IL128902A - תולדות - n- (-2בנזותיאזוליל)--1 פיפרידינאתאנאמין, הכנתן ותכשירי רוקחות המכילים אותן - Google Patents

תולדות - n- (-2בנזותיאזוליל)--1 פיפרידינאתאנאמין, הכנתן ותכשירי רוקחות המכילים אותן

Info

Publication number
IL128902A
IL128902A IL12890297A IL12890297A IL128902A IL 128902 A IL128902 A IL 128902A IL 12890297 A IL12890297 A IL 12890297A IL 12890297 A IL12890297 A IL 12890297A IL 128902 A IL128902 A IL 128902A
Authority
IL
Israel
Prior art keywords
general formula
compound
methyl
mixture
benzothiazolyl
Prior art date
Application number
IL12890297A
Other languages
English (en)
Other versions
IL128902A0 (en
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of IL128902A0 publication Critical patent/IL128902A0/xx
Publication of IL128902A publication Critical patent/IL128902A/he

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
IL12890297A 1996-10-01 1997-09-26 תולדות - n- (-2בנזותיאזוליל)--1 פיפרידינאתאנאמין, הכנתן ותכשירי רוקחות המכילים אותן IL128902A (he)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (fr) 1996-10-01 1996-10-01 Derives de n-(benzothiazol-2-yl) piperidine-1-ethanamine, leur preparation et leur application en therapeutique
PCT/FR1997/001692 WO1998014444A1 (fr) 1996-10-01 1997-09-26 Derives de n-(benzothiazol-2-yl)piperidine-1-ethanamine, leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
IL128902A0 IL128902A0 (en) 2000-02-17
IL128902A true IL128902A (he) 2001-07-24

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12890297A IL128902A (he) 1996-10-01 1997-09-26 תולדות - n- (-2בנזותיאזוליל)--1 פיפרידינאתאנאמין, הכנתן ותכשירי רוקחות המכילים אותן

Country Status (23)

Country Link
EP (1) EP0929550A1 (he)
JP (1) JP2001501217A (he)
KR (1) KR20000048767A (he)
CN (1) CN1230959A (he)
AR (1) AR009105A1 (he)
AU (1) AU722147B2 (he)
BG (1) BG103271A (he)
BR (1) BR9711842A (he)
CA (1) CA2266510A1 (he)
CO (1) CO4650030A1 (he)
CZ (1) CZ112699A3 (he)
EE (1) EE9900135A (he)
FR (1) FR2753970B1 (he)
HU (1) HUP9904091A3 (he)
IL (1) IL128902A (he)
NO (1) NO991581L (he)
NZ (1) NZ334553A (he)
PL (1) PL332648A1 (he)
SK (1) SK42299A3 (he)
TR (1) TR199900634T2 (he)
TW (1) TW438800B (he)
WO (1) WO1998014444A1 (he)
ZA (1) ZA978772B (he)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
ATE385794T1 (de) 2000-06-21 2008-03-15 Hoffmann La Roche Benzothiazolderivate zur behandlung von alzheimer und parkinson
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
SG131946A1 (en) * 2003-10-24 2007-05-28 Hoffmann La Roche Ccr3 receptor antagonists
CA2567703C (en) 2004-05-24 2013-03-05 F. Hoffmann-La Roche Ag 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide
ES2309814T3 (es) 2004-11-05 2008-12-16 F. Hoffmann-La Roche Ag Proceso para la obtencion de derivados del acido isonicotinico.
SI1863818T1 (sl) 2005-03-23 2010-05-31 Hoffmann La Roche Derivati acetilenil pirazolo pirimidina kot antagonisti mglur
BRPI0616571A2 (pt) 2005-09-27 2011-06-21 Hoffmann La Roche oxadiazolil pirazol-piridiminas como antagonistas de mglur2, processo para sua preparação, composição farmacêutica que os contém e uso dos mesmo

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법

Also Published As

Publication number Publication date
NO991581L (no) 1999-06-01
AU722147B2 (en) 2000-07-20
FR2753970B1 (fr) 1998-10-30
AR009105A1 (es) 2000-03-08
HUP9904091A3 (en) 2000-07-28
JP2001501217A (ja) 2001-01-30
CA2266510A1 (en) 1998-04-09
NO991581D0 (no) 1999-03-30
BR9711842A (pt) 1999-08-24
CN1230959A (zh) 1999-10-06
TR199900634T2 (xx) 1999-06-21
WO1998014444A1 (fr) 1998-04-09
ZA978772B (en) 1998-03-27
EP0929550A1 (fr) 1999-07-21
BG103271A (en) 2000-05-31
HUP9904091A2 (hu) 2000-05-28
TW438800B (en) 2001-06-07
IL128902A0 (en) 2000-02-17
AU4463897A (en) 1998-04-24
NZ334553A (en) 2000-11-24
CO4650030A1 (es) 1998-09-03
CZ112699A3 (cs) 1999-06-16
EE9900135A (et) 1999-12-15
PL332648A1 (en) 1999-09-27
FR2753970A1 (fr) 1998-04-03
KR20000048767A (ko) 2000-07-25
SK42299A3 (en) 1999-12-10

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FF Patent granted
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