FR2966151B1 - Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met - Google Patents

Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met

Info

Publication number
FR2966151B1
FR2966151B1 FR1058393A FR1058393A FR2966151B1 FR 2966151 B1 FR2966151 B1 FR 2966151B1 FR 1058393 A FR1058393 A FR 1058393A FR 1058393 A FR1058393 A FR 1058393A FR 2966151 B1 FR2966151 B1 FR 2966151B1
Authority
FR
France
Prior art keywords
triazolopyridazine
sulfanyl
medicaments
cycloalkyl
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR1058393A
Other languages
English (en)
Other versions
FR2966151A1 (fr
Inventor
Eric Bacque
Dominique Damour
Conception Nemecek
Antonio Ugolini
Sylvie Wentzler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Aventis France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France
Priority to FR1058393A priority Critical patent/FR2966151B1/fr
Priority to PCT/FR2011/050682 priority patent/WO2011121223A1/fr
Priority to TW100110835A priority patent/TW201202242A/zh
Priority to UY0001033299A priority patent/UY33299A/es
Publication of FR2966151A1 publication Critical patent/FR2966151A1/fr
Application granted granted Critical
Publication of FR2966151B1 publication Critical patent/FR2966151B1/fr
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
FR1058393A 2010-03-30 2010-10-14 Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met Expired - Fee Related FR2966151B1 (fr)

Priority Applications (4)

Application Number Priority Date Filing Date Title
FR1058393A FR2966151B1 (fr) 2010-10-14 2010-10-14 Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met
PCT/FR2011/050682 WO2011121223A1 (fr) 2010-03-30 2011-03-29 Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met
TW100110835A TW201202242A (en) 2010-03-30 2011-03-29 6-(alkyl-or cycloalkyl-triazolopyridazine-sulfanyl)benzo-thiazole derivatives: preparation, and use as medicaments and as MET inhibitors
UY0001033299A UY33299A (es) 2010-03-30 2011-03-30 Derivados de 6-(alquil-o cicloalquil-triazolopiridacina-silfanil)benzotiazoles:preparacion, aplicación como medicamentos y utilizacion como inhibidores de la met

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR1058393A FR2966151B1 (fr) 2010-10-14 2010-10-14 Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met

Publications (2)

Publication Number Publication Date
FR2966151A1 FR2966151A1 (fr) 2012-04-20
FR2966151B1 true FR2966151B1 (fr) 2012-11-09

Family

ID=43778298

Family Applications (1)

Application Number Title Priority Date Filing Date
FR1058393A Expired - Fee Related FR2966151B1 (fr) 2010-03-30 2010-10-14 Derives de 6-(alkyl- ou cycloalkyl-triazolopyridazine-sulfanyl) benzothiazoles: preparation, application comme medicaments et utilisation comme inhibiteurs de met

Country Status (1)

Country Link
FR (1) FR2966151B1 (fr)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PA8792501A1 (es) * 2007-08-09 2009-04-23 Sanofi Aventis Nuevos derivados de 6-triazolopiridacina-sulfanil benzotiazol y bencimidazol,su procedimiento de preparación,su aplicación como medicamentos,composiciones farmacéuticas y nueva utilización principalmente como inhibidores de met.
EA201170222A1 (ru) * 2008-07-18 2011-08-30 Санофи-Авентис НОВЫЕ ПРОИЗВОДНЫЕ ТРИАЗОЛО[4,3-a]ПИРИДИНА, СПОСОБ ИХ ПОЛУЧЕНИЯ, ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ЛЕКАРСТВЕННЫХ СРЕДСТВ, ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ И НОВОЕ ПРИМЕНЕНИЕ, В ЧАСТНОСТИ, В КАЧЕСТВЕ ИНГИБИТОРОВ МЕТ
US20110257171A1 (en) * 2008-07-18 2011-10-20 Sanofi-Aventis Novel imidazo[1,2-a]pyridine derivatives, method for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use in particular as met inhibitors
FR2941952B1 (fr) * 2009-02-06 2011-04-01 Sanofi Aventis Derives de 6-(6-substitue-triazolopyridazine-sulfanyl) 5-fluoro-benzothiazoles et 5-fluoro-benzimidazoles : preparation, application comme medicaments et utilisation comme inhibiteurs de met.

Also Published As

Publication number Publication date
FR2966151A1 (fr) 2012-04-20

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Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20160630