ES2039242T3 - Un procedimiento para la preparacion de nuevos derivados de piperidina. - Google Patents
Un procedimiento para la preparacion de nuevos derivados de piperidina.Info
- Publication number
- ES2039242T3 ES2039242T3 ES198787307632T ES87307632T ES2039242T3 ES 2039242 T3 ES2039242 T3 ES 2039242T3 ES 198787307632 T ES198787307632 T ES 198787307632T ES 87307632 T ES87307632 T ES 87307632T ES 2039242 T3 ES2039242 T3 ES 2039242T3
- Authority
- ES
- Spain
- Prior art keywords
- procedure
- preparation
- piperidine derivatives
- new piperidine
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/26—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms
Abstract
LA INVENCION SE REFIERE A UN COMPUESTO DE FORMULA (I) O A UNA SAL O SOLVATO DE EL, EN LA QUE R.CO ES UN GRUPO ACILO Y R TIENE LA FORMULA (II) EN LA QUE R3 ES BR, NO2 O CF3; Y R1 Y R2 SON INDEPENDIENTEMENTE ALQUILO DE 1 A 6 C, O JUNTOS FORMAN UN GRUPO POLIMETILENO O ALQUILENO DE 3 A 6 C. EL COMPUESTO ES UTIL COMO ANALGESICO.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB868621134A GB8621134D0 (en) | 1986-09-02 | 1986-09-02 | Compounds |
GB868629642A GB8629642D0 (en) | 1986-12-11 | 1986-12-11 | Compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2039242T3 true ES2039242T3 (es) | 1993-09-16 |
Family
ID=26291239
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES198787307632T Expired - Lifetime ES2039242T3 (es) | 1986-09-02 | 1987-08-28 | Un procedimiento para la preparacion de nuevos derivados de piperidina. |
Country Status (9)
Country | Link |
---|---|
US (1) | US4826819A (es) |
EP (1) | EP0260041B1 (es) |
AU (1) | AU601763B2 (es) |
DE (1) | DE3767816D1 (es) |
DK (1) | DK456987A (es) |
ES (1) | ES2039242T3 (es) |
GR (1) | GR3001411T3 (es) |
NZ (1) | NZ221621A (es) |
PT (1) | PT85628B (es) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0232612B1 (en) * | 1985-12-23 | 1990-04-04 | Dr. Lo. Zambeletti S.p.A. | Azacyclic compounds, processes for their preparation, and their use as pharmaceuticals |
PT86427B (pt) * | 1986-12-22 | 1990-11-20 | Zambeletti Spa L | Processo para a preparacao de derivados de piperidina |
GB8803259D0 (en) * | 1988-02-12 | 1988-03-09 | Zambeletti Spa L | Compounds |
GB8804104D0 (en) * | 1988-02-23 | 1988-03-23 | Glaxo Group Ltd | Chemical compounds |
JPH01308229A (ja) * | 1988-02-23 | 1989-12-12 | Glaxo Group Ltd | 複素環誘導体 |
GB8804014D0 (en) * | 1988-02-23 | 1988-03-23 | Humphreys & Glasgow Ltd | Synthesis gas production |
DK247789A (da) * | 1988-05-23 | 1989-11-24 | Glaxo Group Ltd | Piperazinderivater |
US5270327A (en) * | 1988-08-24 | 1993-12-14 | Sankyo Company, Limited | Analgesic compounds, their preparation, and pharmaceutical compositions containing them |
US5021413B1 (en) * | 1988-08-24 | 1994-12-13 | Sankyo Co | Analgesic thiomorpholins, their preparation, and pharmaceutical compositions containing them |
US5512567A (en) * | 1988-08-24 | 1996-04-30 | Sankyo Company, Limited | Analgesic compounds, their preparation, and pharmaceutical compositions containing them |
DE68924751T2 (de) * | 1988-09-26 | 1996-04-11 | Smithkline Beecham Farma | Azacyclische Verbindungen, verwendbar als Arzneimittel. |
GB8824400D0 (en) * | 1988-10-18 | 1988-11-23 | Glaxo Group Ltd | Chemical compounds |
US5063242A (en) * | 1989-04-21 | 1991-11-05 | Warner-Lambert Company | 7-((substituted)amino)-8-((substituted)carbonyl)-methylamino-1-oxaspiro[4,5]decanes as diuretics antiinflammatory, and cerebrovascular agents |
US4965278A (en) | 1989-04-21 | 1990-10-23 | Warner-Lambert Company | 7-(substituted)amino)-8-((substituted)carbonyl)-methylamino)-1-oxaspiro[4,5]decanes as diuretics antiiflammatory, and cerebrovascular agents |
PT94070A (pt) * | 1989-05-18 | 1991-01-08 | Glaxo Group Ltd | Processo para a preparacao de derivados de piperazina |
GB8926560D0 (en) * | 1989-11-24 | 1990-01-17 | Zambeletti Spa L | Pharmaceuticals |
EP0447704A1 (en) * | 1990-03-21 | 1991-09-25 | Smithkline Beecham Farmaceutici S.p.A. | N-Acylated azacyclic compounds, processes for their preparations and their use as medications |
US5428042A (en) * | 1990-04-28 | 1995-06-27 | Dr Lo Zambeletti S.P.A. | 1-(2H-1-oxo-3,4-dihydronaphtyl-6-yl)-acetyl-piperidines as kappa agonists |
GB9011656D0 (en) * | 1990-05-24 | 1990-07-11 | Zambeletti Spa L | Novel compounds |
AU1532492A (en) * | 1991-04-18 | 1992-11-17 | Dr. Lo Zambeletti S.P.A. | Use of heterocyclic compounds for the treatment of inflammatory pain |
US5317028A (en) * | 1992-09-08 | 1994-05-31 | Warner-Lambert Co. | 7-((substituted)amino)-8((substituted)carbonyl)-methylamino-1-oxaspiro(4,5)decanes useful in Parkinson's disease, dystonia, and other movement disorders |
ES2319265T3 (es) * | 2001-03-30 | 2009-05-06 | Toray Industries, Inc. | Farmacos para el sindrome de piernas inquietas. |
BRPI0510746A (pt) * | 2004-06-10 | 2007-11-20 | Univ Michigan State | sìntese de caprolactama a partir de lisina |
WO2008103366A2 (en) * | 2007-02-20 | 2008-08-28 | Board Of Trustees Of Michigan State University | Catalytic deamination for carprolactam production |
JP2011529087A (ja) * | 2008-07-24 | 2011-12-01 | ドラス コーポレイション | 環状アミドモノマーを作製する方法、ならびに関連する誘導体および方法 |
WO2011103126A1 (en) * | 2010-02-17 | 2011-08-25 | Ampla Pharmaceuticals Inc. | Treatment of metabolic syndrome with piperidine amides |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0052311A1 (en) * | 1980-11-19 | 1982-05-26 | Sterling Drug Inc. | 1-((Benzoylphenyl) - lower-alkyl) piperidines and carbinol analogs and preparation thereof |
GB8531615D0 (en) * | 1985-12-23 | 1986-02-05 | Zambeletti Spa L | Compounds |
EP0232612B1 (en) * | 1985-12-23 | 1990-04-04 | Dr. Lo. Zambeletti S.p.A. | Azacyclic compounds, processes for their preparation, and their use as pharmaceuticals |
PT86427B (pt) * | 1986-12-22 | 1990-11-20 | Zambeletti Spa L | Processo para a preparacao de derivados de piperidina |
-
1987
- 1987-08-28 EP EP87307632A patent/EP0260041B1/en not_active Expired - Lifetime
- 1987-08-28 ES ES198787307632T patent/ES2039242T3/es not_active Expired - Lifetime
- 1987-08-28 DE DE8787307632T patent/DE3767816D1/de not_active Expired - Fee Related
- 1987-08-31 PT PT85628A patent/PT85628B/pt not_active IP Right Cessation
- 1987-08-31 NZ NZ221621A patent/NZ221621A/xx unknown
- 1987-08-31 AU AU77711/87A patent/AU601763B2/en not_active Ceased
- 1987-08-31 US US07/091,275 patent/US4826819A/en not_active Expired - Fee Related
- 1987-09-01 DK DK456987A patent/DK456987A/da not_active Application Discontinuation
-
1991
- 1991-01-31 GR GR91400071T patent/GR3001411T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
DE3767816D1 (de) | 1991-03-07 |
DK456987D0 (da) | 1987-09-01 |
AU601763B2 (en) | 1990-09-20 |
PT85628A (en) | 1987-09-01 |
US4826819A (en) | 1989-05-02 |
AU7771187A (en) | 1988-03-10 |
PT85628B (pt) | 1990-05-31 |
EP0260041A1 (en) | 1988-03-16 |
DK456987A (da) | 1988-03-03 |
GR3001411T3 (en) | 1992-09-25 |
EP0260041B1 (en) | 1991-01-30 |
NZ221621A (en) | 1990-07-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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