GT200600082A - Derivados del 2-(1,5-difenil-1h-pirazol-3-il)-1,3,4-oxadiazol, su preparacion y su aplicacion en terapeutica - Google Patents

Derivados del 2-(1,5-difenil-1h-pirazol-3-il)-1,3,4-oxadiazol, su preparacion y su aplicacion en terapeutica

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Publication number
GT200600082A
GT200600082A GT200600082A GT200600082A GT200600082A GT 200600082 A GT200600082 A GT 200600082A GT 200600082 A GT200600082 A GT 200600082A GT 200600082 A GT200600082 A GT 200600082A GT 200600082 A GT200600082 A GT 200600082A
Authority
GT
Guatemala
Prior art keywords
difenil
pirazol
oxadiazol
therapeutics
derivatives
Prior art date
Application number
GT200600082A
Other languages
English (en)
Inventor
Barth Francis
Congy Christian
Gueule Patrick
Rinaldi-Carmona Murielle
Van Broeck Didier
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079215&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT200600082(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT200600082A publication Critical patent/GT200600082A/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Addiction (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Vascular Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A COMPUESTOS DE LA FÓRMULA GENERAL I EN LA QUE R1,R2,R3,R4, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE. ESTOS COMPUESTOS TIENEN UNA AMPLIA UTILIDAD EN DIVERSAS PATOLOGÍAS TALES COMO TRASTORNOS DEL APETITO, GASTROINTESTINALES, INFLAMATORIOS, PSICÓTICOS, DEPENDENCIA ALCOHÓLICA Y NICOTÍNICA.
GT200600082A 2005-02-21 2006-02-20 Derivados del 2-(1,5-difenil-1h-pirazol-3-il)-1,3,4-oxadiazol, su preparacion y su aplicacion en terapeutica GT200600082A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0501860A FR2882365B1 (fr) 2005-02-21 2005-02-21 Derives de 2-(1,5-diphenyl-1h-pyrazol-3-yl)-1,3,4-oxadiazole leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
GT200600082A true GT200600082A (es) 2006-10-19

Family

ID=35079215

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200600082A GT200600082A (es) 2005-02-21 2006-02-20 Derivados del 2-(1,5-difenil-1h-pirazol-3-il)-1,3,4-oxadiazol, su preparacion y su aplicacion en terapeutica

Country Status (25)

Country Link
US (1) US7632852B2 (es)
EP (1) EP1853595A1 (es)
JP (1) JP4812778B2 (es)
KR (1) KR20070107053A (es)
CN (1) CN101119990A (es)
AR (1) AR055560A1 (es)
AU (1) AU2006215443A1 (es)
BR (1) BRPI0606845A2 (es)
CA (1) CA2597359A1 (es)
DO (1) DOP2006000045A (es)
EA (1) EA200701779A1 (es)
FR (1) FR2882365B1 (es)
GT (1) GT200600082A (es)
IL (1) IL185163A0 (es)
MA (1) MA29261B1 (es)
MX (1) MX2007009994A (es)
NO (1) NO20074763L (es)
NZ (1) NZ560790A (es)
PA (1) PA8663901A1 (es)
PE (1) PE20061038A1 (es)
SV (1) SV2007002422A (es)
TW (1) TW200640916A (es)
UY (1) UY29388A1 (es)
WO (1) WO2006087480A1 (es)
ZA (1) ZA200706953B (es)

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JP2010500300A (ja) 2006-08-08 2010-01-07 サノフィ−アベンティス アリールアミノアリール−アルキル−置換イミダゾリジン−２，４−ジオン、それらの製造法、それらの化合物を含有する薬剤、およびそれらの使用
EP2097410A4 (en) * 2006-09-29 2009-11-25 Green Cross Corp HETEROYL-PYRAZOLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS
US7875647B2 (en) 2006-09-29 2011-01-25 Green Cross Corporation Heteroaryl-pyrazole derivatives as cannabinoid CB1 receptor antagonists
US20080207704A1 (en) * 2007-02-27 2008-08-28 The Green Cross Corporation Heteroaryl-imidazole derivatives as cannabinoid cb1 receptor antagonists
US7705024B2 (en) 2007-04-12 2010-04-27 National Health Research Institutes Oxadiazole compounds
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
WO2009078498A1 (en) * 2007-12-17 2009-06-25 Green Cross Corporation Biarylpyrazole 4-carboxamides as cannabinoid cb1 receptor ligands
EP2310372B1 (en) 2008-07-09 2012-05-23 Sanofi Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof
US8309584B2 (en) * 2008-09-25 2012-11-13 Green Cross Corporation Sulfur containing pyrazole-heterocycle derivatives as cannabinoid CB1 receptor antagonists
WO2010068601A1 (en) 2008-12-08 2010-06-17 Sanofi-Aventis A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof
US8785608B2 (en) 2009-08-26 2014-07-22 Sanofi Crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use
WO2011157827A1 (de) 2010-06-18 2011-12-22 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
EP2683705B1 (de) 2011-03-08 2015-04-22 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8710050B2 (en) 2011-03-08 2014-04-29 Sanofi Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
EP2683704B1 (de) 2011-03-08 2014-12-17 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2766349B1 (de) 2011-03-08 2016-06-01 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683700B1 (de) 2011-03-08 2015-02-18 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
CN109651350B (zh) * 2019-01-11 2022-05-24 贵州大学 一类杂环取代的1,3,4-噁(噻)二唑类化合物及其制备方法和用途
CN109942567B (zh) * 2019-04-30 2023-04-07 贵州大学 一种1,3,4-噁(噻)二唑基的咪唑类化合物及其制备方法和用途

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FR2758723B1 (fr) * 1997-01-28 1999-04-23 Sanofi Sa Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
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FR2882365A1 (fr) 2006-08-25
AU2006215443A1 (en) 2006-08-24
PE20061038A1 (es) 2006-11-24
MA29261B1 (fr) 2008-02-01
SV2007002422A (es) 2007-01-17
JP2008530188A (ja) 2008-08-07
UY29388A1 (es) 2006-10-02
FR2882365B1 (fr) 2007-09-07
US7632852B2 (en) 2009-12-15
CA2597359A1 (fr) 2006-08-24
EA200701779A1 (ru) 2008-02-28
PA8663901A1 (es) 2006-12-07
DOP2006000045A (es) 2006-11-15
JP4812778B2 (ja) 2011-11-09
US20080039510A1 (en) 2008-02-14
EP1853595A1 (fr) 2007-11-14
KR20070107053A (ko) 2007-11-06
NO20074763L (no) 2007-11-16
ZA200706953B (en) 2009-03-25
AR055560A1 (es) 2007-08-22
IL185163A0 (en) 2007-12-03
WO2006087480A1 (fr) 2006-08-24
BRPI0606845A2 (pt) 2009-07-21
MX2007009994A (es) 2007-10-10
CN101119990A (zh) 2008-02-06
TW200640916A (en) 2006-12-01

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