EA201491530A1 - Модуляторы рецепторов эстрогенов и их применение - Google Patents

Модуляторы рецепторов эстрогенов и их применение

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Publication number
EA201491530A1
EA201491530A1 EA201491530A EA201491530A EA201491530A1 EA 201491530 A1 EA201491530 A1 EA 201491530A1 EA 201491530 A EA201491530 A EA 201491530A EA 201491530 A EA201491530 A EA 201491530A EA 201491530 A1 EA201491530 A1 EA 201491530A1
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EA
Eurasian Patent Office
Prior art keywords
estrogen receptors
modulators
application
compounds
estrogen
Prior art date
Application number
EA201491530A
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English (en)
Inventor
Николас Д. Смит
Стивен П. Говек
Мехмет Караман
Джэкэлин Д. Жулиен
Джонни Ю. Нагасава
Каренса Л. Дуглас
Селин Боннефус
Андилли Г. Лай
Original Assignee
Серагон Фармасьютикалс, Инк.
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Publication date
Application filed by Серагон Фармасьютикалс, Инк. filed Critical Серагон Фармасьютикалс, Инк.
Publication of EA201491530A1 publication Critical patent/EA201491530A1/ru

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Abstract

В настоящей заявке раскрываются соединения, представляющие собой модуляторы рецепторов эстрогенов. Также описываются фармацевтические композиции и лекарственные препараты, которые включают соединения по настоящему изобретению, а также способы применения таких модуляторов рецепторов эстрогенов, самостоятельно или в комбинации с другими соединениями, для лечения заболеваний или патологических состояний, которые опосредуются от рецепторов эстрогенов или являются зависимыми от рецепторов эстрогенов.
EA201491530A 2012-03-20 2013-03-14 Модуляторы рецепторов эстрогенов и их применение EA201491530A1 (ru)

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US201261613442P 2012-03-20 2012-03-20
PCT/US2013/031507 WO2013142266A1 (en) 2012-03-20 2013-03-14 Estrogen receptor modulators and uses thereof

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US (1) US9499538B2 (ru)
EP (1) EP2828243B1 (ru)
JP (1) JP6154887B2 (ru)
KR (1) KR20140138296A (ru)
CN (1) CN104220426B (ru)
AU (1) AU2013235499A1 (ru)
CA (1) CA2866891A1 (ru)
CO (1) CO7170179A2 (ru)
CR (1) CR20140479A (ru)
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IL (1) IL234487A0 (ru)
MX (1) MX2014011217A (ru)
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