HRP20170179T1 - Oblici 4-amino-2-(2,6-dioksopiperidin-3-il)izoindolin-1,3-diona - Google Patents

Oblici 4-amino-2-(2,6-dioksopiperidin-3-il)izoindolin-1,3-diona

Info

Publication number
HRP20170179T1
HRP20170179T1 HRP20170179TT HRP20170179T HRP20170179T1 HR P20170179 T1 HRP20170179 T1 HR P20170179T1 HR P20170179T T HRP20170179T T HR P20170179TT HR P20170179 T HRP20170179 T HR P20170179T HR P20170179 T1 HRP20170179 T1 HR P20170179T1
Authority
HR
Croatia
Prior art keywords
dioxopiperidine
isoindoline
dione
formulations
amino
Prior art date
Application number
HRP20170179TT
Other languages
English (en)
Inventor
Anthony Tutino
Michael T. Kelly
Original Assignee
Celgene Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42635489&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20170179(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Celgene Corporation filed Critical Celgene Corporation
Publication of HRP20170179T1 publication Critical patent/HRP20170179T1/hr

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • A—HUMAN NECESSITIES
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P33/00—Antiparasitic agents
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    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Neurology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Hematology (AREA)
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  • Tropical Medicine & Parasitology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
HRP20170179TT 2009-05-19 2017-02-02 Oblici 4-amino-2-(2,6-dioksopiperidin-3-il)izoindolin-1,3-diona HRP20170179T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17967809P 2009-05-19 2009-05-19
PCT/US2010/035357 WO2010135396A2 (en) 2009-05-19 2010-05-19 Formulations of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione
EP10720107.1A EP2391355B1 (en) 2009-05-19 2010-05-19 Formulations of 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione

Publications (1)

Publication Number Publication Date
HRP20170179T1 true HRP20170179T1 (hr) 2017-04-07

Family

ID=42635489

Family Applications (2)

Application Number Title Priority Date Filing Date
HRP20170179TT HRP20170179T1 (hr) 2009-05-19 2017-02-02 Oblici 4-amino-2-(2,6-dioksopiperidin-3-il)izoindolin-1,3-diona
HRP20191094TT HRP20191094T1 (hr) 2009-05-19 2019-06-17 Formulacije 4-amino-2-(2,6-dioksopiperidin-3-il)izoindolin-1,3-diona

Family Applications After (1)

Application Number Title Priority Date Filing Date
HRP20191094TT HRP20191094T1 (hr) 2009-05-19 2019-06-17 Formulacije 4-amino-2-(2,6-dioksopiperidin-3-il)izoindolin-1,3-diona

Country Status (34)

Country Link
US (6) US8828427B2 (hr)
EP (3) EP3199149A1 (hr)
JP (1) JP5752677B2 (hr)
KR (1) KR101381060B1 (hr)
CN (3) CN102333525A (hr)
AU (1) AU2010249615B2 (hr)
BR (1) BRPI1007855B1 (hr)
CA (1) CA2752550C (hr)
CL (1) CL2011001969A1 (hr)
CO (1) CO6430422A2 (hr)
CR (1) CR20110435A (hr)
CY (2) CY1118632T1 (hr)
DK (2) DK2391355T3 (hr)
EC (1) ECSP11011317A (hr)
ES (2) ES2615511T3 (hr)
HR (2) HRP20170179T1 (hr)
HU (2) HUE033115T2 (hr)
IL (2) IL214644A (hr)
LT (2) LT3351240T (hr)
MX (2) MX2011008554A (hr)
NI (1) NI201100158A (hr)
NZ (1) NZ594557A (hr)
PE (1) PE20120654A1 (hr)
PH (1) PH12015501523A1 (hr)
PL (2) PL2391355T3 (hr)
PT (2) PT3351240T (hr)
RU (1) RU2479307C1 (hr)
SG (1) SG174137A1 (hr)
SI (2) SI3351240T1 (hr)
SM (1) SMT201700097B (hr)
TR (1) TR201905423T4 (hr)
UA (1) UA102582C2 (hr)
WO (1) WO2010135396A2 (hr)
ZA (1) ZA201105962B (hr)

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US8404716B2 (en) 2002-10-15 2013-03-26 Celgene Corporation Methods of treating myelodysplastic syndromes with a combination therapy using lenalidomide and azacitidine
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