DZ3493A1 - N-(2-arylethyl)benzylamines comme antagonistes du recepteur 5-ht6 - Google Patents
N-(2-arylethyl)benzylamines comme antagonistes du recepteur 5-ht6Info
- Publication number
- DZ3493A1 DZ3493A1 DZ023493A DZ023493A DZ3493A1 DZ 3493 A1 DZ3493 A1 DZ 3493A1 DZ 023493 A DZ023493 A DZ 023493A DZ 023493 A DZ023493 A DZ 023493A DZ 3493 A1 DZ3493 A1 DZ 3493A1
- Authority
- DZ
- Algeria
- Prior art keywords
- arylethyl
- benzylamines
- receptor antagonists
- antagonists
- receptor
- Prior art date
Links
- 108091005435 5-HT6 receptors Proteins 0.000 title abstract 2
- 150000003939 benzylamines Chemical class 0.000 title 1
- 239000002464 receptor antagonist Substances 0.000 title 1
- 229940044551 receptor antagonist Drugs 0.000 title 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
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- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/64—One oxygen atom attached in position 2 or 6
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61P25/22—Anxiolytics
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- C07C211/52—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
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- C07C211/54—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to two or three six-membered aromatic rings
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- C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
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- C07C311/30—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/37—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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- C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
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- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/31—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atom of at least one of the thio groups bound to a carbon atom of a six-membered aromatic ring of the carbon skeleton
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- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
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- C07D209/82—Carbazoles; Hydrogenated carbazoles
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- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
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US27992801P | 2001-03-29 | 2001-03-29 | |
US32944901P | 2001-10-15 | 2001-10-15 | |
PCT/US2002/005115 WO2002078693A2 (fr) | 2001-03-29 | 2002-03-15 | N-(2-arylethyl)benzylamines utilisees en tant qu'antagonistes du recepteur 5-ht6 |
Publications (1)
Publication Number | Publication Date |
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DZ3493A1 true DZ3493A1 (fr) | 2002-10-10 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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DZ023493A DZ3493A1 (fr) | 2001-03-29 | 2002-03-15 | N-(2-arylethyl)benzylamines comme antagonistes du recepteur 5-ht6 |
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US (3) | US7157488B2 (fr) |
EP (1) | EP1379239B1 (fr) |
JP (1) | JP2004532209A (fr) |
KR (1) | KR100894189B1 (fr) |
CN (1) | CN1610547A (fr) |
AT (1) | ATE372768T1 (fr) |
AU (1) | AU2002303094B2 (fr) |
BR (1) | BR0208179A (fr) |
CA (1) | CA2442114C (fr) |
CY (1) | CY1110362T1 (fr) |
CZ (1) | CZ305838B6 (fr) |
DE (1) | DE60222396T2 (fr) |
DK (2) | DK1379239T3 (fr) |
DZ (1) | DZ3493A1 (fr) |
EA (1) | EA007493B1 (fr) |
ES (2) | ES2292758T3 (fr) |
HK (1) | HK1061649A1 (fr) |
HR (1) | HRP20030771B1 (fr) |
HU (1) | HU230322B1 (fr) |
IL (3) | IL157651A0 (fr) |
MX (1) | MXPA03008726A (fr) |
NO (1) | NO326160B1 (fr) |
NZ (1) | NZ527815A (fr) |
PL (1) | PL220721B1 (fr) |
PT (2) | PT1859798E (fr) |
SI (1) | SI1859798T1 (fr) |
SK (1) | SK287463B6 (fr) |
WO (1) | WO2002078693A2 (fr) |
ZA (1) | ZA200306795B (fr) |
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- 2002-03-15 CA CA2442114A patent/CA2442114C/fr not_active Expired - Lifetime
- 2002-03-15 AT AT02731094T patent/ATE372768T1/de active
- 2002-03-15 EA EA200301073A patent/EA007493B1/ru not_active IP Right Cessation
- 2002-03-15 US US10/472,741 patent/US7157488B2/en not_active Expired - Lifetime
- 2002-03-15 SK SK1205-2003A patent/SK287463B6/sk unknown
- 2002-03-15 WO PCT/US2002/005115 patent/WO2002078693A2/fr active IP Right Grant
- 2002-03-15 BR BR0208179-2A patent/BR0208179A/pt not_active Application Discontinuation
- 2002-03-15 HU HU0303651A patent/HU230322B1/hu unknown
- 2002-03-15 KR KR1020037012694A patent/KR100894189B1/ko active IP Right Grant
- 2002-03-15 CN CNA028105435A patent/CN1610547A/zh active Pending
- 2002-03-15 IL IL15765102A patent/IL157651A0/xx unknown
- 2002-03-15 DZ DZ023493A patent/DZ3493A1/fr active
- 2002-03-15 JP JP2002576959A patent/JP2004532209A/ja active Pending
- 2002-03-15 DK DK02731094T patent/DK1379239T3/da active
- 2002-03-15 DE DE60222396T patent/DE60222396T2/de not_active Expired - Lifetime
- 2002-03-15 PT PT02731094T patent/PT1379239E/pt unknown
- 2002-03-15 EP EP02731094A patent/EP1379239B1/fr not_active Expired - Lifetime
- 2002-03-15 NZ NZ527815A patent/NZ527815A/en not_active IP Right Cessation
- 2002-03-15 DK DK07015058.6T patent/DK1859798T3/en active
- 2002-03-15 AU AU2002303094A patent/AU2002303094B2/en not_active Expired
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2003
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- 2003-08-29 ZA ZA2003/06795A patent/ZA200306795B/en unknown
- 2003-09-24 HR HR20030771A patent/HRP20030771B1/xx not_active IP Right Cessation
- 2003-09-25 NO NO20034289A patent/NO326160B1/no not_active IP Right Cessation
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2004
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2006
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2007
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2009
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