HUP0003978A3 - Guanidinylation reagents - Google Patents

Guanidinylation reagents

Info

Publication number
HUP0003978A3
HUP0003978A3 HU0003978A HUP0003978A HUP0003978A3 HU P0003978 A3 HUP0003978 A3 HU P0003978A3 HU 0003978 A HU0003978 A HU 0003978A HU P0003978 A HUP0003978 A HU P0003978A HU P0003978 A3 HUP0003978 A3 HU P0003978A3
Authority
HU
Hungary
Prior art keywords
guanidinylation reagents
guanidinylation
reagents
Prior art date
Application number
HU0003978A
Other languages
English (en)
Original Assignee
Univ California
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ California filed Critical Univ California
Publication of HUP0003978A2 publication Critical patent/HUP0003978A2/hu
Publication of HUP0003978A3 publication Critical patent/HUP0003978A3/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24Y being a hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/04Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
    • C07C279/14Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/50Compounds containing any of the groups, X being a hetero atom, Y being any atom
    • C07C311/52Y being a hetero atom
    • C07C311/64X and Y being nitrogen atoms, e.g. N-sulfonylguanidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/006General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length of peptides containing derivatised side chain amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C07K1/064General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for omega-amino or -guanidino functions
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Analytical Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
HU0003978A 1997-05-22 1998-05-21 Guanidinylation reagents HUP0003978A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/861,942 US6072075A (en) 1997-05-22 1997-05-22 Guanidinylation reagents
PCT/US1998/010669 WO1998052917A2 (en) 1997-05-22 1998-05-21 Guanidinylation reagents

Publications (2)

Publication Number Publication Date
HUP0003978A2 HUP0003978A2 (en) 2001-03-28
HUP0003978A3 true HUP0003978A3 (en) 2002-03-28

Family

ID=25337171

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0003978A HUP0003978A3 (en) 1997-05-22 1998-05-21 Guanidinylation reagents

Country Status (15)

Country Link
US (3) US6072075A (hu)
EP (1) EP0983232B1 (hu)
JP (1) JP2002502378A (hu)
KR (1) KR20010012732A (hu)
AT (1) ATE227705T1 (hu)
AU (1) AU736072B2 (hu)
BR (1) BR9809859A (hu)
CA (1) CA2288196A1 (hu)
DE (1) DE69809412D1 (hu)
HU (1) HUP0003978A3 (hu)
IL (1) IL132773A0 (hu)
NO (1) NO995693L (hu)
PL (1) PL336996A1 (hu)
SK (1) SK157099A3 (hu)
WO (1) WO1998052917A2 (hu)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6525182B1 (en) * 2000-01-21 2003-02-25 Regents Of The University Of California Guanidinylation, guanidinoglycosides, uses, and methods of assaying their activity
FR2822463B1 (fr) 2001-03-21 2004-07-30 Lipha Derives bicycliques de guanidines et leurs applications en therapeutique
US20060264608A1 (en) * 2001-08-03 2006-11-23 Wender Paul A Bi-directional synthesis of oligoguanidine transport agents
CA2455951A1 (en) * 2001-08-03 2003-02-20 The Board Of Trustees Of The Leland Stanford Junior University Bi-directional synthesis of oligoguanidine transport agents
PL195917B1 (pl) * 2001-10-31 2007-11-30 Inst Farmaceutyczny Nowe peptydy - analogi ludzkiego hormonu uwalniającego hormon wzrostu
US7022214B2 (en) * 2004-01-21 2006-04-04 Bio-Rad Laboratories, Inc. Carrier ampholytes of high pH range
JP4777225B2 (ja) * 2006-12-04 2011-09-21 キヤノン株式会社 吐出用液体及び吐出方法
US9248089B2 (en) 2011-11-07 2016-02-02 Grf (Wuhan) Biotechnology Inc. Peptide-based compounds as inhibitors of neurotransmitter secretion
CN106132926B (zh) * 2014-03-28 2019-05-21 株式会社钟化 三苄氧羰基精氨酸的制造方法
CN107236056A (zh) * 2017-07-27 2017-10-10 山东百玛海洋生物科技有限公司 胍基化壳聚糖衍生物、纳米粒及其制备方法
CN107266610A (zh) * 2017-07-27 2017-10-20 山东百玛海洋生物科技有限公司 胍基化壳聚糖衍生物以及纳米粒的应用
US20200323962A1 (en) * 2017-09-19 2020-10-15 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Lipophilic peptide prodrugs
CN114907241B (zh) * 2021-02-09 2024-05-17 中宏鑫投资控股(深圳)有限公司 一种含氟磺酰基的胍类化合物及其制备方法和应用

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US1677235A (en) * 1928-07-17 Balph v
US1681806A (en) * 1928-08-21 Ments
US1953494A (en) * 1926-08-26 1934-04-03 Ig Farbenindustrie Ag Process of preparing substituted guanidines
US1795738A (en) * 1927-09-12 1931-03-10 Scheringkahlbaum A G Method of producing substituted guanidines
US2898369A (en) * 1956-02-23 1959-08-04 Mcneilab Inc N,n,n',n'' tetraethyl guanidine and its acid addition salts
US3062805A (en) * 1957-03-08 1962-11-06 Sterling Drug Inc Peptide synthesis and intermediates therefor
US3062804A (en) * 1957-03-08 1962-11-06 Sterling Drug Inc Peptide synthesis and intermediates therefor
US3117994A (en) * 1959-12-03 1964-01-14 Monsanto Canada Ltd Nu, nu', nu'-trisubstituted guanidines
US3301755A (en) * 1962-04-18 1967-01-31 Ciba Geigy Corp Allylic guanidines
US3479437A (en) * 1963-08-26 1969-11-18 Stauffer Chemical Co Guanidine complexes as fungicides
US3320229A (en) * 1963-08-26 1967-05-16 Stauffer Chemical Co Complexes of guanidines with completely halogenated acetones
CH426863A (de) * 1963-08-30 1966-12-31 Sandoz Ag Verfahren zur Herstellung von Arginin enthaltenden Polypeptiden
US3609164A (en) * 1968-03-27 1971-09-28 Tanabe Seiyaku Co Process for preparing {11 -butoxycarbonyl compounds
US3551490A (en) * 1968-05-21 1970-12-29 American Cyanamid Co Method for preparing tetramethyl-guanidine
US3646029A (en) * 1968-09-25 1972-02-29 Monsanto Co Piperazino methyl 1 3 diarylguandines
IL38933A0 (en) * 1971-03-17 1972-05-30 Ciba Geigy Ag New carbamates,their manufacture and their use in plant protection
DE2315271C3 (de) * 1973-03-27 1975-09-11 Max-Planck-Gesellschaft Zur Foerderung Der Wissenschaften E.V., 3400 Goettingen L- Norleucin-13-Motilin, Verfahren zu dessen Herstellung und dasselbe enthaltendes Mittel
US4014915A (en) * 1975-04-22 1977-03-29 Fujisawa Pharmaceutical Co., Ltd. Oxime carbonates
DE2544348C3 (de) * 1975-10-03 1979-12-13 Max-Planck-Gesellschaft Zur Foerderung Der Wissenschaften E.V., 3400 Goettingen L-Leucin-13-Motilin, Verfahren zu dessen Herstellung und dasselbe enthaltendes Mittel
US4358613A (en) * 1979-12-26 1982-11-09 General Electric Company Process for the preparation of substituted guanidines
FR2509724B1 (fr) * 1981-07-15 1985-10-25 Centre Nat Rech Scient Nouvelles guanidines a fort encombrement sterique et procedes pour leur preparation
US4956388A (en) * 1986-12-22 1990-09-11 Eli Lilly And Company 3-aryloxy-3-substituted propanamines
JPH0692357B2 (ja) * 1989-10-18 1994-11-16 キヤノン株式会社 グアニジン化合物およびグアニジン化合物を含有する静電荷像現像用トナー
US5262568A (en) * 1990-03-02 1993-11-16 State Of Oregon Tri- and tetra-substituted guanidines and their use as excitatory amino acid antagonists
EP0646573A1 (en) * 1993-09-30 1995-04-05 Hoechst Aktiengesellschaft Preparation of protected and unprotected guanidino-substituted carboxylic acids

Also Published As

Publication number Publication date
JP2002502378A (ja) 2002-01-22
BR9809859A (pt) 2000-12-19
AU7798498A (en) 1998-12-11
IL132773A0 (en) 2001-03-19
WO1998052917A2 (en) 1998-11-26
US6072075A (en) 2000-06-06
NO995693L (no) 2000-01-18
NO995693D0 (no) 1999-11-19
PL336996A1 (en) 2000-07-31
CA2288196A1 (en) 1998-11-26
EP0983232B1 (en) 2002-11-13
SK157099A3 (en) 2000-06-12
WO1998052917A3 (en) 1999-04-22
ATE227705T1 (de) 2002-11-15
US6380358B1 (en) 2002-04-30
US20030055214A1 (en) 2003-03-20
AU736072B2 (en) 2001-07-26
EP0983232A2 (en) 2000-03-08
DE69809412D1 (de) 2002-12-19
HUP0003978A2 (en) 2001-03-28
KR20010012732A (ko) 2001-02-26

Similar Documents

Publication Publication Date Title
GB9703094D0 (en) Assay device
IL133233A0 (en) Position determination
GB9808145D0 (en) Assay
GB9815224D0 (en) Assay
HUP0003978A3 (en) Guanidinylation reagents
GB2366463B (en) Position determination
GB9715522D0 (en) Assays
GB9707743D0 (en) Analysis
GB9721240D0 (en) Assay
GB9410044D0 (en) Assay
GB9803156D0 (en) Assay
GB9727277D0 (en) Assay
GB9701050D0 (en) Structural member
PL340723A1 (en) Structural member
GB9408607D0 (en) Assay
GB9719428D0 (en) Assay
IL136525A0 (en) Agents
GR3036946T3 (en) Immunoassay
GB9420218D0 (en) Combined assay
GB9719809D0 (en) Assay
GB9716453D0 (en) Assay
GB9707040D0 (en) Assay
GB9714874D0 (en) Assay
GB9726747D0 (en) Assay
GB9725231D0 (en) Assay