ECSP077421A - Compuestos y composiciones como inhibidores de la actividad del receptor canabinoide 1 - Google Patents
Compuestos y composiciones como inhibidores de la actividad del receptor canabinoide 1Info
- Publication number
- ECSP077421A ECSP077421A EC2007007421A ECSP077421A ECSP077421A EC SP077421 A ECSP077421 A EC SP077421A EC 2007007421 A EC2007007421 A EC 2007007421A EC SP077421 A ECSP077421 A EC SP077421A EC SP077421 A ECSP077421 A EC SP077421A
- Authority
- EC
- Ecuador
- Prior art keywords
- compounds
- activity
- canabinoid
- compositions
- inhibitors
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D473/32—Nitrogen atom
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- C07D498/04—Ortho-condensed systems
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- Medicinal Chemistry (AREA)
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Abstract
La invención proporciona compuestos, composiciones farmacéuticas que comprenden tales compuestos, y métodos para utilizar tales compuestos con el fin de tratar o prevenir enfermedades o trastornos asociados con la actividad del Receptor Canabinoide 1 (CB1).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US62250804P | 2004-10-26 | 2004-10-26 | |
US67267005P | 2005-04-18 | 2005-04-18 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP077421A true ECSP077421A (es) | 2007-05-30 |
Family
ID=36228382
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2007007421A ECSP077421A (es) | 2004-10-26 | 2007-04-26 | Compuestos y composiciones como inhibidores de la actividad del receptor canabinoide 1 |
Country Status (19)
Country | Link |
---|---|
US (2) | US8158634B2 (es) |
EP (1) | EP1807429A4 (es) |
JP (2) | JP2008518016A (es) |
KR (1) | KR100919524B1 (es) |
CN (2) | CN101048408B (es) |
AR (1) | AR051596A1 (es) |
AU (2) | AU2005299421B2 (es) |
BR (1) | BRPI0517015A (es) |
CA (2) | CA2730374A1 (es) |
EC (1) | ECSP077421A (es) |
IL (1) | IL182527A0 (es) |
MA (1) | MA28937B1 (es) |
MX (1) | MX2007004936A (es) |
NO (1) | NO20072352L (es) |
PE (1) | PE20060599A1 (es) |
RU (1) | RU2431635C2 (es) |
TN (1) | TNSN07161A1 (es) |
TW (1) | TW200630096A (es) |
WO (1) | WO2006047516A2 (es) |
Families Citing this family (74)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA011009B1 (ru) | 2003-01-14 | 2008-12-30 | Арена Фармасьютикалз Инк. | 1,2,3-тризамещённые арильные и гетероарильные производные в качестве модуляторов метаболизма и профилактика и лечение расстройств, связанных с ним, таких как диабет и гипергликемия |
AR045697A1 (es) | 2003-07-14 | 2005-11-09 | Arena Pharm Inc | Aril y heteroaril derivados fusionados como moduladores del metabolismo y la prevencion y tratamiento de trastornos relacionados con el mismo |
WO2005074643A2 (en) * | 2004-01-30 | 2005-08-18 | Smithkline Beecham Corporation | Benzamide compounds useful as rock inhibitors |
AR051596A1 (es) * | 2004-10-26 | 2007-01-24 | Irm Llc | Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios |
GB0506147D0 (en) * | 2005-03-24 | 2005-05-04 | Merck Sharp & Dohme | Therapeutic agents |
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2005
- 2005-10-24 AR ARP050104440A patent/AR051596A1/es not_active Application Discontinuation
- 2005-10-25 PE PE2005001251A patent/PE20060599A1/es not_active Application Discontinuation
- 2005-10-25 TW TW094137369A patent/TW200630096A/zh unknown
- 2005-10-26 US US11/718,016 patent/US8158634B2/en not_active Expired - Fee Related
- 2005-10-26 MX MX2007004936A patent/MX2007004936A/es not_active Application Discontinuation
- 2005-10-26 JP JP2007539039A patent/JP2008518016A/ja not_active Withdrawn
- 2005-10-26 CA CA2730374A patent/CA2730374A1/en not_active Abandoned
- 2005-10-26 RU RU2007119449/04A patent/RU2431635C2/ru not_active IP Right Cessation
- 2005-10-26 CN CN2005800368900A patent/CN101048408B/zh not_active Expired - Fee Related
- 2005-10-26 EP EP05813001A patent/EP1807429A4/en not_active Withdrawn
- 2005-10-26 BR BRPI0517015-0A patent/BRPI0517015A/pt not_active IP Right Cessation
- 2005-10-26 AU AU2005299421A patent/AU2005299421B2/en not_active Ceased
- 2005-10-26 WO PCT/US2005/038361 patent/WO2006047516A2/en active Application Filing
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- 2005-10-26 CA CA2581225A patent/CA2581225C/en not_active Expired - Fee Related
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2007
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- 2007-04-18 MA MA29834A patent/MA28937B1/fr unknown
- 2007-04-25 TN TNP2007000161A patent/TNSN07161A1/fr unknown
- 2007-04-25 KR KR1020077009370A patent/KR100919524B1/ko not_active IP Right Cessation
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- 2007-05-07 NO NO20072352A patent/NO20072352L/no not_active Application Discontinuation
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2009
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2011
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CN101048408A (zh) | 2007-10-03 |
KR100919524B1 (ko) | 2009-10-01 |
EP1807429A2 (en) | 2007-07-18 |
RU2431635C2 (ru) | 2011-10-20 |
CA2581225A1 (en) | 2006-05-04 |
WO2006047516A2 (en) | 2006-05-04 |
MX2007004936A (es) | 2007-06-25 |
CN101048408B (zh) | 2011-07-06 |
JP2011190281A (ja) | 2011-09-29 |
IL182527A0 (en) | 2007-09-20 |
WO2006047516A3 (en) | 2006-10-12 |
AU2005299421B2 (en) | 2010-01-28 |
US20120225869A1 (en) | 2012-09-06 |
CA2730374A1 (en) | 2006-05-04 |
US20090247517A1 (en) | 2009-10-01 |
JP2008518016A (ja) | 2008-05-29 |
TNSN07161A1 (en) | 2008-11-21 |
KR20070057980A (ko) | 2007-06-07 |
AR051596A1 (es) | 2007-01-24 |
CA2581225C (en) | 2011-10-25 |
TW200630096A (en) | 2006-09-01 |
PE20060599A1 (es) | 2006-08-22 |
US8158634B2 (en) | 2012-04-17 |
NO20072352L (no) | 2007-05-31 |
AU2009251216A1 (en) | 2010-01-28 |
MA28937B1 (fr) | 2007-10-01 |
BRPI0517015A (pt) | 2008-09-30 |
AU2005299421A1 (en) | 2006-05-04 |
EP1807429A4 (en) | 2010-03-24 |
CN102241680A (zh) | 2011-11-16 |
RU2007119449A (ru) | 2008-12-10 |
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