IL96891A0 - Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them - Google Patents

Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL96891A0
IL96891A0 IL96891A IL9689191A IL96891A0 IL 96891 A0 IL96891 A0 IL 96891A0 IL 96891 A IL96891 A IL 96891A IL 9689191 A IL9689191 A IL 9689191A IL 96891 A0 IL96891 A0 IL 96891A0
Authority
IL
Israel
Prior art keywords
indole
substituted
membered heteroaromatic
preparation
heteroaromatic compounds
Prior art date
Application number
IL96891A
Other languages
English (en)
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB909001018A external-priority patent/GB9001018D0/en
Priority claimed from GB909008587A external-priority patent/GB9008587D0/en
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Publication of IL96891A0 publication Critical patent/IL96891A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL96891A 1990-01-17 1991-01-07 Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them IL96891A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB909001018A GB9001018D0 (en) 1990-01-17 1990-01-17 Therapeutic agents
GB909008587A GB9008587D0 (en) 1990-04-17 1990-04-17 Therapeutic agents

Publications (1)

Publication Number Publication Date
IL96891A0 true IL96891A0 (en) 1992-03-29

Family

ID=26296509

Family Applications (1)

Application Number Title Priority Date Filing Date
IL96891A IL96891A0 (en) 1990-01-17 1991-01-07 Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them

Country Status (15)

Country Link
EP (1) EP0438230B1 (xx)
JP (1) JPH06100558A (xx)
KR (1) KR910014373A (xx)
CN (1) CN1053429A (xx)
AT (1) ATE152110T1 (xx)
AU (1) AU6944091A (xx)
CA (1) CA2034189A1 (xx)
CS (1) CS8691A2 (xx)
DE (1) DE69125731T2 (xx)
FI (1) FI910228A (xx)
HU (1) HU910128D0 (xx)
IE (1) IE910139A1 (xx)
IL (1) IL96891A0 (xx)
NO (1) NO910187L (xx)
PT (1) PT96477A (xx)

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US6380233B1 (en) 1992-04-07 2002-04-30 Pfizer Inc Indole derivatives as 5-HT1 agonists
RU2101283C1 (ru) 1992-04-07 1998-01-10 Пфайзер Инк. Производные индола или их фармацевтически приемлемые соли
ATE148465T1 (de) * 1992-04-10 1997-02-15 Pfizer Acylaminoindolderivate als 5-ht1 agonisten
GB9207930D0 (en) * 1992-04-10 1992-05-27 Pfizer Ltd Indoles
GB9208161D0 (en) * 1992-04-14 1992-05-27 Pfizer Ltd Indoles
GB9208463D0 (en) * 1992-04-16 1992-06-03 Merck Sharp & Dohme Therapeutic agents
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TW251284B (xx) * 1992-11-02 1995-07-11 Pfizer
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ES2070087B1 (es) * 1993-08-13 1996-02-16 Pfizer Derivados de indol
JP2860603B2 (ja) * 1993-08-31 1999-02-24 ファイザー・インク． ５−アリールインドール誘導体
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US4833153A (en) * 1985-11-08 1989-05-23 Glaxo Group Limited Indole derivatives
GB8724912D0 (en) * 1987-10-23 1987-11-25 Wellcome Found Indole derivatives
NZ227841A (en) * 1988-02-12 1991-08-27 Merck Sharp & Dohme Heterocyclic compounds with at least two non-condensed five membered rings and pharmaceutical compositions

Also Published As

Publication number Publication date
IE910139A1 (en) 1991-07-17
HU910128D0 (en) 1991-08-28
PT96477A (pt) 1991-10-15
CN1053429A (zh) 1991-07-31
ATE152110T1 (de) 1997-05-15
EP0438230A3 (en) 1992-02-12
DE69125731D1 (de) 1997-05-28
CA2034189A1 (en) 1991-07-18
FI910228A0 (fi) 1991-01-16
DE69125731T2 (de) 1997-11-27
NO910187L (no) 1991-07-18
KR910014373A (ko) 1991-08-31
EP0438230A2 (en) 1991-07-24
AU6944091A (en) 1991-07-25
EP0438230B1 (en) 1997-04-23
FI910228A (fi) 1991-07-18
CS8691A2 (en) 1991-09-15
JPH06100558A (ja) 1994-04-12
NO910187D0 (no) 1991-01-16

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