IT1301968B1 - Derivati di eritromicina ad attivita' antibiotica - Google Patents

Derivati di eritromicina ad attivita' antibiotica

Info

Publication number
IT1301968B1
IT1301968B1 IT1998MI001776A ITMI981776A IT1301968B1 IT 1301968 B1 IT1301968 B1 IT 1301968B1 IT 1998MI001776 A IT1998MI001776 A IT 1998MI001776A IT MI981776 A ITMI981776 A IT MI981776A IT 1301968 B1 IT1301968 B1 IT 1301968B1
Authority
IT
Italy
Prior art keywords
erythromycin derivatives
antibiotic activity
erythromycin
derivatives
preparing
Prior art date
Application number
IT1998MI001776A
Other languages
English (en)
Inventor
Franco Pellacini
Daniela Botta
Enrico Albini
Domenico Ungheri
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of ITMI981776A0 publication Critical patent/ITMI981776A0/it
Priority to IT1998MI001776A priority Critical patent/IT1301968B1/it
Priority to US09/744,244 priority patent/US6468979B1/en
Priority to DE69915487T priority patent/DE69915487T2/de
Priority to EP99938386A priority patent/EP1100762B1/en
Priority to AU52901/99A priority patent/AU5290199A/en
Priority to PCT/EP1999/005485 priority patent/WO2000006606A2/en
Priority to AT99938386T priority patent/ATE261425T1/de
Priority to ES99938386T priority patent/ES2215396T3/es
Publication of ITMI981776A1 publication Critical patent/ITMI981776A1/it
Application granted granted Critical
Publication of IT1301968B1 publication Critical patent/IT1301968B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IT1998MI001776A 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica IT1301968B1 (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IT1998MI001776A IT1301968B1 (it) 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica
AU52901/99A AU5290199A (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
DE69915487T DE69915487T2 (de) 1998-07-30 1999-07-27 Erythromycin-derivate mit antibiotischer wirkung
EP99938386A EP1100762B1 (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
US09/744,244 US6468979B1 (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
PCT/EP1999/005485 WO2000006606A2 (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
AT99938386T ATE261425T1 (de) 1998-07-30 1999-07-27 Erythromycin-derivate mit antibiotischer wirkung
ES99938386T ES2215396T3 (es) 1998-07-30 1999-07-27 Derivados de eritromicina con actividad antibiotica.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1998MI001776A IT1301968B1 (it) 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica

Publications (3)

Publication Number Publication Date
ITMI981776A0 ITMI981776A0 (it) 1998-07-30
ITMI981776A1 ITMI981776A1 (it) 2000-01-30
IT1301968B1 true IT1301968B1 (it) 2000-07-20

Family

ID=11380563

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1998MI001776A IT1301968B1 (it) 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica

Country Status (8)

Country Link
US (1) US6468979B1 (it)
EP (1) EP1100762B1 (it)
AT (1) ATE261425T1 (it)
AU (1) AU5290199A (it)
DE (1) DE69915487T2 (it)
ES (1) ES2215396T3 (it)
IT (1) IT1301968B1 (it)
WO (1) WO2000006606A2 (it)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6947844B2 (en) * 2000-08-09 2005-09-20 Yale University Modulators of ribosomal function and identification thereof
US6638908B1 (en) * 2000-08-09 2003-10-28 Yale University Crystals of the large ribosomal subunit
US6952650B2 (en) 2001-08-03 2005-10-04 Yale University Modulators of ribosomal function and identification thereof
IL151012A0 (en) * 2001-08-03 2003-02-12 Ribosomes Structure And Protei Ribosomes structure and protein synthesis inhibitors
AR043050A1 (es) * 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
CN1780846A (zh) * 2003-03-05 2006-05-31 Rib-X医药品有限公司 双官能杂环化合物及其制备和使用方法
NZ543202A (en) 2003-05-31 2008-04-30 Micromet Ag Pharmaceutical composition comprising a bispecific antibody for epcam
WO2005042554A1 (en) * 2003-10-30 2005-05-12 Rib-X Pharmaceuticals, Inc. Bifunctional macrolide heterocyclic compounds and methods of making and using the same
JP2007512256A (ja) * 2003-11-18 2007-05-17 リブ−エックス ファーマシューティカルズ,インコーポレイテッド 二官能性マクロライド複素環化合物ならびにこれらを製造する方法およびこれらを使用する方法
CN102816194A (zh) * 2004-02-27 2012-12-12 瑞伯-X医药品有限公司 大环化合物以及其制作和使用方法
WO2007025098A2 (en) 2005-08-24 2007-03-01 Rib-X Pharmaceuticals, Inc. Triazole compounds and methods of making and using the same
BR112013009823A2 (pt) 2010-10-22 2016-07-05 Bayer Ip Gmbh novos compostos heterocíclicos como pesticidas
BR112017025851A2 (pt) * 2015-06-01 2018-10-16 Bantam Pharmaceutical, Llc compostos de pirazol e pirrol substituídos e métodos para usar os mesmos para inibição de iniciação de tradução e tratamento de doenças e distúrbios relacionados aos mesmo
MX2019006299A (es) 2016-11-30 2019-11-12 Bantam Pharmaceutical Llc Compuestos de pirazola sustituida y metodos para usarlos para el tratamiento de enfermedades hiperproliferativas.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1276901B1 (it) * 1994-12-13 1997-11-03 Zambon Spa Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica

Also Published As

Publication number Publication date
ATE261425T1 (de) 2004-03-15
ITMI981776A1 (it) 2000-01-30
AU5290199A (en) 2000-02-21
WO2000006606A3 (en) 2000-05-04
ES2215396T3 (es) 2004-10-01
EP1100762A2 (en) 2001-05-23
DE69915487T2 (de) 2005-02-17
ITMI981776A0 (it) 1998-07-30
WO2000006606A2 (en) 2000-02-10
EP1100762B1 (en) 2004-03-10
US6468979B1 (en) 2002-10-22
DE69915487D1 (de) 2004-04-15

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Legal Events

Date Code Title Description
0001 Granted