GB1001822A - Improvements in or relating to homothiaxanthenes - Google Patents

Improvements in or relating to homothiaxanthenes

Info

Publication number
GB1001822A
GB1001822A GB2959761A GB2959761A GB1001822A GB 1001822 A GB1001822 A GB 1001822A GB 2959761 A GB2959761 A GB 2959761A GB 2959761 A GB2959761 A GB 2959761A GB 1001822 A GB1001822 A GB 1001822A
Authority
GB
United Kingdom
Prior art keywords
alkyl
hydrogen
compounds
acid addition
addition salts
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB2959761A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz Patent Ltd
Sandoz AG
Original Assignee
Sandoz Patent Ltd
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH968460A external-priority patent/CH384589A/en
Application filed by Sandoz Patent Ltd, Sandoz AG filed Critical Sandoz Patent Ltd
Publication of GB1001822A publication Critical patent/GB1001822A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/10—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D337/12—[b,e]-condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention comprises compounds of general formula <FORM:1001822/C2/1> wherein each of R1, R2 and R3 is hydrogen or alkyl (1-4 C), and R4 and R5 are alkyl (1-4 C) or -NR4R5 signifies morpholino or piperidino, with the proviso that, when two of R1, R2 and R3 are hydrogen, R4 together with the remaining substituent R1, R2 and R3 may represent alkylene (2-4 C) (but excluding 1-dimethyl-amino-3-homothiaxanthylidene-(41) - propane); and their acid addition salts; and their preparation by treating a corresponding 4-substituted-4-hydroxy -homothiaxanthene with a dehydrating agent. Pharmaceutical compositions comprise compounds I and their acid addition salts with inert carriers. The compounds inhibit biogenic amines and have neuroplegic and antidepressant activities. Specifications 1,001,823 and 1,001,825 also are referred to.
GB2959761A 1960-08-26 1961-08-16 Improvements in or relating to homothiaxanthenes Expired GB1001822A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH968460A CH384589A (en) 1960-08-26 1960-08-26 Process for the preparation of heterocyclic compounds
CH1189560 1960-10-25
CH643261 1961-06-01

Publications (1)

Publication Number Publication Date
GB1001822A true GB1001822A (en) 1965-08-18

Family

ID=27175493

Family Applications (2)

Application Number Title Priority Date Filing Date
GB193765A Expired GB1001823A (en) 1960-08-26 1961-08-16 Improvements in or relating to 4-hydroxy homothiaxanthenes
GB2959761A Expired GB1001822A (en) 1960-08-26 1961-08-16 Improvements in or relating to homothiaxanthenes

Family Applications Before (1)

Application Number Title Priority Date Filing Date
GB193765A Expired GB1001823A (en) 1960-08-26 1961-08-16 Improvements in or relating to 4-hydroxy homothiaxanthenes

Country Status (2)

Country Link
ES (1) ES270093A1 (en)
GB (2) GB1001823A (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004052847A2 (en) * 2002-06-26 2004-06-24 Eli Lilly And Company Tricyclic steroid hormone nuclear receptor modulators

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004052847A2 (en) * 2002-06-26 2004-06-24 Eli Lilly And Company Tricyclic steroid hormone nuclear receptor modulators
WO2004052847A3 (en) * 2002-06-26 2004-09-10 Lilly Co Eli Tricyclic steroid hormone nuclear receptor modulators
US7411072B2 (en) 2002-06-26 2008-08-12 Eli Lilly And Company Tricyclic steroid hormone nuclear receptor modulators

Also Published As

Publication number Publication date
ES270093A1 (en) 1962-05-01
GB1001823A (en) 1965-08-18

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