IT1301968B1 - Derivati di eritromicina ad attivita' antibiotica - Google Patents
Derivati di eritromicina ad attivita' antibioticaInfo
- Publication number
- IT1301968B1 IT1301968B1 IT1998MI001776A ITMI981776A IT1301968B1 IT 1301968 B1 IT1301968 B1 IT 1301968B1 IT 1998MI001776 A IT1998MI001776 A IT 1998MI001776A IT MI981776 A ITMI981776 A IT MI981776A IT 1301968 B1 IT1301968 B1 IT 1301968B1
- Authority
- IT
- Italy
- Prior art keywords
- erythromycin derivatives
- antibiotic activity
- erythromycin
- derivatives
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Priority Applications (8)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1998MI001776A IT1301968B1 (it) | 1998-07-30 | 1998-07-30 | Derivati di eritromicina ad attivita' antibiotica |
AU52901/99A AU5290199A (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
DE69915487T DE69915487T2 (de) | 1998-07-30 | 1999-07-27 | Erythromycin-derivate mit antibiotischer wirkung |
EP99938386A EP1100762B1 (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
US09/744,244 US6468979B1 (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
PCT/EP1999/005485 WO2000006606A2 (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
AT99938386T ATE261425T1 (de) | 1998-07-30 | 1999-07-27 | Erythromycin-derivate mit antibiotischer wirkung |
ES99938386T ES2215396T3 (es) | 1998-07-30 | 1999-07-27 | Derivados de eritromicina con actividad antibiotica. |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT1998MI001776A IT1301968B1 (it) | 1998-07-30 | 1998-07-30 | Derivati di eritromicina ad attivita' antibiotica |
Publications (3)
Publication Number | Publication Date |
---|---|
ITMI981776A0 ITMI981776A0 (it) | 1998-07-30 |
ITMI981776A1 ITMI981776A1 (it) | 2000-01-30 |
IT1301968B1 true IT1301968B1 (it) | 2000-07-20 |
Family
ID=11380563
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT1998MI001776A IT1301968B1 (it) | 1998-07-30 | 1998-07-30 | Derivati di eritromicina ad attivita' antibiotica |
Country Status (8)
Country | Link |
---|---|
US (1) | US6468979B1 (it) |
EP (1) | EP1100762B1 (it) |
AT (1) | ATE261425T1 (it) |
AU (1) | AU5290199A (it) |
DE (1) | DE69915487T2 (it) |
ES (1) | ES2215396T3 (it) |
IT (1) | IT1301968B1 (it) |
WO (1) | WO2000006606A2 (it) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6947844B2 (en) * | 2000-08-09 | 2005-09-20 | Yale University | Modulators of ribosomal function and identification thereof |
US6638908B1 (en) * | 2000-08-09 | 2003-10-28 | Yale University | Crystals of the large ribosomal subunit |
US6952650B2 (en) | 2001-08-03 | 2005-10-04 | Yale University | Modulators of ribosomal function and identification thereof |
IL151012A0 (en) * | 2001-08-03 | 2003-02-12 | Ribosomes Structure And Protei | Ribosomes structure and protein synthesis inhibitors |
AR043050A1 (es) * | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
CN1780846A (zh) * | 2003-03-05 | 2006-05-31 | Rib-X医药品有限公司 | 双官能杂环化合物及其制备和使用方法 |
NZ543202A (en) | 2003-05-31 | 2008-04-30 | Micromet Ag | Pharmaceutical composition comprising a bispecific antibody for epcam |
WO2005042554A1 (en) * | 2003-10-30 | 2005-05-12 | Rib-X Pharmaceuticals, Inc. | Bifunctional macrolide heterocyclic compounds and methods of making and using the same |
JP2007512256A (ja) * | 2003-11-18 | 2007-05-17 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | 二官能性マクロライド複素環化合物ならびにこれらを製造する方法およびこれらを使用する方法 |
CN102816194A (zh) * | 2004-02-27 | 2012-12-12 | 瑞伯-X医药品有限公司 | 大环化合物以及其制作和使用方法 |
WO2007025098A2 (en) | 2005-08-24 | 2007-03-01 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
BR112013009823A2 (pt) | 2010-10-22 | 2016-07-05 | Bayer Ip Gmbh | novos compostos heterocíclicos como pesticidas |
BR112017025851A2 (pt) * | 2015-06-01 | 2018-10-16 | Bantam Pharmaceutical, Llc | compostos de pirazol e pirrol substituídos e métodos para usar os mesmos para inibição de iniciação de tradução e tratamento de doenças e distúrbios relacionados aos mesmo |
MX2019006299A (es) | 2016-11-30 | 2019-11-12 | Bantam Pharmaceutical Llc | Compuestos de pirazola sustituida y metodos para usarlos para el tratamiento de enfermedades hiperproliferativas. |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1276901B1 (it) * | 1994-12-13 | 1997-11-03 | Zambon Spa | Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica |
-
1998
- 1998-07-30 IT IT1998MI001776A patent/IT1301968B1/it active IP Right Grant
-
1999
- 1999-07-27 AT AT99938386T patent/ATE261425T1/de not_active IP Right Cessation
- 1999-07-27 US US09/744,244 patent/US6468979B1/en not_active Expired - Fee Related
- 1999-07-27 ES ES99938386T patent/ES2215396T3/es not_active Expired - Lifetime
- 1999-07-27 WO PCT/EP1999/005485 patent/WO2000006606A2/en active IP Right Grant
- 1999-07-27 AU AU52901/99A patent/AU5290199A/en not_active Abandoned
- 1999-07-27 DE DE69915487T patent/DE69915487T2/de not_active Expired - Fee Related
- 1999-07-27 EP EP99938386A patent/EP1100762B1/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
ATE261425T1 (de) | 2004-03-15 |
ITMI981776A1 (it) | 2000-01-30 |
AU5290199A (en) | 2000-02-21 |
WO2000006606A3 (en) | 2000-05-04 |
ES2215396T3 (es) | 2004-10-01 |
EP1100762A2 (en) | 2001-05-23 |
DE69915487T2 (de) | 2005-02-17 |
ITMI981776A0 (it) | 1998-07-30 |
WO2000006606A2 (en) | 2000-02-10 |
EP1100762B1 (en) | 2004-03-10 |
US6468979B1 (en) | 2002-10-22 |
DE69915487D1 (de) | 2004-04-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MX9602837A (es) | Composiciones cosmeticas o farmaceuticas que contienen mangiferina o sus derivados. | |
SE9504661D0 (sv) | New compounds | |
CO5720000A2 (es) | Derivados de macrolidos con actividad antiinflamatoria, su procedimiento de sintesis y composiciones farmaceuticas que los contienen | |
AR066982A2 (es) | Compuestos heteroaromaticos sustituidos como inhibidoress tirosin quinasa, composiciones farmaceuticas que los contiene y su uso en la preparacion de medicamentos | |
KR970006279A (ko) | 약제학적 활성 성분으로서의 6-디메틸아미노메틸-1-페닐-사이클로헥산 화합물 | |
AP9801378A0 (en) | 9-amino-3- keto erythromycin derivatives. | |
PT876388E (pt) | Derivados de eritromicina triciclica | |
IT1301968B1 (it) | Derivati di eritromicina ad attivita' antibiotica | |
CA2326222A1 (en) | Medicinal compositions | |
ES2104845T3 (es) | Composiciones lipofilas de sales de antibioticos oligosacaridos. | |
ATE222243T1 (de) | Pharmazeutisch wirksame benzochinazolin verbindungen | |
HU229443B1 (en) | Betha-carboline particulate form, pharmaceutical compositions containing it, their preparations and their use | |
AP9801321A0 (en) | 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-h-indole derivatives. | |
NO942952L (no) | 11-benzaldoksin-17 ater, fremgangsmåte for deres fremstilling samt legemiddel inneholdende slike | |
ITMI20022292A1 (it) | 9a-azalidi ad attivita' antiinfiammatoria. | |
IT1230703B (it) | Derivati imidazolonici ad attivita' antiipertensiva, loro metodi di preparazione e composizioni farmaceutiche che li contengono. | |
DE69222698D1 (de) | 4-desoxy-4-epipodophyllotoxinderivate oder deren pharmazeutisch akzeptierbaren salze | |
ES2062137T3 (es) | Utilizacion de 5'-deoxi-5'-metil-tioadenosina, s-adenosilmetionina y sus sales para la preparacion de composiciones farmaceuticas reductoras de seborrea. | |
EE9400070A (et) | Bioloogiliselt aktiivsed eburnameniini derivaadid, neid sisaldavad farmatseutilised segud ja nende valmistamise protsess | |
ES2097736T3 (es) | Peptido ciclico con actividad antagonista de sustancia p y sustancia k. | |
SE9504662D0 (sv) | New compounds | |
DE69813263T2 (de) | Hydrazono-benzazulen-derivate, pharmazeutische zusammensetzungen und zwischenprodukte | |
FI945164A0 (fi) | Biologisesti aktiivisesti ureidojohdannaiset, jotka ovat käyttökelpoisia antimetastaattisina aineina | |
NO940844D0 (no) | Farmasöytisk aktive hydroksykarboksylsyrederivater | |
SE9902742D0 (sv) | New pharmaceutical formultion |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
0001 | Granted |