FI964114A - Uusia 1-(5-metaanisulfonamidoindolyyli-2-karbonyyli)-4-(3-(1-metyylietyyliamino)-2-pyridinyyli)piperatsiinin kiteisiä muotoja - Google Patents

Uusia 1-(5-metaanisulfonamidoindolyyli-2-karbonyyli)-4-(3-(1-metyylietyyliamino)-2-pyridinyyli)piperatsiinin kiteisiä muotoja Download PDF

Info

Publication number
FI964114A
FI964114A FI964114A FI964114A FI964114A FI 964114 A FI964114 A FI 964114A FI 964114 A FI964114 A FI 964114A FI 964114 A FI964114 A FI 964114A FI 964114 A FI964114 A FI 964114A
Authority
FI
Finland
Prior art keywords
methanesulfonamidoindolyl
methylethylamino
pyridinyl
carbonyl
piperazine
Prior art date
Application number
FI964114A
Other languages
English (en)
Swedish (sv)
Other versions
FI964114A0 (fi
FI111364B (fi
Inventor
Jeffrey L Havens
Donald P Smith
Michael S Bergren
Mark A Lyster
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FI964114A0 publication Critical patent/FI964114A0/fi
Publication of FI964114A publication Critical patent/FI964114A/fi
Application granted granted Critical
Publication of FI111364B publication Critical patent/FI111364B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Indole Compounds (AREA)
FI964114A 1994-04-15 1996-10-14 Uusia 1-[5-metaanisulfonamidoindolyyli-2-karbonyyli]-4-[3-(1-metyylietyyliamino)-2-pyridinyyli]piperatsiinin kidemuotoja FI111364B (fi)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US22786094A 1994-04-15 1994-04-15
US22786094 1994-04-15
US31178094A 1994-09-23 1994-09-23
US31178094 1994-09-23
US9502166 1995-03-01
PCT/US1995/002166 WO1995028398A1 (en) 1994-04-15 1995-03-01 Novel crystal forms of 1-[5-methanesulfonamidoindolyl-2-carbonyl]-4-[3-(1-methylethylamino)-2-pyridinyl]piperazine

Publications (3)

Publication Number Publication Date
FI964114A0 FI964114A0 (fi) 1996-10-14
FI964114A true FI964114A (fi) 1996-10-14
FI111364B FI111364B (fi) 2003-07-15

Family

ID=26921831

Family Applications (1)

Application Number Title Priority Date Filing Date
FI964114A FI111364B (fi) 1994-04-15 1996-10-14 Uusia 1-[5-metaanisulfonamidoindolyyli-2-karbonyyli]-4-[3-(1-metyylietyyliamino)-2-pyridinyyli]piperatsiinin kidemuotoja

Country Status (26)

Country Link
US (1) US6452007B1 (fi)
EP (1) EP0755393B1 (fi)
JP (1) JP3817261B2 (fi)
KR (1) KR100364941B1 (fi)
CN (1) CN1147253A (fi)
AT (1) ATE207481T1 (fi)
AU (1) AU693939B2 (fi)
CA (1) CA2184598C (fi)
CZ (1) CZ287164B6 (fi)
DE (1) DE69523447T2 (fi)
DK (1) DK0755393T3 (fi)
ES (1) ES2164147T3 (fi)
FI (1) FI111364B (fi)
HU (1) HU226827B1 (fi)
IL (1) IL113162A (fi)
LV (1) LV12957B (fi)
MX (1) MX9604831A (fi)
MY (1) MY116830A (fi)
NO (1) NO310024B1 (fi)
NZ (1) NZ282211A (fi)
PL (1) PL180776B1 (fi)
PT (1) PT755393E (fi)
RU (1) RU2136677C1 (fi)
SK (1) SK282424B6 (fi)
TW (1) TW393478B (fi)
WO (1) WO1995028398A1 (fi)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4827296B2 (ja) 1998-06-11 2011-11-30 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー デラビルジン錠製剤
US6872811B1 (en) 1998-09-30 2005-03-29 Millennium Pharmaceuticals, Inc. HRPCa9 and HRPCa10 nucleic acids and polypeptides
DE102011113749A1 (de) * 2011-09-14 2013-03-14 Aicuris Gmbh & Co. Kg Sulfonsäuresalze Heterocyclylamid-substituiertr Imidazole

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3565924A (en) 1968-07-01 1971-02-23 Wisconsin Alumni Res Found 25-hydroxycholfcalciferol
US3833622A (en) 1969-03-17 1974-09-03 Upjohn Co Crystalline 25-hydroxycholecalciferol hydrate and structurally related compounds
GB1532682A (en) 1976-04-27 1978-11-22 Bristol Myers Co Process for the preparation of cephadroxil
IL63968A (en) 1980-10-01 1985-10-31 Glaxo Group Ltd Form 2 ranitidine hydrochloride,its preparation and pharmaceutical compositions containing it
US5563142A (en) * 1989-12-28 1996-10-08 The Upjohn Company Diaromatic substituted compounds as anti-HIV-1 agents
ATE142621T1 (de) * 1989-12-28 1996-09-15 Upjohn Co Diaromatische substituierte verbindungen gegen den aids-virus
US5599930A (en) * 1991-07-03 1997-02-04 The Upjohn Company Substituted indoles as anti-AIDS pharmaceuticals

Also Published As

Publication number Publication date
EP0755393B1 (en) 2001-10-24
AU3513695A (en) 1995-11-10
MY116830A (en) 2004-04-30
NO964386L (no) 1996-10-15
JPH09512007A (ja) 1997-12-02
SK282424B6 (sk) 2002-01-07
JP3817261B2 (ja) 2006-09-06
CN1147253A (zh) 1997-04-09
WO1995028398A1 (en) 1995-10-26
NZ282211A (en) 1997-10-24
PL180776B1 (pl) 2001-04-30
HUT76467A (en) 1997-09-29
CZ287164B6 (en) 2000-10-11
TW393478B (en) 2000-06-11
SK122996A3 (en) 1997-05-07
US6452007B1 (en) 2002-09-17
CZ294296A3 (en) 1997-01-15
KR970702275A (ko) 1997-05-13
CA2184598C (en) 2005-05-03
DK0755393T3 (da) 2001-12-17
ES2164147T3 (es) 2002-02-16
HU9602857D0 (en) 1996-12-30
AU693939B2 (en) 1998-07-09
PL316688A1 (en) 1997-02-03
EP0755393A1 (en) 1997-01-29
IL113162A0 (en) 1995-06-29
KR100364941B1 (ko) 2003-02-19
DE69523447T2 (de) 2002-05-16
ATE207481T1 (de) 2001-11-15
FI964114A0 (fi) 1996-10-14
PT755393E (pt) 2002-04-29
RU2136677C1 (ru) 1999-09-10
IL113162A (en) 1999-04-11
NO964386D0 (no) 1996-10-15
CA2184598A1 (en) 1995-10-26
LV12957B (en) 2003-04-20
NO310024B1 (no) 2001-05-07
HU226827B1 (en) 2009-11-30
DE69523447D1 (de) 2001-11-29
MX9604831A (es) 1998-05-31
FI111364B (fi) 2003-07-15

Similar Documents

Publication Publication Date Title
DE69328975T2 (de) Aminomethylen substituierte heterocyclische verbindungen und ihre verwendung alssubstanz p antagonisten
BG101112A (en) The use of heterocyclic compounds
NO992770L (no) Nye heterocyklisk substituerte benzamider og deres anvendelse ved bekjempelse av sykdommer
ES2123149T3 (es) Derivados de perhidroisoindol como antagonistas de la substancia p.
FI894911A0 (fi) En terapeutiskt vaerdefull foerening.
BG101110A (en) Substituted pyrimidine compounds and their application
MX9605741A (es) Clorhidrato cristalino del (r)-(-)-2-{n-[4-(1,1-dioxido-3-oxo-2,3-dihidro-benzisotiazol-2-il)-butil ]-aminometil} cromano.
DK0696281T3 (da) Hidtil ukendte 5-pyrrolyl-2-pyridylmethylsulfinylbenzimidazolderivater
TR200201684T2 (tr) Fenilpiperazinil türevleri
ATE178886T1 (de) 1-aryl-2-acylamino-ethan-verbindungen und ihre verwendung als neurokinin- insbesondere als neurokinin-1-antagonisten
CA2298461A1 (en) Heterocyclic substituted 4-benzoyl-pyrazole as herbicides
DE59410304D1 (de) N-substituierte azabicycloheptan-derivate und ihre verwendung, z.b., als neuroleptika
FI964114A0 (fi) Uusia 1-(5-metaanisulfonamidoindolyyli-2-karbonyyli)-4-(3-(1-metyylietyyliamino)-2-pyridinyyli)piperatsiinin kiteisiä muotoja
FI955387A (fi) 4(p-fluorifenyyli)-3-((3,4-(metyleenioksi)fenoksi)metyyli)-piperidiinin N-p-halobentsoyylimetyylijohdannaiset
BG105247A (en) N-substituted azabicycloheptane derivatives, production and use thereof
NO993650L (no) Nye forbindelser med hemoregulerende effekt
YU41908B (en) Process for proucing the crystalline form of 1-(4-amino-6,7-dimethoxy-2-quinazoliyl)-4-(2-furoyl)-piperazine hydrochloride
BG105329A (en) N-substituted azabicycloheptane derivatives, production and use thereof

Legal Events

Date Code Title Description
MA Patent expired