HUP0102935A3 - N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres and pharmaceutical compositions containing them - Google Patents
N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres and pharmaceutical compositions containing themInfo
- Publication number
- HUP0102935A3 HUP0102935A3 HU0102935A HUP0102935A HUP0102935A3 HU P0102935 A3 HUP0102935 A3 HU P0102935A3 HU 0102935 A HU0102935 A HU 0102935A HU P0102935 A HUP0102935 A HU P0102935A HU P0102935 A3 HUP0102935 A3 HU P0102935A3
- Authority
- HU
- Hungary
- Prior art keywords
- pharmaceutical compositions
- compositions containing
- carboxylic acid
- carboxylic acids
- acid isosteres
- Prior art date
Links
- 150000001732 carboxylic acid derivatives Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 229940124530 sulfonamide Drugs 0.000 title 1
- 150000003456 sulfonamides Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4906—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom
- A61K8/4913—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q7/00—Preparations for affecting hair growth
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Birds (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8784298P | 1998-06-03 | 1998-06-03 | |
PCT/US1998/025572 WO1999062880A1 (en) | 1998-06-03 | 1998-12-03 | N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0102935A2 HUP0102935A2 (en) | 2001-12-28 |
HUP0102935A3 true HUP0102935A3 (en) | 2002-01-28 |
Family
ID=22207576
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0102935A HUP0102935A3 (en) | 1998-06-03 | 1998-12-03 | N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres and pharmaceutical compositions containing them |
Country Status (17)
Country | Link |
---|---|
US (3) | US7459473B2 (hu) |
EP (1) | EP1084106A1 (hu) |
JP (1) | JP2002516904A (hu) |
KR (1) | KR20010052503A (hu) |
CN (1) | CN1295561A (hu) |
AU (1) | AU1708099A (hu) |
BG (1) | BG105012A (hu) |
BR (1) | BR9815882A (hu) |
CA (1) | CA2334002A1 (hu) |
EA (1) | EA200001247A1 (hu) |
HU (1) | HUP0102935A3 (hu) |
IL (1) | IL140040A0 (hu) |
NO (1) | NO20006078L (hu) |
PL (1) | PL348661A1 (hu) |
SK (1) | SK18302000A3 (hu) |
WO (1) | WO1999062880A1 (hu) |
ZA (1) | ZA9811060B (hu) |
Families Citing this family (26)
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ATE330950T1 (de) | 2000-12-13 | 2006-07-15 | Wyeth Corp | Heterocyclische sulfonamide als inhibitoren der beta-amyloid-produktion |
SE0100902D0 (sv) * | 2001-03-15 | 2001-03-15 | Astrazeneca Ab | Compounds |
CN1173960C (zh) * | 2001-12-06 | 2004-11-03 | 中国人民解放军军事医学科学院毒物药物研究所 | 取代六元氮杂环类化合物及其作为神经调节剂的用途 |
CA2364985A1 (en) * | 2001-12-14 | 2003-06-14 | John W. Gillard | Imidazo(2,1-b)thiadiazole sulfonamides |
GB0209995D0 (en) * | 2002-05-01 | 2002-06-12 | Merck Sharp & Dohme | Therapeutic agents |
SE0202539D0 (sv) | 2002-08-27 | 2002-08-27 | Astrazeneca Ab | Compounds |
US7648992B2 (en) | 2004-07-05 | 2010-01-19 | Astrazeneca Ab | Hydantoin derivatives for the treatment of obstructive airway diseases |
SE0401763D0 (sv) * | 2004-07-05 | 2004-07-05 | Astrazeneca Ab | Compounds |
SE0401762D0 (sv) | 2004-07-05 | 2004-07-05 | Astrazeneca Ab | Novel compounds |
SE0403086D0 (sv) | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Compounds |
SE0403085D0 (sv) | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Novel componds |
CN101277949A (zh) | 2005-04-22 | 2008-10-01 | 阿兰托斯制药控股公司 | 二肽基肽酶-ⅳ抑制剂 |
DE102005050377A1 (de) * | 2005-10-21 | 2007-04-26 | Bayer Healthcare Ag | Heterocyclische Verbindungen und ihre Verwendung |
TW200831488A (en) * | 2006-11-29 | 2008-08-01 | Astrazeneca Ab | Novel compounds |
US8791128B2 (en) * | 2008-09-16 | 2014-07-29 | University Of Central Florida Research Foundation, Inc. | Compositions for treating or delaying the onset of hair loss |
JP2012041325A (ja) * | 2010-08-23 | 2012-03-01 | Bayer Cropscience Ag | オキサジアゾリノン誘導体およびその有害生物の防除用途 |
TWI534142B (zh) | 2011-03-15 | 2016-05-21 | 大正製藥股份有限公司 | Azole derivatives |
WO2013134562A1 (en) | 2012-03-09 | 2013-09-12 | Inception 2, Inc. | Triazolone compounds and uses thereof |
EP2935228B9 (en) | 2012-12-20 | 2017-12-06 | Inception 2, Inc. | Triazolone compounds and uses thereof |
CA2921420A1 (en) | 2013-09-06 | 2015-03-12 | Inception 2, Inc. | Triazolone compounds and uses thereof |
WO2015112902A2 (en) * | 2014-01-23 | 2015-07-30 | Sova Pharmaceuticals, Inc. | CYSTATHIONINE-(gamma)-LYASE (CSE) INHIBITORS FOR TREATING PAIN |
JP6541118B1 (ja) * | 2018-04-27 | 2019-07-10 | 株式会社成和化成 | 化粧品基材および該化粧品基材を含有する毛髪用化粧品、美白剤 |
WO2022270628A1 (ja) * | 2021-06-25 | 2022-12-29 | 国立大学法人 大分大学 | Rsウイルス感染症の処置および/または予防用医薬としてのヘテロシクロアルキル置換ポリヘテロアゾール誘導体 |
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-
1998
- 1998-12-03 AU AU17080/99A patent/AU1708099A/en not_active Abandoned
- 1998-12-03 IL IL14004098A patent/IL140040A0/xx unknown
- 1998-12-03 US US09/204,236 patent/US7459473B2/en not_active Expired - Fee Related
- 1998-12-03 SK SK1830-2000A patent/SK18302000A3/sk unknown
- 1998-12-03 PL PL98348661A patent/PL348661A1/xx unknown
- 1998-12-03 HU HU0102935A patent/HUP0102935A3/hu unknown
- 1998-12-03 EA EA200001247A patent/EA200001247A1/ru unknown
- 1998-12-03 JP JP2000552092A patent/JP2002516904A/ja active Pending
- 1998-12-03 BR BR9815882-1A patent/BR9815882A/pt not_active Application Discontinuation
- 1998-12-03 KR KR1020007013637A patent/KR20010052503A/ko not_active Application Discontinuation
- 1998-12-03 EP EP98961865A patent/EP1084106A1/en not_active Withdrawn
- 1998-12-03 CN CN98814096A patent/CN1295561A/zh active Pending
- 1998-12-03 ZA ZA9811060A patent/ZA9811060B/xx unknown
- 1998-12-03 WO PCT/US1998/025572 patent/WO1999062880A1/en not_active Application Discontinuation
- 1998-12-03 CA CA002334002A patent/CA2334002A1/en not_active Abandoned
-
2000
- 2000-11-30 NO NO20006078A patent/NO20006078L/no not_active Application Discontinuation
- 2000-12-01 BG BG105012A patent/BG105012A/xx unknown
-
2001
- 2001-02-26 US US09/791,660 patent/US20020052514A1/en not_active Abandoned
-
2003
- 2003-06-24 US US10/601,607 patent/US7078424B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
IL140040A0 (en) | 2002-02-10 |
PL348661A1 (en) | 2002-06-03 |
NO20006078L (no) | 2001-02-05 |
AU1708099A (en) | 1999-12-20 |
KR20010052503A (ko) | 2001-06-25 |
JP2002516904A (ja) | 2002-06-11 |
WO1999062880A1 (en) | 1999-12-09 |
US20020052514A1 (en) | 2002-05-02 |
EP1084106A1 (en) | 2001-03-21 |
BR9815882A (pt) | 2002-09-17 |
HUP0102935A2 (en) | 2001-12-28 |
US7078424B2 (en) | 2006-07-18 |
SK18302000A3 (sk) | 2001-06-11 |
BG105012A (en) | 2001-08-31 |
CA2334002A1 (en) | 1999-12-09 |
CN1295561A (zh) | 2001-05-16 |
ZA9811060B (en) | 1999-12-03 |
US20040082622A1 (en) | 2004-04-29 |
EA200001247A1 (ru) | 2001-08-27 |
NO20006078D0 (no) | 2000-11-30 |
US20020052510A1 (en) | 2002-05-02 |
US7459473B2 (en) | 2008-12-02 |
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