DK2038288T3 - 4-amino-3-(azolylphenoxymethyl)thieno[3,2]pyridin-7-carboxylsyrederivater - Google Patents

4-amino-3-(azolylphenoxymethyl)thieno[3,2]pyridin-7-carboxylsyrederivater

Info

Publication number
DK2038288T3
DK2038288T3 DK07730300.6T DK07730300T DK2038288T3 DK 2038288 T3 DK2038288 T3 DK 2038288T3 DK 07730300 T DK07730300 T DK 07730300T DK 2038288 T3 DK2038288 T3 DK 2038288T3
Authority
DK
Denmark
Prior art keywords
azolylphenoxymethyl
thieno
pyridine
amino
carboxylic acid
Prior art date
Application number
DK07730300.6T
Other languages
English (en)
Inventor
Yi Chen
Kin-Chun Thomas Luk
Pamela Loreen Rossman
Sung-Sau So
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of DK2038288T3 publication Critical patent/DK2038288T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Materials For Medical Uses (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
DK07730300.6T 2006-06-29 2007-06-22 4-amino-3-(azolylphenoxymethyl)thieno[3,2]pyridin-7-carboxylsyrederivater DK2038288T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81761606P 2006-06-29 2006-06-29
PCT/EP2007/056241 WO2008000697A1 (en) 2006-06-29 2007-06-22 Novel 4-amino-3-(-azolyl-phenoxymethyl)-thieno[3,2]pyridine-7-carboxylic acid derivatives

Publications (1)

Publication Number Publication Date
DK2038288T3 true DK2038288T3 (da) 2011-01-03

Family

ID=38514272

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07730300.6T DK2038288T3 (da) 2006-06-29 2007-06-22 4-amino-3-(azolylphenoxymethyl)thieno[3,2]pyridin-7-carboxylsyrederivater

Country Status (16)

Country Link
US (1) US7932390B2 (da)
EP (1) EP2038288B1 (da)
JP (1) JP4933617B2 (da)
KR (1) KR101143286B1 (da)
CN (1) CN101479278B (da)
AT (1) ATE489391T1 (da)
BR (1) BRPI0713041A8 (da)
CA (1) CA2655398C (da)
DE (1) DE602007010779D1 (da)
DK (1) DK2038288T3 (da)
ES (1) ES2354637T3 (da)
IL (1) IL195897A (da)
MX (1) MX2008016068A (da)
PL (1) PL2038288T3 (da)
PT (1) PT2038288E (da)
WO (1) WO2008000697A1 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9540322B2 (en) 2008-08-18 2017-01-10 Yale University MIF modulators
CN102884060B (zh) * 2010-03-24 2019-07-19 阿米泰克治疗方案公司 用于抑制激酶的杂环化合物

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2732970B1 (fr) 1995-04-14 1997-05-16 Hoechst Schering Agrevo Sa Nouveaux derives de l'acide beta-methoxy acrylique, leur procede de preparation et leur application comme pesticides
US6232320B1 (en) 1998-06-04 2001-05-15 Abbott Laboratories Cell adhesion-inhibiting antiinflammatory compounds
UA60365C2 (uk) 1998-06-04 2003-10-15 Пфайзер Продактс Інк. Похідні ізотіазолу, спосіб їх одержання, фармацевтична композиція та спосіб лікування гіперпроліферативного захворювання у ссавця
HN2000000051A (es) 1999-05-19 2001-02-02 Pfizer Prod Inc Derivados heterociclicos utiles como agentes anticancerosos
OA12532A (en) 2000-11-28 2006-06-02 Pfizer Prod Inc Salts of a isothiazole-4-carboxamide and their useas anti-hyperproliferation agents.
CA2480638C (en) 2002-03-29 2013-02-12 Chiron Corporation Substituted benzazoles and use thereof as raf kinase inhibitors
WO2004041285A1 (en) 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
US7592352B2 (en) 2003-05-06 2009-09-22 Smithkline Beecham Corporation Substituted thieno and furo-pyridines
US20050026944A1 (en) 2003-07-24 2005-02-03 Patrick Betschmann Thienopyridine and furopyridine kinase inhibitors
US20050020619A1 (en) 2003-07-24 2005-01-27 Patrick Betschmann Thienopyridine kinase inhibitors
US7202363B2 (en) 2003-07-24 2007-04-10 Abbott Laboratories Thienopyridine and furopyridine kinase inhibitors
US7119102B2 (en) 2003-12-05 2006-10-10 Boehringer Ingelheim Pharmaceuticals, Inc. Substituted 3-amino-thieno[2,3-b]pyridine-2-carboxylic acid amide compounds and processes for preparing and their uses
US20050256154A1 (en) 2004-05-04 2005-11-17 Kin-Chun Luk 4-Amino-thieno[3,2-c]pyridine-7-carboxylic acid amides

Also Published As

Publication number Publication date
BRPI0713041A8 (pt) 2019-01-15
US7932390B2 (en) 2011-04-26
BRPI0713041A2 (pt) 2012-04-17
CN101479278B (zh) 2011-12-07
EP2038288B1 (en) 2010-11-24
JP4933617B2 (ja) 2012-05-16
KR20090021195A (ko) 2009-02-27
ATE489391T1 (de) 2010-12-15
CA2655398C (en) 2014-07-29
ES2354637T3 (es) 2011-03-16
MX2008016068A (es) 2009-01-15
US20080009515A1 (en) 2008-01-10
DE602007010779D1 (en) 2011-01-05
CA2655398A1 (en) 2008-01-03
IL195897A0 (en) 2009-09-01
IL195897A (en) 2016-04-21
AU2007263770A1 (en) 2008-01-03
JP2009541424A (ja) 2009-11-26
WO2008000697A1 (en) 2008-01-03
PL2038288T3 (pl) 2011-05-31
CN101479278A (zh) 2009-07-08
EP2038288A1 (en) 2009-03-25
KR101143286B1 (ko) 2012-05-24
PT2038288E (pt) 2011-01-12

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