EG24142A - Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition - Google Patents

Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition

Info

Publication number
EG24142A
EG24142A EG20011058A EG20011058A EG24142A EG 24142 A EG24142 A EG 24142A EG 20011058 A EG20011058 A EG 20011058A EG 20011058 A EG20011058 A EG 20011058A EG 24142 A EG24142 A EG 24142A
Authority
EG
Egypt
Prior art keywords
preparing
preparation
pharmaceutical composition
crystalline monohydrate
monohydrate
Prior art date
Application number
EG20011058A
Inventor
Banholzer Rolf
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EG24142(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Application granted granted Critical
Publication of EG24142A publication Critical patent/EG24142A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • C07D451/10Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
EG20011058A 2000-10-12 2001-10-09 Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition EG24142A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12

Publications (1)

Publication Number Publication Date
EG24142A true EG24142A (en) 2008-08-06

Family

ID=7659568

Family Applications (1)

Application Number Title Priority Date Filing Date
EG20011058A EG24142A (en) 2000-10-12 2001-10-09 Crystalline monohydrate, process for the preparation thereof and the use thereof for preparing a pharmaceutical composition

Country Status (47)

Country Link
EP (2) EP1326862B1 (en)
JP (1) JP3764422B2 (en)
KR (1) KR100823860B1 (en)
CN (2) CN1221549C (en)
AP (1) AP1572A (en)
AR (2) AR034389A1 (en)
AT (1) ATE276253T1 (en)
AU (2) AU2002214996B2 (en)
BG (1) BG66161B1 (en)
BR (1) BR0114584A (en)
CA (1) CA2425539C (en)
CR (1) CR6938A (en)
CZ (1) CZ301841B6 (en)
DE (1) DE50103666D1 (en)
DK (1) DK1326862T3 (en)
DZ (1) DZ3478A1 (en)
EA (1) EA004381B1 (en)
EC (1) ECSP034540A (en)
EE (1) EE04567B1 (en)
EG (1) EG24142A (en)
ES (1) ES2228965T3 (en)
GE (1) GEP20063905B (en)
HK (2) HK1060567A1 (en)
HR (1) HRP20030276B1 (en)
HU (1) HU226830B1 (en)
IL (2) IL155335A0 (en)
IS (1) IS2339B (en)
MA (1) MA25842A1 (en)
ME (2) ME00243B (en)
MX (1) MXPA03003221A (en)
MY (1) MY126931A (en)
NO (1) NO328465B1 (en)
NZ (1) NZ525733A (en)
OA (1) OA12403A (en)
PE (1) PE20020422A1 (en)
PL (1) PL207870B1 (en)
PT (1) PT1326862E (en)
RS (1) RS50218B (en)
SA (1) SA01220412B1 (en)
SI (1) SI1326862T1 (en)
SK (1) SK287009B6 (en)
TR (1) TR200402579T4 (en)
TW (1) TW589313B (en)
UA (1) UA74215C2 (en)
UY (2) UY26962A1 (en)
WO (1) WO2002030928A1 (en)
ZA (1) ZA200302500B (en)

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JP5165244B2 (en) 2003-11-03 2013-03-21 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Method for producing tiotropium salt, tiotropium salt and pharmaceutical composition containing the same
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AU2006243238B2 (en) 2005-05-02 2012-05-24 Boehringer Ingelheim International Gmbh Novel crystalline forms of tiotropium bromide
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DE102005030733A1 (en) 2005-07-01 2007-01-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg New drug combinations for the treatment of respiratory diseases containing long-acting beta-2 agonists and at least one other active ingredient
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US20070086957A1 (en) 2005-10-10 2007-04-19 Thierry Bouyssou Combination of medicaments for the treatment of respiratory diseases
US7423146B2 (en) 2005-11-09 2008-09-09 Boehringer Ingelheim International Gmbh Process for the manufacturing of pharmaceutically active 3,1-benzoxazine-2-ones
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MX2007012313A (en) 2006-04-19 2007-11-21 Boehringer Ingelheim Int Dihydrothienopyrimidines for the treatment of inflammatory diseases.
EP1847543A1 (en) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidines for the treatment of inflammatory diseases
US20080051582A1 (en) 2006-07-10 2008-02-28 Sicor Inc. Process for the preparation of tiotropium bromide
EP2051714B1 (en) 2006-08-07 2011-04-13 Boehringer Ingelheim International GmbH Drug combinations for the treatment of respiratory tract diseases
UY30550A1 (en) 2006-08-22 2008-03-31 Boehringer Ingelheim Int NEW BETA-AGANISTAS ENANTIOMÉRICAMENTE PUROS, PROCEDURES FOR ITS PREPARATION AND ITS USE AS MEDICATIONS
EP1923393A1 (en) * 2006-11-17 2008-05-21 Boehringer Ingelheim Pharma GmbH & Co. KG Crystalline form of tiotropium bromide and urea
EP1925295A1 (en) 2006-11-22 2008-05-28 Boehringer Ingelheim Pharma GmbH & Co. KG Stable powder formulation containing a new antichinolinergic agent
GB0716026D0 (en) * 2007-08-16 2007-09-26 Norton Healthcare Ltd An inhalable medicament
WO2009050248A1 (en) 2007-10-19 2009-04-23 Boehringer Ingelheim International Gmbh Substituted piperidino-dihydrothienopyrimidines
EP2093219A1 (en) 2008-02-22 2009-08-26 Boehringer Ingelheim International Gmbh Crystalline enantiomer free salt form of a betamimetic and its use as medicine
WO2010011813A1 (en) * 2008-07-23 2010-01-28 Alkermes, Inc. Complex of trospium and pharmaceutical compositions thereof
ES2551557T3 (en) 2008-12-19 2015-11-19 Boehringer Ingelheim International Gmbh Cyclic pyrimidin-4-carboxamides as CCR2 receptor antagonists for the treatment of inflammations, asthma and COPD
EP2201934A1 (en) 2008-12-23 2010-06-30 CHIESI FARMACEUTICI S.p.A. Tiotropium aerosol formulation products with improved chemical stability
EP2403851B1 (en) 2009-03-06 2015-06-17 Mahmut Bilgic New crystalline forms of tiotropium bromide
WO2011015883A1 (en) 2009-08-07 2011-02-10 Generics [Uk] Limited Dichloromethane solvate of tiotropium bromide and its use
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EP2513086B1 (en) 2009-12-17 2015-04-29 Boehringer Ingelheim International GmbH Novel antagonists for ccr2 and uses thereof
ES2524829T3 (en) 2009-12-17 2014-12-12 Boehringer Ingelheim International Gmbh New CCR2 receptor antagonists and uses thereof
EP2528915B1 (en) 2010-01-29 2015-10-28 Boehringer Ingelheim International GmbH Substituted naphthyridines and their use as syk kinase inhibitors
JP5646736B2 (en) 2010-05-12 2014-12-24 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Novel CCR2 receptor antagonists, methods for their preparation, and their use as drugs
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Also Published As

Publication number Publication date
OA12403A (en) 2006-04-18
MXPA03003221A (en) 2004-12-03
CN100519558C (en) 2009-07-29
PE20020422A1 (en) 2002-06-28
HU226830B1 (en) 2009-11-30
CZ301841B6 (en) 2010-07-07
AU2002214996B2 (en) 2007-03-15
HUP0301022A3 (en) 2005-12-28
CA2425539C (en) 2007-04-03
NO20031694L (en) 2003-04-11
CR6938A (en) 2004-10-28
NO328465B1 (en) 2010-02-22
RS50218B (en) 2009-07-15
ATE276253T1 (en) 2004-10-15
NZ525733A (en) 2005-01-28
HRP20030276A2 (en) 2005-02-28
EA004381B1 (en) 2004-04-29
DE50103666D1 (en) 2004-10-21
PL366041A1 (en) 2005-01-24
PT1326862E (en) 2004-11-30
UA74215C2 (en) 2005-11-15
KR100823860B1 (en) 2008-04-21
AU1499602A (en) 2002-04-22
MY126931A (en) 2006-10-31
NO20031694D0 (en) 2003-04-11
CN1733761A (en) 2006-02-15
EA200300457A1 (en) 2003-10-30
EP1326862A1 (en) 2003-07-16
HK1086557A1 (en) 2006-09-22
YU27303A (en) 2006-05-25
SK4362003A3 (en) 2003-08-05
UY26962A1 (en) 2002-06-20
EP1326862B1 (en) 2004-09-15
BG66161B1 (en) 2011-09-30
AR034389A1 (en) 2004-02-25
HRP20030276B1 (en) 2006-02-28
PL207870B1 (en) 2011-02-28
ES2228965T3 (en) 2005-04-16
CA2425539A1 (en) 2003-04-11
SI1326862T1 (en) 2005-02-28
AR068527A2 (en) 2009-11-18
ME00243B (en) 2011-05-10
CN1469877A (en) 2004-01-21
AP2003002775A0 (en) 2003-03-31
BG107687A (en) 2003-09-30
WO2002030928A1 (en) 2002-04-18
IS2339B (en) 2008-02-15
EP1468998A1 (en) 2004-10-20
SK287009B6 (en) 2009-09-07
IL155335A (en) 2009-02-11
EE04567B1 (en) 2005-12-15
TR200402579T4 (en) 2004-12-21
SA01220412B1 (en) 2006-11-05
DZ3478A1 (en) 2002-04-18
HUP0301022A2 (en) 2003-10-28
IL155335A0 (en) 2003-11-23
GEP20063905B (en) 2006-08-25
HK1060567A1 (en) 2004-08-13
BR0114584A (en) 2003-08-26
IS6772A (en) 2003-04-09
DK1326862T3 (en) 2004-11-22
TW589313B (en) 2004-06-01
JP2004526668A (en) 2004-09-02
JP3764422B2 (en) 2006-04-05
ECSP034540A (en) 2003-07-25
CN1221549C (en) 2005-10-05
EE200300171A (en) 2003-06-16
KR20030042008A (en) 2003-05-27
MEP40008A (en) 2011-02-10
AP1572A (en) 2006-02-13
ZA200302500B (en) 2004-04-22
MA25842A1 (en) 2003-07-01
UY34901A (en) 2015-02-27

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