FR2826004B1 - Procede de preparation de derives estrogenes - Google Patents
Procede de preparation de derives estrogenesInfo
- Publication number
- FR2826004B1 FR2826004B1 FR0107711A FR0107711A FR2826004B1 FR 2826004 B1 FR2826004 B1 FR 2826004B1 FR 0107711 A FR0107711 A FR 0107711A FR 0107711 A FR0107711 A FR 0107711A FR 2826004 B1 FR2826004 B1 FR 2826004B1
- Authority
- FR
- France
- Prior art keywords
- preparation
- estrogenic derivatives
- estrogenic
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
- C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
- C07J73/003—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by oxygen as hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Priority Applications (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0107711A FR2826004B1 (fr) | 2001-06-13 | 2001-06-13 | Procede de preparation de derives estrogenes |
EP02747527A EP1404701A1 (fr) | 2001-06-13 | 2002-06-12 | Procede de preparation de derives estrogenes |
JP2003503646A JP2004534796A (ja) | 2001-06-13 | 2002-06-12 | エストロゲン誘導体の製造方法 |
US10/480,618 US7381718B2 (en) | 2001-06-13 | 2002-06-12 | Method for preparing oestrogen derivatives |
PCT/FR2002/002001 WO2002100880A1 (fr) | 2001-06-13 | 2002-06-12 | Procede de preparation de derives estrogenes |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0107711A FR2826004B1 (fr) | 2001-06-13 | 2001-06-13 | Procede de preparation de derives estrogenes |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2826004A1 FR2826004A1 (fr) | 2002-12-20 |
FR2826004B1 true FR2826004B1 (fr) | 2008-03-28 |
Family
ID=8864249
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0107711A Expired - Fee Related FR2826004B1 (fr) | 2001-06-13 | 2001-06-13 | Procede de preparation de derives estrogenes |
Country Status (5)
Country | Link |
---|---|
US (1) | US7381718B2 (fr) |
EP (1) | EP1404701A1 (fr) |
JP (1) | JP2004534796A (fr) |
FR (1) | FR2826004B1 (fr) |
WO (1) | WO2002100880A1 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
USH1511H (en) * | 1992-09-10 | 1995-12-05 | Chappell; Charles W. | Absorbent articles having improved longitudinal fluid movement |
GB0307067D0 (en) | 2002-12-17 | 2003-04-30 | Aventis Pharma Inc | Use of thiazolobenzoheterocycles for treating multiple sclerosis |
FR2854402B1 (fr) * | 2003-04-29 | 2008-07-04 | Aventis Pharma Sa | Nouveau procede et intermediaires de preparation de composes 19-nor-steroides |
US10385093B2 (en) | 2012-12-10 | 2019-08-20 | Northeastern University | Estrogen receptor imaging agents |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2377419A1 (fr) * | 1977-01-13 | 1978-08-11 | Roussel Uclaf | Nouveaux derives steroides 11b-substitues 1,3,5 (10) trieniques, leur procede de preparation et leur application comme medicament |
FR2377418A1 (fr) * | 1977-01-13 | 1978-08-11 | Roussel Uclaf | Nouveaux derives steroides 4,9-dieniques 11b-substitues, leur procede de preparation et leur application comme medicaments |
ZA8231B (en) * | 1981-01-09 | 1982-11-24 | Roussel Uclaf | New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained |
FR2528434B1 (fr) * | 1982-06-11 | 1985-07-19 | Roussel Uclaf | Nouveaux 19-nor steroides substitues en 11b et eventuellement en 2, leur procede de preparation et leur application comme medicament |
FR2640977A2 (en) * | 1982-06-11 | 1990-06-29 | Roussel Uclaf | New position-11 substituted 19-norsteroids and their application as medicinal products. |
FR2598421B1 (fr) * | 1986-05-06 | 1988-08-19 | Roussel Uclaf | Nouveaux produits 19-nor ou 19-nor d-homo steroides substitues en position 11b par un radical phenyle portant un radical alkynyle, leur procede de preparation, leur application comme medicaments et les compositions les renfermant |
FR2643638B1 (fr) * | 1989-02-24 | 1991-06-14 | Roussel Uclaf | Nouveaux 19-nor steroides ayant en position 11beta une chaine carbonee comportant une fonction amide ou carbamate, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
US5929262A (en) * | 1995-03-30 | 1999-07-27 | The United States Of America As Represented By The Department Of Health And Human Services | Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates |
FR2757519B1 (fr) * | 1996-12-23 | 1999-06-11 | Hoechst Marion Roussel Inc | Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant |
FR2761992B1 (fr) * | 1997-04-09 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux steroides 4-halogenes, leur procede et intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant |
FR2771096B1 (fr) * | 1997-11-17 | 2000-08-11 | Hoechst Marion Roussel Inc | Nouveaux 19-nor steroides, substitues en position 11beta, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant |
-
2001
- 2001-06-13 FR FR0107711A patent/FR2826004B1/fr not_active Expired - Fee Related
-
2002
- 2002-06-12 WO PCT/FR2002/002001 patent/WO2002100880A1/fr active Application Filing
- 2002-06-12 US US10/480,618 patent/US7381718B2/en not_active Expired - Lifetime
- 2002-06-12 JP JP2003503646A patent/JP2004534796A/ja active Pending
- 2002-06-12 EP EP02747527A patent/EP1404701A1/fr not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
FR2826004A1 (fr) | 2002-12-20 |
US7381718B2 (en) | 2008-06-03 |
WO2002100880A1 (fr) | 2002-12-19 |
US20040171595A1 (en) | 2004-09-02 |
JP2004534796A (ja) | 2004-11-18 |
EP1404701A1 (fr) | 2004-04-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |
Effective date: 20160229 |