FR2730491B1 - Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent - Google Patents
Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennentInfo
- Publication number
- FR2730491B1 FR2730491B1 FR9501489A FR9501489A FR2730491B1 FR 2730491 B1 FR2730491 B1 FR 2730491B1 FR 9501489 A FR9501489 A FR 9501489A FR 9501489 A FR9501489 A FR 9501489A FR 2730491 B1 FR2730491 B1 FR 2730491B1
- Authority
- FR
- France
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- transferase inhibitors
- farnesyl transferase
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
- C07K5/1013—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/07—Tetrapeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Priority Applications (18)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9501489A FR2730491B1 (fr) | 1995-02-09 | 1995-02-09 | Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
AU47227/96A AU4722796A (en) | 1995-02-09 | 1996-02-07 | Novel farnesyl transferase inhibitors, preparation thereof, and pharmaceutical compositions containing same |
CN96191867A CN1173874A (zh) | 1995-02-09 | 1996-02-07 | 新的法呢基转移酶抑制剂,其制法及其药物组合物 |
BR9607317A BR9607317A (pt) | 1995-02-09 | 1996-02-07 | Peptídios e composição farmacêutica |
KR1019970705443A KR19980702048A (ko) | 1995-02-09 | 1996-02-07 | 신규한 파르네실 트랜스퍼라아제 억제제, 이의 제조방법 및 이를 함유하는 약학 조성물 |
EP96903061A EP0808328A1 (fr) | 1995-02-09 | 1996-02-07 | Inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
CA002210955A CA2210955A1 (fr) | 1995-02-09 | 1996-02-07 | Inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
SK1087-97A SK108797A3 (en) | 1995-02-09 | 1996-02-07 | Novel farnesyl transferase inhibitors, preparation thereof, and pharmaceutical compositions containing same |
TR97/00727T TR199700727T1 (xx) | 1995-02-09 | 1996-02-07 | Farnesil transferaz�n�n yeni inhibit�rleri. |
PCT/FR1996/000198 WO1996024611A1 (fr) | 1995-02-09 | 1996-02-07 | Inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
JP8524037A JPH10513467A (ja) | 1995-02-09 | 1996-02-07 | ファルネシル転移酵素阻害剤、これらの調製、及びこれらを含む製薬学的組成物 |
PL96321675A PL321675A1 (en) | 1995-02-09 | 1996-02-07 | Novel inhibitors of farnesil transferase, their production and pharmaceutic compositions containing them |
CZ972498A CZ249897A3 (en) | 1995-02-09 | 1996-02-07 | Novel inhibitors of farnesyl transferase, process of their preparation and pharmaceutical compositions containing such inhibitors |
US08/875,752 US5856439A (en) | 1995-02-09 | 1996-02-07 | Farnesyl transferase inhibitors, preparation thereof, and pharmaceutical compositions containing same |
ZA961072A ZA961072B (en) | 1995-02-09 | 1996-02-09 | New farnesyl transferase inhibitors their preparation and the pharmaceutical compositions which contain them |
NO973608A NO973608L (no) | 1995-02-09 | 1997-08-05 | Nye farnesyltransferaseinhibitorer, deres fremstilling samt farmasöytiske preparater inneholdende forbindelsene |
MXPA/A/1997/006015A MXPA97006015A (en) | 1995-02-09 | 1997-08-06 | Novedous inhibitors of farnesil transferase, supreparation and pharmaceutical compositions chelos contie |
FI973278A FI973278A (fi) | 1995-02-09 | 1997-08-08 | Uudet farnesyylitransferaasin inhibiittorit, niiden valmistus ja niitä sisältävät farmaseuttiset valmisteet |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9501489A FR2730491B1 (fr) | 1995-02-09 | 1995-02-09 | Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2730491A1 FR2730491A1 (fr) | 1996-08-14 |
FR2730491B1 true FR2730491B1 (fr) | 1997-03-14 |
Family
ID=9475979
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR9501489A Expired - Fee Related FR2730491B1 (fr) | 1995-02-09 | 1995-02-09 | Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
Country Status (17)
Country | Link |
---|---|
US (1) | US5856439A (fr) |
EP (1) | EP0808328A1 (fr) |
JP (1) | JPH10513467A (fr) |
KR (1) | KR19980702048A (fr) |
CN (1) | CN1173874A (fr) |
AU (1) | AU4722796A (fr) |
BR (1) | BR9607317A (fr) |
CA (1) | CA2210955A1 (fr) |
CZ (1) | CZ249897A3 (fr) |
FI (1) | FI973278A (fr) |
FR (1) | FR2730491B1 (fr) |
NO (1) | NO973608L (fr) |
PL (1) | PL321675A1 (fr) |
SK (1) | SK108797A3 (fr) |
TR (1) | TR199700727T1 (fr) |
WO (1) | WO1996024611A1 (fr) |
ZA (1) | ZA961072B (fr) |
Families Citing this family (55)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2730491B1 (fr) * | 1995-02-09 | 1997-03-14 | Rhone Poulenc Rorer Sa | Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
WO2006123182A2 (fr) | 2005-05-17 | 2006-11-23 | Merck Sharp & Dohme Limited | Sulfones de cyclohexyle pour le traitement du cancer |
GB0603041D0 (en) | 2006-02-15 | 2006-03-29 | Angeletti P Ist Richerche Bio | Therapeutic compounds |
WO2008039327A2 (fr) | 2006-09-22 | 2008-04-03 | Merck & Co., Inc. | Procédé de traitement utilisant des inhibiteurs de synthèse d'acide gras |
US20110218176A1 (en) | 2006-11-01 | 2011-09-08 | Barbara Brooke Jennings-Spring | Compounds, methods, and treatments for abnormal signaling pathways for prenatal and postnatal development |
AU2008204380B2 (en) | 2007-01-10 | 2013-08-15 | Msd Italia S.R.L. | Amide substituted indazoles as poly(ADP-ribose)polymerase (PARP) inhibitors |
CN101679266B (zh) | 2007-03-01 | 2015-05-06 | 诺华股份有限公司 | Pim激酶抑制剂及其应用方法 |
BRPI0812159A2 (pt) | 2007-05-21 | 2017-05-02 | Novartis Ag | inibidores de csf-1r, composições e métodos de uso |
US8389553B2 (en) | 2007-06-27 | 2013-03-05 | Merck Sharp & Dohme Corp. | 4-carboxybenzylamino derivatives as histone deacetylase inhibitors |
US7932036B1 (en) | 2008-03-12 | 2011-04-26 | Veridex, Llc | Methods of determining acute myeloid leukemia response to treatment with farnesyltransferase |
EP2413932A4 (fr) | 2009-04-01 | 2012-09-19 | Merck Sharp & Dohme | Inhibiteurs de l'activité akt |
JP6073677B2 (ja) | 2009-06-12 | 2017-02-01 | デイナ ファーバー キャンサー インスティチュート,インコーポレイテッド | 縮合複素環式化合物およびそれらの使用 |
BR112012008849A2 (pt) | 2009-10-14 | 2015-09-22 | Schering Corp | composto, composição farmacêutica, e, uso de um composto |
CA2784807C (fr) | 2009-12-29 | 2021-12-14 | Dana-Farber Cancer Institute, Inc. | Inhibiteurs de kinase raf de type ii |
BR112012023021A2 (pt) | 2010-03-16 | 2016-05-31 | Dana Farber Cancer Inst Inc | compostos de indazol e seus usos |
EP2584903B1 (fr) | 2010-06-24 | 2018-10-24 | Merck Sharp & Dohme Corp. | Nouveaux composés hétérocycliques utilisés comme inhibiteurs de erk |
WO2012016021A2 (fr) | 2010-07-28 | 2012-02-02 | Veridex, Llc | Procédés de détermination de réponse de la leucémie myéloïde aiguë à traitement par inhibiteurs de la farnésyltransférase |
JP6043285B2 (ja) | 2010-08-02 | 2016-12-14 | サーナ・セラピューティクス・インコーポレイテッドSirna Therapeutics,Inc. | 低分子干渉核酸(siNA)を用いたカテニン(カドヘリン結合型タンパク質)β1(CTNNB1)遺伝子発現のRNA干渉媒介性阻害 |
HUE044815T2 (hu) | 2010-08-17 | 2019-11-28 | Sirna Therapeutics Inc | Hepatitisz B vírus (HBV) génexpressziójának RNS-interferencia közvetített gátlása, rövid interferáló nukleinsav (SINS) alkalmazásával |
EP2608669B1 (fr) | 2010-08-23 | 2016-06-22 | Merck Sharp & Dohme Corp. | Nouveaux dérivés de pyrazolo[1,5-a]pyrimidine utilisés comme inhibiteurs de mtor |
EP2613782B1 (fr) | 2010-09-01 | 2016-11-02 | Merck Sharp & Dohme Corp. | Dérivés d'indazole utilisables en tant qu'inhibiteurs de la voie erk |
WO2012036997A1 (fr) | 2010-09-16 | 2012-03-22 | Schering Corporation | Dérivés condensés de pyrazole utilisés comme nouveaux inhibiteurs erk |
US9260471B2 (en) | 2010-10-29 | 2016-02-16 | Sirna Therapeutics, Inc. | RNA interference mediated inhibition of gene expression using short interfering nucleic acids (siNA) |
WO2012087772A1 (fr) | 2010-12-21 | 2012-06-28 | Schering Corporation | Dérivés d'indazole utiles en tant qu'inhibiteurs de erk |
US20140045847A1 (en) | 2011-04-21 | 2014-02-13 | Piramal Enterprises Limited | Crystalline form of a salt of a morpholino sulfonyl indole derivative and a process for its preparation |
WO2013063214A1 (fr) | 2011-10-27 | 2013-05-02 | Merck Sharp & Dohme Corp. | Nouveaux composés qui sont des inhibiteurs d'erk |
WO2013074986A1 (fr) | 2011-11-17 | 2013-05-23 | Dana-Farber Cancer Institute, Inc. | Inhibiteurs de la kinase c-jun-n-terminale (jnk) |
EP3919620A1 (fr) | 2012-05-02 | 2021-12-08 | Sirna Therapeutics, Inc. | Compositions d'acide nucléique interférent court (sina) |
US9233979B2 (en) | 2012-09-28 | 2016-01-12 | Merck Sharp & Dohme Corp. | Compounds that are ERK inhibitors |
US10112927B2 (en) | 2012-10-18 | 2018-10-30 | Dana-Farber Cancer Institute, Inc. | Inhibitors of cyclin-dependent kinase 7 (CDK7) |
WO2014063054A1 (fr) | 2012-10-19 | 2014-04-24 | Dana-Farber Cancer Institute, Inc. | Inhibiteurs de kinase moelle osseuse sur chromosome x (bmx) et leurs utilisations |
US9758522B2 (en) | 2012-10-19 | 2017-09-12 | Dana-Farber Cancer Institute, Inc. | Hydrophobically tagged small molecules as inducers of protein degradation |
BR112015012295A8 (pt) | 2012-11-28 | 2023-03-14 | Merck Sharp & Dohme | Uso de um inibidor de wee1, e, kit para identificar um paciente com câncer |
BR112015013611A2 (pt) | 2012-12-20 | 2017-11-14 | Merck Sharp & Dohme | composto, e, composição farmacêutica |
EP2951180B1 (fr) | 2013-01-30 | 2018-05-02 | Merck Sharp & Dohme Corp. | Purines 2,6,7,8-substituées utilisées en tant qu'inhibiteurs de hdm2 |
EP3041938A1 (fr) | 2013-09-03 | 2016-07-13 | Moderna Therapeutics, Inc. | Polynucléotides circulaires |
JP6491202B2 (ja) | 2013-10-18 | 2019-03-27 | デイナ ファーバー キャンサー インスティチュート,インコーポレイテッド | サイクリン依存性キナーゼ7(cdk7)の多環阻害剤 |
WO2015058126A1 (fr) | 2013-10-18 | 2015-04-23 | Syros Pharmaceuticals, Inc. | Composés hétéroaromatiques utiles dans le traitement de maladies prolifératives |
US9862688B2 (en) | 2014-04-23 | 2018-01-09 | Dana-Farber Cancer Institute, Inc. | Hydrophobically tagged janus kinase inhibitors and uses thereof |
WO2015164614A1 (fr) | 2014-04-23 | 2015-10-29 | Dana-Farber Cancer Institute, Inc. | Inhibiteurs de janus kinase et leurs utilisations |
JO3589B1 (ar) | 2014-08-06 | 2020-07-05 | Novartis Ag | مثبطات كيناز البروتين c وطرق استخداماتها |
AU2015371251B2 (en) | 2014-12-23 | 2020-06-11 | Dana-Farber Cancer Institute, Inc. | Inhibitors of cyclin-dependent kinase 7 (CDK7) |
WO2016160617A2 (fr) | 2015-03-27 | 2016-10-06 | Dana-Farber Cancer Institute, Inc. | Inhibiteurs de kinases cycline-dépendantes |
EP3307728A4 (fr) | 2015-06-12 | 2019-07-17 | Dana Farber Cancer Institute, Inc. | Thérapie d'association utilisant des inhibiteurs de transcription et des inhibiteurs de kinases |
HUE057306T2 (hu) | 2015-08-17 | 2022-04-28 | Kura Oncology Inc | Módszerek rákos páciensek kezelésére farneziltranszferáz inhibitorokkal |
EP3347018B1 (fr) | 2015-09-09 | 2021-09-01 | Dana-Farber Cancer Institute, Inc. | Inhibiteurs de kinases cycline-dépendantes |
JOP20190055A1 (ar) | 2016-09-26 | 2019-03-24 | Merck Sharp & Dohme | أجسام مضادة ضد cd27 |
EA201991091A1 (ru) | 2016-11-03 | 2019-11-29 | Способы лечения пациентов со злокачественными новообразованиями с применением ингибиторов фарнезилтрансферазы | |
JP7160833B2 (ja) | 2017-04-13 | 2022-10-25 | サイロパ ビー.ブイ. | 抗sirpアルファ抗体 |
WO2019094311A1 (fr) | 2017-11-08 | 2019-05-16 | Merck Sharp & Dohme Corp. | Inhibiteurs de prmt5 |
WO2019113269A1 (fr) | 2017-12-08 | 2019-06-13 | Kura Oncology, Inc. | Méthodes de traitement de patients cancéreux avec des inhibiteurs de la farnésyltransférase |
WO2019148412A1 (fr) | 2018-02-01 | 2019-08-08 | Merck Sharp & Dohme Corp. | Anticorps bispécifiques anti-pd-1/lag3 |
EP3833667B1 (fr) | 2018-08-07 | 2024-03-13 | Merck Sharp & Dohme LLC | Inhibiteurs de prmt5 |
WO2020033282A1 (fr) | 2018-08-07 | 2020-02-13 | Merck Sharp & Dohme Corp. | Inhibiteurs de prmt5 |
US20220143006A1 (en) | 2019-03-15 | 2022-05-12 | Kura Oncology, Inc. | Methods of treating cancer with farnesyltransferase inhibitors |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5141851A (en) * | 1990-04-18 | 1992-08-25 | Board Of Regents, The University Of Texas System | Isolated farnesyl protein transferase enzyme |
CA2044333A1 (fr) * | 1990-06-12 | 1991-12-13 | Jackson B. Gibbs | Agents chimiotherapeutiques |
CA2072033A1 (fr) * | 1991-06-28 | 1992-12-29 | Jackson B. Gibbs | Inhibiteur de la farnesyl-proteine-transferase ne se rapportant pas a un substrat |
CA2118985A1 (fr) * | 1993-04-02 | 1994-10-03 | Dinesh V. Patel | Inhibiteurs heterocycliques de la farnesyl proteine transferase |
JPH09500615A (ja) * | 1993-05-14 | 1997-01-21 | ジェネンテク,インコーポレイテッド | Ras−ファルネシル転移酵素阻害剤 |
US5439918A (en) * | 1994-03-14 | 1995-08-08 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
FR2730492B1 (fr) * | 1995-02-09 | 1997-03-14 | Rhone Poulenc Rorer Sa | Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
FR2730491B1 (fr) * | 1995-02-09 | 1997-03-14 | Rhone Poulenc Rorer Sa | Nouveaux inhibiteurs de farnesyl transferase, leur preparation et les compositions pharmaceutiques qui les contiennent |
-
1995
- 1995-02-09 FR FR9501489A patent/FR2730491B1/fr not_active Expired - Fee Related
-
1996
- 1996-02-07 CA CA002210955A patent/CA2210955A1/fr not_active Abandoned
- 1996-02-07 JP JP8524037A patent/JPH10513467A/ja active Pending
- 1996-02-07 TR TR97/00727T patent/TR199700727T1/xx unknown
- 1996-02-07 WO PCT/FR1996/000198 patent/WO1996024611A1/fr not_active Application Discontinuation
- 1996-02-07 CZ CZ972498A patent/CZ249897A3/cs unknown
- 1996-02-07 CN CN96191867A patent/CN1173874A/zh active Pending
- 1996-02-07 AU AU47227/96A patent/AU4722796A/en not_active Abandoned
- 1996-02-07 BR BR9607317A patent/BR9607317A/pt not_active Application Discontinuation
- 1996-02-07 SK SK1087-97A patent/SK108797A3/sk unknown
- 1996-02-07 PL PL96321675A patent/PL321675A1/xx unknown
- 1996-02-07 EP EP96903061A patent/EP0808328A1/fr not_active Ceased
- 1996-02-07 US US08/875,752 patent/US5856439A/en not_active Expired - Fee Related
- 1996-02-07 KR KR1019970705443A patent/KR19980702048A/ko not_active Application Discontinuation
- 1996-02-09 ZA ZA961072A patent/ZA961072B/xx unknown
-
1997
- 1997-08-05 NO NO973608A patent/NO973608L/no unknown
- 1997-08-08 FI FI973278A patent/FI973278A/fi not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
PL321675A1 (en) | 1997-12-22 |
FI973278A0 (fi) | 1997-08-08 |
JPH10513467A (ja) | 1998-12-22 |
CZ249897A3 (en) | 1997-11-12 |
NO973608D0 (no) | 1997-08-05 |
CA2210955A1 (fr) | 1996-08-15 |
ZA961072B (en) | 1996-08-20 |
AU4722796A (en) | 1996-08-27 |
EP0808328A1 (fr) | 1997-11-26 |
FI973278A (fi) | 1997-08-08 |
CN1173874A (zh) | 1998-02-18 |
TR199700727T1 (xx) | 1998-02-21 |
WO1996024611A1 (fr) | 1996-08-15 |
NO973608L (no) | 1997-08-05 |
US5856439A (en) | 1999-01-05 |
FR2730491A1 (fr) | 1996-08-14 |
KR19980702048A (ko) | 1998-07-15 |
MX9706015A (es) | 1997-11-29 |
SK108797A3 (en) | 1997-12-10 |
BR9607317A (pt) | 1997-12-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |