IL139865A0 - A liver selective glucocorticoid antagonist and pharmaceutical compositions containing the same - Google Patents
A liver selective glucocorticoid antagonist and pharmaceutical compositions containing the sameInfo
- Publication number
- IL139865A0 IL139865A0 IL13986599A IL13986599A IL139865A0 IL 139865 A0 IL139865 A0 IL 139865A0 IL 13986599 A IL13986599 A IL 13986599A IL 13986599 A IL13986599 A IL 13986599A IL 139865 A0 IL139865 A0 IL 139865A0
- Authority
- IL
- Israel
- Prior art keywords
- same
- pharmaceutical compositions
- compositions containing
- selective glucocorticoid
- glucocorticoid antagonist
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Diabetes (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9812314.4A GB9812314D0 (en) | 1998-06-08 | 1998-06-08 | Treatment of diabetes |
GBGB9815149.1A GB9815149D0 (en) | 1998-07-13 | 1998-07-13 | Treatment of diabetes |
PCT/IB1999/001175 WO1999063976A2 (en) | 1998-06-08 | 1999-06-07 | Liver-selective glucocorticoid antagonist for treating diabetes |
Publications (1)
Publication Number | Publication Date |
---|---|
IL139865A0 true IL139865A0 (en) | 2002-02-10 |
Family
ID=26313822
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL13986599A IL139865A0 (en) | 1998-06-08 | 1999-06-07 | A liver selective glucocorticoid antagonist and pharmaceutical compositions containing the same |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1143948A3 (de) |
JP (1) | JP2002527355A (de) |
KR (1) | KR20010052431A (de) |
AU (1) | AU751569B2 (de) |
CA (1) | CA2334116A1 (de) |
IL (1) | IL139865A0 (de) |
WO (1) | WO1999063976A2 (de) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9816935D0 (en) * | 1998-08-05 | 1998-09-30 | Karobio Ab | Novel glucocortoid and thyroid receptor ligands for the treatment of metabolic disorders |
GB9907048D0 (en) | 1999-03-27 | 1999-05-19 | Karobio Ab | Novel glucocorticoid receptor ligands for the treatment of meta bolic disorders |
GB9928805D0 (en) * | 1999-12-07 | 2000-02-02 | Karobio Ab | Compounds active at the Glucocorticoid and Thyroid Hormone Receptors |
ES2246292T3 (es) | 2000-10-30 | 2006-02-16 | Pfizer Products Inc. | Moduladores de receptor glucocorticoide. |
GB0029100D0 (en) * | 2000-11-29 | 2001-01-10 | Karobio Ab | Compounds active at the glucocorticoid receptor |
GB0029102D0 (en) | 2000-11-29 | 2001-01-10 | Karobio Ab | Compounds active at the glucocorticoid receptor |
JP2004519439A (ja) * | 2000-12-20 | 2004-07-02 | ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | グルココルチコイド関連副作用の治療用の解離したグルココルチコイドレセプターアンタゴニスト |
US6583180B2 (en) | 2001-02-14 | 2003-06-24 | Abbott Laboratories | Glucocorticoid receptor modulators |
ATE437853T1 (de) * | 2001-02-14 | 2009-08-15 | Karobio Ab | Glucocorticoid-rezeptoren-modulatoren |
EP1285927A3 (de) | 2001-08-16 | 2005-06-29 | Schering Aktiengesellschaft | Verwendung von Glucocorticoid-Rezeptorantagonisten zur Vorbeugung und Behandlung von Erkrankungen des männlichen Reproduktionssystems |
WO2003059253A2 (en) * | 2001-12-21 | 2003-07-24 | Smithkline Beecham Corporation | Compositions and methods for altering glucose production |
MXPA04009329A (es) | 2002-03-26 | 2005-01-25 | Boehringer Ingelheim Pharma | Mimeticos de glucocorticoides, metodos para su preparacion, composiciones farmaceuticas y usos de los mismos. |
US7186864B2 (en) | 2002-05-29 | 2007-03-06 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
US7074806B2 (en) | 2002-06-06 | 2006-07-11 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
US8097606B2 (en) | 2003-07-23 | 2012-01-17 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of catatonia |
US7527829B2 (en) | 2003-07-31 | 2009-05-05 | Soken Chemical & Engineering Co., Ltd. | Fluid colloid crystal and process for producing three-dimensional aligned particle mass therefrom |
UY28526A1 (es) | 2003-09-24 | 2005-04-29 | Boehringer Ingelheim Pharma | Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos |
US7795272B2 (en) | 2004-03-13 | 2010-09-14 | Boehringer Ingelheim Pharmaceutical, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof |
US7741361B2 (en) | 2004-12-27 | 2010-06-22 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
WO2008070507A2 (en) | 2006-12-06 | 2008-06-12 | Boehringer Ingelheim International Gmbh | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
AU2009256289A1 (en) | 2008-06-06 | 2009-12-10 | Boehringer Ingelheim International Gmbh | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
US8138189B2 (en) * | 2009-03-26 | 2012-03-20 | Hoffman-La Roche Inc. | Substituted benzene compounds as modulators of the glucocorticoid receptor |
EP2459524A2 (de) | 2009-07-31 | 2012-06-06 | Cadila Healthcare Limited | Neuartige verbindungen als glucocorticoidrezeptor-modulatoren |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4374148A (en) * | 1980-10-21 | 1983-02-15 | Pfizer Inc. | Carboxylic acid therapeutic agents |
WO1998027986A1 (en) * | 1996-12-24 | 1998-07-02 | Zymogenetics, Inc. | Treatment agents and methods for treating type ii diabetes and symptoms of type ii diabetes |
-
1999
- 1999-06-07 KR KR1020007013430A patent/KR20010052431A/ko not_active Application Discontinuation
- 1999-06-07 AU AU41606/99A patent/AU751569B2/en not_active Ceased
- 1999-06-07 JP JP2000553045A patent/JP2002527355A/ja active Pending
- 1999-06-07 WO PCT/IB1999/001175 patent/WO1999063976A2/en not_active Application Discontinuation
- 1999-06-07 EP EP99925232A patent/EP1143948A3/de not_active Withdrawn
- 1999-06-07 IL IL13986599A patent/IL139865A0/xx unknown
- 1999-06-07 CA CA002334116A patent/CA2334116A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AU4160699A (en) | 1999-12-30 |
KR20010052431A (ko) | 2001-06-25 |
AU751569B2 (en) | 2002-08-22 |
CA2334116A1 (en) | 1999-12-16 |
JP2002527355A (ja) | 2002-08-27 |
EP1143948A3 (de) | 2002-09-11 |
EP1143948A2 (de) | 2001-10-17 |
WO1999063976A3 (en) | 2001-12-20 |
WO1999063976A2 (en) | 1999-12-16 |
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