EA200602016A1 - ПОРОШКОВЫЕ КОМПОЗИЦИИ ДЛЯ ИНГАЛЯЦИИ, СОДЕРЖАЩИЕ ЭНАНТИОМЕРНОЧИСТЫЕ β-АГОНИСТЫ - Google Patents
ПОРОШКОВЫЕ КОМПОЗИЦИИ ДЛЯ ИНГАЛЯЦИИ, СОДЕРЖАЩИЕ ЭНАНТИОМЕРНОЧИСТЫЕ β-АГОНИСТЫInfo
- Publication number
- EA200602016A1 EA200602016A1 EA200602016A EA200602016A EA200602016A1 EA 200602016 A1 EA200602016 A1 EA 200602016A1 EA 200602016 A EA200602016 A EA 200602016A EA 200602016 A EA200602016 A EA 200602016A EA 200602016 A1 EA200602016 A1 EA 200602016A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- enantiomerna
- agentists
- clean
- powder compositions
- inhalation containing
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
Abstract
В заявке описаны порошковые композиции для ингаляции, содержащие энантиомерночистые соединения общей формулы ()в которой остатки R, R, Rи Rмогут иметь указанные в формуле изобретения и описании значения, необязательно в виде их фармацевтически приемлемых кислотно-аддитивных солей, а также необязательно в сочетании с фармацевтически приемлемым вспомогательным веществом, а также описаны способ их получения и их применение в качестве лекарственных средств, прежде всего в качестве лекарственных средств для лечения заболеваний дыхательных путей.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102004024451A DE102004024451A1 (de) | 2004-05-14 | 2004-05-14 | Pulverformulierungen für die Inhalation, die Enantiomerenreine Betaagonisten enthalten |
PCT/EP2005/005078 WO2005110359A1 (de) | 2004-05-14 | 2005-05-11 | Pulverformulierungen für die inhalation, die enantiomerenreine betaagonisten enthalten |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200602016A1 true EA200602016A1 (ru) | 2007-06-29 |
EA012582B1 EA012582B1 (ru) | 2009-10-30 |
Family
ID=35058202
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200602016A EA012582B1 (ru) | 2004-05-14 | 2005-05-11 | ПОРОШКОВЫЕ КОМПОЗИЦИИ ДЛЯ ИНГАЛЯЦИИ, СОДЕРЖАЩИЕ ЭНАНТИОМЕРНОЧИСТЫЕ β-АГОНИСТЫ |
Country Status (24)
Country | Link |
---|---|
EP (1) | EP1809236B1 (ru) |
JP (1) | JP4891899B2 (ru) |
KR (1) | KR101270449B1 (ru) |
CN (1) | CN1984638A (ru) |
AR (1) | AR048899A1 (ru) |
AU (1) | AU2005244424B2 (ru) |
BR (1) | BRPI0511136A (ru) |
CA (1) | CA2565915C (ru) |
DE (1) | DE102004024451A1 (ru) |
DK (1) | DK1809236T3 (ru) |
EA (1) | EA012582B1 (ru) |
ES (1) | ES2401786T3 (ru) |
IL (1) | IL179215A (ru) |
MX (1) | MXPA06013221A (ru) |
MY (1) | MY145838A (ru) |
NO (1) | NO20065078L (ru) |
PE (1) | PE20060239A1 (ru) |
PL (1) | PL1809236T3 (ru) |
SG (1) | SG152258A1 (ru) |
TW (1) | TW200607508A (ru) |
UA (1) | UA86807C2 (ru) |
UY (1) | UY28896A1 (ru) |
WO (1) | WO2005110359A1 (ru) |
ZA (1) | ZA200607785B (ru) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102004024452A1 (de) * | 2004-05-14 | 2005-12-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Aerosolformulierung für die Inhalation von Betaagonisten |
GB0516313D0 (en) | 2005-08-08 | 2005-09-14 | Argenta Discovery Ltd | Azole derivatives and their uses |
NZ566068A (en) | 2005-08-08 | 2011-03-31 | Argenta Discovery Ltd | Bicyclo[2.2.1]hept-7-ylamine derivatives and their uses |
JP5270343B2 (ja) | 2005-08-15 | 2013-08-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ベータミメティックスの製造方法 |
US8236786B2 (en) | 2008-08-07 | 2012-08-07 | Pulmagen Therapeutics (Inflammation) Limited | Respiratory disease treatment |
US8362064B2 (en) | 2008-12-30 | 2013-01-29 | Pulmagen Theraputics (Inflammation) Limited | Sulfonamide compounds for the treatment of respiratory disorders |
WO2010150014A1 (en) | 2009-06-24 | 2010-12-29 | Pulmagen Therapeutics (Inflammation) Limited | 5r- 5 -deuterated glitazones for respiratory disease treatment |
GB0918923D0 (en) | 2009-10-28 | 2009-12-16 | Vantia Ltd | Aminothiazole derivatives |
GB0918922D0 (en) | 2009-10-28 | 2009-12-16 | Vantia Ltd | Aminopyridine derivatives |
GB0918924D0 (en) | 2009-10-28 | 2009-12-16 | Vantia Ltd | Azaindole derivatives |
WO2011098746A1 (en) | 2010-02-09 | 2011-08-18 | Pulmagen Therapeutics (Inflammation) Limited | Crystalline acid addition salts of ( 5r) -enanti0mer of pioglitazone |
GB201002224D0 (en) | 2010-02-10 | 2010-03-31 | Argenta Therapeutics Ltd | Respiratory disease treatment |
GB201002243D0 (en) | 2010-02-10 | 2010-03-31 | Argenta Therapeutics Ltd | Respiratory disease treatment |
JP2015533131A (ja) | 2012-10-09 | 2015-11-19 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 咳を治療するためのベータ2−アドレナリン受容体作動薬 |
WO2018108669A1 (en) | 2016-12-12 | 2018-06-21 | Boehringer Ingelheim International Gmbh | Nintedanib for use in methods for the treatment of interstitial lung diseases by coadministration with olodaterol |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3134590A1 (de) * | 1981-09-01 | 1983-03-10 | Boehringer Ingelheim KG, 6507 Ingelheim | Neue benzo-heterocyclen |
US4460581A (en) * | 1982-10-12 | 1984-07-17 | Boehringer Ingelheim Kg | (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones |
DE4318455A1 (de) | 1993-06-03 | 1994-12-08 | Boehringer Ingelheim Kg | Kapselhalterung |
BR0110331A (pt) * | 2000-04-27 | 2003-01-07 | Boehringer Ingelheim Pharma | Substâncias que mimetizam beta que têm uma atividade de longa duração, processos para prepará-las e o uso das mesmas como medicamentos |
GB0107106D0 (en) * | 2001-03-21 | 2001-05-09 | Boehringer Ingelheim Pharma | Powder inhaler formulations |
DE10141377A1 (de) * | 2001-08-23 | 2003-03-13 | Boehringer Ingelheim Pharma | Aufstreuverfahren zur Herstellung von Pulverformulierungen |
DE10212264A1 (de) | 2002-03-20 | 2003-10-02 | Boehringer Ingelheim Pharma | Kristallines Mikronisat, Verfahren zu dessen Herstellung und dessen Verwendung zur Herstellung eines Arzneimittels |
UA80123C2 (en) | 2002-04-09 | 2007-08-27 | Boehringer Ingelheim Pharma | Inhalation kit comprising inhalable powder of tiotropium |
DE10253282A1 (de) * | 2002-11-15 | 2004-05-27 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung |
-
2004
- 2004-05-14 DE DE102004024451A patent/DE102004024451A1/de not_active Withdrawn
-
2005
- 2005-05-11 CN CNA2005800154329A patent/CN1984638A/zh active Pending
- 2005-05-11 JP JP2007512080A patent/JP4891899B2/ja active Active
- 2005-05-11 EA EA200602016A patent/EA012582B1/ru not_active IP Right Cessation
- 2005-05-11 AU AU2005244424A patent/AU2005244424B2/en not_active Ceased
- 2005-05-11 EP EP05747562A patent/EP1809236B1/de active Active
- 2005-05-11 MX MXPA06013221A patent/MXPA06013221A/es active IP Right Grant
- 2005-05-11 UA UAA200612950A patent/UA86807C2/ru unknown
- 2005-05-11 PL PL05747562T patent/PL1809236T3/pl unknown
- 2005-05-11 ES ES05747562T patent/ES2401786T3/es active Active
- 2005-05-11 BR BRPI0511136-6A patent/BRPI0511136A/pt not_active IP Right Cessation
- 2005-05-11 CA CA2565915A patent/CA2565915C/en not_active Expired - Fee Related
- 2005-05-11 DK DK05747562.6T patent/DK1809236T3/da active
- 2005-05-11 WO PCT/EP2005/005078 patent/WO2005110359A1/de active Application Filing
- 2005-05-11 KR KR1020067026352A patent/KR101270449B1/ko not_active IP Right Cessation
- 2005-05-11 SG SG200902738-4A patent/SG152258A1/en unknown
- 2005-05-12 PE PE2005000530A patent/PE20060239A1/es not_active Application Discontinuation
- 2005-05-12 MY MYPI20052155A patent/MY145838A/en unknown
- 2005-05-12 UY UY28896A patent/UY28896A1/es not_active Application Discontinuation
- 2005-05-13 AR ARP050101958A patent/AR048899A1/es unknown
- 2005-05-13 TW TW094115490A patent/TW200607508A/zh unknown
-
2006
- 2006-09-18 ZA ZA200607785A patent/ZA200607785B/en unknown
- 2006-11-03 NO NO20065078A patent/NO20065078L/no not_active Application Discontinuation
- 2006-11-13 IL IL179215A patent/IL179215A/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
KR101270449B1 (ko) | 2013-06-04 |
PE20060239A1 (es) | 2006-03-27 |
WO2005110359A1 (de) | 2005-11-24 |
KR20070016169A (ko) | 2007-02-07 |
AU2005244424B2 (en) | 2010-12-23 |
CN1984638A (zh) | 2007-06-20 |
ZA200607785B (en) | 2008-07-30 |
UY28896A1 (es) | 2005-12-30 |
SG152258A1 (en) | 2009-05-29 |
IL179215A (en) | 2011-04-28 |
JP2007537195A (ja) | 2007-12-20 |
EP1809236B1 (de) | 2012-12-26 |
MY145838A (en) | 2012-04-30 |
IL179215A0 (en) | 2007-03-08 |
UA86807C2 (ru) | 2009-05-25 |
AR048899A1 (es) | 2006-06-07 |
DK1809236T3 (da) | 2013-02-11 |
EA012582B1 (ru) | 2009-10-30 |
PL1809236T3 (pl) | 2013-05-31 |
NO20065078L (no) | 2006-11-28 |
ES2401786T3 (es) | 2013-04-24 |
MXPA06013221A (es) | 2007-02-08 |
DE102004024451A1 (de) | 2005-12-22 |
CA2565915A1 (en) | 2005-11-24 |
CA2565915C (en) | 2013-12-10 |
TW200607508A (en) | 2006-03-01 |
JP4891899B2 (ja) | 2012-03-07 |
BRPI0511136A (pt) | 2007-11-27 |
EP1809236A1 (de) | 2007-07-25 |
AU2005244424A1 (en) | 2005-11-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ KZ KG MD TJ TM |
|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): BY |
|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): RU |