IT1318636B1 - Derivati dell'acido 2- o 3- tenoico ad attivita' antagonista deirecettori del glutammato. - Google Patents
Derivati dell'acido 2- o 3- tenoico ad attivita' antagonista deirecettori del glutammato.Info
- Publication number
- IT1318636B1 IT1318636B1 IT2000MI001667A ITMI20001667A IT1318636B1 IT 1318636 B1 IT1318636 B1 IT 1318636B1 IT 2000MI001667 A IT2000MI001667 A IT 2000MI001667A IT MI20001667 A ITMI20001667 A IT MI20001667A IT 1318636 B1 IT1318636 B1 IT 1318636B1
- Authority
- IT
- Italy
- Prior art keywords
- acid derivatives
- antagonist activity
- glutamate receptors
- tenoic acid
- tenoic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT2000MI001667A IT1318636B1 (it) | 2000-07-21 | 2000-07-21 | Derivati dell'acido 2- o 3- tenoico ad attivita' antagonista deirecettori del glutammato. |
PCT/IB2001/001295 WO2002008220A1 (en) | 2000-07-21 | 2001-07-20 | 2-thenoic acid (thiophene) derivatives having glutamate receptor antagonistic activity |
AU2001275767A AU2001275767A1 (en) | 2000-07-21 | 2001-07-20 | 2-thenoic acid (thiophene) derivatives having glutamate receptor antagonistic activity |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT2000MI001667A IT1318636B1 (it) | 2000-07-21 | 2000-07-21 | Derivati dell'acido 2- o 3- tenoico ad attivita' antagonista deirecettori del glutammato. |
Publications (3)
Publication Number | Publication Date |
---|---|
ITMI20001667A0 ITMI20001667A0 (it) | 2000-07-21 |
ITMI20001667A1 ITMI20001667A1 (it) | 2002-01-21 |
IT1318636B1 true IT1318636B1 (it) | 2003-08-27 |
Family
ID=11445531
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT2000MI001667A IT1318636B1 (it) | 2000-07-21 | 2000-07-21 | Derivati dell'acido 2- o 3- tenoico ad attivita' antagonista deirecettori del glutammato. |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU2001275767A1 (it) |
IT (1) | IT1318636B1 (it) |
WO (1) | WO2002008220A1 (it) |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK124393D0 (da) * | 1993-11-03 | 1993-11-03 | Lundbeck & Co As H | Compounds |
US5962521A (en) * | 1997-04-04 | 1999-10-05 | Guilford Pharmaceuticals Inc. | Hydroxamic acid derivatives |
UA54403C2 (uk) * | 1996-10-01 | 2003-03-17 | Н'Юросерч А/С | Похідні індол-2,3-діон-3-оксиму, фармацевтична композиція, спосіб лікування розладу чи захворювання ссавців, у тому числі людини та спосіб одержання похідних індол-2,3-діон-3-оксиму |
GB9626151D0 (en) * | 1996-12-17 | 1997-02-05 | Lilly Industries Ltd | Pharmaceutical compounds |
PE20000942A1 (es) * | 1998-07-31 | 2000-09-28 | Lilly Co Eli | Derivados de amida, carbamato y urea |
AU5233699A (en) * | 1998-07-31 | 2000-02-21 | Eli Lilly And Company | Sulfonamide derivatives |
TW593241B (en) * | 1999-04-20 | 2004-06-21 | Hoffmann La Roche | Carbamic acid derivatives |
-
2000
- 2000-07-21 IT IT2000MI001667A patent/IT1318636B1/it active
-
2001
- 2001-07-20 AU AU2001275767A patent/AU2001275767A1/en not_active Abandoned
- 2001-07-20 WO PCT/IB2001/001295 patent/WO2002008220A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
ITMI20001667A0 (it) | 2000-07-21 |
ITMI20001667A1 (it) | 2002-01-21 |
AU2001275767A1 (en) | 2002-02-05 |
WO2002008220A1 (en) | 2002-01-31 |
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