HRP20050432A2 - Novel medicaments for the treatment of chronic obstructive pulmonary diseases - Google Patents
Novel medicaments for the treatment of chronic obstructive pulmonary diseasesInfo
- Publication number
- HRP20050432A2 HRP20050432A2 HR20050432A HRP20050432A HRP20050432A2 HR P20050432 A2 HRP20050432 A2 HR P20050432A2 HR 20050432 A HR20050432 A HR 20050432A HR P20050432 A HRP20050432 A HR P20050432A HR P20050432 A2 HRP20050432 A2 HR P20050432A2
- Authority
- HR
- Croatia
- Prior art keywords
- treatment
- chronic obstructive
- obstructive pulmonary
- pulmonary diseases
- novel medicaments
- Prior art date
Links
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 title abstract 3
- 239000003814 drug Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
Abstract
Predloženi izum odnosi se na upotrebu spojeva opće formule 1,u kojoj radikali R1, R2 i R3 mogu imati značenja navedena u patentnim zahtjevima i u opisu, za proizvodnju lijeka za liječenje COPD-a (kronična opstrukcijska bolest pluća, e. chronic obstructive pulmonarv disease), kao i na nove spojeve opće formule 1 kao takove.The present invention relates to the use of compounds of general formula 1, in which the radicals R1, R2 and R3 may have the meanings given in the claims and in the description, for the manufacture of a medicament for the treatment of COPD (chronic obstructive pulmonary disease). , as well as to novel compounds of general formula 1 as such.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10253282A DE10253282A1 (en) | 2002-11-15 | 2002-11-15 | Treatment of chronic obstructive pulmonary disease, using new or known N-substituted 2-amino-1-(benz-(1,4)-oxazin-3-on-8-yl)-ethanol derivative beta-mimetic agents, suitable for once-daily administration |
PCT/EP2003/012565 WO2004045618A2 (en) | 2002-11-15 | 2003-11-11 | Novel medicaments for the treatment of chronic obstructive pulmonary diseases |
Publications (2)
Publication Number | Publication Date |
---|---|
HRP20050432A2 true HRP20050432A2 (en) | 2006-06-30 |
HRP20050432B1 HRP20050432B1 (en) | 2012-01-31 |
Family
ID=32185709
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20050432A HRP20050432B1 (en) | 2002-11-15 | 2005-05-13 | Novel medicaments for the treatment of chronic obstructive pulmonary diseases |
Country Status (38)
Country | Link |
---|---|
EP (2) | EP1562603B3 (en) |
JP (1) | JP4317138B2 (en) |
KR (1) | KR101092247B1 (en) |
CN (3) | CN101735166A (en) |
AR (2) | AR041969A1 (en) |
AT (1) | ATE430569T1 (en) |
AU (1) | AU2003285326B2 (en) |
BE (1) | BE2014C016I2 (en) |
BR (1) | BRPI0316264B8 (en) |
CA (1) | CA2506082C (en) |
CO (1) | CO5570670A2 (en) |
CY (2) | CY1110500T1 (en) |
DE (2) | DE10253282A1 (en) |
DK (1) | DK1562603T3 (en) |
EA (1) | EA008665B1 (en) |
EC (1) | ECSP055774A (en) |
ES (1) | ES2326878T7 (en) |
FR (1) | FR14C0049I2 (en) |
HR (1) | HRP20050432B1 (en) |
HU (1) | HUS1400011I1 (en) |
IL (1) | IL167900A (en) |
LT (1) | LTC1562603I2 (en) |
LU (1) | LU92433I2 (en) |
ME (1) | ME00354B (en) |
MX (1) | MXPA05005081A (en) |
MY (1) | MY136034A (en) |
NL (1) | NL300650I2 (en) |
NO (2) | NO334314B1 (en) |
NZ (1) | NZ540661A (en) |
PE (1) | PE20040694A1 (en) |
PL (1) | PL212238B1 (en) |
PT (1) | PT1562603E (en) |
RS (1) | RS51607B (en) |
SI (1) | SI1562603T1 (en) |
TW (1) | TWI343812B (en) |
UA (1) | UA81276C2 (en) |
WO (1) | WO2004045618A2 (en) |
ZA (1) | ZA200502246B (en) |
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Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3134590A1 (en) * | 1981-09-01 | 1983-03-10 | Boehringer Ingelheim KG, 6507 Ingelheim | NEW BENZO HETEROCYCLES |
US4460581A (en) | 1982-10-12 | 1984-07-17 | Boehringer Ingelheim Kg | (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones |
DE3743265A1 (en) * | 1987-12-19 | 1989-06-29 | Boehringer Ingelheim Kg | NEW AMMONIUM COMPOUNDS, THEIR MANUFACTURE AND USE |
BR0110331A (en) * | 2000-04-27 | 2003-01-07 | Boehringer Ingelheim Pharma | Beta-mimicking substances that have long-lasting activity, processes for preparing them and their use as medicines |
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2002
- 2002-11-15 DE DE10253282A patent/DE10253282A1/en not_active Withdrawn
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2003
- 2003-11-11 JP JP2004552561A patent/JP4317138B2/en not_active Expired - Lifetime
- 2003-11-11 EP EP03778312.3A patent/EP1562603B3/en not_active Expired - Lifetime
- 2003-11-11 PT PT03778312T patent/PT1562603E/en unknown
- 2003-11-11 BR BRPI0316264A patent/BRPI0316264B8/en active IP Right Grant
- 2003-11-11 AU AU2003285326A patent/AU2003285326B2/en active Active
- 2003-11-11 ME MEP-2008-536A patent/ME00354B/en unknown
- 2003-11-11 ES ES03778312.3T patent/ES2326878T7/en active Active
- 2003-11-11 DK DK03778312T patent/DK1562603T3/en active
- 2003-11-11 CN CN200910266327A patent/CN101735166A/en active Pending
- 2003-11-11 NZ NZ540661A patent/NZ540661A/en not_active IP Right Cessation
- 2003-11-11 KR KR1020057008679A patent/KR101092247B1/en active IP Right Grant
- 2003-11-11 AT AT03778312T patent/ATE430569T1/en active
- 2003-11-11 SI SI200331634T patent/SI1562603T1/en unknown
- 2003-11-11 DE DE50311502T patent/DE50311502D1/en not_active Expired - Lifetime
- 2003-11-11 EA EA200500715A patent/EA008665B1/en active Protection Beyond IP Right Term
- 2003-11-11 PL PL375270A patent/PL212238B1/en unknown
- 2003-11-11 EP EP08169872A patent/EP2025338A1/en not_active Withdrawn
- 2003-11-11 CN CNA2003801030945A patent/CN1713914A/en active Pending
- 2003-11-11 CA CA2506082A patent/CA2506082C/en not_active Expired - Lifetime
- 2003-11-11 UA UAA200505926A patent/UA81276C2/en unknown
- 2003-11-11 CN CN201010004697A patent/CN101817800A/en active Pending
- 2003-11-11 MX MXPA05005081A patent/MXPA05005081A/en active IP Right Grant
- 2003-11-11 WO PCT/EP2003/012565 patent/WO2004045618A2/en active Application Filing
- 2003-11-11 RS YU20050361A patent/RS51607B/en unknown
- 2003-11-13 MY MYPI20034360A patent/MY136034A/en unknown
- 2003-11-13 PE PE2003001147A patent/PE20040694A1/en active IP Right Grant
- 2003-11-14 TW TW092132031A patent/TWI343812B/en active
- 2003-11-14 AR ARP030104201A patent/AR041969A1/en active Pending
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2005
- 2005-03-17 ZA ZA2005/02246A patent/ZA200502246B/en unknown
- 2005-04-07 IL IL167900A patent/IL167900A/en active Protection Beyond IP Right Term
- 2005-05-02 EC EC2005005774A patent/ECSP055774A/en unknown
- 2005-05-13 HR HR20050432A patent/HRP20050432B1/en not_active IP Right Cessation
- 2005-06-14 CO CO05057641A patent/CO5570670A2/en not_active Application Discontinuation
- 2005-06-14 NO NO20052883A patent/NO334314B1/en not_active IP Right Cessation
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2009
- 2009-08-04 CY CY20091100826T patent/CY1110500T1/en unknown
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2012
- 2012-07-19 AR ARP120102613A patent/AR087241A2/en active Pending
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2014
- 2014-02-27 BE BE2014C016C patent/BE2014C016I2/fr unknown
- 2014-03-06 LT LTPA2014012C patent/LTC1562603I2/en unknown
- 2014-03-07 NL NL300650C patent/NL300650I2/en unknown
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