SG11201704523WA - A process for the manufacture of idalopirdine - Google Patents

A process for the manufacture of idalopirdine

Info

Publication number: SG11201704523WA
Authority: SG; Singapore
Prior art keywords: idalopirdine; manufacture
Prior art date: 2014-12-12

Application number

SG11201704523WA

Inventor

Mikkel Fog Jacobsen

Ole Nielsen

Original Assignee

H Lundbeck As

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2014-12-12

Filing date

2015-12-10

Publication date

2017-07-28

2015-12-10 Application filed by H Lundbeck As filed Critical H Lundbeck As

2017-07-28 Publication of SG11201704523WA publication Critical patent/SG11201704523WA/en

Links

YBAWYTYNMZWMMJ-UHFFFAOYSA-N 2-(6-fluoro-1h-indol-3-yl)-n-[[3-(2,2,3,3-tetrafluoropropoxy)phenyl]methyl]ethanamine Chemical compound FC(F)C(F)(F)COC1=CC=CC(CNCCC=2C3=CC=C(F)C=C3NC=2)=C1 YBAWYTYNMZWMMJ-UHFFFAOYSA-N 0.000 title 1
229950005109 idalopirdine Drugs 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
238000000034 method Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines

SG11201704523WA 2014-12-12 2015-12-10 A process for the manufacture of idalopirdine SG11201704523WA (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DK201400721		2014-12-12
PCT/EP2015/079209 WO2016091997A1 (en)	2014-12-12	2015-12-10	A process for the manufacture of idalopirdine

Publications (1)

Publication Number	Publication Date
SG11201704523WA true SG11201704523WA (en)	2017-07-28

Family

ID=55077474

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SG11201704523WA SG11201704523WA (en)	2014-12-12	2015-12-10	A process for the manufacture of idalopirdine

Country Status (5)

Country	Link
US (1)	US20160168089A1 (en)
AR (1)	AR102980A1 (en)
SG (1)	SG11201704523WA (en)
TW (1)	TW201630881A (en)
WO (1)	WO2016091997A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT3231793T (en)	2014-12-12	2020-05-06	Japan Tobacco Inc	Dihydropyrimidine-2-one compounds and medicinal uses thereof
US9975850B2 (en)	2016-04-08	2018-05-22	H. Lundbeck A/S	Process for the manufacture of idalopirdine via hydrogenation of an imine
WO2018013686A1 (en) *	2016-07-12	2018-01-18	Concert Pharmaceuticals, Inc.	Deuterated idalopirdine
EP3760616A4 (en)	2018-02-28	2021-11-03	Japan Tobacco Inc.	4-methyldihydropyrimidinone compound and medicinal use thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3042685A (en) *		1962-07-03		Process of making g-fluoro tryptamine
EP0807631B1 (en) *	1996-05-15	2003-03-12	Sankyo Company Limited	Tricyclic compounds having fungicidal activity, their preparation and their use
SI1859798T1 (en)	2001-03-29	2016-07-29	Eli Lilly And Company	N-(2-arylethyl) benzylamines as antagonists of the 5-ht6 receptor
US7022645B2 (en) *	2003-08-04	2006-04-04	Catalytic Distillation Technologies	Ni hydrogenation catalysts, manufacture and use
AR065804A1 (en) *	2007-03-23	2009-07-01	Smithkline Beecham Corp	COMPOSITE OF INDOL CARBOXAMIDE, PHARMACEUTICAL COMPOSITION THAT UNDERSTANDS IT AND USE OF THIS COMPOUND TO PREPARE A MEDICINAL PRODUCT
WO2008130553A1 (en) *	2007-04-16	2008-10-30	Mallinckrodt Inc.	Novel opiate reduction utilizing catalytic hydrogen transfer reaction
TW201139370A (en)	2009-12-23	2011-11-16	Lundbeck & Co As H	Processes for the manufacture of a pharmaceutically active agent

2015
- 2015-12-10 WO PCT/EP2015/079209 patent/WO2016091997A1/en active Application Filing
- 2015-12-10 TW TW104141485A patent/TW201630881A/en unknown
- 2015-12-10 US US14/965,308 patent/US20160168089A1/en not_active Abandoned
- 2015-12-10 SG SG11201704523WA patent/SG11201704523WA/en unknown
- 2015-12-11 AR ARP150104048A patent/AR102980A1/en unknown

Also Published As

Publication number	Publication date
WO2016091997A1 (en)	2016-06-16
US20160168089A1 (en)	2016-06-16
TW201630881A (en)	2016-09-01
AR102980A1 (en)	2017-04-05

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