DK1943243T3 - Kinase-inhibitorer - Google Patents

Kinase-inhibitorer

Info

Publication number
DK1943243T3
DK1943243T3 DK06826650.1T DK06826650T DK1943243T3 DK 1943243 T3 DK1943243 T3 DK 1943243T3 DK 06826650 T DK06826650 T DK 06826650T DK 1943243 T3 DK1943243 T3 DK 1943243T3
Authority
DK
Denmark
Prior art keywords
kinase inhibitors
kinase
inhibitors
Prior art date
Application number
DK06826650.1T
Other languages
English (en)
Inventor
Jolie Anne Bastian
De Blas Jesus Andres Blas
Dios Alfonso De
Kevin John Hudziak
Tiechao Li
Mary Margaret Mader
Michael Ray Myers
Mark Andrew Pobanz
Chuan Shih
Boyu Zhong
De Uralde-Garmendia Beatriz Lopez
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43298635&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1943243(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK1943243T3 publication Critical patent/DK1943243T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
DK06826650.1T 2005-10-28 2006-10-25 Kinase-inhibitorer DK1943243T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US73160405P 2005-10-28 2005-10-28
EP06380151 2006-06-02
US82196306P 2006-08-10 2006-08-10
PCT/US2006/041644 WO2007053394A1 (en) 2005-10-28 2006-10-25 Kinase inhibitors

Publications (1)

Publication Number Publication Date
DK1943243T3 true DK1943243T3 (da) 2011-03-07

Family

ID=43298635

Family Applications (1)

Application Number Title Priority Date Filing Date
DK06826650.1T DK1943243T3 (da) 2005-10-28 2006-10-25 Kinase-inhibitorer

Country Status (19)

Country Link
US (1) US7652015B2 (da)
EP (1) EP1943243B1 (da)
KR (1) KR101004156B1 (da)
AR (1) AR056582A1 (da)
AT (1) ATE493403T1 (da)
AU (1) AU2006309044B2 (da)
BR (1) BRPI0616901A2 (da)
CA (1) CA2627673A1 (da)
DK (1) DK1943243T3 (da)
DO (1) DOP2006000234A (da)
EA (1) EA015189B1 (da)
PE (1) PE20070795A1 (da)
PL (1) PL1943243T3 (da)
PT (1) PT1943243E (da)
RS (1) RS51949B (da)
SI (1) SI1943243T1 (da)
TN (1) TNSN08191A1 (da)
TW (1) TWI325423B (da)
WO (1) WO2007053394A1 (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0905955D0 (en) 2009-04-06 2009-05-20 Respivert Ltd Novel compounds
JP5787977B2 (ja) 2010-04-08 2015-09-30 レスピバート・リミテツド P38mapキナーゼ阻害剤
WO2011158044A2 (en) 2010-06-17 2011-12-22 Respivert Limited Respiratory formulations and compounds for use therein
CA2842976A1 (en) 2011-07-26 2013-01-31 Grunenthal Gmbh Substituted bicyclic aromatic carboxamide and urea derivatives as vanilloid receptor ligands
US20150210722A1 (en) 2012-08-29 2015-07-30 Respivert Limited Kinase inhibitors
WO2014033447A2 (en) 2012-08-29 2014-03-06 Respivert Limited Kinase inhibitors
EP2890701B1 (en) 2012-08-29 2017-03-29 Respivert Limited Kinase inhibitors
EP2925742B1 (en) 2012-11-16 2016-10-26 Respivert Limited Kinase inhibitors
WO2014162121A1 (en) 2013-04-02 2014-10-09 Topivert Pharma Limited Kinase inhibitors based upon n-alkyl pyrazoles
EP2981535B8 (en) 2013-04-02 2021-03-10 Oxular Acquisitions Limited Urea derivatives useful as kinase inhibitors
WO2015092423A1 (en) 2013-12-20 2015-06-25 Respivert Limited Urea derivatives useful as kinase inhibitors
HUE060660T2 (hu) 2014-03-07 2023-04-28 Biocryst Pharm Inc Szubsztituált pirazolok mint humán plazma kallikrein-gátlók
MA40775A (fr) 2014-10-01 2017-08-08 Respivert Ltd Dérivé d'acide 4-(4-(4-phényluréido-naphtalén -1-yl) oxy-pyridin-2-yl) amino-benzoïque utilisé en tant qu'inhibiteur de la kinase p38
CA3015978A1 (en) 2016-04-06 2017-10-12 Topivert Pharma Limited Kinase inhibitors
PT3691620T (pt) 2017-10-05 2022-10-06 Fulcrum Therapeutics Inc Os inibidores da quinase p38 reduzem a expressão de dux4 e genes a jusante para o tratamento de fshd
US10342786B2 (en) 2017-10-05 2019-07-09 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD
LT3700902T (lt) 2017-10-27 2023-06-26 Boehringer Ingelheim International Gmbh Trpc6 inhibitoriai

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL136768A0 (en) * 1997-12-22 2001-06-14 Bayer Ag INHIBITION OF p38 KINASE ACTIVITY USING ARYL AND HETEROARYL SUBSTITUTED HETEROCYCLIC UREAS
SI1761520T1 (sl) * 2004-06-23 2008-10-31 Lilly Co Eli Inhibitorji kinaze

Also Published As

Publication number Publication date
TWI325423B (en) 2010-06-01
AU2006309044A1 (en) 2007-05-10
EP1943243B1 (en) 2010-12-29
EP1943243A1 (en) 2008-07-16
AU2006309044B2 (en) 2011-10-13
US20080269244A1 (en) 2008-10-30
KR101004156B1 (ko) 2010-12-27
AR056582A1 (es) 2007-10-10
RS51949B (en) 2012-02-29
DOP2006000234A (es) 2007-05-31
SI1943243T1 (sl) 2011-04-29
TNSN08191A1 (en) 2009-10-30
EA015189B1 (ru) 2011-06-30
CA2627673A1 (en) 2007-05-10
ATE493403T1 (de) 2011-01-15
US7652015B2 (en) 2010-01-26
PE20070795A1 (es) 2007-08-24
BRPI0616901A2 (pt) 2011-07-05
KR20080053394A (ko) 2008-06-12
EA200801199A1 (ru) 2008-08-29
PL1943243T3 (pl) 2011-05-31
WO2007053394A1 (en) 2007-05-10
PT1943243E (pt) 2011-01-11
TW200800184A (en) 2008-01-01

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