GB1351719A - Triazolobenzodiazepines - Google Patents
TriazolobenzodiazepinesInfo
- Publication number
- GB1351719A GB1351719A GB3731672A GB3731672A GB1351719A GB 1351719 A GB1351719 A GB 1351719A GB 3731672 A GB3731672 A GB 3731672A GB 3731672 A GB3731672 A GB 3731672A GB 1351719 A GB1351719 A GB 1351719A
- Authority
- GB
- United Kingdom
- Prior art keywords
- reacting
- alkyl
- prepared
- triazolobenzodiazepines
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Fodder In General (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
1351719 Triazolobenzodiazepines UPJOHN CO 10 Aug 1972 [13 Sept 1971] 37316/72 Heading C2C Compounds of the general formula (R 1 = H, C 1-3 alkyl; R 2 = pyridyl, 2-pyrimidyl, furyl, pyrryl, thienyl, C 1-3 alkyl, C 2-3 alkenyl- C 5-7 cycloalkyl or cycloalkenyl; R 3 = H, halo, gen, NO 2 , CF 3 , C 1-3 alkoxy or alkylthio, di-(C 1-3 alkyl) amino) and their acid addition salts are prepared by reacting a compound of the formula with trifluoroacetic acid, optionally followed by salt formation. The starting materials are prepared by reacting the corresponding thione with hydrazine hydrate; the thiones are obtained by reacting the ketone with phosphorus pentasulphide. The above compounds are sedatives, hypnotics, anticonvulsants, tranquillizers and muscle relaxants, and increased growth rate and feed efficiency of livestock. They may be administered in the form of pharmaceutical or veterinary preparations or food premixes containing them in association with a carrier.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18011271A | 1971-09-13 | 1971-09-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1351719A true GB1351719A (en) | 1974-05-01 |
Family
ID=22659243
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB3731672A Expired GB1351719A (en) | 1971-09-13 | 1972-08-10 | Triazolobenzodiazepines |
Country Status (4)
| Country | Link |
|---|---|
| JP (1) | JPS4836194A (en) |
| DE (1) | DE2244571A1 (en) |
| FR (1) | FR2154495B1 (en) |
| GB (1) | GB1351719A (en) |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1955349C2 (en) * | 1969-11-04 | 1982-01-28 | Takeda Chemical Industries, Ltd., Osaka | s-Triazolo [4,3-a] [1,4] benzodiazepines |
-
1972
- 1972-08-10 GB GB3731672A patent/GB1351719A/en not_active Expired
- 1972-09-08 JP JP47089685A patent/JPS4836194A/ja active Pending
- 1972-09-11 DE DE19722244571 patent/DE2244571A1/en active Pending
- 1972-09-12 FR FR7232260A patent/FR2154495B1/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| FR2154495B1 (en) | 1976-04-23 |
| JPS4836194A (en) | 1973-05-28 |
| DE2244571A1 (en) | 1973-03-22 |
| FR2154495A1 (en) | 1973-05-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| PLNP | Patent lapsed through nonpayment of renewal fees |