis citrella), immobilized leaflet Persimmon fruit moth (Stathmopoda masinissa), Peach fruit moth (Carposina sasakii), Allium leafminer (Acrolepiopsis sapporensis), Yami leafminer (Acrolepiopsis suzukiella), Peach fruit moth (Pel fruit) ), Diamondback moth (Plutella xylostella), red stem borer (Chilo suppressalis), Shibatatsuga Bluegrass webworm (Parapediasia teterrella) Cabbage webworm (Hellula undalis), Rice leaf roller (Cnaphalocrocis medinalis), Yellow moth moth (Conogethes punctiferalis), Cotton moth (Diaphania indica), Mulberry pyras (Mulberry pyras) Ostrinia furnacalis), European corn borer (Ostrinia nubilalis), Azuki bean borer (Ostrinia scapulalis), Sorghum moth Lesser corn stalk borer (Elasmopalpus lignosellus), ella borer L Tree borer Peach tree borer (Synanthedon exitiosa), Cosca Shiba Cherry tree borer (Synanthedon hector), Kubiakasukashiba (Toleria romanovi), Iraga Oriental moth (Monema flavescens), Aura Iga (Parasa consocia), Hiloheira Oiraga (Parasa) lepida), Parasa siniea, Parana siniea, Artona martini, Illiberis pruni, Illiberis rotundata, Carpenter moth (Cossus insularis), Codlingmon lum, Cydia Fruit moth (Grapholita dimorpha), Oriental fruit moth (Grapholita molesta), Bean pod borer (Leguminivora glycinivorella), Bean podworm (Matsumuraeses phaseoli), Grapeberry moss (Grape berryite moth) Smaller tea tortrix (Adoxophyes honmai), Apple coconut oyster Summer fruit tortrix (Adoxophyes orana fasciata), Apple peach oyster Asiatic leafroller (Archips breviplicanus), Midareka kumamaki Apple tortrix (Archips fuscocupreanus) Oriental tea tortrix (Homona magnanima), Tobihamaki Dark fruit-tree tortrix (Pandemis heparana), Matsukareha Pine moth (Dendrolimus spectabilis), Tsukakareha Jananese hemlock caterpillar (Dendrolimus superans), Takekareha, Japanese bamboo thrix ha Euthrix potatoria, Oriental lappet (Gastropacha orientalis), Kunugia undans, Kunugia yamadai, Tomato hornworm (Manduca quinquemaculata), Tobacco hornworm (Alliga moth) cunea), Mulberry tiger moth (Lemyra imparilis), white flies (Eilema fuscodorsalis), black buckwheat (Eilema laevis), white moths udoconspersa), Swan moth (Sphrageidus similis), Gypsy moth (Lymantria dispar), White-spotted tussock moth (Orgyia thyellina), Rice green caterpillar (Naranga aenescens), Naranga aenescens leaf worm (Aedia leucomelas), mushroom Cabbage armyworm (Mamestra brassicae), Ayayoto Oriental armyworm (Pseudaletia separata), Japanese swordfish Lawn grass cutworm (Spodoptera depravata), Southern army worm Southern armyworm (ex armed worm) Fall army worm Fall armyworm (Spodoptera frugiperda), cotton leaf worm Cotton leafworm (Spodoptera littoralis), common cutworm (Spodoptera litura), giant bollworm (Helicoverpa armigera), tobacco moth Orienta l tobacco budworm (Helicoverpa assulta), tobacco bad worm Tobacco budworm (Heliothis virescens), American tobacco moth Corn earworm (Helicoverpa zea), Japanese red moth Black cutworm (Agrotis ipsilon), Kaburaya moth Turnip moth (Agrotis segetum) ), Honey beetle Threespotted plusia (Ctenoplusia agnata), soy bean looper, soybean looper (Pseudoplusia includens), nettle cabbage cabbage looper (Trichoplusia ni), mugwort Japanese giant looper (Ascotis selenaria), brass white white butterfly Lis , Lepidoptera (Lepidoptera) such as Cabbage white butterfly (Pieris rapae crucivora), Ichimongiseri Straight swift (Parnara guttata), cotton leaf worm cotton leafworm (Alabama argillacea), sugarcane borer (Diatraea sacharalis) Insect,
The fruit fly Melon fly (Bactrocera cucurbitae), the fruit fly Oriental fruit fly (Bactrocera dorsalis), the Queensland fruit fly Queensland fruit fly (Bactrocera tryoni), the fruit fly Japanese orange fly (Bactrocera tsuneonis), the Mediterranean fruit fly Mediterraneitis fly (Anastrepha ludens), ring-fly fly Apple maggot (Rhagoletis pomonella), rice leaf fly Rice leaf miner (Agromyza oryzae), leaf flyer Pea leaf miner (Chromatomyia horticola), oil leaf fly Cabbage leafminer (Liriomyza brassicae) ), Green leaf fly Stone leek leafminer (Liriomyza chinensis), green leaf fly Pea leafminer (Liriomyza huidobrensis), tomato leaf fly Tomato leafminer (Liriomyza sativae), bean leaf fly Serpentine leafminer (Liriom yza trifolii), Japanese fruit fly (Drosophila suzukii), Small leaf rice leaf miner (Hydrellia griseola), Tsetse fly (Glossina morsitans, G. palpalis), White fly, Forest fly (Hippobca) Melophagus ovinus), Onion fly (Delia antiqua), Seed corn maggot (Delia platura), sugar beet fly, Beet leaf miner (Pegomya cunicularia), Lesser house fly (Fannia canicularis), Sheep head fly (Hritae flyfly) ), Sweet fly (Morellia simplex), Face fly (Musca autumnalis), Housefly (Musca domestica), Australian bush fly (Musca vetustissima), Horn flies Horn fly (Haematobia irritans), Stable fly (Stable fly) Stomoxys calci trans, Calliphora lata, Bottle fly (Calliphora vicina), Old world screw-worm fly (Chrysomya bezziana), Blow fly (Chrysomya chloropyga), Oriental latrine fly (Chrysomya, Chrysomya America) New World screw-worm fly (Cochliomyia hominivorax), Black blow fly (Phormia regina), Northern blowfly (Protophormia terraenovae), sheep fly, Australian sheep blowfly (Lucilia cuprina), Green bottle fly (Lucilia illustris) Common green bottle fly (Lucilia sericata), Bot flies (Cuterebra spp.), Human fly botfly (Dermatobia hominis), Horse-nosed bot fly (Gasterophilus haemorrhoidalis), Horse-fly Horis bottest t fly (Gasterophilus nasalis), Bullflies Warble fly (Hypoderma bovis), Common cattle grub (Hypoderma lineatum), Sheep nasal bot fly (Oestrus ovis), Fresh fly Flesh fly (Sarcophaga carnaria), perch Srina ), Splayed deerfly (Chrysops caecutiens), Mekurabu Deer fly (Chrysops suavis), Common horse fly (Haematopota pluvialis), Greenhead horsefly (Greenhead horse fly (Tabanus nigrovittatus)) ), Soybean pod gall midge (Asphondylia yushimai), Hessian fly Hessian fly (Mayetiola destructor), mud wings Orange wheat blossom midge (Sitodiplosis mosellana), chick nuka Biting midge (Culicoides arakawae), L nipponens is), Black-tailed Blackfish (Prosimulium yezoensis), Black fly (Simulium ochraceum), African Malaria mosquito (Anopheles gambiae), Red-backed Shrimp (Anopheles hyrcanus sinesis), Anophelestosi aegypti), Asian tiger mosquito (Aedes albopictus), Chikaeka House mosquito (Culex pipiens molestus), Akaieka House mosquito (Culex pipiens pallens), Culex tritaeniorhynchus, moth P Diptera insects such as Telmatoscopus albipunctatus)
Chicken flea Hen flea (Ceratophyllus gallinae), Japanese flea Chigoe flea (Tunga penetrans), Dog flea Dog flea (Ctenocephalides canis), Cat flea Cat flea (Ctenocephalides felis), Chicken flea Sticktight flea (Echidnopha human ritual) , Siphonaptera insects such as Oriental rat flea (Xenopsylla cheopis),
Tobacco beetle (Lasioderma serricorne), Common bean weevil (Acanthoscelides obtectus), Adzuki bean beetle (Callosobruchus chinensis), Grape borer (Xylotrechus pyrrhoder beetle beetle) White-spotted longicorn beetle (Anoplophora malasiaca), Japanese pine sawyer (Monochamus alternatus), Yellow-spotted longicorn beetle (Psacothea hilaris), Colorado potato beetle Colorado beetle beetle (Phaedon cochleariae), rice leaf beetle Rice leaf beetle (Oulema oryzae), spotted leaf beetle (Demotina fasciculata), leaf beetle Cucurbit leaf beetle (Aulacophora femoralis) Beet flea beetle (Chaetocnema concinna), Northern corn rootworm (Diabrotica barberi), Southern corn rootworm (Diabrotica undecimpunctata), Western corn rootworm Western corn rootworm (Diabrotica virgifera), Triped P flea beetle striolata), Solanum flea beetle (Psylliodes angusticollis), green beetle Mexican been beetle (Epilachna varivestis), large twenty-eight-spotted ladybird (Epilachna vigintioctomawata bird), (Epilachna vigintioctopunctata), Epuraea domina, Pollen beetle (Meligethes aeneus), Peach curculio (Rhynchites heros), Sweetpotato weevil (Cylas formicarius), potato weevil West Indian sweet potato weevil (Euscepes postfasciatus), cotton weevil Boll weevil (Anthonomus grandis), white-flying beetle White-fringed beetle (Graphognatus leucoloma), horned weevil weevil Octopus weevil Alfalfa weevil (Hypera postica), Granary weevil (Sitophilus granarius), Chinese weevil Maize weevil (Sitophilus zeamais), Shibao weevil Hunting billbug (Sphenophorus venatus vestitus), Ezo weevil weevil (Lissohoptrus oryzophilus), yellow mealworm (Tenebrio molitor), red flour beetle (Tribolium castaneum), sweet potato wireworm (Melanotus fortnumi), citrus fruit Tsuruga Sugarcane wireworm (Melanotus tamsuyensis), Coreus crested citrus flower chafer (Gametis jucunda), Nagachakogane, Yellowish elongate chafer (Heptophylla picea), Douganebuibu Cupreous chafer (Anomala cuprea), Japanese beetle ), Coleoptera insects such as Rove beetle (Paederus fuscipes),
Asian citrus psyllid (Diaphorina citri), pear sucker Pear sucker (Psylla pyrisuga), Chatel spiny whitefly (Aleurocanthus camelliae), orange spiny whitefly (Aleurocanthus spiniferus), white leaffly (Aleurocanthus spiniferus) Whitefly Sweetpotato whitefly (Bemisia tabaci), Citrus whitefly (Dialeurodes citri), Greenhouse whitefly (Trialeurodes vaporariorum), Pea aphid (Acyrthosiphon pisum), Bean accura bee crab aphid (Aphis fabae), Soybean Aphid (Aphis glycines), Cotton Aphid (Aphis gossypii), Apple Aphid (Aphis pomi), Spiraea aphid (Aphis pomi) Aphis spiraecola), Foxglove aphid (Aulacorthum solani), Leaf curl plum aphid (Brachycaudus helichrysi), Japanese aphid Cabbage aphid (Brevicoryne brassiae), Walnut aphid Wola Russian wheat aphid (Diuraphis noxia), plantain beetle Rosy apple aphid (Dysaphis plantaginea), peach beetle Mealy plum aphid (Hyalopterus pruni), black pea aphid Turnip aphid (Lipaphis erysimi), tulip beetle aphid Margin door aphid (Monellia caryella), peach aphid Green peach aphid (Myzus persicae), Lettuce aphid (Nasonovia ribisnigri), Nephia Onion aphid (N eotoxoptera formosana), wheat cherry-oat aphid (Rhopalosiphum padi), rice aphid Rice root aphid (Rhopalosiphum rufiabdominalis), wheat leaf aphid (Sitobion akebiae), English grain aito avenae), Greenbug (Schizaphis graminum), Black citrus aphid (Toxoptera aurantii), Brown citrus aphid (Toxoptera citricida), Apple weevil Wooly apple aphid (Eriosoma lanigerum), Grape aphid Viteus vitifolii), hornet beetle Indian wax scale (Ceroplastes ceriferus), ruby weevil Red wax scale (Ceroplastes rubens), citrus scale insect (Coccus pseudomagnoliarum), red beetle California red scale (Aonidiella aurantii), pear Scale scale San jose scale (Comstockaspis perniciosa), scale scale tea scale (Teori scale), scale scale scale Peony scale (Pseudaonidia paeoniae), scale beetle scale Mulberry scale (Pseudaulacaspis pentagona), white scale scale Pula scale pi Citrus snow scale (Unaspis citri), Euonymus scale (Unaspis euonymi), Agarhead scale (Unaspis yanonensis), Giant margarodid scale (Drosicha corottenta scale) purchasi), worm beetle Cotton mealy bug (Phenacoccus solani), citrus mealybug (Citrus mealybug (Planococcus citri)), Japanese mealybug (Planococcus kuraunhiae), stag beetle Comstock me alybug (Pseudococcus comstocki), grape mealybug (Pseudococcus maritimus), brown brown planthopper (Laodelphax striatella), brown rice planthopper (Nilaparvata lugens), white-backedella planta (Gifer) Leafhopper (Epiacanthus stramineus), Indian cotton leafhopper (Amrasca devastans), Greens leafhopper (Bardsley leafhopper (Balclutha saltuella)), Aster leafhopper (Macrosteles fascifrons), Green leafy leafhopper (Macrosteles striifrons) leafhopper (Nephotettix cincticeps), Grape Leafhopper (Arboridia apicalis), Potato Leafhopper (Empoasca fabae), Emporasca nipponica, Chanomi Green leafhopper (Empoasca onukii), Bean's smaller green leafhopper (Empoasca sakaii), Sleek bug (Dolycoris baccarum), Sea turtle Cabbage bug (Eurydema rugosa), Spined whitespot ), White-spotted stink bug (Eysarcoris lewisi), white-spotted stink bug (Eysarcoris ventralis), blue-headed stink bug Sheild bug (Glaucias subpunctatus), brown marmorink stink bug (Halyomorpha haly) Nezara antennata), Southern green stink bug (Nezara viridula), Redbanded stink bug (Piezodorus guildinii), Redbanded shield bug (Piezodorus hybneri), Brown-winged crossota (Brown-winged cross bug) Japanese black rice bug (Scotinophora lurida), Bean bug (Riptortus clavatus), Spider helicopter Rice bug (Leptocorisa chinensis), Japanese stink bug Rice stink bug (Cletus punctiger), Southern bug shrimp bug (Paradasynus spinosus), Red-backed Helicopod Bug Rhopalid bug (Rhopalus maculatus), American Red-footed Beetle True chinch bug (Blissus leucopterus), Japanese Red-headed Bug, Oriental chinch bug (Cavelerius saccharivorus) Red cotton bug (Dysdercus cingulatus), Venezuelan sand turtle Blood-sucking bug (Rhodnius prolixus), Mexican sand turtle Kissing bug (Triatoma dimidiata), Brazilian sand turtle Kissing bug (Triatoma infestans), green stink bug sternumhil Aster ), Blown Stink bag brown stink bug (Euschistus servus), Southern green stink bag (Nezara viridula), Tarnished plant bug (Lygus lineolaris), Stink bag (Dichelops furcatus), Sugarcans pitle bag sugarcane spittlebug (Mahanarva fimbriolata), azalea lace bug (Stephanitis pyrioides), bed bug Bed bug (Cimex lectularius), bluefin turtle Pale greenplant bug (Apolygus spinolae), western tarnished plant bug (Lygus hesperus) Tarnished plant bug (Lygus lineolaris), Nagamushikasikameka Rice stink bug (Stenodema sibiricum), Akasujikasikameka Sorghum plant bug (Stenotus rubrovittatus), Rice fossil turtle Rice leaf bug (Trigonotylus caelestlium) Hemiptera insects such as and fleahopper (Halticus insularis), Cotton fleahopper (Pseudatomoscelis seriatus), Flower thrips (Frankliniella intonsa), Green lizard Yellow tea thrips (Scirtothrips dorsalis), Southern thrips Melon thrips (Thrips palmi), Black thrips Onion thrips (Thrips tabaci), Japanese gall-forming thrips (optonicthrips) ,
Chick shaft louse (Menopon hallid) (Cuclotogaster heterographa), brown fin louse (Goniodes dissmilis), bluefin louse Fluff louse (Goniodes gallinae), large bald larvae Large hen louse (Goniodes gigas), chicken swallow louse (Duru) ), Cat louse Cat louse (Felicola subrostrata), dog lice Dog biting louse (Trichodectes canis), cattle lice Short-nosed cattle louse (Haematopinus eurysternus), cattle lice Tail switch louse (Haematopinus quadripertusus), pig louse L inus suis), buffalo louse (Haematopinus tuberculatus), dog lice Dog sucking louse (Linognathus setosus), bovine white lice Long-nosed cattle louse (Linognathus cattle louse (Haemodipsus ventricosus ), Human louse Head louse (Pediculus humanus), mouse louse Mouse louse (Polyplax serratus), pheasant Crab louse (Pthirus pubis), etc.
Desert locust (Schistocerca gregaria), Australian platypus locust Australian plague locust (Chortoicetes terminifera), locust grasshopper Migratory locust (Locusta migratoria), red-eye locust Lesser paddy grasshopper (Oxya japonica), red-eye grass oxen (Teleogryllus emma), Kela Oriental mole cricket (Gryllotalpa orientalis), etc., Orthoptera insects,
German cockroach (Blattella germanica), American cockroach (Periplaneta americana), Black cockroach Smoky-brown cockroach (Periplaneta jafonica), Japanese cockroach (Periplaneta japonica), Daikokuus tomato (America) Termite Western dry-wood termite (Incisitermes minor), Common termite Formosan subterranean termite (Coptotermes formosanus), Japanese termite Japanese subterranean termite (Reticulitermes speratus), Thai termite Black-winged subterranean termite (Odontotermes formosanus) ,
Rootfeeding springtail (Onychiurus folsomi), Siberian white beetle (Onychiurus sibiricus), Garb spring spring (Bourletiella hortensis), etc.
Isopoda crustaceans such as Pill bug (Armadillidium vulgare), common rough woodlouse (Porcellio scaber),
Butterflyfish (Arguloida) crustaceans such as butterfly (Argulus coregoni), butterfly Japanese fishlouse (Argulus japonicus), sea butterfly (Argulus scutiformis)
Sea louse (Caligus curtus, C. elongatus), Salmon rose Salmon louse (Lepeophtheirus salmonis) and other crustaceans (Siphonostomatoida) crustaceans,
Sayaashi mite Storage mite (Glycyphagus destructor), house ticks mite (Glycyphagus domesticus), wheat mite Brown-legged grain mite (Aleuroglyphus ovatus), black mite Cheese mite (Tyrophagus putrescentiae), spiny mite Tyrophas , Hyugata mite Feather mite (Pterolichus obtusus), chick mite Feather mite (Megninia cubitalis), white house mite American house dust mite (Dermatophagoides farinae), yellow leopard mite bovis), Dog ear mite (Otodectes cynotis), Cattle cypress mite Psoroptic mite (Psoroptes communis), Rabbit ear mite Rabbit ear mite (Psoroptes cuniculi), Sheep cucumber Nhizendani Sheep scab mite (Psoroptes ovis), SENKOU mites Itch mite (Sarcoptes scabiei), cat foraminous mites Cat mange mite (Notoedres cati) mites suborder such as (Astigmata) mites,
Orabatida mites, such as the house salad ni (Haplochthonius simplex)
Sperm tick (Chelacaropsis moorei), cat tick (Cheyletiella blakei), rabbit tick Rabbit fur mite (Cheyletiella parasitovorax), crested tick (Cheyletiella yasguri), crested tick (Cheyletus eruditus), tick mite (Cheyletus eruditus) ), Caterpillar mites Cat follicle mite (Demodex cati), Acne mites Face mite (Demodex folliculorum), Tulip rust mites Wheat curl mite (Aceria tulipae), Black rust mites Pear rust mite (Eriophyes chibaensis), Peach bud insi ), Pearleaf blister mite (Eriophyes pyri), tea rust mite Tea rust mite (Acaphylla theavagrans), tomato rust mite Tomato russet mite (Aculops lycopersici), citrus mite Pink citrus rust mite (Aculops pelekassi) e rust mite (Aculus schlechtendali), Citrus rust mite Citrus rust mite (Phyllocoptruta oleivora), mite broad mite (Polyphagotarsonemus latus), cyclamen mite Cyclamen mite (Phytonemus pallidus), chuone mus mite Mite spider mite Citrus red mite (Panonychus citri), Mite spider mite Spider mite (Panonychus mori), Apple spider mite European red mite (Panonychus ulmi), Kanzawa spider mite Kanzawa spider mite (Tetranychus kanzawai), Nami spider mite Two mite Two-spot mite erythrocephalus), wheat mite Winter grain mite (Penthaleus major), Etsurombicula wichmanni, Miyagata pine tsutsumugi Trombiculid mite (Helenicula miyagawai), red tsutsugamushi (Leptotrombidium akamushi), yellow tsutsugamushi Prostigmata mites, such as Leptotrombidium pallida, Tsutsutsugamushi mite (Leptotrombidium scutellare),
English fowl tick (Argas persicus), tick soft tick (Ornithodoros moubata), relapsing fever tick (Ornithodoros turicata), spinose ear tick (Otobius megnini), Lone star tick (Lone star tick) Amblyomma americanum, Gulf coast tick (Amblyomma maculatum), Tick tick (Haemaphysalis campanulata), Tick tick (Haemaphysalis flava), Bite tick (Haemaphysalis longicornis), Mega physic tick (Haemaphysalis longicornis) aegyptium), Mediterranean tick (Hyalomma marginatum), Tropical cattle tick (Boophilus microplus), Ixodes nipponensis, Yamato tick (Ixodes ovatus), Western black-legge d tick (Ixodes pacifcus), Schulze tick Taiga tick (Ixodes persulcatus), Sheep tick Castor bean tick (Ixodes ricinus), Black-legged tick (Ixodes scapularis), Tropical horse tick (Anocentor nitens), Rocky Mountains Rocky Mountain wood tick (Dermacentor andersoni), Pacific Coast tick (Dermacentor occidentalis), Amikemeka tick Ornate cow tick (Dermacentor reticulatus), American dog tick American dog tick (Dermacentor variabilis), Ripicentor spp. Tick American cattle tick (Rhipicephalus annulatus), Brown dog tick (Rhipicephalus sanguineus) and other ticks (Metastigmata) ticks,
Red mite (Dermanyssus gallinae), house dust mite Tropical rat mite (Ornithonyssus bacoti), northern fowl mite (Ornithonyssus sylviarum), honey bee mite Honeybee mite (Varroa destructor), honeybee mite Varroa mite Varroa mite (Mesostigmata) mites,
Pancreas (Architaenioglossa) gastropod, such as Apple snail (Pomacea canaliculata)
Giant African snail (Achatina fulica), terrestrial slug (Limax marginatus), slug slug (Meghimatium bilineatum), Korean round snail (Acusta despecta sieboldiana), Miss maimai Land snio (Euhadra mai) Eyes (Stylommatophora) gastropods,
Giant kidney worm (Dioctophyma renale), ringed capillary worm Thread worms (Capillaria annulata), torsion capillary nematode Cropworm (Capillaria contorta), liver capillary nematode Capillary liver worm (Capillaria hepatica), penetrating capillary nematode (Capillaria) perforans), Philippine Capillaria philippinensis, Capillaria suis, Caterpillar Whipworm (Trichuris discolor), Whipworm Whipworm (Trichuris ovis), Pig whipworm Pig Whipworm (Trichuris suis), human Enoplida nematodes such as the whipworm Human whipworm (Trichuris trichiura), dog whipworm Dog whipworm (Trichuris vulpis), Trichinella pork worm (Trichinella spiralis),
桿 such as Nipple faecal nematode Intestinal threadworm (Strongyloides papillosus), cat fecal nematode (Strongyloides planiceps), pig fecal nematode Pig threadworm (Strongyloides ransomi), human fecal nematode Threadworm (Strongyloides stercoralis), Micronema spp. Rhabditida nematode,
Brazilian Hookworm (Ancylostoma braziliense), Dog Hookworm Dog hookworm (Ancylostoma caninum), Zubini Hookworm Old World hookworm (Ancylostoma duodenale), Cat Hookworm Cat hookworm (Ancylostoma tubaeforme), Narrowhead Hookworm The Northern hookworm of dogs (Uncinaria stenocephala) Caterpillar Cattle hookworm (Bunostomum phlebotomum), Sheep worm, Small ruminant hookworm (Bunostomum trigonocephalum), American worm New World hookworm (Necator americanus), Cyathostomum spp., Cylicocyclus spyl. spp.), Cylicostephanus spp., Donkeys (Strongylus asini), edentulous (Strongylus edentatus), Horse worms Blood worm (Strongylus equinus), Common worms Blood worm (Strongylus vulgaris) Large-mouthed bowel worm (Chabertia ovina), Indian nodular worm (Oesophagostomum brevic) audatum), Colombian nodule worm (Oesophagostomum columbianum), Nodule worm (Oesophagostomum dentatum), Nodular worm (Oesophagostomum georgianum), Nodular worm (Oesophagostomum columbianum) Nodular worm (Oesophagostomum quadrispinulatum), cattle intestinal nodular worm (Oesophagostomum radiatum), goat intestinal nodular worm (Oesophagostomum venulosum), scrijabin worm (Syngamus skrjabinomorpha), chicken worm moth trachea (Syngamus skrjabinomorpha) Swine kidney worm (Stephanurus dentatus), Couperia cattle bankrupt worm (Cooperia oncophora), red stomach worm (Hyostrongylus rubidus), stomach hair worm (Trichostrongylus axei), serpentine ciliate nematode (Trichostrongylus colubriformis), Oriental ciliate nematode Oriental trichostrongylus (Trichostrongylus orientalis), torsion stomachworm Red stomach worm (Haemonchus co ntortus), cattle stomach worm (Mecistocirrus digitatus), Ostertag stomach worm (Ostertagia ostertagi), filamentous lungworm Common lungworm (Dictyocaulus filaria), bovine lungworm Bovine lungworm (Dictyocaulus viviparus) Insect worms (Nematodirus filicollis), Swine lungworm (Metastrongylus elongatus), Lungworm (Filaroides hirthi), Lungworm (Crenosoma aerophila), Fox lungworm (Crenosoma vulpis) Strong lungida nematodes such as Rat lung worm (Angiostrongylus cantonensis), Schistosoma nematode French heartworm (Angiostrongylus vasorum), Protostrongylus spp.
Rice white nematode (Aphelenchoides besseyi), Pine wood nematode (Bursaphelenchus xylophilus) nematode (Aphelenchida) nematode,
Potato cyst nematode (Globodera rostochiensis), wheat cyst nematode Cereal cyst nematode (Heterodera avenae), soybean cyst nematode (Seterbean cyst nematode (Heterodera glycines)), arenaria root nematode (Peterut root-Menot nematode) -knot nematode (Meloidogyne hapla), Southern root-knot nematode (Meloidogyne incognita), Java root-knot nematode (Meloidogyne javanica), Southern root-kion nematode Coffee root-lesion nematode (Pratylus nechade) Root-lesion nematode (Pratylenchus loosi), Cobb's root-lesion nematode (Pratylenchus penetrans), Crested nematode Walnut root-lesion nematode (Pratylenchus vulnus), etc. lenchida) nematode,
Oxyurida nematodes such as human worm Pinworm (Enterobius vermicularis), horse worm Equine pinworm (Oxyuris equi), rabbit worm Rabbit pinworm (Passalurus ambiguus),
Pig roundworm (Ascaris suum), Horse roundworm Horse roundworm (Parascaris equorum), Dog roundworm Dog roundworm (Toxascaris leonina), Dog roundworm Dog intestinal roundworm (Toxocara canis), Cat roundworm Feline roundworm (Toxocara cati), Cattle roundworm Large cattle roundworm (Toxocara vitulorum), Anisakis spp., Pseudoterranova spp., chicken caecal caecal worm (Heterakis gallinarum), chicken roundworm (Ascaridia galli) and other roundworms (Ascaridida) Nematode,
Medinaworm Guinea worm (Dracunculus medinensis), Dolores jaw-and-mouth beetle (Gnathostoma doloresi), Ganthostoma hispidum, Japanese jaw-and-mouth beetle (Gnathostoma nipponicum), Reddish-coloured worm (Gnathostoma spinigerum) Dog stomach worm (Physaloptera canis), cat stomach worm (Physaloptera felidis, P. praeputialis), lala gastroworm Feline / canine stomach worm (Physaloptera rara), oriental eyeworm Eye worm (Thelazia callipaeda), Bovine eyeworm (Thelazia rhodesi), Large mouth stomach worm (Draschia megastoma), Equine stomach worm (Habronema microstoma), Stomach worm (Habronema muscae), Beautiful esophagus Gullet worm ( Gongylonema pulchrum), Thick stomach worm (Ascarops strongylina), Parafilaria (Parafilaria bovicola), Parafilaria multipapillosa, Stephanofilaria okinawaensis), Bancroft filaria (Wuchereria bancrofti), Malay filamentous worm (Brugia malayi), Neck threadworm (Onchocerca cervicalis), Gibson filamentous worm (Onchocerca gibsoni), Cattle filarial worm (Onchocercer gautum) ), Convolvulus (Onchocerca volvulus), finger filamentous worm Bovine filarial worm (Setaria digitata), equine filamentous peritoneal worm (Setaria equina), papillary larva (Setaria labiatopapillosa), marshall filariae (Setaria marshalli), dog Spirurida nematodes, such as the dog heartworm (Dirofilaria immitis) and the African eye worm (Loa loa),
Bald worms such as Moniliformis moniliformis, Giant thorny-headed worm (Macracanthorhynchus hirudinaceus),
Artificial leaves such as Fish tapeworm (Diphyllobothrium latum), Diphyllobothrium nihonkaiense, Manson tapeworm (Spirometra erinaceieuropaei), Diplogonoporus grandis Eye (Pseudophyllidea) tapeworm,
Wire worms (Mesocestoides lineatus), striped worms Chicken tapeworm (Raillietina cesticillus), spiny cleft worm Fowl tapeworm (Raillietina echinobothrida), square tapeworm Chicken tapeworm (Raillietina tetragona), canine tapeworm (Taenia hydatigena), Canine tapeworm (Taenia multiceps), sheep worm Sheep measles (Taenia ovis), beetle tapeworm Dog tapeworm (Taenia pisiformis), striped beetle Beef tapeworm (Taenia saginata), striped worm Tapeworm (Taenia serialis) ), Rodentworm Pork tapeworm (Taenia solium), caterpillar Feline tapeworm (Taenia taeniaeformis), single tapeworm Hydatid tapeworm (Echinococcus granulosus), multi-budworm, small fox tapeworm (Echinococcus multilocularis), cat (Echinococcus oligarthrus), Vogel's crustacean (Echinococcus vogeli), reduced tapeworm Rat tapeworm (Hymenolepis diminuta), small tapeworm Dwarf tapeworm (Hymenolepis nana), crustacea double-pored dog tapeworm (Dipylidium ca ninum), cuneate tapeworms (Amoebotaenia sphenoides), funnel-like crustaceans (Choanotaenia infundibulum), quail crustaceans (Metroliasthes coturnix), crustacea Equine tapeworm (Anoplocephala magna), phytophyte crustacean Cecal tapeworm (Anoplocephala perfoliata), papillae Insects Dwarf equine tapeworm (Paranoplocephala mamillana), Benedenta taper Common tapeworm (Moniezia benedeni), expanded tapeworm Sheep tapeworm (Moniezia expansa), Stilsia spp.
Striated insects (Pharyngostomum cordatum), Schistosoma haematobium, Schistosoma haematobium, Schistosoma japonicum, Schistosoma japonicum, Schistosoma mansoni, etc.
Echinostoma cinetorchis, Echinostoma hortense, Giant liver fluke (Fasciola gigantica), Liver common liver fluke (Fasciola hepatica), Fasciolopsis buski, Flat belly twin Echinostomida, such as Homalogaster paloniae,
Continental flukes (Dicrocoelium chinensis), moth-type flukes Lancet liver fluke (Dicrocoelium dendriticum), African moth-type flukes African lancet fluke (Dicrocoelium hospes), small pancreatic folds (Eurytrema coelomaticum), pancreatic folds Pancreatic fluke (Eurytrema pancreaticum) Paragonimus miyazakii, Paragonimus ohirai, Westermann Lung fluke (Paragonimus westermani), etc. Platimorchiida
Amphimerus spp., Liver fluke Chinese liver fluke (Clonorchis sinensis), Cat liver fluke Cat liver fluke (Opisthorchis felineus), Thai liver fluke Southeast Aasian liver fluke (Opisthorchis viverrini), Pseudamphistom spp .), Metrochis spp., Parametorchis spp., Malformed fluke (Heterophyes heterophyes), Metagonimus yokokawai, foregut fluke (Pygidiopsis summa), etc. Opisthorchiida) fluke,
Amoeba such as Entamoeba histolytica, E. invadens,
Futago Babesia (Babesia bigemina), Cattle Babesia bovis, Big Horse Babesia caballi, Dog Babesia canis, Cat Babesia felis, Gibson dog Babesia gibsoni, Large Piroplasma (Babesia ovata) ), Cytauxzoon felis, tropical piroplasmosis Tyleria (Theileria annulata), pseudocoastal fever Tyreria (Theileria mutans), small piroplasma (Theileria orientalis), east coast fever Tyrelia (Theileria parva), etc. Piroplasmida sporophytes,
Haemoproteus mansoni, chicken leucocytozone (Leucocytozoon caulleryi), Plasmodium falciparum, Plasmodium malariae, Plasmodium ovale, Plasmodium ovale Haemosporida spores such as Plasmodium vivax,
Caryospora spp., Eimeria acervulina, Eimeria bovis, Eimeria brunetti, Eimeria maxima, Eimeria necatrix, Eimeria necatrix Eimeria ovinoidalis, rabbit liver coccidium (Eimeria stiedae), chicken cecal coccidium (Eimeria tenella), dog isospora canis, feline isospora (Isospora felis), porcine isospora suis (Isospora suis), Tizeria aleni , Tyzzeria anseris, Tyzzeria perniciosa, Wenyonella anatis, Wenyonella gagari, Cryptosporidium canis, cat crypt Cryptosporidium felis, Cryptosporidium hominis, turkey Cryptosporidium meleagridis, Cryptosporidium muris, small Cryptosporidium parvco, sarcosis (Sarcocystis cruzi), Sarcocystis felis, Sarcocystis hominis, Sarcocystis miescheriana, Sarcocystis neurona, Sarcocystis colostis tenis S tenis Sarcocystis ovalis), Toxoplasma gondii, dog hepatozoon (Hepatozoon canis), cat hepatozoon (Hepatozoon felis), etc. cidiorida) spores,
Vestibuliferida ciliates, such as large intestine barantidium coli,
Histomanas meleagridis, Pentatrichomonas hominis, Trichomonas tenax and other Trichomonadida flagellates,
Dipromonads (Diplomonadida) flagellates such as Giardia intestinalis, Giardia muris, turkey hexamita (Hexamita meleagridis), Hexamita parva,
Leishmania donovani, Leishmania infantum, Leishmania major, Leishmania tropica, Trypanosoma brucei gambiense, Trypanosoma brucei cruise, Trypanosoma brucei rhodesi Trypanosoma cruzi, Trypanosoma equiperdum, Trypanosoma evansi, etc. Kinotoplastida flagellates,
However, pests in the field of agriculture and horticulture that can be controlled using the compounds of the present invention and external or internal parasites such as livestock, poultry, and pet animals are not limited to these.

さらに、本発明化合物は、有機燐系化合物、カーバメート系化合物又はピレスロイド系化合物等の既存の殺虫剤に対して抵抗性の発達した有害生物に対しても有効である。   Furthermore, the compound of the present invention is also effective against pests that have developed resistance to existing insecticides such as organophosphorus compounds, carbamate compounds, and pyrethroid compounds.

すなわち、本発明化合物は、粘管目(トビムシ目)、網翅目(ゴキブリ目)、直翅目(バッタ目)、シロアリ目、総翅目(アザミウマ目)、半翅目(カメムシ目及びヨコバイ目)、鱗翅目(チョウ目)、鞘翅目(コウチュウ目)、膜翅目(ハチ目)、双翅目(ハエ目)、等翅目(ノミ目)及びシラミ目等の昆虫類、ダニ類、腹足類及び線虫類等に属する有害生物を低濃度で有効に防除することが出来る。一方、本発明化合物はホ乳類、魚類、甲殻類及び益虫(ミツバチ、マルハナバチ等の有用昆虫やツヤコバチ、アブラバチ、ヤドリバエ、ヒメハナカメムシ、カブリダニ等の天敵)に対してほとんど悪影響の無い極めて有用な特長を有している。   That is, the compound of the present invention is composed of the order of mucous eyes (Coleoptera), reticulates (Roaches), straight moths (Grasshoppers), termites, common moths (Thrips), hemimorphs (stink bugs and leafhoppers). Eyes), Lepidoptera (Lepidoptera), Coleoptera (Coleoptera), Hymenoptera (Hymenoptera), Diptera (Flyidae), Islamic (Flea), Liceid, and other insects, ticks In addition, pests belonging to gastropods and nematodes can be effectively controlled at low concentrations. On the other hand, the compounds of the present invention are extremely useful with little adverse effect on mammals, fish, crustaceans and beneficial insects (beneficial insects such as bees and bumblebees, natural enemies such as honeybees, wasps, mistletoe flies, mosquitoes, and mites). Has features.

本発明化合物を使用するにあたっては、通常適当な固体担体又は液体担体と混合し、更に所望により界面活性剤、浸透剤、展着剤、増粘剤、凍結防止剤、結合剤、固結防止剤、崩壊剤、消泡剤、防腐剤および分解防止剤等を添加して、液剤（soluble concentrate）、乳剤（emulsifiable concentrate）、水和剤（wettable powder）、水溶剤（water soluble powder）、顆粒水和剤（water dispersible granule）、顆粒水溶剤（water soluble granule）、懸濁剤（suspension concentrate）、乳濁剤（concentrated emulsion）、サスポエマルジョン（suspoemulsion）、マイクロエマルジョン（microemulsion）、粉剤（dustable powder）、粒剤（granule）錠剤（tablet）および乳化性ゲル剤（emulsifiable gel）等任意の剤型の製剤にて実用に供することができる。また、省力化および安全性向上の観点から、上記任意の剤型の製剤を、水溶性カプセルおよび水溶性フィルムの袋等の水溶性包装体に封入して供することもできる。   When using the compound of the present invention, it is usually mixed with a suitable solid carrier or liquid carrier, and if desired, a surfactant, penetrant, spreading agent, thickener, antifreezing agent, binder, anti-caking agent , Disintegrating agents, antifoaming agents, preservatives and anti-degradation agents, etc., and soluble concentrate, emulsion (emulsifiable concentrate), wettable powder, water-soluble powder, granular water Water dispersible granule, water soluble granule, suspension concentrate, concentrated emulsion, suspoemulsion, microemulsion, dustable powder ), Granule tablets, and emulsifiable gels, and can be put to practical use. Further, from the viewpoint of labor saving and safety improvement, the preparations of any of the above dosage forms can be provided by being enclosed in a water-soluble package such as a water-soluble capsule and a bag of a water-soluble film.

固体担体としては、例えば石英、方解石、海泡石、ドロマイト、チョーク、カオリナイト、パイロフィライト、セリサイト、ハロサイト、メタハロサイト、木節粘土、蛙目粘土、陶石、ジークライト、アロフェン、シラス、きら、タルク、ベントナイト、活性白土、酸性白土、軽石、アタパルジャイト、ゼオライトおよび珪藻土等の天然鉱物質、例えば焼成クレー、パーライト、シラスバルーン、バーミキュライト、アタパルガスクレーおよび焼成珪藻土等の天然鉱物質の焼成品、例えば炭酸マグネシウム、炭酸カルシウム、炭酸ナトリウム、炭酸水素ナトリウム、硫酸アンモニウム、硫酸ナトリウム、硫酸マグネシウム、リン酸水素二アンモニウム、リン酸二水素アンモニウムおよび塩化カリウム等の無機塩類、例えばブドウ糖、果糖、しょ糖および乳糖などの糖類、例えば澱粉、粉末セルロースおよびデキストリン等の多糖類、例えば尿素、尿素誘導体、安息香酸および安息香酸の塩等の有機物、例えば木粉、コルク粉、トウモロコシ穂軸、クルミ殻およびタバコ茎等の植物類、フライアッシュ、ホワイトカーボン（例えば、含水合成シリカ、無水合成シリカおよび含水合成シリケート等）ならびに肥料等が挙げられる。   Examples of the solid carrier include quartz, calcite, gypsum, dolomite, chalk, kaolinite, pyrophyllite, sericite, halosite, metahalosite, kibushi clay, glazed clay, porcelain stone, siegrite, and allophane. Natural minerals such as shirasu, kira, talc, bentonite, activated clay, acid clay, pumice, attapulgite, zeolite and diatomaceous earth, for example, calcined clay, perlite, shirasu balloon, vermiculite, attapulgus clay and calcined diatomaceous earth Baked products such as magnesium carbonate, calcium carbonate, sodium carbonate, sodium bicarbonate, ammonium sulfate, sodium sulfate, magnesium sulfate, diammonium hydrogen phosphate, ammonium dihydrogen phosphate and potassium chloride, such as glucose, fructose , And Sugars such as sugar and lactose, polysaccharides such as starch, powdered cellulose and dextrin, organic materials such as urea, urea derivatives, benzoic acid and benzoic acid salts, such as wood flour, cork flour, corn cobs, walnut shells and Examples include plants such as tobacco stalks, fly ash, white carbon (for example, hydrous synthetic silica, anhydrous synthetic silica, hydrous synthetic silicate, etc.) and fertilizers.

液体担体としては、例えばキシレン、アルキル（Ｃ₉又はＣ₁₀等）ベンゼン、フェニルキシリルエタンおよびアルキル（Ｃ₁又はＣ₃等）ナフタレン等の芳香族炭化水素類、マシン油、ノルマルパラフィン、イソパラフィンおよびナフテン等の脂肪族炭化水素類、ケロシン等の芳香族炭化水素と脂肪族炭化水素の混合物、エタノール、イソプロパノール、シクロヘキサノール、フェノキシエタノールおよびベンジルアルコール等のアルコール、エチレングリコール、プロピレングリコール、ジエチレングリコール、ヘキシレングリコール、ポリエチレングリコールおよびポリプロピレングリコール等の多価アルコール、プロピルセロソルブ、ブチルセロソルブ、フェニルセロソルブ、プロピレングリコールモノメチルエーテル、プロピレングリコールモノエチルエーテル、プロピレングリコールモノプロピルエーテル、プロピレングリコールモノブチルエーテルおよびプロピレングリコールモノフェニルエーテル等のエーテル、アセトフェノン、シクロヘキサノンおよびγ−ブチロラクトン等のケトン、脂肪酸メチルエステル、コハク酸ジアルキルエステル、グルタミン酸ジアルキルエステル、アジピン酸ジアルキルエステルおよびフタル酸ジアルキルエステル等のエステル、Ｎ−アルキル（Ｃ₁、Ｃ₈又はＣ₁₂等）ピロリドン等の酸アミド、大豆油、アマニ油、ナタネ油、ヤシ油、綿実油およびヒマシ油等の油脂、ジメチルスルホキシドならびに水が挙げられる。 Examples of the liquid carrier include xylene, alkyl (C ₉ or C ₁₀ etc.) benzene, phenyl xylyl ethane and alkyl (C ₁ or C ₃ etc.) naphthalene and other aromatic hydrocarbons, machine oil, normal paraffin, isoparaffin and Aliphatic hydrocarbons such as naphthene, mixtures of aromatic and aliphatic hydrocarbons such as kerosene, alcohols such as ethanol, isopropanol, cyclohexanol, phenoxyethanol and benzyl alcohol, ethylene glycol, propylene glycol, diethylene glycol, hexylene glycol , Polyhydric alcohols such as polyethylene glycol and polypropylene glycol, propyl cellosolve, butyl cellosolve, phenyl cellosolve, propylene glycol monomethyl ether, propylene glycol Ethers such as ethyl monoethyl ether, propylene glycol monopropyl ether, propylene glycol monobutyl ether and propylene glycol monophenyl ether, ketones such as acetophenone, cyclohexanone and γ-butyrolactone, fatty acid methyl esters, dialkyl esters of succinic acid, dialkyl esters of glutamic acid, adipine esters such as dialkyl ester and dialkyl phthalate esters, N- alkyl (C _1, C ₈ or C _12, etc.) acid amide pyrrolidone, soybean oil, linseed oil, rapeseed oil, coconut oil, such as cottonseed oil and castor oil Examples include fats and oils, dimethyl sulfoxide and water.

これら固体および液体担体は、単独で用いても２種以上を併用してもよい。   These solid and liquid carriers may be used alone or in combination of two or more.

界面活性剤としては、例えばポリオキシエチレンアルキルエーテル、ポリオキシエチレンアルキル（モノ又はジ）フェニルエーテル、ポリオキシエチレン（モノ、ジ又はトリ）スチリルフェニルエーテル、ポリオキシエチレンポリオキシプロピレンブロックコポリマー、ポリオキシエチレン脂肪酸（モノ又はジ）エステル、ソルビタン脂肪酸エステル、ポリオキシエチレンソルビタン脂肪酸エステル、ヒマシ油エチレンオキサイド付加物、アセチレングリコール、アセチレンアルコール、アセチレングリコールのエチレンオキサイド付加物、アセチレンアルコールのエチレンオキサイド付加物およびアルキルグリコシド等のノニオン性界面活性剤、アルキル硫酸エステル塩、アルキルベンゼンスルホン酸塩、リグニンスルホン酸塩、アルキルスルホコハク酸塩、ナフタレンスルホン酸塩、アルキルナフタレンスルホン酸塩、ナフタレンスルホン酸のホルマリン縮合物の塩、アルキルナフタレンスルホン酸のホルマリン縮合物の塩、ポリオキシエチレンアルキルエーテル硫酸又は燐酸エステル塩、ポリオキシエチレン（モノ又はジ）アルキルフェニルエーテル硫酸又は燐酸エステル塩、ポリオキシエチレン（モノ、ジ又はトリ）スチリルフェニルエーテル硫酸又は燐酸エステル塩、ポリカルボン酸塩（例えば、ポリアクリル酸塩、ポリマレイン酸塩およびマレイン酸とオレフィンとの共重合物等）およびポリスチレンスルホン酸塩等のアニオン性界面活性剤、アルキルアミン塩およびアルキル４級アンモニウム塩等のカチオン性界面活性剤、アミノ酸型およびベタイン型等の両性界面活性剤、シリコーン系界面活性剤ならびにフッ素系界面活性剤が挙げられる。   Examples of the surfactant include polyoxyethylene alkyl ether, polyoxyethylene alkyl (mono or di) phenyl ether, polyoxyethylene (mono, di or tri) styryl phenyl ether, polyoxyethylene polyoxypropylene block copolymer, polyoxyethylene Ethylene fatty acid (mono or di) ester, sorbitan fatty acid ester, polyoxyethylene sorbitan fatty acid ester, castor oil ethylene oxide adduct, acetylene glycol, acetylene alcohol, ethylene oxide adduct of acetylene glycol, ethylene oxide adduct of acetylene alcohol and alkyl Nonionic surfactants such as glycosides, alkyl sulfate esters, alkylbenzene sulfonates, lignin sulfonates, alkyls Rufosuccinate, naphthalene sulfonate, alkyl naphthalene sulfonate, salt of formalin condensate of naphthalene sulfonic acid, salt of formalin condensate of alkyl naphthalene sulfonic acid, polyoxyethylene alkyl ether sulfate or phosphate ester salt, polyoxyethylene (Mono or di) alkyl phenyl ether sulfate or phosphate ester salt, polyoxyethylene (mono, di or tri) styryl phenyl ether sulfate or phosphate ester salt, polycarboxylate (eg polyacrylate, polymaleate and maleate) Copolymer of acid and olefin, etc.) and anionic surfactants such as polystyrene sulfonate, cationic surfactants such as alkylamine salts and alkyl quaternary ammonium salts, and amphoteric interfaces such as amino acid type and betaine type Sexual agents, silicone-based surfactants and fluorinated surfactants.

これら界面活性剤の含有量は、特に限定されるものではないが、本発明の製剤１００重量部に対し、通常０．０５〜２０重量部の範囲が望ましい。また、これら界面活性剤は、単独で用いても２種以上を併用してもよい。   The content of these surfactants is not particularly limited, but is usually preferably in the range of 0.05 to 20 parts by weight with respect to 100 parts by weight of the preparation of the present invention. These surfactants may be used alone or in combination of two or more.

本発明化合物の施用薬量は適用場面、施用時期、施用方法、栽培作物等により差異は有るが、一般には有効成分量としてヘクタール（ha）当たり０.００５〜５０kg程度が適当である。   The application amount of the compound of the present invention varies depending on the application scene, application time, application method, cultivated crops, etc., but generally 0.005 to 50 kg per hectare (ha) is appropriate as the amount of active ingredient.

一方、家畜及び愛玩動物としての哺乳動物および鳥類の外部又は内部寄生虫の防除に本発明化合物を使用するにあたっては、有効量の本発明化合物を製剤用添加物とともに経口投与、注射（筋肉内、皮下、静脈内、腹腔内）などの非経口投与；浸漬、スプレー、入浴、洗浄、滴下（pouring-on)およびスポッティング(spotting-on)並びにダスティング(dusting)などの経皮投与；経鼻投与により投与することができる。本発明化合物はまた、細片、プレート、バンド、カラー、イヤー・マーク(ear mark)、リム(limb)・バンド、標識装置などを用いた成形製品により投与することができる。投与にあたっては本発明化合物を投与経路に適した任意の剤型とすることができる。   On the other hand, when using the compound of the present invention for the control of the ectoparasites of mammals and birds as domestic animals and pets, an effective amount of the compound of the present invention is administered orally together with injection additives (intramuscular, Parenteral administration such as subcutaneous, intravenous, intraperitoneal; transdermal administration such as immersion, spraying, bathing, washing, pouring-on and spotting-on and dusting; nasal administration Can be administered. The compounds of the present invention can also be administered by molded products using strips, plates, bands, collars, ear marks, limb bands, labeling devices and the like. In administration, the compound of the present invention can be in any dosage form suitable for the administration route.

調製される任意の剤型としては、粉剤、粒剤、水和剤、ペレット、錠剤、大丸薬、カプセル剤、活性化合物を含む成形製品などの固体調製物；注射用液剤、経口用液剤、皮膚上又は体腔中に用いる液剤；滴下（Pour-on)剤、点下(Spot-on)剤、フロアブル剤、乳剤などの溶液調製物；軟膏剤、ゲルなどの半固体調製物などが挙げられる。   Arbitrary forms to be prepared include solid preparations such as powders, granules, wettable powders, pellets, tablets, large pills, capsules, molded products containing active compounds; injection solutions, oral solutions, skin Liquid preparations used above or in body cavities; solution preparations such as Pour-on agents, spot-on agents, flowable agents and emulsions; semi-solid preparations such as ointments and gels.

固体調製物は、主に経口投与あるいは水などで希釈して経皮投与にあるいは環境処理にて用いることができる。固体調製物は、活性化合物を必要ならば補助剤を加えて適当な賦形剤と共に混合し、そして所望の形状に変えることにより調製できる。適当な賦形剤としては、例えば炭酸塩、炭酸水素塩、リン酸塩、酸化アルミニウム、シリカ、粘土などの無機物質、糖、セルロース、粉砕された穀物、澱粉などの有機物質がある。   The solid preparation can be used mainly for oral administration or diluted with water for transdermal administration or environmental treatment. Solid preparations can be prepared by adding the active compound, if necessary, with adjuncts, mixing with appropriate excipients, and converting to the desired shape. Suitable excipients include, for example, inorganic substances such as carbonates, bicarbonates, phosphates, aluminum oxides, silicas, clays, and organic substances such as sugars, cellulose, crushed grains, and starches.

注射用液剤は、静脈内、筋肉内および皮下に投与できる、注射用液剤は、活性化合物を適当な溶媒に溶解させ、そして必要ならば可溶化剤、酸、塩基、緩衝用塩、酸化防止剤および保護剤などの添加剤を加えることにより調製できる。適当な溶媒としては、水、エタノール、ブタノール、ベンジルアルコール、グリセリン、プロピレングリコール、ポリエチレングリコール、Ｎ−メチルピロリドン並びにこれらの混合物、生理学的に許容しうる植物油、注射に適する合成油などがあげられる。可溶化剤としては、ポリビニルピロリドン、ポリオキシエチル化されたヒマシ油およびポリオキシエチル化されたソルビタンエステルなどがあげられる。保護剤には、ベンジルアルコール、トリクロロブタノール、ｐ−ヒドロキシ安息香酸エステルおよびｎ−ブタノールなどがある。   Injection solutions can be administered intravenously, intramuscularly and subcutaneously. Injection solutions dissolve the active compound in a suitable solvent and, if necessary, solubilizers, acids, bases, buffer salts, antioxidants. And can be prepared by adding additives such as protective agents. Suitable solvents include water, ethanol, butanol, benzyl alcohol, glycerin, propylene glycol, polyethylene glycol, N-methylpyrrolidone and mixtures thereof, physiologically acceptable vegetable oils, synthetic oils suitable for injection, and the like. Examples of solubilizers include polyvinylpyrrolidone, polyoxyethylated castor oil, and polyoxyethylated sorbitan ester. Protecting agents include benzyl alcohol, trichlorobutanol, p-hydroxybenzoic acid ester and n-butanol.

経口液剤は直接又は希釈して投与することができる。注射用液剤と同様に調製することができる。   Oral solutions can be administered directly or diluted. It can be prepared in the same manner as an injectable solution.

フロアブル剤、乳剤、などは直接又は希釈して経皮的に、又は環境処理にて投与できる。   Flowables, emulsions, etc. can be administered directly or diluted transdermally or by environmental treatment.

皮膚上で用いる液剤は、滴下し、広げ、すり込み、噴霧し、散布するか、又は浸漬（浸漬、入浴又は洗浄）により塗布することにより投与できる。これらの液剤は注射用液剤と同様に調製できる。   Solutions used on the skin can be administered by dripping, spreading, rubbing, spraying, spraying or applying by dipping (immersion, bathing or washing). These solutions can be prepared in the same manner as injection solutions.

滴下(Pour-on)剤および点下(Spot-on)剤は皮膚の限定された場所に滴下するか、又は噴霧し、これにより活性化合物を皮膚に浸漬させそして全身的に作用させることができる。滴下剤および点下剤は、有効成分を適当な皮膚適合性溶媒又は溶媒混合物に溶解するか、懸濁させるか又は乳化することにより調製できる。必要ならば、界面活性剤、着色剤、吸収促進物質、酸化防止剤、光安定剤および接着剤などの補助剤を加えてもよい。   Pour-on and spot-on agents can be dripped or sprayed onto a limited area of the skin, so that the active compound can be immersed in the skin and act systemically . Drops and drop preparations can be prepared by dissolving, suspending or emulsifying the active ingredient in suitable skin-compatible solvents or solvent mixtures. If necessary, auxiliary agents such as surfactants, colorants, absorption promoting substances, antioxidants, light stabilizers and adhesives may be added.

適当な溶媒としては、水、アルカノール、グリコール、ポリエチレングリコール、ポリプロピレングリコール、グリセリン、ベンジルアルコール、フェニルエタノール、フェノキシエタノール、酢酸エチル、酢酸ブチル、安息香酸ベンジル、ジプロピレングリコールモノメチルエーテル、ジエチレングリコールモノブチルエーテル、アセトン、メチルエチルケトン、芳香族および／又は脂肪族炭化水素、植物又は合成油、ＤＭＦ、流動パラフィン、軽質流動パラフィン、シリコーン、ジメチルアセトアミド、Ｎ−メチルピロリドン又は２，２−ジメチル−４−オキシ−メチレン−１，３−ジオキソランが挙げられる。吸収促進物質には、ＤＭＳＯ、ミリスチン酸イソプロピル、ペラルゴン酸ジプロピレングリコール、シリコーン油、脂肪族エステル、トリグリセリドおよび脂肪アルコールが挙げられる。酸化防止剤には、亜硫酸塩、メタ重亜硫酸塩、アスコルビン酸、ブチルヒドロキシトルエン、ブチルヒドロキシアニソールおよびトコフェロールが挙げられる。   Suitable solvents include water, alkanol, glycol, polyethylene glycol, polypropylene glycol, glycerin, benzyl alcohol, phenylethanol, phenoxyethanol, ethyl acetate, butyl acetate, benzyl benzoate, dipropylene glycol monomethyl ether, diethylene glycol monobutyl ether, acetone, Methyl ethyl ketone, aromatic and / or aliphatic hydrocarbons, vegetable or synthetic oil, DMF, liquid paraffin, light liquid paraffin, silicone, dimethylacetamide, N-methylpyrrolidone or 2,2-dimethyl-4-oxy-methylene-1, 3-dioxolane is mentioned. Absorption enhancers include DMSO, isopropyl myristate, dipropylene glycol pelargonate, silicone oil, aliphatic esters, triglycerides and fatty alcohols. Antioxidants include sulfites, metabisulfites, ascorbic acid, butylhydroxytoluene, butylhydroxyanisole and tocopherol.

乳剤は、経口投与、経皮投与又は注射として投与できる。乳剤は、有効成分を疎水性相又は親水性相に溶解させ、このものを適当な乳化剤により、必要ならばさらに着色剤、吸収促進物質、保護剤、酸化防止剤、遮光剤および増粘物質などの補助剤と共に他の相の溶媒と均質化することにより調製できる。   The emulsion can be administered orally, transdermally or as an injection. In emulsions, active ingredients are dissolved in a hydrophobic phase or a hydrophilic phase, and this is further added with a suitable emulsifier, and if necessary, a colorant, an absorption promoting substance, a protective agent, an antioxidant, a light-shielding agent, a thickening substance, etc. Can be prepared by homogenizing with other phase solvents together with other auxiliary agents.

疎水性相（油）としては、パラフィン油、シリコーン油、ゴマ油、アーモンド油、ヒマシ油、合成トリグリセリド、ステアリン酸エチル、アジピン酸ジーｎ−ブチリル、ラウリル酸ヘキシル、ペラルゴン酸ジプロピレングリコール、分枝鎖状の短鎖長脂肪酸と鎖長Ｃ１６〜Ｃ１８の飽和脂肪酸とのエステル、ミリスチン酸イソプロピル、パルミチン酸イソプロピル、鎖長Ｃ１２〜Ｃ１８の飽和脂肪アルコールのカプリル／カプリン酸エステル、ステアリン酸イソプロピル、オレイン酸オレイル、オレイン酸デシル、オレイン酸エチル、乳酸エチル、ワックス状脂肪酸エステル、フタル酸ジブチル、アジピン酸ジイソプロピル、イソトリデシルアルコール、２−オクチルドデカノール、セチルステアリルアルコール、オレイルアルコールが挙げられる。   As hydrophobic phase (oil), paraffin oil, silicone oil, sesame oil, almond oil, castor oil, synthetic triglyceride, ethyl stearate, di-n-butyryl adipate, hexyl laurate, dipropylene glycol pelargonate, branched chain Of a short fatty acid having a chain length and a saturated fatty acid having a chain length of C16 to C18, isopropyl myristate, isopropyl palmitate, capryl / caprate of a saturated fatty alcohol having a chain length of C12 to C18, isopropyl stearate, oleyl oleate Decyl oleate, ethyl oleate, ethyl lactate, waxy fatty acid ester, dibutyl phthalate, diisopropyl adipate, isotridecyl alcohol, 2-octyldodecanol, cetyl stearyl alcohol, oleyl alcohol It is.

親水性相としては、水、プロピレングリコール、グリセリン、ソルビトールが挙げられる。   Examples of the hydrophilic phase include water, propylene glycol, glycerin, and sorbitol.

乳化剤としては、ポリオキシエチル化されたヒマシ油、ポリオキシエチル化されたモノオレフィン酸ソルビタン、モノステアリン酸ソルビタン、モノステアリン酸グリセリン、ステアリン酸ポリオキシエチル、アルキルフェノールポリグリコールエーテルなどの非イオン性界面活性剤；Ｎ−ラウリル−β−イミノジプロピオン酸二ナトリウム、レシチンなどの両性界面活性剤；ラウリル硫酸ナトリウム、脂肪アルコール硫酸エーテル、モノ／ジアルキルポリグリコールオルトリン酸エステルのモノエタノールアミン塩などの陰イオン性界面活性剤；塩化セチルトリメチルアンモニウムなどの陽イオン性界面活性剤などが挙げられる。   Emulsifiers include nonionic interfaces such as polyoxyethylated castor oil, polyoxyethylated sorbitan monoolefin acid, sorbitan monostearate, glyceryl monostearate, polyoxyethyl stearate, alkylphenol polyglycol ether, etc. Activators; amphoteric surfactants such as disodium N-lauryl-β-iminodipropionate and lecithin; anions such as sodium lauryl sulfate, fatty alcohol sulfate ether, monoethanolamine salt of mono / dialkyl polyglycol orthophosphate Surfactants; cationic surfactants such as cetyltrimethylammonium chloride.

他の補助剤として、カルボキシメチルセルロース、メチルセルロース、ポリアクリレート、アルギネート、ゼラチン、アラビアゴム、ポリビニルピロリドン、ポリビニルアルコール、メチルビニルエーテル、無水マレイン酸の共重合体、ポリエチレングリコール、ワックス、コロイド状シリカが挙げられる。   Other adjuvants include carboxymethyl cellulose, methyl cellulose, polyacrylate, alginate, gelatin, gum arabic, polyvinyl pyrrolidone, polyvinyl alcohol, methyl vinyl ether, a copolymer of maleic anhydride, polyethylene glycol, wax, colloidal silica.

半固体調製物は皮膚上に塗布するか、もしくは広げるか、又は体腔中に導入することにより投与できる。ゲルは注射用液剤について上記したように調製した溶液に、軟膏状の粘稠性を有する透明な物質を生じさせるに十分なシックナーを加えることにより調製できる。   Semi-solid preparations can be administered by application on the skin or spreading or introduction into body cavities. Gels can be prepared by adding sufficient thickener to a solution prepared as described above for an injectable solution to produce a clear material having an ointment-like consistency.

次に本発明化合物を用いる場合の製剤の配合例を示す。但し本発明の配合例は、これらのみに限定されるものではない。なお、以下の配合例において「部」は重量部を意味する。   Next, formulation examples of the preparation when using the compound of the present invention are shown. However, the formulation examples of the present invention are not limited to these. In the following formulation examples, “parts” means parts by weight.

〔水和剤〕
本発明化合物 ０.１〜８０部
固体担体 ５〜９８.９部
界面活性剤 １〜１０部
その他 ０〜５部
その他として、例えば固結防止剤、分解防止剤等があげれらる。 [Wettable powder]
Compound of the present invention 0.1 to 80 parts Solid carrier 5 to 98.9 parts Surfactant 1 to 10 parts Others 0 to 5 parts Other examples include anti-caking agents and decomposition inhibitors.

〔乳 剤〕
本発明化合物 ０.１〜３０部
液体担体 ４５〜９５部
界面活性剤 ４.９〜１５部
その他 ０〜１０部
その他として、例えば展着剤、分解防止剤等が挙げられる。 [Milk]
Compound of the present invention 0.1-30 parts Liquid carrier 45-95 parts Surfactant 4.9-15 parts Others 0-10 parts Others include, for example, spreading agents, decomposition inhibitors, and the like.

〔懸濁剤〕
本発明化合物 ０.１〜７０部
液体担体 １５〜９８.８９部
界面活性剤 １〜１２部
その他 ０.０１〜３０部
その他として、例えば凍結防止剤、増粘剤等が挙げられる。 [Suspension]
Compound of the present invention 0.1 to 70 parts Liquid carrier 15 to 98.89 parts Surfactant 1 to 12 parts Others 0.01 to 30 parts Others include, for example, antifreezing agents and thickeners.

〔顆粒水和剤〕
本発明化合物 ０.１〜９０部
固体担体 ０〜９８.９部
界面活性剤 １〜２０部
その他 ０〜１０部
その他として、例えば結合剤、分解防止剤等が挙げられる。 [Granule wettable powder]
Compound of the present invention 0.1 to 90 parts Solid carrier 0 to 98.9 parts Surfactant 1 to 20 parts Others 0 to 10 parts Others include, for example, binders and decomposition inhibitors.

〔液 剤〕
本発明化合物 ０.０１〜７０部
液体担体 ２０〜９９.９９部
その他 ０〜１０部
その他として、例えば凍結防止剤、展着剤等が挙げられる。 (Liquid)
Compound of the present invention 0.01 to 70 parts Liquid carrier 20 to 99.99 parts Others 0 to 10 parts Other examples include antifreezing agents and spreading agents.

〔粒 剤〕
本発明化合物 ０.０１〜８０部
固体担体 １０〜９９.９９部
その他 ０〜１０部
その他として、例えば結合剤、分解防止剤等が挙げられる。 [Granule]
Compound of the present invention 0.01 to 80 parts Solid carrier 10 to 99.99 parts Others 0 to 10 parts Others include, for example, binders, decomposition inhibitors and the like.

〔粉 剤〕
本発明化合物 ０.０１〜３０部
固体担体 ６５〜９９.９９部
その他 ０〜５部
その他として、例えばドリフト防止剤、分解防止剤等が挙げられる。 [Dust]
Compound of the present invention 0.01 to 30 parts Solid support 65 to 99.99 parts Others 0 to 5 parts Other examples include a drift inhibitor and a decomposition inhibitor.

次に、本発明化合物を有効成分とする製剤例をより具体的に示すが、本発明はこれらに限定されるものではない。   Next, although the formulation example which uses this invention compound as an active ingredient is shown more concretely, this invention is not limited to these.

尚、以下の配合例において、「部」は重量部を意味する。   In the following formulation examples, “parts” means parts by weight.

〔配合例１〕水和剤
本発明化合物No.１-００１ ２０部
パイロフィライト ７４部
ソルポール５０３９ ４部
（非イオン性界面活性剤とアニオン性界面活性剤との混合物：東邦化学工業（株）商品名）
カープレックス＃８０Ｄ ２部
（合成含水珪酸：塩野義製薬（株）商品名）
以上を均一に混合粉砕して水和剤とする。 [Formulation Example 1] wettable powder Compound No.1-001 20 parts pyrophyllite 74 parts Solpol 5039 4 parts (mixture of nonionic surfactant and anionic surfactant: Toho Chemical Co., Ltd.) Product name)
Carplex # 80D 2 parts (Synthetic hydrous silicic acid: Shionogi & Co., Ltd. trade name)
The above is uniformly mixed and ground to obtain a wettable powder.

〔配合例２〕乳 剤
本発明化合物No.１-００１ ５部
キシレン ７５部
Ｎ−メチルピロリドン １５部
ソルポール２６８０ ５部
（非イオン性界面活性剤とアニオン性界面活性剤との混合物：東邦化学工業（株）商品名）
以上を均一に混合して乳剤とする。 [Formulation Example 2] Milk Compound of the present invention No.1-001 5 parts Xylene 75 parts N-methylpyrrolidone 15 parts Solpol 2680 5 parts (mixture of nonionic surfactant and anionic surfactant: Toho Chemical Industry (Product name)
The above is uniformly mixed to obtain an emulsion.

〔配合例３〕懸濁剤
本発明化合物No.１-００１ ２５部
アグリゾールＳ−７１０ １０部
（非イオン性界面活性剤：花王（株）商品名）
ルノックス１０００Ｃ ０.５部
（アニオン性界面活性剤：東邦化学工業（株）商品名）
キサンタンガム ０.２部
水 ６４.３部
以上を均一に混合した後、湿式粉砕して懸濁剤とする。 [Formulation Example 3] Suspension Agent Compound No.1-001 25 parts Agrisol S-710 10 parts (Nonionic Surfactant: Kao Corporation trade name)
LUNOX 1000C 0.5 part (anionic surfactant: Toho Chemical Industries, Ltd. trade name)
Xanthan gum 0.2 parts water 64.3 parts After uniformly mixing the above, wet pulverize to make a suspension.

〔配合例４〕顆粒水和剤
本発明化合物No.１-００１ ７５部
ハイテノールNE-15 ５部
（アニオン性界面活性剤：第一工業製薬（株）商品名）
バニレックスＮ １０部
（アニオン性界面活性剤：日本製紙（株）商品名）
カープレックス＃８０Ｄ １０部
（合成含水珪酸：塩野義製薬（株）商品名）
以上を均一に混合粉砕した後、少量の水を加えて撹拌混合し、押出式造粒機で造粒し、乾燥して顆粒水和剤とする。 [Composition Example 4] Granule wettable powder Compound No.1-001 of the present invention 75 parts Hytenol NE-15 5 parts (anionic surfactant: Daiichi Kogyo Seiyaku Co., Ltd. trade name)
Vanillex N 10 parts (anionic surfactant: Nippon Paper Industries Co., Ltd. trade name)
Carplex # 80D 10 parts (Synthetic hydrous silicic acid: Shionogi Pharmaceutical Co., Ltd. trade name)
After uniformly mixing and pulverizing the above, a small amount of water is added, stirred and mixed, granulated with an extrusion granulator, and dried to obtain a granulated wettable powder.

〔配合例５〕粒 剤
本発明化合物No.１-００１ ５部
ベントナイト ５０部
タルク ４５部
以上を均一に混合粉砕した後、少量の水を加えて撹拌混合し、押出式造粒機で造粒し、乾燥して粒剤とする。 [Formulation Example 5] Granules Invention compound No. 1-101 5 parts Bentonite 50 parts Talc 45 parts And dried into granules.

〔配合例６〕粉 剤
本発明化合物No.１-００１ ３部
カープレックス＃８０Ｄ ０.５部
（合成含水珪酸：塩野義製薬（株）商品名）
カオリナイト ９５部
リン酸ジイソプロピル １.５部
以上を均一に混合粉砕して粉剤とする。 [Composition Example 6] Powder Compound of the present invention No.1-001 3 parts Carplex # 80D 0.5 part (Synthetic hydrous silicic acid: Shionogi Pharmaceutical Co., Ltd. trade name)
Kaolinite 95 parts Diisopropyl phosphate 1.5 parts The above is uniformly mixed and ground to obtain a powder.

使用に際しては、上記製剤を水で１〜１００００倍に希釈して、又は希釈せずに直接散布する。   In use, the above preparation is diluted 1 to 10000 times with water or sprayed directly without dilution.

〔配合例７〕水和剤調製物
本発明化合物No.１-００１ ２５部
ジイソブチルナフタレンスルホン酸ナトリウム １部
ｎ−ドデシルベンゼンスルホン酸カルシウム １０部
アルキルアリール ポリグリコールエーテル １２部
ナフタレンスルホン酸ホルマリン縮合物のナトリウム塩 ３部
エマルジョン型シリコーン １部
二酸化ケイ素 ３部
カオリン ４５部
〔配合例８〕水溶性濃厚剤調製物
本発明化合物No.１-００１ ２０部
ポリオキシエチレンラウリルエーテル ３部
ジオクチルスルホコハク酸ナトリウム ３.５部
ジメチルスルホキシド ３７部
２−プロパノール ３６.５部
〔配合例９〕噴霧用液剤
本発明化合物No.１-００１ ２部
ジメチルスルホキシド １０部
２−プロパノール ３５部
アセトン ５３部
〔配合例１０〕経皮投与用液剤
本発明化合物No.１-００１ ５部
ヘキシレングリコール ５０部
イソプロパノール ４５部
〔配合例１１〕経皮投与用液剤
本発明化合物No.１-００１ ５部
プロピレングリコールモノメチルエーテル ５０部
ジプロピレングリコール ４５部
〔配合例１２〕経皮投与(滴下)用液剤
本発明化合物No.１-００１ ２部
軽質流動パラフィン ９８部
〔配合例１３〕経皮投与(滴下)用液剤
本発明化合物No.１-００１ ２部
軽質流動パラフィン ５８部
オリーブ油 ３０部
ＯＤＯ−Ｈ ９部
信越シリコーン １部
また、本発明化合物を農薬として使用する場合には、必要に応じて製剤時又は散布時に他種の除草剤、各種殺虫剤、殺ダニ剤、殺線虫剤、殺菌剤、植物生長調節剤、共力剤、肥料、土壌改良剤等と混合施用しても良い。 [Formulation Example 7] wettable powder preparation Compound No. 1-001 of the present invention 25 parts sodium diisobutylnaphthalenesulfonate 1 part calcium n-dodecylbenzenesulfonate 10 parts alkylaryl polyglycol ether 12 parts naphthalenesulfonic acid formalin condensate Sodium salt 3 parts Emulsion type silicone 1 part Silicon dioxide 3 parts Kaolin 45 parts [Formulation Example 8] Water-soluble thickener preparation Compound No.1-001 20 parts Polyoxyethylene lauryl ether 3 parts Sodium dioctyl sulfosuccinate 3. 5 parts dimethyl sulfoxide 37 parts 2-propanol 36.5 parts [Formulation Example 9] Solution for spraying the present compound No.1-001 2 parts dimethyl sulfoxide 10 parts 2-propanol 35 parts acetone 53 parts [Formulation Example 10] transdermal Solution for administration The present compound No.1-001 5 Parts hexylene glycol 50 parts isopropanol 45 parts [Formulation Example 11] Solution for transdermal administration Compound No. 1-001 5 parts propylene glycol monomethyl ether 50 parts Dipropylene glycol 45 parts [Formulation example 12] transdermal administration (instillation) ) Solution for the Invention Compound No.1-001 2 parts Light Liquid Paraffin 98 parts [Formulation Example 13] Solution for the transdermal administration (drip) Compound No.1-001 2 parts Light Liquid Paraffin 58 parts Olive Oil 30 parts ODO -H 9 parts Shin-Etsu Silicone 1 part In addition, when the compound of the present invention is used as an agrochemical, other types of herbicides, various insecticides, acaricides, nematicides, You may mix and apply with a disinfectant, a plant growth regulator, a synergist, a fertilizer, a soil conditioner, etc.

特に他の農薬あるいは植物ホルモンと混合施用することにより、施用薬量の低減による低コスト化、混合薬剤の相乗作用による殺虫スペクトラムの拡大やより高い有害生物防除効果が期待できる。この際、同時に複数の公知農薬との組み合わせも可能である。本発明化合物と混合使用する農薬の種類としては、例えばザ・ペスティサイド・マニュアル（The Pesticide Manual）１５版、２００９年に記載されている化合物等が挙げられる。具体的にその一般名を例示すれば次の通りであるが、必ずしもこれらのみに限定されるものではない。   In particular, when mixed with other pesticides or plant hormones, the cost can be reduced by reducing the amount of applied medicine, the insecticidal spectrum can be expanded by the synergistic action of the mixed drugs, and higher pest control effects can be expected. At this time, a combination with a plurality of known agricultural chemicals is also possible. Examples of the type of agricultural chemical used in combination with the compound of the present invention include compounds described in The Pesticide Manual 15th edition, 2009, and the like. Specific examples of common names are as follows, but the general names are not necessarily limited to these.

殺菌剤：アシベンゾラルーＳ−メチル（acibenzolar-S-methyl）、アシルアミノベンザミド(acylaminobenzamide)、アシペタックス(acypetacs)、アルジモルフ(aldimorph)、アミスルブロム(amisulbrom)、アンバム(amobam)、アムプロピルホス（ampropyfos）、アニラジン（anilazine）、アザコナゾール（azaconazole）、アジチラム(azithiram)、アゾキシストロビン（azoxystrobin）、バリウムポリサルファイド(barium polysulfide)、ベナラキシル（benalaxyl）、ベノダニル（benodanil）、ベノミル（benomyl）、ベンキノックス(benquinox)、ベンタルロン(bentaluron)、ベンチアバリカルブ(benthiavalicarb)、ベンチアゾール(benthiazole)、ベンザマクリル（benzamacril）、ベンズアモルフ(benzamorf)、ベトキサジン（bethoxazine）、ビナパクリル（binapacryl）、ビフェニル（biphenyl）、ビテルタノール（bitertanol）、ブラストサイジン−Ｓ（blasticidin-S）、ボルドー液（bordeaux mixture）、ボスカリド(boscalid)、ブロモコナゾール（bromoconazole）、ブピリメート（bupirimate）、ブチオベート（buthiobate）、カルシウムポリスルフィド（calcium polysulfide）、キャプタフォール（captafol）、キャプタン（captan）、カルプロパミド（carpropamid）、カルバモルフ(carbamorph)、カルベンダジン（carbendazim）、カルボキシン（carboxin）、カルボン(carvone)、チェシュントミクスチャ(cheshunt mixture)、キノメチオネート（chinomethionat）、クロベンチアゾン（chlobenthiazone）、クロラニフォルメタン(chloraniformethane)、クロラニル(chloranil)、クロルフェナゾール（chlorfenazol）、クロロネブ（chloroneb）、クロロピクリン(chloropicrin)、クロロタロニル（chlorothalonil）、クロロキノックス(chlorquinox)、クロゾリネート（chlozolinate）、クリムバゾール(climbazole)、クロトリマゾール(clotrimazole)、カッパーアセテイト(copper acetate)、塩基性炭酸銅(copper carbonate, basic)、水酸化第二銅(copper hydroxide)、カッパーナフタレン(copper naphthenate)、カッパーオルアイト(copper oleate)、カッパーオキシクロリド（copper oxychloride）、硫酸銅(copper sulfate)、塩基性硫酸銅(copper sulfate, basic)、カッパージンククロメイト(copper zinc chromate)、クフラネブ（cufraneb）、クプロバム(cuprobam)、シアゾファミド(cyazofamid)、シクラフルアミド(cyclafuramid)、シクロヘキシミド(cycloheximide)、シフルフェナミド(cyflufenamid)、シモキサニル（cymoxanil）、サイペンダゾール(cypendazole)、シプロコナゾール（cyproconazol）、シプロジニル（cyprodinil）、シプロフラム（cyprofuram）、ダゾメット(dazomet)、デバカルブ（debacarb）、デカフェンチン(decafentin)、デハイドロアセテイト(dehydroacetic acid)、ジクロフルアニド（dichlofluanid）、ジクロン(dichlone)、ジクロロフェン（dichlorophen）、ジクロゾリン(dichlozoline)、ジクロブトラゾール（diclobutrazol）、ジクロシメット（diclocymet）、ジクロメジン（diclomedine）、ジクロラン（dicloran）、ジエトフェンカルブ（diethofencarb）、ジフェノコナゾール（difenoconazole）、ジフルメトリン（diflumetorim）、ジメチリモール（dimethirimol）、ジメトモルフ（dimethomorph）、ジモキシストロビン(dimoxystrobin)、ジニコナゾール（diniconazole）、ジニコナゾール−Ｍ（diniconazole-M）、ジノブトン(dinobuton)、ジノカップ（dinocap）、ジノカップ−４(dinocap-4)、ジノカップ−６(dinocap-6)、ジノクトン(dinocton)、ジノスルフォン(dinosulfon)、ジノテルボン(dinoterbon)、ジフェニルアミン（diphenylamine）、ジピリチオン（dipyrithione）、ジタリムホス（ditalimfos）、ジチアノン（dithianon）、ドデモルフ（dodemorph）、ドジン（dodine）、ドラゾクソロン（drazoxolon）、エデフェノホス（edifenphos）、エポキシコナゾール（epoxiconazole）、エタコナゾール（etaconazole）、エテム(etem)、エチリモル（ethirimol）、エトキシキン(ethoxyquin)、エトリジアノール（etridiazole）、ファモキサゾン（famoxadone）、フェナリモル（fenarimol）、フェブコナゾール（febuconazole）、フェナミドン（fenamidone）、フェナミノスルフ(fenaminosulf)、フェナパニル(fenapanil)、フェンダゾスラム(fendazosulam)、フェンフラム（fenfuram）、フェンヘキサミド（fenhexamid）、フェニトロパン(fenitropan)、フェノキサニル(fenoxanil)、フェンピクロニル（fenpiclonil）、フェンプロピジン（fenpropidin）、フェンプロピモルフ（fenpropimorph）、フェンチン（fentin）、フェルバン（ferbam）、フェリムゾン（ferimzone）、フルアジナム（fluazinam）、フルジオキソニル（fludioxonil）、フルメトベル(flumetover)、フルモルフ(flumorph)、フルオピコリド（fluopicolide）、フルオロイミド（fluoroimide）、フルオトリマゾール(fluotrimazole)、フルオキサストロビン(fluoxastrobin)、フルキンコナゾール（fluquinconazole）、フルシラゾール（flusilazole）、フルスルファミド（flusulfamide）、フルトラニル（flutolanil）、フルトリアフォール（flutriafol）、フォルペット（folpet）、フォセチル−アルミニウム（fosetyl-aluminium）、フベリダゾール（fuberidazole）、フララキシル（furalaxyl）、フラメトピル(furametpyr)、フルカルバニル(furcarbanil)、フルコナゾール(furconazole)、フルコナゾール−シス(furconazole-cis)、フルメシクロックス(furmecyclox)、フルファネート(furphanate)、グリオジン(glyodin)、グリセオフルビン(griseofulvin)、グアザチン（guazatine）、ハラクリネイト(halacrinate)、ヘキサクロロベンゼン（hexachlorobenzene）、ヘキサコナゾール（hexaconazole）、ヘキシルチオフォス(hexylthiofos)、ハイドロキシキノリン サルフェイト(8-hydroxyquinoline sulfate)、ヒメキサゾール（hymexazol）、イマザリル（imazalil）、イミベンコナゾール（imibenconazole）、イミノクタジン（iminoctadine）、イプコナゾール（ipconazole）、イプロベンホス（iprobenfos）、イプロジオン（iprodione）、イプロバリカルブ（iprovalicarb）、イソプロチオラン（isoprothiolane）、イソバレジオン(isovaledione)、カスガマイシン（kasugamycin）、クレソキシム−メチル（kresoxim-methyl）、マンカッパー（mancopper）、マンコゼブ（mancozeb）、マンジプロパミド（mandipropamid）、マンネブ（maneb）、メベニル（mebenil）、メカルビンジド（mecarbinzid）、メパニピリム（mepanipyrim）、メプロニル（mepronil）、メタラキシル（metalaxyl）、メタラキシル−Ｍ（metalaxyl-M）、メタム（metam）、メタゾキソロン（metazoxolon）、メトコナゾール（metconazole）、メタスルホカルブ(methasulfocarb)、メトフロキサム（methfuroxam）、メチルイソチオシアネイト（methyl isothiocyanate）、メチラム（metiram）、メトミノストロビン（metominostrobin）、メトラフェノン（metrafenone）、メトスルフォバックス（metsulfovax）、ミルネブ（milneb）、ミクロブタニル（myclobutanil）、ミクロゾリン（myclozolin）、ナバム（nabam）、ナタマイシン（natamycin）、ニッケルビス（ジメチルジチオカーバメート）（nickel bis(dimethyldithiocarbamate)）、ニトロスチレン（nitrostyrene）、ニトロタール−イソプロピル（nitrothal-isopropyl）、ヌアリモル（nuarimol）、オーシーエイチ（OCH）、オクチリノン（octhilinone）、オフレース（ofurace）、オリサストロビン（orysastrobin）、オキサジキシル（oxadixyl）、有機銅（oxine copper）、オキシカルボキシン（oxycarboxin）、オキスポコナゾールフマール酸塩（oxpoconazole fumarate）、ペフラゾエート（pefurzoate）、ペンコナゾール（penconazole）、ペンシクロン（pencycuron）、ペンチオピラド（penthiopyrad）、オルソフェニルフェノール（o-phenylphenol）、フォスジフェン（phosdiphen）、フタライド（phthalide）、ピコキシストロビン（picoxystrobin）、ピペラリン（piperalin）、ポリカーバメート（polycarbamate）、ポリオキシン（polyoxins）、ポリオクソリム（polyoxorim）、ポタシウムアザイド（potassium azide）、炭酸水素カリウム(potassium hydrogen carbonate)、プロキナジド（proquinazid）、プロベナゾール（probenazole）、プロクロラズ（prochloraz）、プロシミドン（procymidone）、プロパモカルブ塩酸塩（propamocarb hydrochloride）、プロピコナゾール（propiconazole）、プロピネブ（propineb）、プロチオカルブ（prothiocarb）、プロチオコナゾール（prothioconazole）、ピラカルボリド（pyracarbolid）、ピラクロストロビン（pyraclostrobin）、ピラゾホス（pyrazophos）、ピリジニトリル（pyridinitril）、ピリフェノックス（pyrifenox）、ピリメタニル（pyrimethanil）、ピロキュロン（pyroquilon）、ピロキシクロル（pyroxychlor）、ピロキシフル（pyroxyfur）、キノメチオネート(quinomethionate)、キノキシフェン（quinoxyfen）、キントゼン（quintozene）、キナセトール・スルフェート（quinacetol-sulfate）、キナザミド（quinazamid）、キンコナゾール（quinconazole）、ラベンザゾール（rabenzazole）、アジ化ナトリウム（sodium azide）、炭酸水素ナトリウム(sodium hydrogen carbonate)、次亜塩素酸ナトリウム(sodium hypochlorite)、硫黄（sulfur）、スピロキサミン（spiroxamine）、サリチルアニリド（salycylanilide）、シルチオファム（silthiofam）、シメコナゾール（simeconazole）、テブコナゾール（tebuconazole）、テクナゼン（tecnazene）、テコラム（tecoram）、テトラコナゾール（tetraconazole）、チアベンダゾール（thiabendazole）、チアジフルオール（thiadifluor）、チシオフェン（thicyofen）、チフルザミド（thifluzamide）、チオクロルフェンフィム（thiochlorfenphim）、チオファネート（thiophanate）、チオファネート−メチル（thiophanate-methyl）、チオキノックス（thioquinox）、チラム（thiram）、チアジニル（tiadinil）、チオキシミド（tioxymid）、トルクロホス−メチル（tolclofos-methyl）、トリルフラニド（tolylfluanid）、トリアジメホン（triadimefon）、トリアジメノール（toriadimenol）、トリアミフォス（triamiphos）、トリアリモル（triarimol）、トリアゾキシド（triazoxide）、トリアズブチル（triazbutil）、トリブチルチンオキサイド（tributyltin oxide）、トリクラミド（trichlamide）、トリシクラゾール（tricyclazole）、トリデモルフ（tridemorph）、トリフロキシストロビン(trifloxystrobin)、トリフルミゾール（triflumizole）、トリホリン（triforine）、トリチコナゾール（triticonazole）、バリダマイシン（validamycin）、ビンクロゾリン（vinclozolin）、ザリルアミド（zarilamide）、硫酸亜鉛(zinc sulfate)、ジネブ（zineb）、ジラム（ziram）、ゾキサミド（zoxamide）及びシイタケ菌糸体抽出物など。   Bactericides: acibenzolar-S-methyl, acylaminobenzamide, acypetacs, aldimorph, amisulbrom, amobam, ampropyfos, Anilazine, azaconazole, azithiram, azoxystrobin, barium polysulfide, benalaxyl, benodanil, benomyl, benquinox , Benthaluron, benthiavalicarb, benthiazole, benzamacril, benzamorf, bethoxazine, binapacryl, biphenyl, bitertanol ,blast Idin-S (blasticidin-S), Bordeaux mixture, boscalid, bromoconazole, bupirimate, buthiobate, calcium polysulfide, captafol , Captan, carpropamid, carbamorph, carbendazim, carboxin, carvone, carvone, cheshunt mixture, chinomethionat, clobenazone (Chlobenthiazone), chloraniformethane, chloranil, chlorfenazol, chloroneb, chloropicrin, chlorothalonil, chlorquinox, clozolinate linate), climbazole, clotrimazole, copper acetate, basic carbonate, copper carbonate, copper hydroxide, copper naphthenate , Copper oleate, copper oxychloride, copper sulfate, copper sulfate, basic, copper zinc chromate, cufraneb, Cuprobam, cyazofamid, cyclafuramid, cycloheximide, cyflufenamid, cymoxanil, cypendazole, cyproconazol, din , Cyprofuram, dazomet, debacarb, decafenci Decafentin, dehydroacetic acid, dichlofluanid, dichlone, dichlorophen, dichlorophenoline, diclobutrazol, diclocymet, Diclomedine, dicloran, diethofencarb, difenoconazole, diflumetorim, dimethirimol, dimethomorph, dimethomorph, dimoxystrobin, dimoxystrobin M (diniconazole-M), dinobuton, dinocap, dinocap-4, dinocap-6, dinoton, dinosulfon, dinoterbon , Diphenylamine mine, dipyrithione, ditalimfos, dithianon, dodemorph, dodine, drazoxolone, edifenphos, epoxiconazole, etaconazole, eta Etem, ethirimol, ethoxyquin, etridiazole, famoxadone, fenarimol, febuconazole, fenamidone, fenaminosulf, fenilil ), Fendazosulam, fenfuram, fenhexamid, fenitropan, fenoxanil, fenpiclonil, fenpropidin, fenproidin Morph (fenpropimorph), fentin, ferbam, ferimzone, fluazinam, fludioxonil, flumetover, flumetover, flumorph, fluopicolide, fluoroimide , Fluotrimazole, fluoxastrobin, fluquinconazole, flusilazole, flusulfamide, flutolanil, flutriafol, folpet , Fosetyl-aluminium, fuberidazole, furalaxyl, furametpyr, furcarbanil, furconanol, fluconazole-cis, furconazole-cis Memecyclox, furphanate, glyodin, griseofulvin, guazatine, halacrineate, hexachlorobenzene, hexaconazole, hexylthiofos , Hydroxyquinoline sulfate, hymexazol, imazalil, imibenconazole, iminoctadine, ipconazole, iprobenfos, iprobenfos, proprobion (Iprovalicarb), isoprothiolane, isovaledione, kasugamycin, kresoxim-methyl, mancopper, mancozeb ozeb, mandipropamid, maneb, mebenil, mecarbinzid, mepanipyrim, mepronil, metalaxyl, metalaxyl-M, metalaxyl-M ), Metazoxolon, metconazole, methasulfocarb, metfuroxam, methyl isothiocyanate, metiram, metinofenstro, metolafenone, metrafenone Metsulfovax, milneb, microbutanil, myclozolin, nabam, natamycin, nickel bis (dimethyldithiocarbamate), Nitrostyrene, nitrothal-isopropyl, nuarimol, ochirinone, octhilinone, offurace, orysastrobin, oxadixyl, organic copper ( oxine copper, oxycarboxin, oxpoconazole fumarate, pefurzoate, penconazole, pencycuron, penthiopyrad, ortho-phenylphenol ), Phosdiphen, phthalide, picoxystrobin, piperalin, polycarbamate, polyoxins, polyoxorim, potassium azide potassium azide, potassium hydrogen carbonate, proquinazid, probenazir, prochloraz, prochlorazone, promomidone, propamocarb hydrochloride, propiconazole, propiconazole (propiconazole) propineb, prothiocarb, prothioconazole, pyracarbolid, pyraclostrobin, pyrazophos, pyridiinitril, pyrifenox, pyrimethanil, piroculanil (Pyroquilon), pyroxychlor, pyroxyfur, quinomethionate, quinoxyfen, quintozene, quinacetosulfate (quinaceto) l-sulfate), quinazamid, quinconazole, rabenzazole, sodium azide, sodium hydrogen carbonate, sodium hypochlorite, sulfur ( sulfur, spiroxamine, salicylanilide, silthiofam, simeconazole, tebuconazole, tecnazene, tecoram, tetraconazole, thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole thiabendazole th , Thiadifluor, thicyofen, thifluzamide, thiochlorfenphim, thiophanate, thiophanate-methyl, thioquinox, thira (Thiram), thiadinil, tioxymid, tolclofos-methyl, tolylfluanid, triadimefon, triadimenol, triamiphos, triarimol, Triazoxide, triazbutil, tributyltin oxide, trichlamide, tricyclazole, triridemorph, trifloxystrobin, triflumizole, triphorin (triflumizole) triforine, triticonazole, validamycin, vinclozolin, zalilamide, zinc sulfate, zineb, ziram, zoxamid e) and shiitake mycelium extract.

殺バクテリア剤：ベンザルコニウムクロライド(benzalkonium chloride)、ビチオノール(bithionol)、ブロノポール（bronopol）、クレゾール(cresol)、ホルムアルデヒド（formaldehyde）、ニトラピリン（nitrapyrin）、オキソリニックアシド（oxolinic acid）、オキシテトラサイクリン（oxyterracycline）、ストレプトマイシン（streptomycin）及びテクロフタラム(tecloftalam)など。   Bactericides: benzalkonium chloride, bithionol, bronopol, cresol, formaldehyde, nitrapyrin, oxolinic acid, oxyterracycline , Streptomycin and tecloftalam.

殺線虫剤：アルドキシカルブ（aldoxycarb）、カズサホス（cadusafos）、デービーシーピー(DBCP)、ジクロフェンチオン（dichlofenthion）、デーエスピー（DSP）、エトプロホス（ethoprophos）、フェナミホス（fenamiphos）、フェンスルホチオン（fensulfothion）、フォスチアゼート（fosthiazate）、フォスチエタン（fosthietan）、イミシアホス（imicyafos）、イサミドホス（isamidofos）、イサゾホス（isazofos）、オキサミル（oxamyl）及びチオナジン（thionazin）など。   Nematicides: aldoxycarb, cadusafos, DDBCP, dichlofenthion, DSP (DSP), etoprophos, fenamiphos, fensulfothion, fostiazeto (Fosthiazate), fosthietan, imiciafos, isamifos, isazofos, oxamyl and thionazin.

殺ダニ剤：アセキノシル（acequinocyl）、アクリナトリン（acrinathrin）、アミトラズ（amitraz）、ＢＣＩ−０３３（試験名）、ビフェナゼート（bifenazate）、ブロモプロピレート（bromopropylate）、チノメチオネート（chinomethionat）、クロロベンジラート（chlorobezilate）、クロフェンテジン（clofentezine）、シエノピラフェン（cyenopyrafen）、シフルメトフェン（cyflumetofen）、サイヘキサチン（cyhexatine）、ジコフォール（dicofol）、ジエノクロール（dienochlor）、デーエヌオーシー(DNOC)、エトキサゾール（etoxazole）、フェナザキン（fenazaquin）、フェンブタチンオキシド（fenbutatin oxide）、フェノチオカルブ（fenothiocarb）、フェンプロパトリン（fenpropathrin）、フェンピロキシメート（fenpyroximate）、フルアクリピリム（fluacrypyrim）、ハルフェンプロックス（halfenprox）、ヘキシチアゾックス（hexythiazox）、ミルベメクチン（milbemectin）、プロパルギット（propargite）、ピリダベン（pyridaben）、ピリミジフェン（pyrimidifen）、Ｓ−１８７０（試験名）、スピロジクロフェン（spirodiclofen）、スピロメシフェン（spyromesifen）及びテブフェンピラド（tebufenpyrad）など。   Acaricide: acequinocyl, acrinathrin, amitraz, BCI-033 (test name), bifenazate, bromopropylate, chinomethionat, chlorobezilate , Clofentezine, cyenopyrafen, cyflumetofen, cyhexatine, dicofol, dienochlor, denochlor (DNOC), etoxazole, quinazaquin (fenaza) Fenbutatin oxide, fenothiocarb, fenpropathrin, fenpyroximate, fluacrypyrim, halfenprox (halfenpro) x), hexythiazox, milbemectin, propargite, pyridaben, pyrimidifen, S-1870 (test name), spirodiclofen, spiromesifen ( spyromesifen) and tebufenpyrad.

殺虫剤：アバメクチン（abamectin）、アセフェート（acephate）、アセタミピリド（acetamipirid）、アラニカルブ（alanycarb）、アルディカルブ（aldicarb）、アレスリン（allethrin）、アジンホス−メチル（azinphos-methyl）、バチルスチューリンゲシス（bacillus thuringiensis）、ベンジオカルブ（bendiocarb）、ベンフラカルブ（benfuracarb）、ベンスルタップ（bensultap）、ビフェントリン（bifenthrin）、ブプロフェジン（buprofezin）、ブトカルボキシン（butocarboxim）、カルバリル（carbaryl）、カルボフラン（carbofuran）、カルボスルファン（carbosulfan）、カルタップ（cartap）、クロルアントラニリプロール（chlorantraniliprole）、クロルフェナピル（chlorfenapyr）、クロルフェンビンホス（chlorfenvinphos）、クロルフルアズロン（chlorfluazuron）、クロルピリホス（chlorpyrifos）、クロピリホス−メチル（chlorpyrifos-methyl）、クロマフェノジド（chromafenozide）、クロチアニジン（clothianidin）、シクロプロトリン（cycloprothrin）、シフルメトフェン（cyflumetofen）、シフルトリン（cyfluthrin）、ベータ−シフルトリン（beta-cyfluthrin）、シハロトリン（cyhalothrin）、ラムダ−シハロトリン（lambda-cyhalothrin）、シペルメトリン（cypermethrin）、シロマジン（cyromazine）、デルタメトリン（deltamethrin）、ジアクロデン（diacloden）、ジアフェンチウロン（diafenthiuron）、ダイアジノン（diazinon）、ジクロルボス（dichlorvos）、ジフルベンズロン（diflubenzuron）、ジメチルビンホス（dimethylvinphos）、ジノテフラン（dinotefuran）、ジオフェノラン（diofenolan）、ジスルフォトン（disulfoton）、ジメトエート（dimethoate）、エマメクチンベンゾエート（emamectin-benzoate）、イーピーエヌ（EPN）、エスフェンバレレート（esfenvalerate）、エチオフェンカルブ（ethiofencarb）、エチプロール（ethiprole）、エトフェンプロックス（etofenprox）、エトリムホス（etrimfos）、フェニトロチオン（fenitrothion）、フェノブカルブ（fenobucarb）、フェノキシカーブ（fenoxycarb）、フェンプロパトリン（fenpropathrin）、フェンチオン（fenthion）、フェンバレレート（fenvalerate）、フィプロニル（fipronil）、フロニカミド（flonicamid）、フルベンジアミド（flubendiamide）、フルシトリネート（flucythrinate）、フルフェネリム（flufenerim）、フルフェノクスウロン（flufenoxuron）、フルフェンプロックス（flufenprox）、フルバリネート（fluvalinate）、タウ−フルバリネート（tau-fluvalinate）、ホノホス（fonophos）、フォルメタネート（formetanate）、フォルモチオン（formothion）、フラチオカルブ（furathiocarb）、ハロフェノジド（halofenozide）、ヘキサフルムロン（hexaflumuron）、ヒドラメチルノン（hydramethylnon）、イミダクロプリド（imidacloprid）、イソフェンホス（isofenphos）、インドキサカルブ（indoxacarb）、イソプロカルブ（isoprocarb）、イソキサチオン（isoxathion）、レピメクチン（lepimectin）、ルフェヌウロン（lufenuron）、マラチオン（malathion）、メタルデヒド（metaldehyde）、メタミドホス（methamidophos）、メチダチオン（methidathion）、メタクリホス（methacrifos）、メタフルミゾン（metaflumizone）、メタルカルブ（metalcarb）、メソミル（methomyl）、メソプレン（methoprene）、メトキシクロール（methoxychlor）、メトキシフェノジド（methoxyfenozide）、メチルブロマイド（methyl bromide）、モノクロトホス（monocrotophos）、ムスカルーレ（muscalure）、ニテンピラム（nitenpyram）、ノバルロン（novaluron）、オメトエート（omethoate）、オキサミル（oxamyl）、オキシデメトン−メチル（oxydemeton-methyl）、オキシデプロホス（oxydeprofos）、パラチオン（parathion）、パラチオン−メチル（parathion-methyl）、ペンタクロロフェノール（pentachlorophenol(PCP)）、ペルメトリン（permethrin）、フェントエート（phenthoate）、フォキシム（phoxim）、ホレート（phorate）、ホサロン（phosalone）、ホスメット（phosmet）、ホスファミドン（phosphamidon）、ピリミカルブ（pirimicarb）、ピリミホス−メチル（pirimiphos-methyl）、プロフェノホス（profenofos）、プロチオホス（prothiofos）、プロパホス（propaphos）、プロトリフェンブト（protrifenbute）、ピメトロジン（pymetrozine）、ピラクロホス（pyraclofos）、ピリダリル（pyridalyl）、ピリフルキナゾン（pyrifluquinazon）、ピリプロキシフェン（pyriproxyfen）、ロテノン（rotenone）、ＳＩ−０４０５（試験名）、スルプロホス（sulprofos）、シラフルオフェン（silafluofen）、スピネトラム（spinetoram）、スピノサド（spinosad）、スピロテトラマート（spirotetramat）、スルホテップ（sulfotep）、ＳＹＪ−１５９（試験名）、テブフェノジド（tebfenozide）、テフルベンズロン（teflubenzuron）、テフルトリン（tefluthorin）、テルブホス（terbufos）、テトラクロロビンホス（tetrachlorvinphos）、チアクロプリド（thiacloprid）、チオシクラム（thiocyclam）、チオジカルブ（thiodicarb）、チアメトキサム（thiamethoxam）、チオファノックス（thiofanox）、チオメトン（thiometon）、トルフェンピラド（tolfenpyrad）、トラロメスリン（tralomethrin）、トリクロルホン（trichlorfon）、トリアズロン（triazuron）、トリフルムロン（triflumuron）及びバミドチオン（vamidothion）など。   Insecticides: abamectin, acephate, acetamipirid, alanycarb, aldicarb, allethrin, azinphos-methyl, bacillus thuringiensis ), Bendiocarb, benfuracarb, bensultap, bifenthrin, buprofezin, butocarboxim, carbaryl, carbofuran, carbosulfan , Cartap, chlorantraniliprole, chlorfenapyr, chlorfenvinphos, chlorfluazuron, chlorpyrifos, chlorpyrifos, chlorpyrifos, chlorpyrifos Pyrifos-methyl, chromafenozide, clothianidin, cycloprothrin, cyflumetofen, cyfluthrin, beta-cyfluthrin, cyhalothrin, cyhalothrin Lambda-cyhalothrin, cypermethrin, cyromazine, deltamethrin, diacloden, diafenthiuron, diazinon, dichlorvos, diflubenzuron diflubenzuron, dimethylvinphos, dinotefuran, diofenolan, disulfoton, dimethoate, emamectin-benzoat e), EPN, esfenvalerate, ethiofencarb, ethiprole, etofenprox, etrimfos, fenitrothion, fenobucarb, phenoxy curve fenoxycarb), fenpropathrin, fenthion, fenvalerate, fipronil, flonicamid, flubendiamide, flucythrinate, flufenerim, flufenerim Flufenoxuron, flufenprox, fluvalinate, tau-fluvalinate, fonophos, formetanate, formoti ON, formothion, furathiocarb, halofenozide, hexaflumuron, hydramethylnon, imidacloprid, isofenphos, indoxacarb, isoprocarb , Isoxathion, lepimectin, lufenuron, malathion, metalaldehyde, metamidophos, methidathion, methacrifos, metaflumizone, metaflumizone , Metomyl, metoprene, methoxychlor, methoxyfenozide, methyl bromide, monocrotophos Muscalure, nitenpyram, novaluron, omethoate, oxamyl, oxydemeton-methyl, oxydeprofos, parathion, parathion-methyl ( parathion-methyl, pentachlorophenol (PCP), permethrin, phenthoate, phenthoate, phoxim, phorate, phosalone, phosmet, phosphamidon, Pirimicarb, pirimiphos-methyl, profenfos, prothiofos, propaphos, protrifenbute, pymetrozine, pyraclofos, pyridali (Pyridalyl), pyrifluquinazon, pyriproxyfen, rotenone, SI-0405 (study name), sulprofos, silafluofen, spintoram, spinosad, spirosad Tetramart (spirotetramat), sulfotep (sulfotep), SYJ-159 (test name), tebfenozide (tebfenozide), teflubenzuron (teflubenzuron), tefluthorin (tefluthorin), terbufos (terbufos), tetrachlorovinphos (tetrachlorvinphos), thiacloprid (thiacloprid) ), Thiocyclam, thiodicarb, thiamethoxam, thiofanox, thiometon, tolfenpyrad, tralomethrin, triclometh Hong (trichlorfon), Toriazuron (triazuron), such as triflumuron (triflumuron) and vamidothion (vamidothion).

以下に本発明化合物の合成例、試験例を実施例として具体的に述べることで、本発明をさらに詳しく説明するが、本発明はこれらによって限定されるものではない。   Hereinafter, the present invention will be described in more detail by specifically describing synthesis examples and test examples of the compounds of the present invention as examples, but the present invention is not limited thereto.

合成例に記載したプロトン核磁気共鳴ケミカルシフト値は、基準物質としてＭｅ_４Ｓｉ（テトラメチルシラン）を用い、３００ＭＨｚにて測定した。 The proton nuclear magnetic resonance chemical shift value described in the synthesis example was measured at 300 MHz using Me ₄ Si (tetramethylsilane) as a reference substance.

合成例に記載した中圧分取液体クロマトグラフィーは、山善株式会社中圧分取装置；ＹＦＬＣ−Ｗｐｒｅｐ（流速１８ｍｌ／ｍｉｎ、シリカゲル４０μｍのカラム）を使用した。   The medium pressure preparative liquid chromatography described in the synthesis example used an intermediate pressure preparative apparatus (Yamazen Co., Ltd.);

［合成例］
合成例１
１−｛３−メチル−１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝エタノン Ｏ−メチル オキシムの製造（本発明化合物１−００３）
工程１
１−｛３−メチル−１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝エタノンの製造
３−ヨードピリジン１２．６ｇのＮ，Ｎ−ジメチルホルムアミド１００ｍｌ溶液に、別途調整した１−（３−メチル−１Ｈ−ピラゾール−４−イル）エタノン７．０８ｇのＮ，Ｎ−ジメチルホルムアミド２０ｍｌ溶液及び炭酸セシウム４６．３ｇを順次添加した。添加終了後、反応容器中を窒素ガスで置換した後に、ヨウ化銅（１価）２．３ｇを添加し、室温にて３０分攪拌した。攪拌終了後、１２０℃に昇温し、同温度で１５時間攪拌を継続した。反応終了後、該反応混合物を室温まで放冷した。放冷後に該反応混合物中に析出した不溶物を、減圧下にてセライトろ過により除去した後、ろ液に酢酸エチル２００ｍｌを添加した。得られた有機層を飽和食塩水、無水硫酸ナトリウムの順で洗浄・乾燥し、減圧下にて溶媒を留去した。得られた残渣をｎ−ヘキサン−酢酸エチル〔１：１〜１：９のグラジエント（体積比、以下同じである）〕にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物７．８ｇを白色固体として得た。
^１Ｈ ＮＭＲ（測定溶媒ＣＤＣｌ_３）δ８．９８（ｄ，Ｊ＝３．３Ｈｚ，１Ｈ），８．６０（ｄ，Ｊ＝４．８Ｈｚ，１Ｈ），８．３３（ｓ，１Ｈ），８．０５−８．１０（ｍ，１Ｈ），７．４３（ｄｄ，Ｊ＝４．８，８．４Ｈｚ，１Ｈ），２．５８（ｓ，３Ｈ），２．５０（ｓ，３Ｈ）
工程２
１−｛３−メチル−１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝エタノン Ｏ−メチル オキシムの製造
１−｛３−メチル−１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝エタノン２００ｍｇのメタノール１ｍｌ溶液に、Ｏ−メチルヒドロキシルアミン 塩酸塩９９．６ｍｇ添加し、室温にて一晩撹拌した。反応終了後、該反応混合物に水５ｍｌを添加し、酢酸エチル５ｍｌにて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。得られた固体を、クロロホルムで洗浄し目的物８２ｍｇを白色固体として得た。
融点；１５５−１５６℃
合成例２
３−［４−｛（トリメチルシリル）エチニル｝−１Ｈ−ピラゾール−１−イル］ピリジンの製造（本発明化合物２−００１）
３−（４−ヨード−１Ｈ−ピラゾール−１−イル）ピリジン１．０ｇのＮ，Ｎ−ジメチルホルムアミド２０ｍｌ溶液に、トリメチルシリルアセチレン７２５ｍｇ、ヨウ化銅（１価）５０ｍｇ、ジクロロビストリフェニルホスフィンパラジウム５０ｍｇ及びトリエチルアミン７４５ｍｇを順次添加した後、８０℃にて５時間撹拌した。反応終了後、該反応混合物に水３０ｍｌを添加し、酢酸エチル５０ｍｌにて抽出した。得られた有機層を、無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。得られた残渣をｎ−ヘキサン−酢酸エチル（４：６）にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物４００ｍｇを淡黄色固体として得た。
^１Ｈ ＮＭＲ（測定溶媒ＣＤＣｌ_３）δ８．９７（ｂｓ，１Ｈ），８．６０（ｄ，Ｊ＝３．６Ｈｚ，１Ｈ），８．０９（ｓ，１Ｈ），８．０４（ｄ，Ｊ＝８．１Ｈｚ，１Ｈ），７．８４（ｓ，１Ｈ），７．４３（ｄｄ，Ｊ＝８．１，４．８Ｈｚ，１Ｈ），０．２５（ｓ，９Ｈ）
融点；７９−８１℃
合成例３
３−（４−エチニル−１Ｈ−ピラゾール−１−イル）ピリジンの製造（本発明化合物２−００２）
３−［４−｛（トリメチルシリル）エチニル｝−１Ｈ−ピラゾール−１−イル］ピリジン２．３ｇのメタノール１０ｍｌ溶液に、炭酸カリウム２．０ｇを添加し、室温で２時間３０分撹拌した。反応終了後、該反応混合物に水２０ｍｌを添加し、酢酸エチル６０ｍｌにて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。得られた固体をｎ−ヘキサンで洗浄し、目的物１．５６ｇを薄黄白色固体として得た。
融点；１１２−１１４℃
合成例４
３−［４−｛３−（メチルチオ）プロピン−１−イル｝−１Ｈ−ピラゾール−１−イル］ピリジンの製造（本発明化合物２−００１）
３−（４−エチニル−１Ｈ−ピラゾール−１−イル）ピリジン２００ｍｇのテトラヒドロフラン５ｍｌ溶液を、窒素雰囲気下にて−７８℃に冷却した。次いで、１．６Ｍ ｎ−ブチルリチウム ｎ−ヘキサン溶液１．２ｍｌを滴下した。滴下終了後、−７８℃にて３０分撹拌した後、クロロジメチルスルフィド２６２ｍｇを添加した。添加終了後、室温まで昇温した後、ヨウ化カリウム１ｍｇを添加し、更に室温にて２３時間撹拌を継続した。反応終了後、該反応混合物に水５ｍｌを添加し、酢酸エチル１５ｍｌにて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。溶媒を留去した後に得られた残渣をクロロホルム−メタノール（９：１）にて溶出する薄層クロマトグラフにて精製し、目的物４６ｍｇを茶褐色固体として得た。
融点；４５−４７℃
合成例５
３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝−Ｎ−（２，２，２−トリフルオロエチル）アクリルアミドの製造（本発明化合物３−００３）
工程１
エチル ３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝アクリレートの製造
３−（４−ヨード−１Ｈ−ピラゾール−１−イル）ピリジン３．０ｇのＮ，Ｎ−ジメチルホルムアミド５０ｍｌ溶液に、アクリル酸エチル１．６６ｇ、［１，１’−ビス（ジフェニルホスフィノ）フェロセン］パラジウム（ＩＩ）ジクロリド ジクロロメタン付加物９５０ｍｇ及びトリエチルアミン２．３６ｇを順次添加し、窒素雰囲気下１２０℃にて２時間撹拌した。反応終了後、該反応混合物に水５０ｍｌを添加し、酢酸エチル１００ｍｌにて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。得られた残渣をｎ−ヘキサン−酢酸エチル（１：１）にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物１．０ｇを薄茶色固体として得た。
^１Ｈ ＮＭＲ（測定溶媒ＣＤＣｌ_３）δ８．９９（ｄ，Ｊ＝２．４Ｈｚ，１Ｈ），８．６０（ｍ，１Ｈ），８．１２（ｍ，１Ｈ），８．００−８．１０（ｍ，１Ｈ），７．９７（ｓ，１Ｈ），７．６３（ｄ，１５．９Ｈｚ，１Ｈ），７．４４（ｄｄ，Ｊ＝８．４，４．９Ｈｚ，１Ｈ），６．３１（ｄ，１５．９Ｈｚ，１Ｈ），４．２６（ｑ，７．２Ｈｚ，２Ｈ），１．３４（ｔ，７．２Ｈｚ，３Ｈ）
工程２
エチル ３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝アクリル酸の製造
エチル ３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝アクリレート０．９ｇのエタノール１０ｍｌ溶液に、水酸化カリウム０．４５ｇ及び水５ｍｌを順次添加し、５０℃にて１時間撹拌した。反応終了後、該反応混合物に２Ｎ塩酸水溶液を添加し、反応混合物のｐＨを３とした。減圧下溶媒を留去し、目的物及び塩化カリウムを含む混合物物１．２ｇを白色固体として得た。 [Synthesis example]
Synthesis example 1
1- {3-Methyl-1- (pyridin-3-yl) -1H-pyrazol-4-yl} ethanone Production of O-methyl oxime (present compound 1-003)
Process 1
Preparation of 1- {3-methyl-1- (pyridin-3-yl) -1H-pyrazol-4-yl} ethanone 1 separately prepared in a solution of 12.6 g of 3-iodopyridine in 100 ml of N, N-dimethylformamide -(3-Methyl-1H-pyrazol-4-yl) ethanone 7.08 g in 20 ml of N, N-dimethylformamide and 46.3 g of cesium carbonate were sequentially added. After the addition was completed, the reaction vessel was replaced with nitrogen gas, 2.3 g of copper iodide (monovalent) was added, and the mixture was stirred at room temperature for 30 minutes. After completion of the stirring, the temperature was raised to 120 ° C., and stirring was continued for 15 hours at the same temperature. After completion of the reaction, the reaction mixture was allowed to cool to room temperature. The insoluble matter precipitated in the reaction mixture after being allowed to cool was removed by Celite filtration under reduced pressure, and 200 ml of ethyl acetate was added to the filtrate. The obtained organic layer was washed and dried in the order of saturated brine and anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate [gradient of 1: 1 to 1: 9 (volume ratio, the same shall apply hereinafter)], and target product 7 .8 g was obtained as a white solid.
¹ H NMR (measurement solvent CDCl ₃ ) δ 8.98 (d, J = 3.3 Hz, 1H), 8.60 (d, J = 4.8 Hz, 1H), 8.33 (s, 1H), 8. 05-8.10 (m, 1H), 7.43 (dd, J = 4.8, 8.4 Hz, 1H), 2.58 (s, 3H), 2.50 (s, 3H)
Process 2
1- {3-Methyl-1- (pyridin-3-yl) -1H-pyrazol-4-yl} ethanone Preparation of O-methyl oxime 1- {3-Methyl-1- (pyridin-3-yl) -1H -Pyrazol-4-yl} ethanone To a solution of 200 mg of methanol in 1 ml of methanol was added 99.6 mg of O-methylhydroxylamine hydrochloride and stirred overnight at room temperature. After completion of the reaction, 5 ml of water was added to the reaction mixture and extracted with 5 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained solid was washed with chloroform to obtain 82 mg of the objective compound as a white solid.
Melting point: 155-156 ° C
Synthesis example 2
Production of 3- [4-{(trimethylsilyl) ethynyl} -1H-pyrazol-1-yl] pyridine (present compound 2-001)
To a solution of 1.0 g of 3- (4-iodo-1H-pyrazol-1-yl) pyridine in 20 ml of N, N-dimethylformamide, 725 mg of trimethylsilylacetylene, 50 mg of copper iodide (monovalent), 50 mg of dichlorobistriphenylphosphine palladium and After sequentially adding 745 mg of triethylamine, the mixture was stirred at 80 ° C. for 5 hours. After completion of the reaction, 30 ml of water was added to the reaction mixture and extracted with 50 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (4: 6) to obtain 400 mg of the desired product as a pale yellow solid.
¹ H NMR (measurement solvent CDCl ₃ ) δ 8.97 (bs, 1H), 8.60 (d, J = 3.6 Hz, 1H), 8.09 (s, 1H), 8.04 (d, J = 8.1 Hz, 1H), 7.84 (s, 1H), 7.43 (dd, J = 8.1, 4.8 Hz, 1H), 0.25 (s, 9H)
Melting point: 79-81 ° C
Synthesis example 3
Production of 3- (4-ethynyl-1H-pyrazol-1-yl) pyridine (the present compound 2-002)
To a 10 ml methanol solution of 2.3 g of 3- [4-{(trimethylsilyl) ethynyl} -1H-pyrazol-1-yl] pyridine, 2.0 g of potassium carbonate was added and stirred at room temperature for 2 hours 30 minutes. After completion of the reaction, 20 ml of water was added to the reaction mixture and extracted with 60 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained solid was washed with n-hexane to obtain 1.56 g of the desired product as a pale yellowish white solid.
Melting point: 112-114 ° C
Synthesis example 4
Production of 3- [4- {3- (methylthio) propin-1-yl} -1H-pyrazol-1-yl] pyridine (Compound 2-001 of the present invention)
A solution of 200 mg of 3- (4-ethynyl-1H-pyrazol-1-yl) pyridine in 5 ml of tetrahydrofuran was cooled to −78 ° C. under a nitrogen atmosphere. Then, 1.2 ml of 1.6M n-butyllithium n-hexane solution was added dropwise. After completion of the dropwise addition, the mixture was stirred at −78 ° C. for 30 minutes, and 262 mg of chlorodimethyl sulfide was added. After completion of the addition, the temperature was raised to room temperature, 1 mg of potassium iodide was added, and stirring was further continued at room temperature for 23 hours. After completion of the reaction, 5 ml of water was added to the reaction mixture and extracted with 15 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The residue obtained after distilling off the solvent was purified by thin layer chromatography eluting with chloroform-methanol (9: 1) to obtain 46 mg of the desired product as a brown solid.
Melting point: 45-47 ° C
Synthesis example 5
Production of 3- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} -N- (2,2,2-trifluoroethyl) acrylamide (present compound 3-003)
Process 1
Preparation of ethyl 3- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} acrylate 3- (4-iodo-1H-pyrazol-1-yl) pyridine 3.0 g of N, N-dimethyl 1.66 g of ethyl acrylate, 950 mg of [1,1′-bis (diphenylphosphino) ferrocene] palladium (II) dichloride dichloromethane adduct and 2.36 g of triethylamine are sequentially added to a 50 ml solution of formamide, and 120 ° C. under a nitrogen atmosphere. For 2 hours. After completion of the reaction, 50 ml of water was added to the reaction mixture and extracted with 100 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (1: 1) to obtain 1.0 g of the objective product as a light brown solid.
¹ H NMR (measurement solvent CDCl ₃ ) δ 8.99 (d, J = 2.4 Hz, 1H), 8.60 (m, 1H), 8.12 (m, 1H), 8.00-8.10 ( m, 1H), 7.97 (s, 1H), 7.63 (d, 15.9 Hz, 1H), 7.44 (dd, J = 8.4, 4.9 Hz, 1H), 6.31 ( d, 15.9 Hz, 1 H), 4.26 (q, 7.2 Hz, 2 H), 1.34 (t, 7.2 Hz, 3 H)
Process 2
Preparation of ethyl 3- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} acrylic acid Ethyl 3- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} acrylate 0 0.45 g of potassium hydroxide and 5 ml of water were sequentially added to a solution of .9 g of ethanol in 10 ml and stirred at 50 ° C. for 1 hour. After completion of the reaction, 2N hydrochloric acid aqueous solution was added to the reaction mixture to adjust the pH of the reaction mixture to 3. The solvent was distilled off under reduced pressure to obtain 1.2 g of a mixture containing the target product and potassium chloride as a white solid.

工程３
３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝−Ｎ−（２，２，２−トリフルオロエチル）アクリルアミドの製造
工程２で合成したエチル ３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝アクリル酸０．４ｇをジクロロメタン１５ｍｌに懸濁させ、１−エチル−３−（３−ジメチルアミノプロピル）カルボジイミド塩酸塩０．５ｇ、トリフルオロエチルアミン０．３ｇ及びトリエチルアミン１．０ｇを順次添加し、室温にて１５時間撹拌した。反応終了後、該反応混合物に水２０ｍｌを添加し、酢酸エチル３０ｍｌにて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥後、減圧下にて溶媒を留去した。得られた固体をｎ−ヘキサン−酢酸エチル（１：１）にて洗浄し、目的物０．１５ｇを白色固体として得た。
融点；２２８−２３０℃
合成例６
Ｎ−メチル−Ｎ’−[１−｛３−メチル−１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝エチリデン]−３−（メチルチオ）プロパンヒドラジドの製造（本発明化合物４−００１）
１−｛３−メチル−１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝エタノン３００ｍｇのエタノール１０ｍｌ溶液に、３−（メチルチオ）プロパンヒドラジド３００ｍｇを添加し、９０℃にて８時間撹拌した。反応終了後、溶媒を留去し、得られた残留物にＮ，Ｎ−ジメチルホルムアミド１０ｍｌを添加した。該反応溶液に６０重量％水素化ナトリウム（鉱油中に分散）４５．５ｍｇ次いでトリフルオロメタンスルホン酸メチル１８７ｍｇを添加し、７０℃にて２日間撹拌した。反応終了後、該反応溶液に水３０ｍｌを添加し、酢酸エチル３０ｍｌで抽出した。得られた有機層を無水硫酸ナトリウムで脱水し、減圧下にて溶媒を留去した。得られた残留物をｎ−ヘキサン−酢酸エチル（１：１〜１：９のグラジエント）にて溶出する中圧分取液体クロマトグラフィーにて精製し、目的物７ｍｇを褐色固体として得た。
融点；６０−６５℃
合成例７
ターシャリーブチル ［２−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝ビニル］カーバメートの製造（本発明化合物３−０１０）
３−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝アクリル酸０．９ｇのテトラヒドロフラン３０ｍｌ溶液にターシャリーブタノール０．３７ｇ、トリメチルシリルアジド０．５３ｇ、プロピルホスホニックアンヒドリド ジメチルホルムアミド溶液（１．６ｍｏｌ／Ｌ）２．９ｍｌ、トリエチルアミン０．７ｇを順次加え、窒素雰囲気下で８０℃にて４時間撹拌した。攪拌終了後、該反応混合物を室温まで冷却し、減圧下にて溶媒を留去した。得られた残留物に水３０ｍｌを添加し、酢酸エチル（５０ｍｌ）にて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥し、減圧下にて溶媒を留去した。得られた残留物をｎ−ヘキサン−酢酸エチル（１：１）にて溶出するシリカゲルカラムクロマトグラフィーで精製し、目的物０．２５ｇを白色固体として得た。
融点９３−９７℃
合成例８
ターシャリーブチル メチル［２−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝ビニル］カーバメートの合成（本発明化合物３−０１１）
ターシャリーブチル［２−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝ビニル］カーバメート０．２５ｇをＮ，Ｎ−ジメチルホルムアミド５ｍｌに溶解させた。該反応混合物に、０℃にて６０重量％水素化ナトリウム（鉱油中に分散）０．０４ｇを添加した。添加終了後、同温度で１０分間攪拌した。攪拌終了後、該反応混合物に０℃にてジメチル硫酸０．１２ｇを添加した。添加終了後、室温にて３時間攪拌を継続した。反応終了後、該反応混合物に水２０ｍｌを添加し、酢酸エチル（３０ｍｌ）にて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥し、減圧下にて溶媒を留去した。得られた残留物をｎ−ヘキサン−酢酸エチル（１：１）にて溶出するシリカゲルカラムクロマトグラフィーで精製し、目的物０．２０ｇを淡黄色固体として得た。
融点１２０−１２１℃
合成例９
Ｎ−メチル−２−（メチルチオ）−Ｎ−［２−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝ビニル］プロパンアミドの合成（本発明化合物３−０１２）
ターシャリーブチル メチル［２−｛１−（ピリジン−３−イル）−１Ｈ−ピラゾール−４−イル｝ビニル］カーバメート０．２ｇに塩酸 １，４−ジオキサン溶液（４ｍｏｌ／Ｌ）１０ｍｌを添加し、室温にて３時間撹拌した。反応終了後、減圧下にて、該反応混合物から蟻酸を留去した。得られた残渣にジクロロメタン１０ｍｌを加え懸濁させた。別途、２−（メチルチオ）プロパン酸３００ｍｇのジクロロメタン５ｍｌ溶液に塩化オキサリル０．１ｇ及びジメチルホルムアミド０．０５ｇを加えて室温下で３０分間攪拌して調製した２−（メチルチオ）プロパノイルクロリドを該反応溶液に添加した。次いで、トリエチルアミン２ｍｌ、４−Ｎ，Ｎ−ジメチルアミノピリジン０．０５ｇを添加し、室温にて１時間撹拌した。反応終了後、該反応溶液に水１０ｍｌを添加し、酢酸エチル（２０ｍｌ）にて抽出した。得られた有機層を無水硫酸ナトリウムで脱水・乾燥し、減圧下にて溶媒を留去した。得られた残渣をｎ−ヘキサン−酢酸エチル（１：１）にて溶出するシリカゲルカラムクロマトグラフィーで精製し、目的物０．０３ｇを白色固体として得た。
融点１４３−１４５℃
本発明化合物は、前記製造法及び実施例に準じて製造することができる。 Process 3
Preparation of 3- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} -N- (2,2,2-trifluoroethyl) acrylamide Ethyl 3- {1- ( 0.4 g of pyridin-3-yl) -1H-pyrazol-4-yl} acrylic acid was suspended in 15 ml of dichloromethane, 0.5 g of 1-ethyl-3- (3-dimethylaminopropyl) carbodiimide hydrochloride, trifluoro 0.3 g of ethylamine and 1.0 g of triethylamine were sequentially added and stirred at room temperature for 15 hours. After completion of the reaction, 20 ml of water was added to the reaction mixture and extracted with 30 ml of ethyl acetate. The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained solid was washed with n-hexane-ethyl acetate (1: 1) to obtain 0.15 g of the desired product as a white solid.
Melting point: 228-230 ° C
Synthesis Example 6
Production of N-methyl-N ′-[1- {3-methyl-1- (pyridin-3-yl) -1H-pyrazol-4-yl} ethylidene] -3- (methylthio) propanehydrazide (Compound 4 of the present invention) -001)
1- {3-Methyl-1- (pyridin-3-yl) -1H-pyrazol-4-yl} ethanone 300 mg of 3- (methylthio) propane hydrazide was added to a solution of 300 mg of ethanol in 8 mg at 90 ° C. Stir for hours. After completion of the reaction, the solvent was distilled off, and 10 ml of N, N-dimethylformamide was added to the obtained residue. To the reaction solution, 45.5 mg of 60 wt% sodium hydride (dispersed in mineral oil) and then 187 mg of methyl trifluoromethanesulfonate were added and stirred at 70 ° C. for 2 days. After completion of the reaction, 30 ml of water was added to the reaction solution, and extracted with 30 ml of ethyl acetate. The obtained organic layer was dehydrated with anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by medium pressure preparative liquid chromatography eluting with n-hexane-ethyl acetate (1: 1 to 1: 9 gradient) to obtain 7 mg of the objective product as a brown solid.
Melting point: 60-65 ° C
Synthesis example 7
Production of tertiary butyl [2- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} vinyl] carbamate (present compound 3-010)
To a solution of 0.9 g of 3- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} acrylic acid in 30 ml of tetrahydrofuran, 0.37 g of tertiary butanol, 0.53 g of trimethylsilyl azide, dimethyl propylphosphonic anhydride dimethyl 2.9 ml of a formamide solution (1.6 mol / L) and 0.7 g of triethylamine were sequentially added, and the mixture was stirred at 80 ° C. for 4 hours under a nitrogen atmosphere. After completion of the stirring, the reaction mixture was cooled to room temperature, and the solvent was distilled off under reduced pressure. 30 ml of water was added to the obtained residue, and the mixture was extracted with ethyl acetate (50 ml). The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by silica gel column chromatography eluting with n-hexane-ethyl acetate (1: 1) to obtain 0.25 g of the desired product as a white solid.
Melting point 93-97 ° C
Synthesis example 8
Synthesis of tertiary butyl methyl [2- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} vinyl] carbamate (present compound 3-011)
0.25 g of tertiary butyl [2- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} vinyl] carbamate was dissolved in 5 ml of N, N-dimethylformamide. To the reaction mixture was added 0.04 g of 60 wt% sodium hydride (dispersed in mineral oil) at 0 ° C. After completion of the addition, the mixture was stirred at the same temperature for 10 minutes. After completion of the stirring, 0.12 g of dimethyl sulfate was added to the reaction mixture at 0 ° C. After completion of the addition, stirring was continued at room temperature for 3 hours. After completion of the reaction, 20 ml of water was added to the reaction mixture and extracted with ethyl acetate (30 ml). The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by silica gel column chromatography eluting with n-hexane-ethyl acetate (1: 1) to obtain 0.20 g of the desired product as a pale yellow solid.
Melting point 120-121 ° C
Synthesis Example 9
Synthesis of N-methyl-2- (methylthio) -N- [2- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} vinyl] propanamide (present compound 3-012)
10 ml of 1,4-dioxane hydrochloric acid solution (4 mol / L) was added to 0.2 g of tertiary butyl methyl [2- {1- (pyridin-3-yl) -1H-pyrazol-4-yl} vinyl] carbamate, Stir at room temperature for 3 hours. After completion of the reaction, formic acid was distilled off from the reaction mixture under reduced pressure. To the obtained residue, 10 ml of dichloromethane was added and suspended. Separately, 2- (methylthio) propanoyl chloride prepared by adding 0.1 g of oxalyl chloride and 0.05 g of dimethylformamide to a solution of 300 mg of 2- (methylthio) propanoic acid in 5 ml of dichloromethane and stirring at room temperature for 30 minutes was added to the reaction. Added to the solution. Subsequently, 2 ml of triethylamine and 0.05 g of 4-N, N-dimethylaminopyridine were added and stirred at room temperature for 1 hour. After completion of the reaction, 10 ml of water was added to the reaction solution, and extracted with ethyl acetate (20 ml). The obtained organic layer was dehydrated and dried over anhydrous sodium sulfate, and the solvent was distilled off under reduced pressure. The obtained residue was purified by silica gel column chromatography eluting with n-hexane-ethyl acetate (1: 1) to obtain 0.03 g of the desired product as a white solid.
Melting point 143-145 ° C
This invention compound can be manufactured according to the said manufacturing method and an Example.

合成例１乃至合成例９と同様に製造した本発明化合物の例を第7表乃至第１０表に示すが、本発明はこれらのみに限定されるものではない。なお、表中、Ｄ２−７ｂ、Ｄ２−３２ａ、Ｄ２−３２ｂ、Ｄ２−３４ａ、Ｄ２−１０８ａ、Ｄ２−１０８ｂで表される構造は下記の構造を表し、Ｄ２−７ｂ、Ｄ２−３２ｂ、Ｄ１０８ｂの構造式に記された番号は、Ｘの置換位置を表す。また、表中、＊１は「樹脂状」を表し、(decomp.)は、融点測定後に化合物が分解したことをそれぞれ意味する。   Examples of the compounds of the present invention produced in the same manner as in Synthesis Examples 1 to 9 are shown in Tables 7 to 10, but the present invention is not limited to these. In the table, the structures represented by D2-7b, D2-32a, D2-32b, D2-34a, D2-108a, D2-108b represent the following structures, and D2-7b, D2-32b, D108b The number written in the structural formula represents the substitution position of X. In the table, * 1 represents “resinous”, and (decomp.) Means that the compound was decomposed after the melting point measurement.

本発明化合物のうち、融点の記載のない化合物の１Ｈ ＮＭＲデータを第１１表に示す。なお、表中の記号はそれぞれ、下記の意味を表す。
ｓ：シングレット、ｄ：ダブレット、ｔ：トリプレット、ｑ：カルテット、ｍ：マルチプレット。 Among the compounds of the present invention, Table 1 shows 1H NMR data of compounds having no melting point. In addition, each symbol in the table represents the following meaning.
s: singlet, d: doublet, t: triplet, q: quartet, m: multiplet.

〔第７表〕 [Table 7]

―――――――――――――――――――――――――――――――――――――
No. R³ R^a R^b m.p.(℃)
―――――――――――――――――――――――――――――――――――――
1-001 Me Me CH₂CF₃ 161-167
1-002 Me Me CH₂(D2-32a) 125-127
1-003 Me Me Me 155-156
1-004 -CH₂CH₂CH₂- CH₂CF₃ 110-115
1-005 -CH₂CH₂CH₂- CH₂(D2-34a) 100-108
1-006 Me Me CH₂(D2-34a) 131-133
1-007 H H CH₂CF₃ 45-46
1-008 H C(O)NHCH₂CF₃ Me 173-174
1-009 Me D2-7b(X=3-CF₂CF₃) Me *1
1-010 H C(O)OEt Me 59-60
1-011 Cl Me CH₂CF₃ 130-131
1-012 Cl Me CH₂SMe 121-123
1-013 H NHCH₂CF₃ Me 75-76
―――――――――――――――――――――――――――――――――――――
〔第８表〕 ―――――――――――――――――――――――――――――――――――――
No. R ³ R ^a R ^b mp (℃)
―――――――――――――――――――――――――――――――――――――
1-001 Me Me CH ₂ CF ₃ 161-167
1-002 Me Me CH ₂ (D2-32a) 125-127
1-003 Me Me Me 155-156
1-004 -CH ₂ CH ₂ CH ₂ -CH ₂ CF ₃ 110-115
1-005 -CH ₂ CH ₂ CH ₂ -CH ₂ (D2-34a) 100-108
1-006 Me Me CH ₂ (D2-34a) 131-133
1-007 HH CH ₂ CF ₃ 45-46
1-008 HC (O) NHCH ₂ CF ₃ Me 173-174
1-009 Me D2-7b (X = 3-CF ₂ CF ₃ ) Me * 1
1-010 HC (O) OEt Me 59-60
1-011 Cl Me CH ₂ CF ₃ 130-131
1-012 Cl Me CH ₂ SMe 121-123
1-013 H NHCH ₂ CF ₃ Me 75-76
―――――――――――――――――――――――――――――――――――――
[Table 8]

――――――――――――――――――――――――――――
No. R³ R^c m.p.(℃)
――――――――――――――――――――――――――――
2-001 H Si(Me)₃ 79-81
2-002 H H 112-114
2-003 H C(O)NHEt 141-143
2-004 H CH₂SMe 45-47
2-005 H SMe 89-90
2-006 H S(O)Me 184-186
2-007 H S(O)₂Me 123-124
2-008 H D2-32b(X=5-CF₃) 162-163
2-009 H C(O)SMe 121-122
2-010 H CH₂CH₂OH 85-86
2-011 H CH₂CH₂OS(O)₂CH₃ 91-92
2-012 H CH₂CH₂SCH₃ 60-61
――――――――――――――――――――――――――――
〔第９表〕 ――――――――――――――――――――――――――――
No. R ³ R ^c mp (℃)
――――――――――――――――――――――――――――
2-001 H Si (Me) ₃ 79-81
2-002 HH 112-114
2-003 HC (O) NHEt 141-143
2-004 H CH ₂ SMe 45-47
2-005 H SMe 89-90
2-006 HS (O) Me 184-186
2-007 HS (O) ₂ Me 123-124
2-008 H D2-32b (X = 5-CF ₃ ) 162-163
2-009 HC (O) SMe 121-122
2-010 H CH ₂ CH ₂ OH 85-86
2-011 H CH ₂ CH ₂ OS (O) ₂ CH ₃ 91-92
2-012 H CH ₂ CH ₂ SCH ₃ 60-61
――――――――――――――――――――――――――――
[Table 9]

―――――――――――――――――――――――――――――――――――――
No. R³ R^e R^f m.p.(℃)
―――――――――――――――――――――――――――――――――――――
3-001 H H D2-108a 130-133
3-002 H H D2-108b(X=4-CF₃) 143-146
3-003 H H C(O)NHCH₂CF₃ 228-230
3-004 H H C(O)OEt 112-114
3-005 H H C(O)N(Me)CH₂CF₃ 179-181
3-006 H H SMe *1
3-007 H H D2-7b(X=3-CF₂CF₃) 135-136
3-008 H -CH₂CH₂N(CH₂CF₃)C(O)- 200-210
3-009 H -CH₂CH₂NHC(O)- 220(decomp.)
3-010 H H NHC(O)OC(CH₃)₃ 93-97
3-011 H H N(CH₃)C(O)OC(CH₃)₃ 120-121
3-012 H H N(CH₃)C(O)CH(CH₃)SCH₃ 143-145
―――――――――――――――――――――――――――――――――――――
〔第１０表〕 ―――――――――――――――――――――――――――――――――――――
^{No. R 3 R e R f mp} (℃)
―――――――――――――――――――――――――――――――――――――
3-001 HH D2-108a 130-133
3-002 HH D2-108b (X = 4-CF ₃ ) 143-146
3-003 HHC (O) NHCH ₂ CF ₃ 228-230
3-004 HHC (O) OEt 112-114
3-005 HHC (O) N (Me) CH ₂ CF ₃ 179-181
3-006 HH SMe * 1
3-007 HH D2-7b (X = 3-CF ₂ CF ₃ ) 135-136
3-008 H -CH ₂ CH ₂ N (CH ₂ CF ₃ ) C (O)-200 -210
3-009 H -CH ₂ CH ₂ NHC (O)-220 (decomp.)
3-010 HH NHC (O) OC (CH ₃ ) ₃ 93-97
3-011 HHN (CH ₃ ) C (O) OC (CH ₃ ) ₃ 120-121
3-012 HHN (CH ₃ ) C (O) CH (CH ₃ ) SCH ₃ 143-145
―――――――――――――――――――――――――――――――――――――
[Table 10]

―――――――――――――――――――――――――――――――――――――
No. R³ R^a R^g R^g2 m.p.(℃)
―――――――――――――――――――――――――――――――――――――
4-001 Me Me C(O)CH₂CH₂SCH₃ Me 60-65
―――――――――――――――――――――――――――――――――――――
〔第１１表〕
―――――――――――――――――――――――――――――――――――――――
Ｎｏ． プロトン核磁気共鳴ケミカルシフト値（ＣＤＣｌ_３中）：σ（ｐｐｍ）
―――――――――――――――――――――――――――――――――――――――
３−００６
９．００（ｄ，Ｊ＝２．４Ｈｚ，１Ｈ），８．５４（ｄｄ，Ｊ＝４．８，１．５Ｈｚ，１Ｈ），８．１８（ｓ，１Ｈ），８．０５（ｄｄｄ，Ｊ＝８．４，２．７，１．２，Ｈｚ，１Ｈ），７．８６（ｓ，１Ｈ），７．４０（ｄｄ，Ｊ＝８．４，４．８Ｈｚ，１Ｈ），６．３４（ｄ，Ｊ＝１０．５Ｈｚ，１Ｈ），６．１５（ｄ，Ｊ＝１０．２Ｈｚ，１Ｈ），２．４６（ｓ，３Ｈ）
―――――――――――――――――――――――――――――――――――――――
［試験例］
次に、本発明化合物の有害生物防除剤としての有用性について、以下の試験例において具体的に説明するが、本発明はこれらのみに限定されるものではない。
試験例１ トビイロウンカに対する殺虫試験
本発明化合物の１０％乳剤（化合物によっては１０％水和剤を供試）を展着剤の入った水で希釈して、５００ｐｐｍ濃度の薬液を調製した。この薬液中にイネの葉鞘を約１０秒間浸漬し、風乾後試験管に入れ、この中にトビイロウンカ（Ｎｉｌａｐａｒｖａｔａ ｌｕｇｅｎｓ）の２齢幼虫を試験管当たり５頭放虫し、スポンジで蓋をして２５℃恒温室に収容した。６日後の死虫数を調査し、死虫率(％)(死虫数÷供試虫数×１００)を算出した。尚、試験は２連制で行なった。 ―――――――――――――――――――――――――――――――――――――
No. R ³ R ^a R ^g R ^g2 mp (℃)
―――――――――――――――――――――――――――――――――――――
4-001 Me Me C (O) CH ₂ CH ₂ SCH ₃ Me 60-65
―――――――――――――――――――――――――――――――――――――
[Table 11]
―――――――――――――――――――――――――――――――――――――――
No. Proton nuclear magnetic resonance chemical shift value (in CDCl ₃ ): σ (ppm)
―――――――――――――――――――――――――――――――――――――――
3-006
9.00 (d, J = 2.4 Hz, 1H), 8.54 (dd, J = 4.8, 1.5 Hz, 1H), 8.18 (s, 1H), 8.05 (ddd, J = 8.4, 2.7, 1.2, Hz, 1H), 7.86 (s, 1H), 7.40 (dd, J = 8.4, 4.8 Hz, 1H), 6.34 ( d, J = 10.5 Hz, 1H), 6.15 (d, J = 10.2 Hz, 1H), 2.46 (s, 3H)
―――――――――――――――――――――――――――――――――――――――
[Test example]
Next, the usefulness of the compound of the present invention as a pest control agent will be specifically described in the following test examples, but the present invention is not limited to these.
Test Example 1 Insecticidal test against brown planthopper A 10% emulsion of the compound of the present invention (depending on the compound, 10% wettable powder) was diluted with water containing a spreading agent to prepare a chemical solution having a concentration of 500 ppm. Rice leaf sheaths are immersed in this chemical solution for about 10 seconds, air-dried and placed in a test tube, and 5 second-instar larvae of Nilaparvata lugens are released per test tube, covered with a sponge and 25 Housed in a constant temperature room. The number of dead insects after 6 days was investigated, and the death rate (%) (number of dead insects ÷ number of test insects × 100) was calculated. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が９０％以上の死虫率を示した。
本発明化合物：１−００１〜１−０１１、２−００１、２−００２、２−００４、３−００１、３−００２、３−００３、３−００５〜３−００８、３−０１０、３−０１２、４−００１
試験例２ シルバーリーフコナジラミに対する殺虫試験
内径７ｃｍのスチロールカップに湿った濾紙を敷き、その上に３ｃｍに切り取ったインゲンの葉を置いた。本発明化合物の１０％乳剤（化合物によっては１０％水和剤を供試）を展着剤の入った水で希釈して、５００ｐｐｍ濃度の薬液を調製し、回転式散布塔を用いて薬液をスチロールカップ当たり２．５ｍｌずつ散布した（２．５ｍｇ／ｃｍ２）。葉を風乾後、シルバーリーフコナジラミ（Ｂｅｍｉｓｉａ ａｒｇｅｎｔｉｆｏｌｉｉ）の成虫を放虫し、蓋をして２５℃恒温室に収容した。５日後の死虫数を調査し、試験例１と同様の計算式から死虫率を算出した。尚、試験は２連制で行なった。 As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001 to 1-011, 2-001, 2-002, 2-004, 3-001, 3-002, 3-003, 3-005 to 3-008, 3-010, 3- 012, 4-001
Test Example 2 Insecticidal test for silver leaf whitefly A moist filter paper was laid on a styrene cup having an inner diameter of 7 cm, and a green leaf cut into 3 cm was placed thereon. A 10% emulsion of a compound of the present invention (depending on the compound, 10% wettable powder) is diluted with water containing a spreading agent to prepare a chemical solution with a concentration of 500 ppm, and the chemical solution is prepared using a rotary spray tower. 2.5 ml was sprayed per styrene cup (2.5 mg / cm 2). After the leaves were air-dried, adults of silver leaf whiteflies (Bemisia argentifolii) were released, covered, and housed in a thermostatic chamber at 25 ° C. The number of dead insects after 5 days was investigated, and the dead insect rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が９０％以上の死虫率を示した。
本発明化合物：１−００４、１−００９、１−０１１、２−００１、
試験例３ モモアカアブラムシに対する殺虫試験
内径3cmのガラスシャーレに湿った脱脂綿を敷き、その上に同径に切り取ったカンランの葉を置き、モモアカアブラムシ（Ｍｙｚｕｓ ｐｅｒｓｉｃａｅ）無翅成虫を４頭放虫した。１日後、本発明化合物の１０％乳剤（化合物によっては１０％水和剤を供試）を展着剤の入った水で希釈して、５００ppm濃度の薬液を調製し、回転式散布塔にて薬液を散布(2.5mg/cm2)、蓋をして２５℃恒温室に収容した。６日後の死虫数を調査し、試験例１と同様の計算式から死虫率を算出した。尚、試験は２連制で行なった。 As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
The present compound: 1-004, 1-009, 1-011, 2-001,
Test Example 3 Insecticidal test against peach aphid A moist absorbent cotton was laid on a glass petri dish with an inner diameter of 3 cm, and kanran leaves cut out to the same diameter were placed on it. did. One day later, a 10% emulsion of the compound of the present invention (depending on the compound, 10% wettable powder) was diluted with water containing a spreading agent to prepare a chemical solution with a concentration of 500 ppm. The chemical solution was sprayed (2.5 mg / cm 2), covered, and stored in a constant temperature room at 25 ° C. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が９０％以上の死虫率を示した。
本発明化合物：１−００１〜１−０１１、２−００１〜２−００４、３−００１、３−００２、３−００３、３−００５、３−００６、３−００８、３−０１０、３−０１２、４−００１
試験例４ ワタアブラムシに対する殺虫試験
内径3cmのガラスシャーレに湿った脱脂綿を敷き、その上に同径に切り取ったキュウリの葉を置き、ワタアブラムシ（Ａｐｈｉｓ ｇｏｓｓｙｐｉｉ）無翅成虫を４頭放虫した。１日後、本発明化合物の１０％乳剤（化合物によっては１０％水和剤を供試）を展着剤の入った水で希釈して、５００ppm濃度の薬液を調製し、回転式散布塔にて薬液を散布(2.5mg/cm2)、蓋をして２５℃恒温室に収容した。６日後の死虫数を調査し、試験例１と同様の計算式から死虫率を算出した。尚、試験は２連制で行なった。 As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001 to 1-011, 2-001 to 2-004, 3-001, 3-002, 3-003, 3-005, 3-006, 3-008, 3-010, 3- 012, 4-001
Test Example 4 Insecticidal test for cotton aphids Wet cotton wool with a 3 cm inner diameter petri dish and a cucumber leaf cut out to the same diameter was placed on the cotton aphid, and four cotton aphids (Aphis gossypi) adults were released. One day later, a 10% emulsion of the compound of the present invention (depending on the compound, 10% wettable powder) was diluted with water containing a spreading agent to prepare a chemical solution with a concentration of 500 ppm. The chemical solution was sprayed (2.5 mg / cm 2), covered, and stored in a constant temperature room at 25 ° C. The number of dead insects after 6 days was investigated, and the death rate was calculated from the same calculation formula as in Test Example 1. In addition, the test was performed by 2 continuous systems.

その結果、供試した化合物の内、下記の化合物が９０％以上の死虫率を示した。
本発明化合物：１−００１、１−００８、１−００９、１−０１１、２−００１、２−００２、２−００４、３−００１、３−００２、３−００３、３−００５、３−００７、３−００８、３−０１０、３−０１２、４−００１
試験例５ モモアカアブラムシに対する土壌潅注処理試験
本発明化合物の１０％乳剤を水道水で希釈して、濃度が１００ｐｐｍの薬液を調製した。 As a result, among the compounds tested, the following compounds showed a death rate of 90% or more.
Compounds of the present invention: 1-001, 1-008, 1-009, 1-011, 2-001, 2-002, 2-004, 3-001, 3-002, 3-003, 3-005, 3- 007, 3-008, 3-010, 3-012, 4-001
Test Example 5 Soil irrigation treatment test for peach aphid A 10% emulsion of the compound of the present invention was diluted with tap water to prepare a chemical solution having a concentration of 100 ppm.

プラスチックカップ植えキャベツ苗（２．５本葉期）の株元土壌部分に１０ｍｌの薬液を潅注処理し、温室内に放置した。潅注処理１日後にモモアカアブラムシ（Ｍｙｚｕｓ ｐｅｒｓｉｃａｅ）の成虫を２０頭／株で放虫し、その後温室内に放置した。放虫６日後の生存虫数を調査し、下記の計算式から対照値を算出した。
対照値(％)＝｛1-(Cb×Tai)/(Cai×Tb)｝×100
式中の文字は下記を表している。
Cb：無処理区における処理前の虫の数
Cai：無処理区における最終調査時の生存虫数
Tb：処理区における処理前の虫の数
Cai：処理区における最終調査時の生存虫数
その結果、供試した化合物の内、下記の化合物が９０％以上の対照値を示した。
本発明化合物：３−００３ 10 ml of the chemical solution was irrigated to the stock soil portion of the plastic cup planted cabbage seedling (2.5 true leaf stage) and left in the greenhouse. One day after the irrigation treatment, 20 mosquitoes / strain of adult peach aphid (Myzus persicae) were released and then left in the greenhouse. The number of surviving insects 6 days after the release was examined, and a control value was calculated from the following formula.
Control value (%) = {1- (Cb × Tai) / (Cai × Tb)} × 100
The characters in the formula represent the following:
Cb: Number of insects before treatment in the untreated area
Cai: Number of surviving insects at the final survey in the untreated area
Tb: Number of insects before treatment in the treatment area
Cai: Number of live worms at the final survey in the treated group As a result, among the compounds tested, the following compounds showed a control value of 90% or more.
Compound of the present invention: 3-003

本発明における新規なピラゾール誘導体は、優れた有害生物防除活性、特に殺虫・殺ダニ活性を示し、且つ、ホ乳動物、魚類及び益虫等の非標的生物に対してほとんど悪影響の無い、極めて有用な化合物である。   The novel pyrazole derivative in the present invention exhibits excellent pest control activity, particularly insecticidal / miticidal activity, and is extremely useful with little adverse effect on non-target organisms such as mammals, fish and beneficial insects. A compound.

Claims (10)

式（１）：

〔式中、Ａ^１は、−Ｎ（−Ｏ）_ｍ２又は−ＣＲ^１を表し、
Ｒ^１、Ｒ^３及びＲ^４は、各々独立して水素原子、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、Ｃ_１〜Ｃ_６アルキル、Ｒ^２８ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_３〜Ｃ_８ハロシクロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６ハロアルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルチオカルボニル、Ｃ_１〜Ｃ_６アルコキシチオカルボニル、Ｃ_１〜Ｃ_６アルキルジチオカルボニル、Ｃ_１〜Ｃ₆アルキルアミノカルボニル、Ｃ_１〜Ｃ₆ハロアルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノカルボニル、トリ（Ｃ_１〜Ｃ_６アルキル）シリル、Ｃ_１〜Ｃ₆アルキルアミノスルホニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、Ｃ_１〜Ｃ_６アルキルスルホニルオキシ、Ｃ_１〜Ｃ_６ハロアルキルスルホニルオキシ、Ｃ_１〜Ｃ_６アルキルアミノ、ジ（Ｃ_１〜Ｃ_６アルキル）アミノ、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^２は、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、Ｃ_１〜Ｃ_６アルキル、Ｒ^２８ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^２８ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^２８ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_３〜Ｃ_８ハロシクロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６ハロアルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルチオカルボニル、Ｃ_１〜Ｃ_６アルコキシチオカルボニル、Ｃ_１〜Ｃ_６アルキルジチオカルボニル、Ｃ_１〜Ｃ₆アルキルアミノカルボニル、Ｃ_１〜Ｃ₆ハロアルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノカルボニル、トリ（Ｃ_１〜Ｃ_６アルキル）シリル、Ｃ_１〜Ｃ₆アルキルアミノスルホニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、Ｃ_１〜Ｃ_６アルキルスルホニルオキシ、Ｃ_１〜Ｃ_６ハロアルキルスルホニルオキシ、Ｃ_１〜Ｃ_６アルキルアミノ、ジ（Ｃ_１〜Ｃ_６アルキル）アミノ、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、ｎが２以上の整数を表すとき、各々のＲ^２は互いに同一であっても又は互いに相異なってもよく、
Ａ^２は、−Ｃ（Ｒ^ａ）＝ＮＯＨ、−Ｃ（Ｒ^ａ）＝ＮＯＲ^ｂ、−Ｃ≡ＣＲ^ｃ、−Ｃ（Ｒ^ｄ）＝Ｃ（Ｒ^ｅ）Ｒ^ｆ又は−Ｃ（Ｒ^ａ）＝ＮＮ（Ｒ^ｇ）Ｒ^ｇ２を表し、
Ｒ^ａは、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、或いは、Ｒ^ａはＲ^３と一緒になってＣ_２〜Ｃ_５のアルキレン鎖又はＣ_２〜Ｃ_５アルケニレン鎖を形成することにより、Ｒ^ａが結合する炭素原子及びＲ^３が結合する炭素原子と共に５〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１又は２個含んでもよく、且つハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−ＯＨ，−ＯＲ^１１、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１１、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^ｂは、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^ｃは、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^ｄは、水素原子、ハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ又は−Ｃ（Ｏ）Ｒ^７を表し、
Ｒ^ｅ及びＲ^ｆは、各々独立して水素原子、−ＯＨ、−ＯＲ^６、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^６、−Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、或いは、Ｒ^ｅはＲ^ｆと一緒になってＣ_２〜Ｃ_７のアルキレン鎖を形成することにより、Ｒ^ｅ及びＲ^ｆが結合する炭素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖は酸素原子、硫黄原子又は窒素原子を１又は２個個含んでもよく、且つハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−ＯＨ，−ＯＲ^１１、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１１、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^ｇ及びＲ^ｇ２は、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^５で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^５で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｓ）ＯＲ^６ａ、−Ｃ（Ｓ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｒ^７、−Ｃ（Ｓ）Ｒ^７、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｃ（Ｓ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓ（Ｏ）_ｒＮ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^５は、ハロゲン原子、シアノ、Ｃ_３〜Ｃ_８シクロアルキル、−ＯＨ、−ＯＲ^１１、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１１、−Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｃ（Ｏ）ＯＲ^１１ａ、−Ｃ（Ｓ）ＯＲ^１１ａ、−Ｃ（Ｏ）ＳＲ^１１ａ、−Ｃ（Ｓ）ＳＲ^１１ａ、−Ｃ（Ｏ）Ｒ^１２、−Ｃ（Ｓ）Ｒ^１２、−Ｃ（Ｏ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｃ（Ｓ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｓ（Ｏ）_ｒＮ（Ｒ^１３ａ）Ｒ^１３、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^６及びＲ^６ａは、各々独立してＣ_１〜Ｃ_６アルキル又はＲ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^７は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^８及びＲ^８ａは、各々独立して水素原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｒ^１４で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、−Ｓ（Ｏ）_ｒＲ^１１、−Ｃ（Ｏ）ＯＲ^１１ａ、−Ｃ（Ｓ）ＯＲ^１１ａ、−Ｃ（Ｏ）ＳＲ^１１ａ、−Ｃ（Ｓ）ＳＲ^１１ａ、−Ｃ（Ｏ）Ｒ^１２、−Ｃ（Ｓ）Ｒ^１２、−Ｃ（Ｏ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｃ（Ｓ）Ｎ（Ｒ^１３ａ）Ｒ^１３、−Ｓ（Ｏ）_ｒＮ（Ｒ^１３ａ）Ｒ^１３、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、、或いは、Ｒ^８はＲ^８ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^８及びＲ^８ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、且つハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、フェニル、（Ｚ^２）_ｑ２によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^９、Ｒ^９ａ及びＲ^９ｂは、各々独立してＣ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６アルコキシ又はフェニルを表し、
Ｒ^１１は、−Ｓ（Ｏ）_２Ｒ^１５ａ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１１ａ及びＲ^１２は、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１３及びＲ^１３ａは、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１４ａで任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１４ａで任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、、或いは、Ｒ^１３はＲ^１３ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^１３及びＲ^１３ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、且つハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、フェニル、（Ｚ^２）_ｑ２によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^１４及びＲ^１４ａは、各々独立してハロゲン原子、シアノ、ニトロ、Ｃ_３〜Ｃ_８シクロアルキル、Ｃ_３〜Ｃ_８ハロシクロアルキル、Ｃ_３〜Ｃ_８シクロアルケニル、Ｃ_３〜Ｃ_８ハロシクロアルケニル、−ＯＨ、−ＯＲ^１５、−ＳＨ、−Ｓ（Ｏ）_ｒＲ^１５、−Ｎ（Ｒ^１７ａ）Ｒ^１７、−Ｃ（Ｏ）ＯＲ^１５、−Ｃ（Ｏ）ＳＲ^１５、−Ｃ（Ｓ）ＯＲ^１５、−Ｃ（Ｓ）ＳＲ^１５、−Ｃ（Ｏ）Ｒ^１６、−Ｃ（Ｏ）Ｎ（Ｒ^１７ａ）Ｒ^１７、−Ｃ（Ｓ）Ｎ（Ｒ^１７ａ）Ｒ^１７、−Ｓ（Ｏ）_ｒＮ（Ｒ^１７ａ）Ｒ^１７、−Ｃ（＝ＮＲ^１７）ＯＲ^１５、−Ｃ（＝ＮＲ^１７）Ｓ（Ｏ）_ｒＲ^１５、−Ｃ（＝ＮＲ^１７）Ｒ^１６、−Ｃ（＝ＮＯＨ）Ｒ^１６、−Ｃ（＝ＮＯＲ^１５）Ｒ^１６、−Ｃ｛＝ＮＮ（Ｒ^１７ａ）Ｒ^１７｝Ｒ^１６、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、を表し、
Ｒ^１５及びＲ^１５ａは、各々独立してＣ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１６は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｒ^１７及びＲ^１７ａは、各々独立して水素原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^１８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｃ_２〜Ｃ_６シクロアルケニル、Ｒ^１８で任意に置換された（Ｃ_２〜Ｃ_６）シクロアルケニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表すか、或いは、Ｒ^１７はＲ^１７ａと一緒になってＣ_２〜Ｃ_７のアルキレン鎖又はＣ_２〜Ｃ_７のアルケニレン鎖を形成することにより、Ｒ^１７及びＲ^１７ａが結合する窒素原子と共に３〜８員環を形成してもよく、このときこのアルキレン鎖又はアルケニレン鎖は酸素原子、硫黄原子又は窒素原子を１個含んでもよく、且つハロゲン原子、シアノ、Ｃ_１〜Ｃ_６アルキル、Ｒ^１８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、フェニル、（Ｚ^２）_ｑ２によって置換されたフェニル、オキソ基又はチオキソ基によって任意に置換されてもよく、
Ｒ^１８は、ハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、−Ｓｉ（Ｒ^９ｂ）（Ｒ^９ａ）Ｒ^９、フェニル、ナフチル、（Ｚ^２）_ｑ２で置換されたフェニル、（Ｚ^２）_ｑ２で置換されたナフチル又はＤ２−１〜Ｄ２−１０２を表し、
Ｄ２−１〜Ｄ２−１０２は、それぞれ下記の構造式で表される環を表し、




Ｘ^２は、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、−Ｃ（Ｏ）ＮＨ_２、−Ｃ（Ｓ）ＮＨ_２、−Ｓ（Ｏ）_２ＮＨ_２又はＲ^２０を表し、ｔ１、ｔ２又はｔ４が２以上の整数を表すとき、各々のＸ^２は互いに同一であっても又は互いに異なってもよく、更に、２つのＸ^２が隣接する場合には、隣接する２つのＸ^２は、−ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＯＣＨ_２−，−ＯＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２Ｓ−，−ＣＨ_２ＳＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２ＯＣＨ_２−，−ＣＨ_２ＯＣＨ_２Ｏ−，−ＯＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２ＣＨ_２Ｓ−又は−ＯＣＨ_２ＣＨ_２Ｓ−を形成することにより、それぞれのＸ^２が結合する炭素原子と共に５員環又は６員環を形成してもよく、このとき環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル基、Ｃ_１〜Ｃ_６ハロアルキル基、Ｃ_１〜Ｃ_６アルコキシ基、Ｃ_１〜Ｃ_６アルキルチオ基、Ｃ_１〜Ｃ_６アルキルスルフィニル基又はＣ_１〜Ｃ_６アルキルスルホニル基によって任意に置換されてもよく、
Ｘ^２ａは、水素原子、シアノ、−ＯＨ、−ＮＨ_２、−ＣＨＯ又はＲ^２０を表し、Ｘ^２ａの隣接位にＸ^２が存在する場合には、隣接するＸ^２ａとＸ^２は、−ＣＨ_２ＣＨ_２ＣＨ_２ＣＨ_２−、−ＣＨ＝ＣＨＣＨ＝ＣＨ−、−Ｎ＝ＣＨＣＨ＝ＣＨ−、−ＣＨ＝Ｎ−ＣＨ＝ＣＨ−、−ＣＨ＝ＣＨ−Ｎ＝ＣＨ−又は−ＣＨ＝ＣＨ−ＣＨ＝Ｎ−を形成することにより、Ｘ^２ａ及びＸ^２のそれぞれが結合する原子と共に６員環を形成してもよく、このとき、環を形成する各々の炭素原子に結合する水素原子は、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル基、Ｃ_１〜Ｃ_６ハロアルキル基、Ｃ_１〜Ｃ_６アルコキシ基、Ｃ_１〜Ｃ_６アルキルチオ基、Ｃ_１〜Ｃ_６アルキルスルフィニル基又はＣ_１〜Ｃ_６アルキルスルホニル基によって任意に置換されてもよく、
Ｘ^２ｂは、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、−Ｃ（Ｏ）ＮＨ_２、−Ｃ（Ｓ）ＮＨ_２、−Ｓ（Ｏ）_２ＮＨ_２、−ＣＨＯ又はＲ^２０を表し、ｕ１、ｕ２、ｕ４、ｕ５、ｕ６、ｕ７、ｕ８又はｕ９が２以上の整数を表すとき、各々のＸ^２ｂは互いに同一であっても、又は互いに相異なってもよく、更に、２つのＸ^２ｂが同一の炭素上に置換している場合、２つのＸ^２ｂは一緒になってオキソ、チオキソ、イミノ、Ｃ_１〜Ｃ_６アルキルイミノ、Ｃ_１〜Ｃ_６アルコキシイミノ又はＣ_１〜Ｃ_６アルキリデンを形成してもよく、
Ｚ^２は、ハロゲン原子、シアノ、ニトロ、−ＯＨ、−ＳＨ、−ＮＨ_２、−Ｃ（Ｏ）ＮＨ_２、−Ｃ（Ｓ）ＮＨ_２、−Ｓ（Ｏ）_２ＮＨ_２又はＲ^２０を表し、ｑ２が２以上の整数を表すとき、各々のＺ^２は互いに同一であっても又は互いに異なってもよく、更に、２つのＺ^２が隣接する場合には、隣接する２つのＺ^２は−ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＯＣＨ_２−，−ＯＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２Ｓ−，−ＣＨ_２ＳＣＨ_２−，−ＣＨ_２ＣＨ_２Ｎ（Ｘ^２ａ）−，−ＣＨ_２Ｎ（Ｘ^２ａ）ＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２ＣＨ_２−，−ＣＨ_２ＣＨ_２ＣＨ_２Ｏ−，−ＣＨ_２ＣＨ_２ＯＣＨ_２−，−ＣＨ_２ＯＣＨ_２Ｏ−，−ＯＣＨ_２ＣＨ_２Ｏ−，−ＯＣＨ_２ＣＨ_２Ｓ−，−ＣＨ_２ＣＨ＝ＣＨ−，−ＯＣＨ＝ＣＨ−，−ＳＣＨ＝ＣＨ−，−Ｎ（Ｘ^２ａ）ＣＨ＝ＣＨ−，−ＯＣＨ＝Ｎ−，−ＳＣＨ＝Ｎ−，−Ｎ（Ｘ^２ａ）ＣＨ＝Ｎ−，−Ｎ（Ｘ^２ａ）Ｎ＝ＣＨ−，−ＯＣＨ_２ＣＨ＝ＣＨ−，−Ｎ＝ＣＨＣＨ＝ＣＨ−，−ＣＨ＝ＮＣＨ＝ＣＨ−，−Ｎ＝ＮＣＨ＝ＣＨ−，−ＣＨ＝ＮＮ＝ＣＨ−，−Ｎ＝ＣＨＣＨ＝Ｎ−又は−Ｎ＝ＣＨＮ＝ＣＨ−を形成することにより、それぞれのＺ^２が結合する炭素原子と共に５員環又は６員環を形成してもよく、このとき、環を形成する各々の炭素原子に結合した水素原子は、ハロゲン原子、Ｃ_１〜Ｃ_６アルキル基、Ｃ_１〜Ｃ_６ハロアルキル基、Ｃ_１〜Ｃ_６アルコキシ基、Ｃ_１〜Ｃ_６アルキルチオ基、Ｃ_１〜Ｃ_６アルキルスルフィニル基又はＣ_１〜Ｃ_６アルキルスルホニル基によって任意に置換されてもよく、
Ｒ^２０は、Ｃ_１〜Ｃ_６アルキル、Ｃ_２〜Ｃ_６アルケニル、Ｃ_２〜Ｃ_６アルキニル、Ｃ_３〜Ｃ_８シクロアルキル、Ｒ^２８で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、Ｒ^２８で任意に置換された（Ｃ_２〜Ｃ_６）アルケニル、Ｒ^２８で任意に置換された（Ｃ_２〜Ｃ_６）アルキニル、Ｒ^２８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルキル、Ｒ^２８で任意に置換された（Ｃ_３〜Ｃ_８）シクロアルケニル、−ＯＲ^２５、−Ｓ（Ｏ）_ｒＲ^２５、−Ｃ（Ｏ）ＯＲ^２５、−Ｃ（Ｏ）Ｒ^２６、−Ｎ（Ｒ^２７ａ）Ｒ^２７、−Ｃ（Ｏ）Ｎ（Ｒ^２７ａ）Ｒ^２７、−Ｃ（Ｓ）Ｎ（Ｒ^２７ａ）Ｒ^２７、−Ｓ（Ｏ）_ｒＮ（Ｒ^２７ａ）Ｒ^２７、フェニル、Ｃ_１〜Ｃ_６アルキル又はハロゲン原子で任意に置換されたフェニルを表し、
Ｒ^２５、Ｒ^２６及びＲ^２７ａは、各々独立して水素原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６ハロアルキル又はＣ_３〜Ｃ_８シクロアルキルを表し、
Ｒ^２７は、水素原子、Ｃ_１〜Ｃ_６アルキル、Ｃ_１〜Ｃ_６ハロアルキル、Ｃ_３〜Ｃ_８シクロアルキル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル又はＣ_１〜Ｃ_６ハロアルコキシカルボニルを表し、
Ｒ^２８及びＲ^２８ａは、各々独立してハロゲン原子、シアノ、ニトロ、Ｃ_１〜Ｃ_６アルコキシ、Ｃ_１〜Ｃ_６ハロアルコキシ、Ｃ_２〜Ｃ_６アルケニルオキシ、Ｃ_１〜Ｃ_６アルキルチオ、Ｃ_１〜Ｃ_６アルキルスルフィニル、Ｃ_１〜Ｃ_６アルキルスルホニル、Ｃ_１〜Ｃ_６ハロアルキルチオ、Ｃ_１〜Ｃ_６ハロアルキルスルフィニル、Ｃ_１〜Ｃ_６ハロアルキルスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニル、Ｃ_３〜Ｃ_８シクロアルキルカルボニル、Ｃ_１〜Ｃ_６ハロアルキルカルボニル、Ｃ_３〜Ｃ_８ハロシクロアルキルカルボニル、Ｃ_１〜Ｃ_６アルコキシカルボニル、Ｃ_１〜Ｃ_６ハロアルコキシカルボニル、Ｃ_１〜Ｃ_６アルキルチオカルボニル、Ｃ_１〜Ｃ_６アルコキシチオカルボニル、Ｃ_１〜Ｃ_６アルキルジチオカルボニル、Ｃ_１〜Ｃ₆アルキルアミノカルボニル、Ｃ_１〜Ｃ₆ハロアルキルアミノカルボニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノカルボニル、トリ（Ｃ_１〜Ｃ_６アルキル）シリル、Ｃ_１〜Ｃ₆アルキルアミノスルホニル、ジ（Ｃ_１〜Ｃ_６アルキル）アミノスルホニル、Ｃ_１〜Ｃ_６アルキルカルボニルオキシ、Ｃ_１〜Ｃ_６アルキルスルホニルオキシ、Ｃ_１〜Ｃ_６ハロアルキルスルホニルオキシ、Ｃ_１〜Ｃ_６アルキルアミノ又はジ（Ｃ_１〜Ｃ_６アルキル）アミノを表し、
ｎ、ｔ１及びｕ１は、各々独立して０、１、２又は３の整数を表し、
ｔ２及びｕ２は、各々独立して０、１又は２の整数を表し、
ｔ３は、０又は１の整数を表し、
ｔ４及びｕ４は、各々独立して０、１、２、３又は４の整数を表し、
ｕ５は、０、１、２、３、４又は５の整数を表し、
ｕ６は、各々独立して０、１、２、３、４、５又は６の整数を表し、
ｕ７は、各々独立して０、１、２、３、４、５、６又は７の整数を表し、
ｕ８は、０、１、２、３、４、５、６、７又は８の整数を表し、
ｕ９は、０、１、２、３、４、５、６、７、８又は９の整数を表し、
ｑ２は、１、２、３、４又は５の整数を表し、
ｍ１、ｍ２及びｍ４は、各々独立して０又は１の整数を表し、
ｒ、ｒ２及びｒ３は、各々独立して０、１又は２の整数を表す〕で表されるピラゾール誘導体又はその塩。 Formula (1):

[Wherein, A ¹ represents —N (—O) _{m 2} or —CR ¹ ;
R ¹ , R ³ and R ⁴ are each independently optionally substituted with a hydrogen atom, a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , C ₁ -C ₆ alkyl, R ^28a ( C ₁ -C ₆ ) alkyl, C ₃ -C ₈ cycloalkyl, optionally substituted with R ^28a (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ alkenyl, optionally substituted with R ^28a ( C ₂ -C _{6) alkenyl,} C 3 -C ₈ ^{cycloalkenyl,} substituted optionally substituted with ^{R 28a} _(C 3 ~C _{8) cycloalkenyl,} C 2 -C ₆ ^alkynyl, optionally with ^{R 28a} ( C ₂ -C _{6) alkynyl,} C 1 -C _{6 alkoxy,} C 1 -C _{6 haloalkoxy,} C 2 -C _{6 alkenyloxy,} C 1 -C _{6 alkylthio,} C 1 -C _{6 alkylsulfinyl, C} 1 ~ _{6 alkylsulfonyl,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 haloalkylsulfonyl,} C 1 -C _{6 alkylcarbonyl,} C 3 -C _{8 cycloalkylcarbonyl,} C 1 -C _{6 haloalkylcarbonyl,} C 3 -C ₈ halocycloalkyl _carbonyl, C 1 -C _{6 alkoxycarbonyl,} C 1 -C _{6 haloalkoxycarbonyl,} C 1 -C _{6 alkylthiocarbonyl,} C 1 -C _{6 alkoxythiocarbonyl, C} 1 ~ C ₆ alkyldithiocarbonyl, C ₁ -C ₆ alkylaminocarbonyl, C ₁ -C ₆ haloalkylaminocarbonyl, di (C ₁ -C ₆ alkyl) aminocarbonyl, tri (C ₁ -C ₆ alkyl) silyl, C _1- C ₆ alkylaminosulfonyl, di _(C 1 ~ ₆ alkyl) _{aminosulfonyl,} C 1 -C _{6 alkylcarbonyloxy,} C 1 -C _{6 alkylsulfonyloxy,} C 1 -C _{6 haloalkylsulfonyloxy,} C 1 -C ₆ alkylamino, di _(C 1 -C ₆ alkyl) represents amino, phenyl, ^naphthyl, phenyl substituted with (Z _{2) ^q2,} naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ² is a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^28a , C ₃ -C _8. ^cycloalkyl, substituted optionally substituted with ^{R 28a} _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ ^alkenyl, optionally with ^{R 28a} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ ^{cycloalkenyl,} optionally substituted with ^{R 28a} _(C 3 ~C _{8) cycloalkenyl,} C 2 -C ₆ ^alkynyl, which is optionally substituted with ^{R 28a} _(C 2 ~C _{6) alkynyl,} C 1 -C _{6 alkoxy,} C 1 -C _{6 haloalkoxy,} C 2 -C _{6 alkenyloxy,} C 1 -C _{6 alkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ C _{Roarukiruchio,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 haloalkylsulfonyl,} C 1 -C _{6 alkylcarbonyl,} C 3 -C _{8 cycloalkylcarbonyl,} C 1 -C _{6 haloalkylcarbonyl,} C 3 -C ₈ halo Cycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, C ₁ -C ₆ alkylthiocarbonyl, C ₁ -C ₆ alkoxythiocarbonyl, C ₁ -C ₆ alkyldithiocarbonyl, C _1- C _{6 alkylaminocarbonyl,} C 1 -C ₆ haloalkylcarbonyl aminocarbonyl, di _(C 1 -C ₆ alkyl) aminocarbonyl, tri _(C 1 -C ₆ alkyl) _silyl, C 1 -C ₆ alkylaminosulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, _{C 1} C _{6 alkylcarbonyloxy,} C 1 -C _{6 alkylsulfonyloxy,} C 1 -C _{6 haloalkylsulfonyloxy,} C 1 -C ₆ alkylamino, di _(C 1 -C ₆ alkyl) amino, phenyl, naphthyl, ^{(Z 2} ) Represents a phenyl substituted with _q2 , (Z ² ) a naphthyl substituted with _q2 , or D2-1 to D2-102, and when n represents an integer of 2 or more, each R ² may be the same as each other Or they may be different from each other,
A ² is —C (R ^a ) = NOH, —C (R ^a ) = NOR ^b , —C≡CR ^c , —C (R ^d ) = C (R ^e ) R ^f or —C (R ^a ) = NN (R ^g ) R ^g2 ,
R ^a is a hydrogen _atom, C 1 -C ₆ alkyl, optionally substituted with ^{R 5} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ cycloalkyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkyl,} C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkenyl,} C 2 -C ₆ alkynyl, optionally substituted with ^{R 5} _(C 2 ~C ₆₎ ^{alkynyl, -OH, -OR 6, -SH,} -S (O) r R 6, ^{-N (R 8a) R 8,} -C (O) OR 6a, -C (O) SR 6a, -C (S) OR 6a, -C (S) SR 6a, -C (O) R 7, - ^{C (S) R 7, -C} (O) N (R 8a) R 8, -C (S) N (R 8a) R 8, - _{^{(O) r N (R 8a}} ) R 8, -Si (R 9a) (R 9b) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, naphthyl substituted with (Z _{2) q2} or represents a D2-1～D2-102, or, ^{R a} is by forming an alkylene chain or _C 2 -C ₅ alkenylene chain of _C 2 -C ₅ taken together with ^{R 3, R a} is a bond And a carbon atom to which R ³ is bonded may form a 5- to 8-membered ring, in which case the alkylene chain or alkenylene chain may contain one or two oxygen atoms, sulfur atoms or nitrogen atoms, and halogen atoms, cyano, _nitro, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 14} _(C 1 ~C ₆₎ ^{alkyl, -OH, -OR 11, -SH,} -S (O) r R 11 Oxo group or thioxo Optionally substituted by a group,
R ^b _is, C 1 -C ₆ alkyl, optionally substituted with ^{R 5} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ cycloalkyl, optionally substituted with ^{R 5} _(C 3 ~C ₈ ) _cycloalkyl, C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally substituted with ^{R 5} _(C 3 ~C ₈ ) _{cycloalkenyl,} substituted C 2 -C ₆ alkynyl, optionally with ^{R 5} _(C 2 ~C _{6) ^{alkynyl, -S (O) r R 6}} , -C (O) OR 6a, -C (O) ^{SR 6a, -C (S) OR} 6a, -C (S) SR 6a, -C (O) R 7, -C (S) R 7, -C (O) N (R 8a) R 8, -C _{^{(S) N (R 8a)}} R 8, -S (O) r N (R 8a) R 8, -Si (R 9a) (R 9b) ⁹ represents phenyl, ^naphthyl, phenyl substituted with (Z _{2) ^q2,} naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ^c is hydrogen _atom, C 1 -C ₆ alkyl, optionally substituted with ^{R 5} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ cycloalkyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkyl,} C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally substituted with ^{R 5} _{(C 3} -C _{8) cycloalkenyl,} C 2 -C ₆ alkynyl, optionally substituted with ^{R 5} _(C 2 ~C ₆₎ ^{alkynyl, -OH, -OR 6, -SH,} -S (O) r R 6, ^{-N (R 8a) R 8,} -C (O) OR 6a, -C (O) SR 6a, -C (S) OR 6a, -C (S) SR 6a, -C (O) R 7, - ^{C (S) R 7, -C} (O) N (R 8a) R 8, -C (S) N (R 8a) R 8, - _{^{(O) r N (R 8a}} ) R 8, -Si (R 9a) (R 9b) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, naphthyl substituted with (Z _{2) q2} Or D2-1 to D2-102,
R ^d is a hydrogen atom, a halogen atom, cyano, nitro, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ , —OH, —OR ⁶ , —SH, —S _(O) represents the ^{r R 6, -N (R 8a} ) R 8, -C (O) oR 6a or -C (O) ^{R 7,}
R ^e and R ^f are each independently a hydrogen atom, —OH, —OR ⁶ , —SH, —S (O) _r R ⁶ , —N (R ^8a ) R ⁸ , —C (O) OR ^6a , ^{-C (O) SR 6a, -C} (S) OR 6a, -C (S) SR 6a, -C (O) R 7, -C (S) R 7, -C (O) N (R 8a) _{^{R 8, -C (S) N}} (R 8a) R 8, -S (O) r N (R 8a) R 8, -Si (R 9a) (R 9b) R 9, phenyl, naphthyl, ^{(Z 2} ) Represents phenyl substituted with _q2 , (Z ² ) naphthyl substituted with _q2 or D2-1 to D2-102, or R ^e together with R ^f represents a C _{2 to} C ₇ alkylene chain by forming, they may form a 3-8 membered ring together with the carbon atom to which R ^e and R ^f are bonded, this time the alkylene chain oxygen Hara May contain 1 or 2 individual sulfur atom or a nitrogen atom, and a halogen atom, cyano, _nitro, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 14} _(C 1 ~C ₆₎ alkyl, -OH , —OR ¹¹ , —SH, —S (O) _r R ¹¹ , an oxo group or a thioxo group,
R ^g and R ^g2 are each independently a hydrogen atom, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ , C ₃ -C ₈ cycloalkyl, optional with R ⁵ substituted in _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ alkenyl, optionally substituted with ^{R 5} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl, optionally ^{R 5} (C ₃ -C ₈ ) cycloalkenyl, C ₂ -C ₆ alkynyl, (C ₂ -C ₆ ) alkynyl optionally substituted with R ⁵ , —S (O) _r R ⁶ , —C ( O) OR ^6a , —C (O) SR ^6a , —C (S) OR ^6a , —C (S) SR ^6a , —C (O) R ⁷ , —C (S) R ⁷ , —C (O) ^{N (R 8a) R 8,} -C (S) N (R 8a) R 8, -S (O) r N (R 8a) R ^{, -Si (R 9a) (R} 9b) R 9, represents phenyl, ^naphthyl, phenyl substituted with (Z _{2) ^q2,} naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ⁵ is a halogen atom, cyano, C ₃ -C ₈ cycloalkyl, —OH, —OR ¹¹ , —SH, —S (O) _r R ¹¹ , —N (R ^13a ) R ¹³ , —C (O). OR ^11a , -C (S) OR ^11a , -C (O) SR ^11a , -C (S) SR ^11a , -C (O) R ¹² , -C (S) R ¹² , -C (O) N ( ^{R 13a) R 13, -C (} S) N (R 13a) R 13, -S (O) r N (R 13a) R 13, -Si (R 9a) (R 9b) R 9, phenyl, naphthyl, ^(Z ₂₎ phenyl substituted with ^_q2, represents naphthyl or D2-1~D2-102 substituted with (Z _{2) q2,}
R ⁶ and R ^6a each independently represent C ₁ -C ₆ alkyl or (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ ;
R ⁷ is a hydrogen _atom, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 14} _(C 1 ~C _{6) alkyl,} C 3 -C ₈ ^cycloalkyl, optionally substituted with ^{R 14} _{(C 3} -C _{8) cycloalkyl,} C 2 -C ₆ ^alkenyl, optionally substituted with ^{R 14} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ ^{cycloalkenyl,} optionally substituted with ^{R 14} _{(C 3} -C _{8) cycloalkenyl,} optionally substituted with C 2 -C _{6 ^{alkynyl, R 14 (C 2 ~C 6}} ) alkynyl, phenyl, ^naphthyl, phenyl substituted with ^{_{(Z 2) q2, (Z}} 2) represents naphthyl or D2-1 to D2-102 substituted with _q2 ,
R ⁸ and R ^8a are each independently a hydrogen atom, cyano, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ , C ₃ -C ₈ cycloalkyl, R ^14. optionally substituted _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ ^alkenyl, optionally substituted with ^{R 14} _(C 2 ~C _{6) alkenyl,} C 3 -C ₈ cycloalkenyl ^{in, R 14} optionally substituted _(C 3 ~C _{8) cycloalkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14} _(C 2 ~C ₆₎ alkynyl, -S _(O) ^{r R 11} in, - C (O) OR ^11a , -C (S) OR ^11a , -C (O) SR ^11a , -C (S) SR ^11a , -C (O) R ¹² , -C (S) R ¹² , -C ( O) N (R ^13a ) R ¹³ , —C (S) N (R ^13a ) _{^{R 13, -S (O) r}} N (R 13a) R 13, -Si (R 9a) (R 9b) R 9, phenyl, ^naphthyl, phenyl substituted with ^{_{(Z 2) q2, (Z}} 2) q2 in or represents naphthyl or D2-1~D2-102 substituted ,, Alternatively, ^{R 8} forms a alkenylene chain alkylene chain or _C 2 -C ₇ of _C 2 -C ₇ together with ^{R 8a} In this case, a 3- to 8-membered ring may be formed together with the nitrogen atom to which R ⁸ and R ^8a are bonded, and this alkylene chain or alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, And a halogen atom, cyano, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ , C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ Alkylthio, ₁ -C _{6 haloalkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ haloalkylsulfonyl, ^phenyl, substituted by (Z _{2) q2} Optionally substituted by a phenyl, oxo group or thioxo group,
R ⁹ , R ^9a and R ^9b each independently represent C ₁ -C ₆ alkyl, C ₁ -C ₆ alkoxy or phenyl;
R ¹¹ _is, -S ^{(O) 2} R 15a _substituent, C 1 -C ₆ ^alkyl, which is optionally substituted with ^{R 14a} _(C 1 ~C _{6) alkyl,} C 2 -C ₆ ^alkenyl, optionally with ^{R 14a} been _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14a} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally substituted with ^{R 14a} (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ cycloalkenyl, optionally substituted with (C ₂ -C ₆ ) cycloalkenyl, phenyl, naphthyl, (Z ² ) _q ² optionally substituted with R ^14a Represents phenyl, (Z ² ) _q2 substituted naphthyl or D2-1 to D2-102;
R ^11a and R ¹² are each independently a hydrogen atom, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a , C ₂ -C ₆ alkenyl, optionally with R ^14a substituted substituted _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14a} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally in ^{R 14a} (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ cycloalkenyl, (C ₂ -C ₆ ) cycloalkenyl optionally substituted with R ^14a , phenyl, naphthyl, substituted with (Z ² ) _q ² Naphthyl substituted with phenyl, (Z ² ) _q2 or D2-1 to D2-102,
R ¹³ and R ^13a are each independently a hydrogen atom, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a , C ₂ -C ₆ alkenyl, optionally R ^14a substituted substituted _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 14a} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally in ^{R 14a} (C ₃ -C ₈ ) cycloalkyl, C ₂ -C ₆ cycloalkenyl, (C ₂ -C ₆ ) cycloalkenyl optionally substituted with R ^14a , phenyl, naphthyl, substituted with (Z ² ) _q ^{2 phenyl,} (Z ₂₎ ,, or or represents naphthyl or D2-1~D2-102 substituted with ^{_q2, R 13} is an alkylene chain or _C 2 ~ of _C 2 -C ₇ together with ^{R 13a} C Of by forming the alkenylene chain may form a 3-8 membered ring together with the nitrogen atom to which R ¹³ and R ^13a are attached, this time the alkylene chain or alkenylene chain oxygen atom, a sulfur atom or a nitrogen atom One (1) and halogen atom, cyano, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a , C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy , _C 1 -C _{6 alkylthio,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ haloalkylsulfonyl, phenyl, (Z ² ) optionally substituted by a phenyl, oxo group or thioxo group substituted by _q2 ,
R ¹⁴ and ^{R 14a} are each independently a halogen atom, cyano, _nitro, C 3 -C _{8 cycloalkyl,} C 3 -C _{8 halocycloalkyl,} C 3 -C _{8 cycloalkenyl,} C 3 -C ₈ Haroshikuro Alkenyl, —OH, —OR ¹⁵ , —SH, —S (O) _r R ¹⁵ , —N (R ^17a ) R ¹⁷ , —C (O) OR ¹⁵ , —C (O) SR ¹⁵ , —C (S ^{) OR 15, -C (S)} SR 15, -C (O) R 16, -C (O) N (R 17a) R 17, -C (S) N (R 17a) R 17, -S (O _{^{) r N (R 17a) R}} 17, -C (= NR 17) OR 15, -C (= NR 17) S (O) r R 15, -C (= NR 17) R 16, -C (= NOH ^{) R 16, -C (= NOR} 15) R 16, -C {= NN (R 17a) R 1 ^{} R 16, -Si (R 9b} ) (R 9a) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, (Z ₂₎ is substituted with _q2 naphthyl or D2-1~D2-102 Represents, represents,
R ¹⁵ and ^{R 15a} have been replaced each independently _C 1 -C ₆ ^alkyl, optionally substituted with ^{R 18} _(C 1 ~C _{6) alkyl,} C 2 -C ₆ ^alkenyl, optionally with ^{R 18} _(C 2 _{~C 6) alkenyl,} optionally substituted with C 2 -C ₆ ^alkynyl, which is optionally substituted with ^{R 18} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^{cycloalkyl, R 18} ( C ₃ -C _{8) cycloalkyl,} C 2 -C ₆ ^{cycloalkenyl,} optionally substituted with ^{R 18} _(C 2 ~C ₆₎ ^{cycloalkenyl, -Si (R 9b) (R} 9a) R 9, phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, (Z ₂₎ naphthyl or D2-1~D2-102 substituted with _q2 represent,
R ¹⁶ is a hydrogen _atom, C 1 -C ₆ ^alkyl, optionally substituted with ^{R 18} _(C 1 ~C _{6) alkyl,} C 2 -C ₆ ^alkenyl, optionally substituted with ^{R 18} _(C 2 ~ C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 18} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^cycloalkyl, optionally substituted with ^{R 18} _(C 3 ~C _{8) cycloalkyl,} C 2 -C ₆ ^{cycloalkenyl,} optionally substituted with ^{R 18} _(C 2 ~C ₆₎ ^{cycloalkenyl, -Si (R 9b) (R} 9a) R 9, phenyl, naphthyl, (Z phenyl substituted with ^{2) _q2,} the (Z ₂₎ naphthyl or D2-1~D2-102 substituted with _q2 represent,
R ¹⁷ and R ^17a are each independently a hydrogen atom, cyano, nitro, C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁸ , C ₂ -C ₆ alkenyl, R optionally substituted with ¹⁸ _(C 2 ~C _{6) alkenyl,} C 2 -C ₆ ^alkynyl, optionally substituted with ^{R 18} _(C 2 ~C _{6) alkynyl,} C 3 -C ₈ ^{cycloalkyl, R 18} (C ₃ -C ₈ ) cycloalkyl optionally substituted with, C ₂ -C ₆ cycloalkenyl, (C ₂ -C ₆ ) cycloalkenyl optionally substituted with R ¹⁸ , —Si (R ^9b ) (R ^{9a) R 9,} phenyl, ^naphthyl, (Z ₂₎ phenyl substituted with ^_q2, or represents (Z ₂₎ naphthyl or D2-1~D2-102 substituted with _q2, ^{or, R 17} is a ^{R 17a} Together By forming the alkylene chain or alkenylene chain of _C 2 -C ₇ for ₂ -C ^_7, may form a 3-8 membered ring together with the nitrogen atom ^{to which R 17} and ^{R 17a} are attached, this time the alkylene chain Alternatively, the alkenylene chain may contain one oxygen atom, sulfur atom or nitrogen atom, and (C ₁ -C ₆ ) alkyl optionally substituted with a halogen atom, cyano, C ₁ -C ₆ alkyl, R ¹⁸ , C ₁ -C _{6 alkoxy,} C 1 -C _{6 haloalkoxy,} C 1 -C _{6 alkylthio,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 alkylsulfinyl,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ haloalkylsulfonyl, ^phenyl, (Z ₂₎ phenyl substituted by _q2, oxo group or thioxo group Thus it may be optionally substituted,
R ¹⁸ is a halogen atom, cyano, nitro, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₁ -C ₆ alkylthio, C ₁ -C ₆ haloalkylthio, C ₁ -C ₆ alkylsulfinyl, C 1 ₁ -C _{6 haloalkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C ₆ ^{haloalkylsulfonyl, -Si (R 9b) (R} 9a) R 9, phenyl, ^naphthyl, phenyl substituted with (Z _{2) q2} , (Z ² ) naphthyl substituted with _q2 or D2-1 to D2-102,
D2-1 to D2-102 each represent a ring represented by the following structural formula;




X ² represents a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , —C (O) NH ₂ , —C (S) NH ₂ , —S (O) ₂ NH ₂ or R ²⁰ . , T1, t2 or t4 each represents an integer of 2 or more, each X ² may be the same as or different from each other. Further, when two X ² are adjacent, X ² represents —CH ₂ CH ₂ CH ₂ —, —CH ₂ CH ₂ O—, —CH ₂ OCH ₂ —, —OCH ₂ O—, —CH ₂ CH ₂ S—, —CH ₂ SCH ₂ —, — CH ₂ CH ₂ CH ₂ CH ₂ —, —CH ₂ CH ₂ CH ₂ O—, —CH ₂ CH ₂ OCH ₂ —, —CH ₂ OCH ₂ O—, —OCH ₂ CH ₂ O—, —CH ₂ CH ₂ by CH ₂ S- or form a -OCH ₂ CH ₂ S-, it A 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each X ² is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is a halogen atom, C _{1 to} C _6. alkyl _group, C 1 -C ₆ haloalkyl _group, C 1 -C ₆ alkoxy _group, C 1 -C ₆ alkylthio _group, optionally substituted by C 1 -C ₆ alkylsulfinyl group or a _C 1 -C ₆ alkylsulfonyl group Well,
X ^2a is a hydrogen atom, cyano, _-OH, an -NH 2, -CHO or ^{R 20, when X 2} is present at the adjacent position to ^{X 2a} is, ^{X 2a} and ^{X 2} the adjacent, -CH ₂ CH ₂ CH ₂ CH ₂ —, —CH═CHCH═CH—, —N═CHCH═CH—, —CH═N—CH═CH—, —CH═CH—N═CH— or —CH═CH— By forming CH═N—, a 6-membered ring may be formed together with the atom to which each of X ^2a and X ² is bonded. At this time, the hydrogen atom bonded to each carbon atom forming the ring is halogen _atom, C 1 -C ₆ alkyl _group, C 1 -C ₆ haloalkyl _group, C 1 -C ₆ alkoxy _group, C 1 -C ₆ alkylthio _group, C 1 -C ₆ alkylsulfinyl group or a _C 1 -C ₆ alkyl Optionally substituted by a sulfonyl group It may be,
X ^2b is a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , —C (O) NH ₂ , —C (S) NH ₂ , —S (O) ₂ NH ₂ , —CHO or R ^When u1, u2, u4, u5, u6, u7, u8 or u9 represent an integer of 2 or more, each X ^2b may be the same as or different from each other, When two X ^2b are substituted on the same carbon, the two X ^2b together are oxo, thioxo, imino, C ₁ -C ₆ alkylimino, C ₁ -C ₆ alkoxyimino or C _1- C ₆ alkylidene may be formed,
Z ² represents a halogen atom, cyano, nitro, —OH, —SH, —NH ₂ , —C (O) NH ₂ , —C (S) NH ₂ , —S (O) ₂ NH ₂ or R ²⁰ . , Q2 represents an integer of 2 or more, each Z ² may be the same as or different from each other, and when two Z ² are adjacent, the two adjacent Z ² are − _{CH 2 CH 2 CH 2 -,} - CH 2 CH 2 O -, - CH 2 OCH 2 -, - OCH 2 O -, - CH 2 CH 2 S -, - CH 2 SCH 2 -, - CH 2 CH 2 N _{^{(X 2a) -, - CH}} 2 N (X 2a) CH 2 -, - CH 2 CH 2 CH 2 CH 2 -, - CH 2 CH 2 CH 2 O -, - CH 2 CH 2 OCH 2 -, - CH ₂ OCH ₂ O—, —OCH ₂ CH ₂ O—, —OCH ₂ CH ₂ S—, —C _{H 2 CH = CH -, -} OCH = CH -, - SCH = CH -, - N (X 2a) CH = CH -, - OCH = N -, - SCH = N -, - N (X 2a) CH = _{^{N -, - N (X 2a}} ) N = CH -, - OCH 2 CH = CH -, - N = CHCH = CH -, - CH = NCH = CH -, - N = NCH = CH -, - CH = NN By forming ═CH—, —N═CHCH═N— or —N═CHN═CH—, a 5-membered ring or a 6-membered ring may be formed together with the carbon atom to which each Z ² is bonded. when the hydrogen atoms bonded to each carbon atom forming the ring, a halogen _atom, C 1 -C ₆ alkyl _group, C 1 -C ₆ haloalkyl _group, C 1 -C ₆ alkoxy _group, C 1 -C ₆ alkylthio _group, C 1 -C ₆ alkylsulfinyl group or a _C 1 -C ₆ Arukirusu It may be optionally substituted by Honiru group,
R ²⁰ is C ₁ -C ₆ alkyl, C ₂ -C ₆ alkenyl, C ₂ -C ₆ alkynyl, C ₃ -C ₈ cycloalkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ²⁸ , optionally substituted with R ²⁸ _(C 2 ~C ₆₎ ^alkenyl, optionally substituted with ^{R 28} _(C 2 ^~C ₆₎ ^alkynyl, optionally substituted with ^{R 28} _(C 3 ^~C ₈₎ cycloalkyl (C ₃ -C ₈ ) cycloalkenyl optionally substituted with alkyl, R ²⁸ , —OR ²⁵ , —S (O) _r R ²⁵ , —C (O) OR ²⁵ , —C (O) R ²⁶ , — ^{N (R 27a) R 27,} -C (O) N (R 27a) R 27, -C (S) N (R 27a) R 27, -S (O) r N (R 27a) R 27, phenyl, phenyl optionally substituted with C ₁ -C ₆ alkyl or halogen atom It represents,
R ²⁵ , R ²⁶ and R ^27a each independently represent a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl or C ₃ -C ₈ cycloalkyl,
R ²⁷ is a hydrogen atom, C ₁ -C ₆ alkyl, C ₁ -C ₆ haloalkyl, C ₃ -C ₈ cycloalkyl, C ₁ -C ₆ alkylcarbonyl, C ₃ -C ₈ cycloalkylcarbonyl, C ₁ -C Represents ₆ haloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl or C ₁ -C ₆ haloalkoxycarbonyl,
R ²⁸ and R ^28a are each independently a halogen atom, cyano, nitro, C ₁ -C ₆ alkoxy, C ₁ -C ₆ haloalkoxy, C ₂ -C ₆ alkenyloxy, C ₁ -C ₆ alkylthio, C ₁ -C _{6 alkylsulfinyl,} C 1 -C _{6 alkylsulfonyl,} C 1 -C _{6 haloalkylthio,} C 1 -C _{6 haloalkylsulfinyl,} C 1 -C _{6 haloalkylsulfonyl,} C 1 -C _{6 alkylcarbonyl,} C 3 -C ₈ cycloalkylcarbonyl, C ₁ -C ₆ haloalkylcarbonyl, C ₃ -C ₈ halocycloalkylcarbonyl, C ₁ -C ₆ alkoxycarbonyl, C ₁ -C ₆ haloalkoxycarbonyl, C ₁ -C ₆ alkylthiocarbonyl, C ₁ -C _{6 alkoxythiocarbonyl,} C 1 -C ₆ alkyl dithio months _Boniru, C 1 -C _{6 alkylaminocarbonyl,} C 1 -C ₆ haloalkylcarbonyl aminocarbonyl, di _(C 1 -C ₆ alkyl) aminocarbonyl, tri _(C 1 -C ₆ alkyl) _silyl, C 1 -C ₆ alkylamino Sulfonyl, di (C ₁ -C ₆ alkyl) aminosulfonyl, C ₁ -C ₆ alkylcarbonyloxy, C ₁ -C ₆ alkylsulfonyloxy, C ₁ -C ₆ haloalkylsulfonyloxy, C ₁ -C ₆ alkylamino or di _(C 1 -C ₆ alkyl) an amino,
n, t1, and u1 each independently represents an integer of 0, 1, 2, or 3;
t2 and u2 each independently represent an integer of 0, 1 or 2;
t3 represents an integer of 0 or 1,
t4 and u4 each independently represent an integer of 0, 1, 2, 3 or 4;
u5 represents an integer of 0, 1, 2, 3, 4 or 5;
u6 each independently represents an integer of 0, 1, 2, 3, 4, 5 or 6;
u7 each independently represents an integer of 0, 1, 2, 3, 4, 5, 6 or 7;
u8 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7 or 8;
u9 represents an integer of 0, 1, 2, 3, 4, 5, 6, 7, 8 or 9,
q2 represents an integer of 1, 2, 3, 4 or 5,
m1, m2 and m4 each independently represents an integer of 0 or 1,
r, r2 and r3 each independently represents an integer of 0, 1 or 2] or a salt thereof. Ａ^１は、−ＣＲ^１を表し、
Ｒ^１、Ｒ^３及びＲ^４は、各々独立して水素原子、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^２は、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表す請求項１記載のピラゾール誘導体又はその塩。 A ¹ represents -CR ¹
R ¹ , R ³ and R ⁴ each independently represents a hydrogen atom, a halogen atom or C ₁ -C ₆ alkyl;
The pyrazole derivative or a salt thereof according to claim ₁ , wherein R ² represents a halogen atom or C ₁ -C ₆ alkyl. Ａ^１は、−Ｎ（−Ｏ）_ｍ２を表し、
Ｒ^２は、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^３及びＲ^４は、各々独立して水素原子、ハロゲン原子又はＣ_１〜Ｃ_６アルキルを表す請求項１記載のピラゾール誘導体又はその塩。 A ¹ represents -N (-O) _m2 ,
R ² represents a halogen atom or C ₁ -C ₆ alkyl,
The pyrazole derivative or a salt thereof according to claim ₁ , wherein R ³ and R ⁴ each independently represent a hydrogen atom, a halogen atom or C ₁ -C ₆ alkyl. Ｒ^１及びＲ^４は、水素原子を表し、
Ａ^２は、−Ｃ（Ｒ^ａ）＝ＮＯＲ^ｂ、−Ｃ≡ＣＲ^ｃ、−Ｃ（Ｒ^ｄ）＝Ｃ（Ｒ^ｅ）Ｒ^ｆ又は−Ｃ（Ｒ^ａ）＝ＮＮ（Ｒ^ｇ）Ｒ^ｇ２を表し、
Ｒ^ａは、水素原子、Ｃ_１〜Ｃ_６アルキル、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｎ（Ｒ^８ａ）Ｒ^８又はＤ２−７を表すか、或いは、Ｒ^ａはＲ^３と一緒になってＣ_３のアルキレン鎖を形成することにより、Ｒ^ａが結合する炭素原子及びＲ^３が結合する炭素原子と共に６員環を形成してもよく、
Ｒ^ｂは、Ｃ_１〜Ｃ_６アルキル、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^ｃは、水素原子、Ｒ^５で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＳＲ^６ａ、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｓｉ（Ｒ^９ａ）（Ｒ^９ｂ）Ｒ^９又はＤ２−３２を表し、
Ｒ^ｄ及びＲ^ｅは、水素原子を表し、
Ｒ^ｆは、−Ｓ（Ｏ）_ｒＲ^６、−Ｃ（Ｏ）ＯＲ^６ａ、−Ｃ（Ｏ）Ｎ（Ｒ^８ａ）Ｒ^８、−Ｎ（Ｒ^８ａ）Ｒ^８、フェニル、（Ｚ^２）_ｑ２で置換されたフェニル又はＤ２−７を表すか、或いは、Ｒ^ｅはＲ^ｆと一緒になってＣ_４のアルキレン鎖を形成することにより、Ｒ^ｅ及びＲ^ｆが結合する炭素原子と共に５員環を形成し、このときこのアルキレン鎖は窒素原子を１個含み、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、オキソ基によって任意に置換されてもよく、
Ｒ^ｇは、−Ｃ（Ｏ）Ｒ^７を表し、
Ｒ^ｇ２は、Ｃ_１〜Ｃ_６アルキルを表し、
Ｒ^５は、ハロゲン原子、−ＯＨ、−ＯＲ^１１、−Ｓ（Ｏ）_ｒＲ^１１又はＤ２−３２又はＤ２−３４を表し、
Ｒ^６及びＲ^６ａは、各々独立してＣ_１〜Ｃ_６アルキルを表し、
Ｒ^７は、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^８は、Ｃ_１〜Ｃ_６アルキル、Ｒ^１４で任意に置換された（Ｃ_１〜Ｃ_６）アルキル、−Ｃ（Ｏ）ＯＲ^１１ａ又は−Ｃ（Ｏ）Ｒ^１２を表し、
Ｒ^８ａは、水素原子又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^１１は、−Ｓ（Ｏ）_２Ｒ^１５ａ又はＣ_１〜Ｃ_６アルキルを表し、
Ｒ^１１ａは、Ｃ_１〜Ｃ_６アルキルを表し、
Ｒ^１２は、Ｒ^１４ａで任意に置換された（Ｃ_１〜Ｃ_６）アルキルを表し、
Ｒ^１４は、ハロゲン原子又は−Ｓ（Ｏ）_ｒＲ^１５を表し、
Ｒ^１４ａは、−Ｓ（Ｏ）_ｒＲ^１５を表し、
Ｒ^１５及びＲ^１５ａは、各々独立してＣ_１〜Ｃ_６アルキルを表し、
Ｘ^２及びＺ^２は、各々独立してＣ_１〜Ｃ_６ハロアルキルを表し、
ｑ２は、０又は１の整数を表し、
ｔ１は、１の整数を表し、
ｔ４は、０又は１の整数を表し、
ｎ、ｍ１及びｍ２は、０を表し、
ｒは、０、１又は２の整数を表す請求項２記載のピラゾール誘導体又はその塩。 R ¹ and R ⁴ represent a hydrogen atom,
A ² represents —C (R ^a ) = NOR ^b , —C≡CR ^c , —C (R ^d ) = C (R ^e ) R ^f or —C (R ^a ) = NN (R ^g ) R ^g2 Represent,
R ^a represents a hydrogen atom, C ₁ -C ₆ alkyl, —C (O) OR ^6a , —C (O) N (R ^8a ) R ⁸ , —N (R ^8a ) R ⁸ or D 2-7. Alternatively, R ^a may form a C ₃ alkylene chain together with R ³ to form a 6-membered ring together with the carbon atom to which R ^a is bonded and the carbon atom to which R ³ is bonded;
R ^b represents C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ ;
R ^c is a hydrogen atom, (C ₁ -C ₆ ) alkyl optionally substituted with R ⁵ , —S (O) _r R ⁶ , —C (O) SR ^6a , —C (O) N (R ^{8a ) R 8, -Si (R 9a} ) ( represents R 9b) ^{R 9} or D2-32,
R ^d and R ^e represent a hydrogen atom,
R ^{f _{is, -S (O) r R 6}} , -C (O) OR 6a, -C (O) N (R 8a) R 8, -N (R 8a) R 8, ^phenyl, (Z _{2) q2} Represents phenyl or D2-7 substituted with R 5, or R ^e together with R ^f forms a C ₄ alkylene chain to form a 5-membered ring together with the carbon atom to which R ^e and R ^f are bonded. Wherein the alkylene chain contains one nitrogen atom and may be optionally substituted by a (C ₁ -C ₆ ) alkyl, oxo group optionally substituted with R ¹⁴ ,
R ^g represents —C (O) R ⁷ ,
R ^g2 represents C ₁ -C ₆ alkyl,
R ⁵ represents a halogen atom, —OH, —OR ¹¹ , —S (O) _r R ¹¹ or D2-32 or D2-34;
R ⁶ and R ^6a each independently represent C ₁ -C ₆ alkyl,
R ⁷ represents (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ ;
R ⁸ represents C ₁ -C ₆ alkyl, (C ₁ -C ₆ ) alkyl optionally substituted with R ¹⁴ , —C (O) OR ^11a or —C (O) R ¹² ,
R ^8a represents a hydrogen atom or C ₁ -C ₆ alkyl;
R ¹¹ represents —S (O) ₂ R ^15a or C ₁ -C ₆ alkyl;
R ^11a represents C ₁ -C ₆ alkyl;
R ¹² represents (C ₁ -C ₆ ) alkyl optionally substituted with R ^14a ,
R ¹⁴ represents a halogen atom or —S (O) _r R ¹⁵ ;
R ^14a represents -S (O) _r R ¹⁵ ;
R ¹⁵ and R ^15a each independently represent C ₁ -C ₆ alkyl;
X ² and Z ² each independently represent C ₁ -C ₆ haloalkyl,
q2 represents an integer of 0 or 1,
t1 represents an integer of 1,
t4 represents an integer of 0 or 1,
n, m1 and m2 represent 0;
The pyrazole derivative or a salt thereof according to claim 2, wherein r represents an integer of 0, 1 or 2. 請求項１〜請求項４記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する有害生物防除剤。   The pest control agent which contains the 1 type (s) or 2 or more types chosen from the pyrazole derivative and its salt of Claims 1-4 as an active ingredient. 請求項１〜請求項４記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する農薬。   An agrochemical containing one or more selected from the pyrazole derivative according to claim 1 and a salt thereof as an active ingredient. 請求項１〜請求項４記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する哺乳動物又は鳥類の内部もしくは外部寄生虫防除剤。   A mammal or avian internal or ectoparasite control agent comprising one or more selected from the pyrazole derivatives and salts thereof according to claim 1 as active ingredients. 請求項１〜請求項４記載のピラゾール誘導体及びその塩から選ばれる１種又は２種以上を有効成分として含有する殺虫剤又は殺ダニ剤。   An insecticide or acaricide containing, as an active ingredient, one or more selected from the pyrazole derivatives and salts thereof according to claim 1. 請求項１〜請求項４記載のピラゾール誘導体及びそれらの塩から選ばれる１種又は２種以上を有効成分として含有する土壌処理剤。   The soil treatment agent which contains the 1 type (s) or 2 or more types chosen from the pyrazole derivative of Claims 1-4, and those salts as an active ingredient. 土壌処理方法が土壌潅注処理である請求項９記載の土壌処理剤。   The soil treatment agent according to claim 9, wherein the soil treatment method is soil irrigation treatment.