FR2205313A1 - - Google Patents
Info
- Publication number
- FR2205313A1 FR2205313A1 FR7339380A FR7339380A FR2205313A1 FR 2205313 A1 FR2205313 A1 FR 2205313A1 FR 7339380 A FR7339380 A FR 7339380A FR 7339380 A FR7339380 A FR 7339380A FR 2205313 A1 FR2205313 A1 FR 2205313A1
- Authority
- FR
- France
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/41—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by hydrogenolysis or reduction of carboxylic groups or functional derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/58—Preparation of carboxylic acid halides
- C07C51/60—Preparation of carboxylic acid halides by conversion of carboxylic acids or their anhydrides or esters, lactones, salts into halides with the same carboxylic acid part
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
- C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D317/18—Radicals substituted by singly bound oxygen or sulfur atoms
- C07D317/24—Radicals substituted by singly bound oxygen or sulfur atoms esterified
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
- C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D317/28—Radicals substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D463/00—Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D463/02—Preparation
- C07D463/06—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/568—Four-membered rings
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US30390572A | 1972-11-06 | 1972-11-06 | |
US39566273A | 1973-09-18 | 1973-09-18 |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2205313A1 true FR2205313A1 (cs) | 1974-05-31 |
FR2205313B1 FR2205313B1 (cs) | 1976-07-02 |
Family
ID=26973713
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7339380A Expired FR2205313B1 (cs) | 1972-11-06 | 1973-11-06 |
Country Status (11)
Country | Link |
---|---|
JP (1) | JPS5632993B2 (cs) |
AT (1) | AT340590B (cs) |
BE (1) | BE806921A (cs) |
CH (1) | CH602723A5 (cs) |
DE (1) | DE2355209A1 (cs) |
ES (1) | ES420271A1 (cs) |
FR (1) | FR2205313B1 (cs) |
GB (1) | GB1455016A (cs) |
HK (1) | HK86679A (cs) |
NL (1) | NL178005C (cs) |
SE (1) | SE417205B (cs) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2388815A1 (fr) * | 1977-04-28 | 1978-11-24 | Shionogi & Co | Procede de preparation d'haloarylmalonamidooxacephalosporines, nouveaux produits ainsi obtenus et leur utilisation pour le traitement de maladies dues aux bacteries |
FR2397419A1 (fr) * | 1977-07-14 | 1979-02-09 | Shionogi & Co | Dihydrotriazinylthiooxacephalosporines et leur utilisation comme agents antimicrobiens |
FR2401165A1 (fr) * | 1977-08-25 | 1979-03-23 | Shionogi & Co | Procede de preparation d'analogues de thiadiazolylcephalosporine et nouveaux produits ainsi obtenus, a activite antibacterienne |
FR2476091A1 (cs) * | 1980-01-22 | 1981-08-21 | Shionogi & Co |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4226866A (en) * | 1972-11-06 | 1980-10-07 | Merck & Co., Inc. | Novel antibiotic analogues of cephalosporins |
US4172199A (en) * | 1975-01-02 | 1979-10-23 | Bristol-Myers Company | O-2-isocephem-4-carboxylic acid derivatives as antibacterial agents |
US4012383A (en) * | 1975-01-02 | 1977-03-15 | Bristol-Myers Company | Δ2,3 -1,4-morpholine-2-carboxylic acids and derivatives thereof useful in preparation of antibacteria agents |
US4166906A (en) * | 1975-04-11 | 1979-09-04 | Bristol-Myers Company | 0-2-Isocephem-4-carboxylic acid derivatives as antibacterial agents |
US4171439A (en) * | 1975-04-11 | 1979-10-16 | Bristol-Myers Company | Antibacterial analogs of isocephalosporins |
US4166905A (en) * | 1975-04-11 | 1979-09-04 | Bristol-Myers Company | O-2-Isocephem-4-carboxylic acid derivatives as antibacterial agents |
US4011216A (en) * | 1975-04-11 | 1977-03-08 | Bristol-Myers Company | Δ2,3-0-2-Isocephem-4-carboxylic acid and derivatives thereof as antibacterial agents |
US4108992A (en) | 1975-05-10 | 1978-08-22 | Beecham Group Limited | Cephalosporin analogues and compositions |
US4013648A (en) * | 1975-07-23 | 1977-03-22 | Bristol-Myers Company | Δ2,3 -0-2-Isocephem-4-carboxylic acid and derivatives as antibacterial agents |
US4171438A (en) * | 1975-07-23 | 1979-10-16 | Bristol-Myers Company | 0-2-Isocephem-4-carboxylic acid derivatives as antibacterial agents |
US4180571A (en) * | 1976-03-25 | 1979-12-25 | Shionogi & Co., Ltd. | Arylmalonamido-1-oxadethiacephalosporins |
CA1085392A (en) | 1976-03-25 | 1980-09-09 | Masayuki Narisada | Arylmalonamido-1-oxadethiacephalosporins |
NO158505C (no) * | 1976-03-25 | 1988-09-21 | Shionogi & Co | Analogifremgangsmaate for fremstilling av et terapeutisk aktivt 7beta-substituert malonamido-1-oksadetia 7alfa-metoksy-3-(1-metyltetrazol-5-yl)-tiometyl cefalosporin. |
JPS607635B2 (ja) * | 1976-04-27 | 1985-02-26 | 塩野義製薬株式会社 | オキサゾリジン化合物 |
JPS604811B2 (ja) * | 1976-07-28 | 1985-02-06 | 塩野義製薬株式会社 | メチルケトンのハロゲン化 |
JPS609515B2 (ja) * | 1976-08-09 | 1985-03-11 | 塩野義製薬株式会社 | 3′−ノルオキサセファロスポリン類 |
CA1076125A (en) * | 1976-08-09 | 1980-04-22 | Masayuki Narisada | Intermediates for cephalosporin analogues |
JPS5331690A (en) * | 1976-09-01 | 1978-03-25 | Shionogi & Co Ltd | Oxadithiacephalosporins |
US4089956A (en) * | 1976-09-08 | 1978-05-16 | Smithkline Corporation | 7-Acylamino-8-oxo-3-oxa-1-azabicyclo[4.2.0]octane-2-carboxylic acid derivatives and bactericidal compositions and use thereof |
JPS5398951A (en) | 1977-02-08 | 1978-08-29 | Shionogi & Co Ltd | Azetidinone derivatives and process for their preparation |
GB1557552A (en) * | 1977-02-15 | 1979-12-12 | Shionogi & Co | 1 oxadethiacepham compounds |
JPS53105491A (en) | 1977-02-25 | 1978-09-13 | Shionogi & Co Ltd | Oxazolinoazethidinylbutyrylic acid derivatives |
JPS53149991A (en) * | 1977-06-01 | 1978-12-27 | Shionogi & Co Ltd | Preparation of 3-heterothiomethyl-1-oxadethia-3-cephem-4-carboxylic acid |
IT1102408B (it) * | 1977-12-23 | 1985-10-07 | Fujisawa Pharmaceutical Co | Composti analoghi della cefalosforina e procedimenti per la loro preparazione |
EP0004134B1 (en) * | 1978-03-04 | 1981-12-30 | Beecham Group Plc | Beta-lactam antibacterial agents, their pharmaceutical compositions and process for their preparation |
JPS5936914B2 (ja) * | 1978-06-24 | 1984-09-06 | 協和醗酵工業株式会社 | セフアロスポリン類縁体 |
US4327093A (en) * | 1978-10-24 | 1982-04-27 | Fujisawa Pharmaceutical Co., Ltd. | 3,7-Disubstituted-2 or 3-cephem-4-carboxylic acid compounds |
JPS5671092A (en) * | 1979-11-14 | 1981-06-13 | Kyowa Hakko Kogyo Co Ltd | Optical active cephalosporin analogous derivative |
JPS5616491A (en) * | 1979-07-19 | 1981-02-17 | Kyowa Hakko Kogyo Co Ltd | Cephalosporin analog |
DE3069524D1 (en) * | 1979-12-20 | 1984-11-29 | Hoechst Uk Ltd | Penem derivatives |
US4304774A (en) * | 1980-09-17 | 1981-12-08 | Eli Lilly And Company | Bis-tetrazolmethyl substituted β-lactam antibiotics |
DE3225269A1 (de) * | 1982-07-06 | 1984-01-12 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von 7-amino-1-dethia-1-oxa-3-hydroxymethyl-cephem-4-carbonsaeuren |
JPS59104389A (ja) * | 1982-12-06 | 1984-06-16 | Shionogi & Co Ltd | オキサセファム誘導体 |
US4717722A (en) * | 1984-05-07 | 1988-01-05 | Merck & Co., Inc. | Substituted 1-oxa-dethiacephalosporins as anti-inflammatory and antidegenerative agents |
US4708956A (en) * | 1985-12-12 | 1987-11-24 | Kyowa Hakko Kogyo Co., Ltd. | 3-position halogenated cephalosporin analogs and pharmaceutical compositions |
US5019571A (en) * | 1988-01-25 | 1991-05-28 | Eli Lilly And Company | 1-carbacephalosporin antibiotics |
JP2004168775A (ja) * | 2002-11-08 | 2004-06-17 | Orchid Chemicals & Pharmaceuticals Ltd | オキサセファロスポリンの改良合成法 |
CN103635478A (zh) * | 2011-04-28 | 2014-03-12 | 盐野义制药株式会社 | 具有儿茶酚或假儿茶酚结构的新颖头孢烯类化合物 |
CN103254215B (zh) * | 2013-05-24 | 2015-06-03 | 浙江东邦药业有限公司 | 一种烯丙基氯代氧头孢化合物的制备方法 |
-
1973
- 1973-10-25 NL NLAANVRAGE7314711,A patent/NL178005C/xx not_active IP Right Cessation
- 1973-10-26 SE SE7314569A patent/SE417205B/xx unknown
- 1973-11-02 CH CH1549273A patent/CH602723A5/xx not_active IP Right Cessation
- 1973-11-05 BE BE137412A patent/BE806921A/xx not_active IP Right Cessation
- 1973-11-05 ES ES420271A patent/ES420271A1/es not_active Expired
- 1973-11-05 GB GB5130173A patent/GB1455016A/en not_active Expired
- 1973-11-05 DE DE19732355209 patent/DE2355209A1/de not_active Ceased
- 1973-11-06 JP JP12486473A patent/JPS5632993B2/ja not_active Expired
- 1973-11-06 FR FR7339380A patent/FR2205313B1/fr not_active Expired
-
1975
- 1975-06-26 AT AT491775A patent/AT340590B/de not_active IP Right Cessation
-
1979
- 1979-12-20 HK HK866/79A patent/HK86679A/xx unknown
Non-Patent Citations (1)
Title |
---|
NEANT * |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2388815A1 (fr) * | 1977-04-28 | 1978-11-24 | Shionogi & Co | Procede de preparation d'haloarylmalonamidooxacephalosporines, nouveaux produits ainsi obtenus et leur utilisation pour le traitement de maladies dues aux bacteries |
FR2397419A1 (fr) * | 1977-07-14 | 1979-02-09 | Shionogi & Co | Dihydrotriazinylthiooxacephalosporines et leur utilisation comme agents antimicrobiens |
FR2401165A1 (fr) * | 1977-08-25 | 1979-03-23 | Shionogi & Co | Procede de preparation d'analogues de thiadiazolylcephalosporine et nouveaux produits ainsi obtenus, a activite antibacterienne |
FR2476091A1 (cs) * | 1980-01-22 | 1981-08-21 | Shionogi & Co |
Also Published As
Publication number | Publication date |
---|---|
BE806921A (fr) | 1974-05-06 |
AT340590B (de) | 1977-12-27 |
DE2355209A1 (de) | 1974-05-16 |
NL178005B (nl) | 1985-08-01 |
ATA491775A (de) | 1977-04-15 |
NL7314711A (cs) | 1974-05-08 |
ES420271A1 (es) | 1976-07-01 |
JPS49133594A (cs) | 1974-12-21 |
SE417205B (sv) | 1981-03-02 |
NL178005C (nl) | 1986-01-02 |
JPS5632993B2 (cs) | 1981-07-31 |
FR2205313B1 (cs) | 1976-07-02 |
HK86679A (en) | 1979-12-28 |
GB1455016A (en) | 1976-11-10 |
CH602723A5 (cs) | 1978-07-31 |