HK1214475A1 - 經取代的 -氟- -亞胺基- -甲基- -側氧基- -二氫嘧啶- -甲酸酯衍生物 - Google Patents

經取代的 -氟- -亞胺基- -甲基- -側氧基- -二氫嘧啶- -甲酸酯衍生物

Info

Publication number
HK1214475A1
HK1214475A1 HK16102490.3A HK16102490A HK1214475A1 HK 1214475 A1 HK1214475 A1 HK 1214475A1 HK 16102490 A HK16102490 A HK 16102490A HK 1214475 A1 HK1214475 A1 HK 1214475A1
Authority
HK
Hong Kong
Prior art keywords
dihydropyrimidine
imino
oxo
fluoro
substituted
Prior art date
Application number
HK16102490.3A
Other languages
English (en)
Inventor
Beth Lorsbach
W John Owen
Chenglin Yao
Lindsay Stelzer
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of HK1214475A1 publication Critical patent/HK1214475A1/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22O-Aryl or S-Aryl esters thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
HK16102490.3A 2012-12-28 2016-03-04 經取代的 -氟- -亞胺基- -甲基- -側氧基- -二氫嘧啶- -甲酸酯衍生物 HK1214475A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261747086P 2012-12-28 2012-12-28
PCT/US2013/077540 WO2014105844A1 (en) 2012-12-28 2013-12-23 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives

Publications (1)

Publication Number Publication Date
HK1214475A1 true HK1214475A1 (zh) 2016-07-29

Family

ID=51022033

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16102490.3A HK1214475A1 (zh) 2012-12-28 2016-03-04 經取代的 -氟- -亞胺基- -甲基- -側氧基- -二氫嘧啶- -甲酸酯衍生物

Country Status (19)

Country Link
US (2) US9622474B2 (zh)
EP (1) EP2938194B1 (zh)
JP (1) JP6324994B2 (zh)
KR (1) KR20150103096A (zh)
CN (2) CN110003118A (zh)
AU (1) AU2013370493B2 (zh)
BR (1) BR102013033709B1 (zh)
CA (1) CA2893778A1 (zh)
CR (1) CR20150382A (zh)
DK (1) DK2938194T3 (zh)
EC (1) ECSP15032859A (zh)
HK (1) HK1214475A1 (zh)
HU (1) HUE047711T2 (zh)
IL (1) IL239561B (zh)
MX (1) MX2015008441A (zh)
PL (1) PL2938194T3 (zh)
RU (1) RU2638556C2 (zh)
UA (1) UA115462C2 (zh)
WO (1) WO2014105844A1 (zh)

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CN110003118A (zh) 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 制备羧酸酯衍生物的方法
EP3689142A1 (en) * 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
EP2945634A4 (en) 2012-12-28 2016-05-25 Dow Agrosciences Llc N- (SUBSTITUTED) -5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDIN-1 (2H) -CARBOXAMIDE DERIVATIVES
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WO2016109288A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Use of picolinamide compounds with fungicidal activity
CA2972034A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamides with fungicidal activity
BR112017013608B8 (pt) 2014-12-30 2022-08-23 Dow Agrosciences Llc Picolinamidas como fungicidas
CA2972403A1 (en) 2014-12-30 2016-07-07 Dow Agrosciences Llc Picolinamide compounds with fungicidal activity
BR122019026066B1 (pt) 2014-12-30 2022-01-18 Dow Agrosciences Llc Compostos de picolinamida

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EP3689142A1 (en) 2012-12-28 2020-08-05 Adama Makhteshim Ltd. 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
EP2945634A4 (en) 2012-12-28 2016-05-25 Dow Agrosciences Llc N- (SUBSTITUTED) -5-FLUORO-4-IMINO-3-METHYL-2-OXO-3,4-DIHYDROPYRIMIDIN-1 (2H) -CARBOXAMIDE DERIVATIVES
PL2953463T3 (pl) 2012-12-31 2022-01-03 Adama Makhteshim Ltd. Pochodne 3-alkilo-5-fluoro-4-podstawione-imino-3,4-dihydropirymidyn-2(1h)-onu jako środki grzybobójcze
AU2014373850A1 (en) 2013-12-31 2016-08-11 Adama Makhteshim Ltd. Synergistic fungicidal mixtures and compositions for fungal control
PE20161174A1 (es) 2013-12-31 2016-10-26 Adama Makhteshim Ltd 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparacion
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Also Published As

Publication number Publication date
UA115462C2 (uk) 2017-11-10
EP2938194A4 (en) 2016-08-31
PL2938194T3 (pl) 2020-09-21
EP2938194B1 (en) 2019-11-27
KR20150103096A (ko) 2015-09-09
MX2015008441A (es) 2015-09-23
EP2938194A1 (en) 2015-11-04
IL239561B (en) 2018-01-31
AU2013370493A1 (en) 2015-07-02
ECSP15032859A (es) 2015-11-30
WO2014105844A1 (en) 2014-07-03
DK2938194T3 (da) 2020-01-02
CR20150382A (es) 2015-08-21
HUE047711T2 (hu) 2020-05-28
US20160192653A1 (en) 2016-07-07
US20170204069A1 (en) 2017-07-20
BR102013033709B1 (pt) 2019-05-14
US9908855B2 (en) 2018-03-06
JP6324994B2 (ja) 2018-05-16
CN104902757B (zh) 2019-01-08
IL239561A0 (en) 2015-08-31
CA2893778A1 (en) 2014-07-03
US9622474B2 (en) 2017-04-18
BR102013033709A2 (pt) 2015-10-06
RU2638556C2 (ru) 2017-12-14
RU2015131095A (ru) 2017-02-06
AU2013370493B2 (en) 2017-08-17
CN110003118A (zh) 2019-07-12
JP2016507512A (ja) 2016-03-10
CN104902757A (zh) 2015-09-09

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