EA201500431A1 - Соединения боронатного эфира и его фармацевтические составы - Google Patents

Соединения боронатного эфира и его фармацевтические составы

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Publication number
EA201500431A1
EA201500431A1 EA201500431A EA201500431A EA201500431A1 EA 201500431 A1 EA201500431 A1 EA 201500431A1 EA 201500431 A EA201500431 A EA 201500431A EA 201500431 A EA201500431 A EA 201500431A EA 201500431 A1 EA201500431 A1 EA 201500431A1
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EA
Eurasian Patent Office
Prior art keywords
bononate
compounds
air
pharmaceutical compositions
provides
Prior art date
Application number
EA201500431A
Other languages
English (en)
Inventor
Эрик Л. Эллиот
Абу Дж. Фердоус
Майкл Дж. Кауфман
Соня А. Комар
Дебра Л. Мазаик
Квентин Дж. Маккаббин
Пхоунг М. Нгуйен
Ваитхианатхан Паланиаппан
Рэймонд Д. Скверчински
Нобель Т. Труонг
Ксанад М. Варга
Питер Н. Заванех
Original Assignee
Милленниум Фармасьютикалз, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41061278&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201500431(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Милленниум Фармасьютикалз, Инк. filed Critical Милленниум Фармасьютикалз, Инк.
Publication of EA201500431A1 publication Critical patent/EA201500431A1/ru

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    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
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Abstract

Изобретение обеспечивает получение новых соединений, применимых в качестве ингибиторов протеасом. Изобретение также обеспечивает получение фармацевтически приемлемых рецептур с содержанием веществ, указанных в изобретении, а также обеспечивает методами использования данных рецептур при лечении различных заболеваний.
EA201500431A 2008-06-17 2009-06-16 Соединения боронатного эфира и его фармацевтические составы EA201500431A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13224408P 2008-06-17 2008-06-17
US21149909P 2009-03-31 2009-03-31

Publications (1)

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EA201500431A1 true EA201500431A1 (ru) 2015-11-30

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Application Number Title Priority Date Filing Date
EA201500431A EA201500431A1 (ru) 2008-06-17 2009-06-16 Соединения боронатного эфира и его фармацевтические составы
EA201500430A EA030685B1 (ru) 2008-06-17 2009-06-16 Способ получения соединения боронатного эфира
EA201170036A EA027346B1 (ru) 2008-06-17 2009-06-16 Соединения боронатного эфира и его фармацевтические составы
EA201500432A EA201500432A1 (ru) 2008-06-17 2009-06-16 Соединения боронатного эфира и его фармацевтические составы

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EA201500430A EA030685B1 (ru) 2008-06-17 2009-06-16 Способ получения соединения боронатного эфира
EA201170036A EA027346B1 (ru) 2008-06-17 2009-06-16 Соединения боронатного эфира и его фармацевтические составы
EA201500432A EA201500432A1 (ru) 2008-06-17 2009-06-16 Соединения боронатного эфира и его фармацевтические составы

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US (17) US20090325903A1 (ru)
EP (6) EP2318419B1 (ru)
JP (9) JP5566380B2 (ru)
KR (5) KR101704694B1 (ru)
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Families Citing this family (80)

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CN103435638A (zh) 2013-12-11
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IL234285B (en) 2018-04-30
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PH12015501193A1 (en) 2016-01-11
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KR101691093B1 (ko) 2016-12-29
ECSP14010763A (es) 2014-07-31
PH12015501192B1 (en) 2016-01-11
ZA201504133B (en) 2016-11-30
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CR20160014A (es) 2016-02-08
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MX358222B (es) 2018-08-10
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US20130165390A1 (en) 2013-06-27
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JP2014169317A (ja) 2014-09-18
US10526351B2 (en) 2020-01-07
MA32471B1 (fr) 2011-07-03
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AR072162A1 (es) 2010-08-11
US11485746B2 (en) 2022-11-01
GEP201706703B (en) 2017-07-25
EA201500432A1 (ru) 2015-11-30
US20160031913A1 (en) 2016-02-04
EP3536693A1 (en) 2019-09-11
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US20210198289A1 (en) 2021-07-01
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