DK260483D0 - Fremgangsmade til fremstilling af pyrrolderivater - Google Patents

Fremgangsmade til fremstilling af pyrrolderivater

Info

Publication number
DK260483D0
DK260483D0 DK2604/83A DK260483A DK260483D0 DK 260483 D0 DK260483 D0 DK 260483D0 DK 2604/83 A DK2604/83 A DK 2604/83A DK 260483 A DK260483 A DK 260483A DK 260483 D0 DK260483 D0 DK 260483D0
Authority
DK
Denmark
Prior art keywords
sub
pyrol
procedure
preparation
hydrogen
Prior art date
Application number
DK2604/83A
Other languages
English (en)
Other versions
DK260483A (da
Inventor
Joseph Martin Muchowski
Robert James Greenhouse
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of DK260483D0 publication Critical patent/DK260483D0/da
Publication of DK260483A publication Critical patent/DK260483A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK260483A 1982-06-08 1983-06-07 Fremgangsmaade til fremstilling af pyrrolderivater DK260483A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/386,174 US4612325A (en) 1982-06-08 1982-06-08 5-Aroyl-6-alkylthio-1,2-dihydro-3H-pyrrolo(1,2-A)pyrrole-1-carboxylic acids and use thereof as analgesics and anti-inflammatories

Publications (2)

Publication Number Publication Date
DK260483D0 true DK260483D0 (da) 1983-06-07
DK260483A DK260483A (da) 1983-12-09

Family

ID=23524483

Family Applications (1)

Application Number Title Priority Date Filing Date
DK260483A DK260483A (da) 1982-06-08 1983-06-07 Fremgangsmaade til fremstilling af pyrrolderivater

Country Status (16)

Country Link
US (1) US4612325A (da)
EP (1) EP0096583B1 (da)
JP (1) JPS595190A (da)
KR (1) KR880000393B1 (da)
AT (1) ATE29497T1 (da)
AU (1) AU556295B2 (da)
CA (1) CA1200244A (da)
DE (1) DE3373474D1 (da)
DK (1) DK260483A (da)
ES (4) ES523063A0 (da)
FI (1) FI77245C (da)
HU (1) HU190106B (da)
IL (1) IL68909A (da)
NO (1) NO162386B (da)
NZ (1) NZ204487A (da)
ZA (1) ZA834137B (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4560699A (en) * 1983-01-17 1985-12-24 Syntex (U.S.A.) Inc. 5-(4-Vinylbenzoyl)-1,2-dihydro-3H-pyrrolo-[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof and use as analgesics and anti-inflammatories
JPH0739418B2 (ja) * 1987-09-10 1995-05-01 久光製薬株式会社 新規な３−アロイル−６，７−ジヒドロ−５Ｈ−ピロロ〔１，２−ｃ〕イミダゾール−７−カルボン酸誘導体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4097579A (en) * 1977-03-31 1978-06-27 Syntex (U.S.A.) Inc. 5-(2-Pyrroyl)-1,2-dihydro-3H-pyrrolo 1,2-a!pyrrole-1-carboxylic acid derivatives and process for the production thereof
US4232038A (en) * 1979-08-31 1980-11-04 Syntex (U.S.A.) Inc. 5-Alkylsulfinylbenzoyl- and 5-alkylsulfonylbenzoyl-1,2-dihydro-3H-pyrrolo[1,]pyrrole-1-carboxylic acids
US4344943A (en) * 1980-06-09 1982-08-17 Syntex (U.S.A.) Inc. 6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) * 1980-11-21 1982-10-12 Syntex (U.S.A.) Inc. Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) * 1982-06-10 1985-04-16 Merck & Co., Inc. 5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents

Also Published As

Publication number Publication date
NZ204487A (en) 1986-06-11
FI77245C (fi) 1989-02-10
NO832053L (no) 1983-12-09
CA1200244A (en) 1986-02-04
ES537694A0 (es) 1985-10-16
IL68909A (en) 1987-02-27
AU1546483A (en) 1983-12-15
IL68909A0 (en) 1983-10-31
FI832045L (fi) 1983-12-09
EP0096583A2 (en) 1983-12-21
ES8600294A1 (es) 1985-10-16
US4612325A (en) 1986-09-16
NO162386B (no) 1989-09-11
FI832045A0 (fi) 1983-06-07
KR880000393B1 (ko) 1988-03-21
HU190106B (en) 1986-08-28
ES537696A0 (es) 1985-10-16
ATE29497T1 (de) 1987-09-15
JPS595190A (ja) 1984-01-12
ES537695A0 (es) 1985-10-16
ES8600296A1 (es) 1985-10-16
ZA834137B (en) 1985-01-30
ES8502999A1 (es) 1985-02-16
ES8600295A1 (es) 1985-10-16
FI77245B (fi) 1988-10-31
DK260483A (da) 1983-12-09
DE3373474D1 (en) 1987-10-15
AU556295B2 (en) 1986-10-30
ES523063A0 (es) 1985-02-16
EP0096583A3 (en) 1985-05-02
KR840005144A (ko) 1984-11-03
EP0096583B1 (en) 1987-09-09

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment