HUP0600239A3 - 5-amino-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine derivatives, process for their preparation, their use as adenosine a2a receptor antagonists and pharmaceutical compositions containing them - Google Patents

5-amino-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine derivatives, process for their preparation, their use as adenosine a2a receptor antagonists and pharmaceutical compositions containing them

Info

Publication number
HUP0600239A3
HUP0600239A3 HU0600239A HUP0600239A HUP0600239A3 HU P0600239 A3 HUP0600239 A3 HU P0600239A3 HU 0600239 A HU0600239 A HU 0600239A HU P0600239 A HUP0600239 A HU P0600239A HU P0600239 A3 HUP0600239 A3 HU P0600239A3
Authority
HU
Hungary
Prior art keywords
triazolo
pyrazolo
adenosine
amino
preparation
Prior art date
Application number
HU0600239A
Other languages
English (en)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of HUP0600239A2 publication Critical patent/HUP0600239A2/hu
Publication of HUP0600239A3 publication Critical patent/HUP0600239A3/hu
Publication of HU230420B1 publication Critical patent/HU230420B1/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HU0600239A 2000-05-26 2001-05-24 Adenozin A2a receptor anatgonisták HU230420B1 (hu)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US20714300P 2000-05-26 2000-05-26
US60/207,143 2000-05-26
PCT/US2001/016954 WO2001092264A1 (en) 2000-05-26 2001-05-24 Adenosine a2a receptor antagonists

Publications (3)

Publication Number Publication Date
HUP0600239A2 HUP0600239A2 (en) 2006-07-28
HUP0600239A3 true HUP0600239A3 (en) 2008-06-30
HU230420B1 HU230420B1 (hu) 2016-05-30

Family

ID=22769372

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0600239A HU230420B1 (hu) 2000-05-26 2001-05-24 Adenozin A2a receptor anatgonisták

Country Status (31)

Country Link
US (4) US6630475B2 (hu)
EP (1) EP1283839B1 (hu)
JP (3) JP4574112B2 (hu)
KR (1) KR100520907B1 (hu)
CN (2) CN100384847C (hu)
AR (1) AR028621A1 (hu)
AT (1) ATE293627T1 (hu)
AU (2) AU2001268089C1 (hu)
BR (1) BRPI0111015B8 (hu)
CA (1) CA2410237C (hu)
CZ (1) CZ303790B6 (hu)
DE (1) DE60110219T2 (hu)
DK (1) DK1283839T3 (hu)
EC (1) ECSP024364A (hu)
ES (1) ES2237576T3 (hu)
HK (1) HK1049007B (hu)
HU (1) HU230420B1 (hu)
IL (3) IL152726A0 (hu)
MX (1) MXPA02011625A (hu)
MY (1) MY132006A (hu)
NO (1) NO325008B1 (hu)
NZ (1) NZ522326A (hu)
PE (1) PE20020062A1 (hu)
PL (1) PL218764B1 (hu)
PT (1) PT1283839E (hu)
RU (1) RU2315053C2 (hu)
SI (1) SI1283839T1 (hu)
SK (1) SK287748B6 (hu)
TW (1) TWI288137B (hu)
WO (1) WO2001092264A1 (hu)
ZA (1) ZA200208898B (hu)

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Also Published As

Publication number Publication date
ES2237576T3 (es) 2005-08-01
CZ20023886A3 (cs) 2003-02-12
BRPI0111015B8 (pt) 2021-05-25
JP2006219497A (ja) 2006-08-24
US20020099061A1 (en) 2002-07-25
USRE44205E1 (en) 2013-05-07
RU2315053C2 (ru) 2008-01-20
PL360472A1 (en) 2004-09-06
ATE293627T1 (de) 2005-05-15
AU6808901A (en) 2001-12-11
HK1049007A1 (en) 2003-04-25
EP1283839B1 (en) 2005-04-20
AU2001268089B2 (en) 2005-04-28
NO325008B1 (no) 2008-01-14
HU230420B1 (hu) 2016-05-30
PE20020062A1 (es) 2002-02-02
DE60110219T2 (de) 2006-03-09
BR0111015A (pt) 2005-01-11
JP2007145875A (ja) 2007-06-14
MY132006A (en) 2007-09-28
HK1049007B (zh) 2005-09-16
IL220174A0 (en) 2012-07-31
IL152726A0 (en) 2003-06-24
SK16712002A3 (sk) 2003-08-05
NZ522326A (en) 2006-03-31
JP2003535094A (ja) 2003-11-25
US7067655B2 (en) 2006-06-27
CN1451007A (zh) 2003-10-22
SK287748B6 (sk) 2011-08-04
ZA200208898B (en) 2004-03-01
US20050026932A1 (en) 2005-02-03
AR028621A1 (es) 2003-05-14
BRPI0111015B1 (pt) 2017-11-07
DE60110219D1 (de) 2005-05-25
US6630475B2 (en) 2003-10-07
US20040023997A1 (en) 2004-02-05
NO20025651L (no) 2003-01-23
TWI288137B (en) 2007-10-11
SI1283839T1 (hu) 2005-08-31
PT1283839E (pt) 2005-08-31
CN100384847C (zh) 2008-04-30
KR100520907B1 (ko) 2005-10-11
JP4938348B2 (ja) 2012-05-23
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DK1283839T3 (da) 2005-07-25
ECSP024364A (es) 2003-03-31
PL218764B1 (pl) 2015-01-30
US6897216B2 (en) 2005-05-24
HUP0600239A2 (en) 2006-07-28
IL220174A (en) 2015-07-30
KR20030003746A (ko) 2003-01-10
EP1283839A1 (en) 2003-02-19
MXPA02011625A (es) 2003-03-27
IL152726A (en) 2012-07-31
AU2001268089C1 (en) 2006-04-13
CZ303790B6 (cs) 2013-05-09
WO2001092264A1 (en) 2001-12-06
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