FR2440362A1 - Nouveaux derives d'acides mercaptoacylpiperazinecarboxyliques, utiles notamment comme hypotenseurs, et leur procede de preparation - Google Patents

Nouveaux derives d'acides mercaptoacylpiperazinecarboxyliques, utiles notamment comme hypotenseurs, et leur procede de preparation

Info

Publication number
FR2440362A1
FR2440362A1 FR7926901A FR7926901A FR2440362A1 FR 2440362 A1 FR2440362 A1 FR 2440362A1 FR 7926901 A FR7926901 A FR 7926901A FR 7926901 A FR7926901 A FR 7926901A FR 2440362 A1 FR2440362 A1 FR 2440362A1
Authority
FR
France
Prior art keywords
mercaptoacylpiperazinecarboxylic
hydropensors
novel
preparation process
acid derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR7926901A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2440362A1 publication Critical patent/FR2440362A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'INVENTION CONCERNE DES MEDICAMENTS DE FORMULE: (CF DESSIN DANS BOPI) DANS LAQUELLE R, R ET R REPRESENTENT CHACUN L'HYDROGENE OU UN GROUPE ALKYLE INFERIEUR; R EST UN GROUPE ALKYLE INFERIEUR; R UN ATOME D'HYDROGENE OU UN GROUPE ALCANOYLE INFERIEUR, BENZOYLE OU (CF DESSIN DANS BOPI) M EST EGAL A 0, 1 OU 2; N EST EGAL A 1, 2 OU 3; LA SOMME MN ETANT EGALE A 1, 2 OU 3; ET LEURS SELS. APPLICATIONS EN TABLETTES, CAPSULES OU ELIXIRS POUR L'ADMINISTRATION ORALE OU EN SOLUTIONS OU SUSPENSIONS STERILES POUR L'ADMINISTRATION PARENTERALE, CONTENANT ENVIRON 10 A 500MG D'INGREDIENT ACTIF.
FR7926901A 1978-10-30 1979-10-30 Nouveaux derives d'acides mercaptoacylpiperazinecarboxyliques, utiles notamment comme hypotenseurs, et leur procede de preparation Withdrawn FR2440362A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/955,854 US4198509A (en) 1978-10-30 1978-10-30 Mercaptoacylpiperazine carboxylic acid compounds

Publications (1)

Publication Number Publication Date
FR2440362A1 true FR2440362A1 (fr) 1980-05-30

Family

ID=25497451

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7926901A Withdrawn FR2440362A1 (fr) 1978-10-30 1979-10-30 Nouveaux derives d'acides mercaptoacylpiperazinecarboxyliques, utiles notamment comme hypotenseurs, et leur procede de preparation

Country Status (6)

Country Link
US (1) US4198509A (fr)
JP (1) JPS5555170A (fr)
DE (1) DE2943809A1 (fr)
FR (1) FR2440362A1 (fr)
GB (1) GB2036723A (fr)
IT (1) IT1164131B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA794723B (en) * 1978-09-11 1980-08-27 Univ Miami Anti-hypertensive agents
US4692458A (en) * 1980-03-05 1987-09-08 University Of Miami Anti-hypertensive agents
JPS6053216B2 (ja) * 1980-05-19 1985-11-25 アイシン精機株式会社 車輛用変速装置
CA1248531A (fr) * 1984-04-17 1989-01-10 Jeffrey C. Watkins Derives de substitution en 4 d'acides piperazine-2- carboxyliques
US5413999A (en) * 1991-11-08 1995-05-09 Merck & Co., Inc. HIV protease inhibitors useful for the treatment of AIDS

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2161910A1 (fr) * 1971-10-07 1973-07-13 Bristol Myers Co

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3147261A (en) * 1962-05-24 1964-09-01 Robert R Mod Nu-acyl-nu'-methylpiperazines
US4105776A (en) * 1976-06-21 1978-08-08 E. R. Squibb & Sons, Inc. Proline derivatives and related compounds
US4046889A (en) * 1976-02-13 1977-09-06 E. R. Squibb & Sons, Inc. Azetidine-2-carboxylic acid derivatives

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2161910A1 (fr) * 1971-10-07 1973-07-13 Bristol Myers Co

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
CA1965 *

Also Published As

Publication number Publication date
IT7950642A0 (it) 1979-10-23
US4198509A (en) 1980-04-15
GB2036723A (en) 1980-07-02
DE2943809A1 (de) 1980-05-14
JPS5555170A (en) 1980-04-22
IT1164131B (it) 1987-04-08

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Legal Events

Date Code Title Description
RE Withdrawal of published application