HK1135703A1 - Piperidine gpcr agonists - Google Patents

Piperidine gpcr agonists

Info

Publication number
HK1135703A1
HK1135703A1 HK10103731.6A HK10103731A HK1135703A1 HK 1135703 A1 HK1135703 A1 HK 1135703A1 HK 10103731 A HK10103731 A HK 10103731A HK 1135703 A1 HK1135703 A1 HK 1135703A1
Authority
HK
Hong Kong
Prior art keywords
gpcr agonists
piperidine
piperidine gpcr
agonists
obesity
Prior art date
Application number
HK10103731.6A
Other languages
English (en)
Inventor
Matthew Colin Thor Fyfe
John Keily
Simon Andrew Swain
Original Assignee
Prosidion Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700123A external-priority patent/GB0700123D0/en
Priority claimed from GB0719760A external-priority patent/GB0719760D0/en
Application filed by Prosidion Ltd filed Critical Prosidion Ltd
Publication of HK1135703A1 publication Critical patent/HK1135703A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
HK10103731.6A 2007-01-04 2010-04-16 Piperidine gpcr agonists HK1135703A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0700123A GB0700123D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0719760A GB0719760D0 (en) 2007-10-10 2007-10-10 GPCR agonists
PCT/GB2008/050010 WO2008081204A1 (en) 2007-01-04 2008-01-04 Piperidine gpcr agonists

Publications (1)

Publication Number Publication Date
HK1135703A1 true HK1135703A1 (en) 2010-06-11

Family

ID=39203133

Family Applications (1)

Application Number Title Priority Date Filing Date
HK10103731.6A HK1135703A1 (en) 2007-01-04 2010-04-16 Piperidine gpcr agonists

Country Status (17)

Country Link
US (1) US20100048632A1 (da)
EP (2) EP2114933B1 (da)
JP (1) JP2010514828A (da)
AT (1) ATE523507T1 (da)
BR (1) BRPI0806498A2 (da)
CA (1) CA2674348A1 (da)
CY (1) CY1112483T1 (da)
DK (1) DK2114933T3 (da)
EA (1) EA015129B1 (da)
ES (1) ES2373181T3 (da)
HK (1) HK1135703A1 (da)
HR (1) HRP20110852T1 (da)
PL (1) PL2114933T3 (da)
PT (1) PT2114933E (da)
RS (1) RS52065B (da)
SI (1) SI2114933T1 (da)
WO (1) WO2008081204A1 (da)

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Also Published As

Publication number Publication date
HRP20110852T1 (hr) 2011-12-31
CA2674348A1 (en) 2008-07-10
EA200900877A1 (ru) 2010-02-26
EP2114933B1 (en) 2011-09-07
US20100048632A1 (en) 2010-02-25
PT2114933E (pt) 2011-12-20
PL2114933T3 (pl) 2012-02-29
JP2010514828A (ja) 2010-05-06
EP2377863A1 (en) 2011-10-19
EP2114933A1 (en) 2009-11-11
BRPI0806498A2 (pt) 2014-04-22
RS52065B (en) 2012-06-30
DK2114933T3 (da) 2012-01-02
SI2114933T1 (sl) 2012-01-31
WO2008081204A1 (en) 2008-07-10
ATE523507T1 (de) 2011-09-15
CY1112483T1 (el) 2015-12-09
ES2373181T3 (es) 2012-02-01
EA015129B1 (ru) 2011-06-30

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Legal Events

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20150104