DK1819670T3 - 12-Aryl-prostaglandinanaloger - Google Patents

12-Aryl-prostaglandinanaloger

Info

Publication number
DK1819670T3
DK1819670T3 DK05853429.8T DK05853429T DK1819670T3 DK 1819670 T3 DK1819670 T3 DK 1819670T3 DK 05853429 T DK05853429 T DK 05853429T DK 1819670 T3 DK1819670 T3 DK 1819670T3
Authority
DK
Denmark
Prior art keywords
aryl
prostaglandin analogues
prostaglandin
analogues
Prior art date
Application number
DK05853429.8T
Other languages
English (en)
Inventor
Yariv Donde
Jeremiah H Nguyen
Original Assignee
Allergan Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan Inc filed Critical Allergan Inc
Application granted granted Critical
Publication of DK1819670T3 publication Critical patent/DK1819670T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/42—Unsaturated compounds containing hydroxy or O-metal groups
    • C07C59/56—Unsaturated compounds containing hydroxy or O-metal groups containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/90—Unsaturated compounds containing keto groups containing singly bound oxygen-containing groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/04—Systems containing only non-condensed rings with a four-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
DK05853429.8T 2004-12-10 2005-12-08 12-Aryl-prostaglandinanaloger DK1819670T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11/009,298 US7091231B2 (en) 2004-12-10 2004-12-10 12-Aryl prostaglandin analogs
PCT/US2005/044501 WO2006063179A1 (en) 2004-12-10 2005-12-08 12-aryl prostaglandin analogs

Publications (1)

Publication Number Publication Date
DK1819670T3 true DK1819670T3 (da) 2012-09-17

Family

ID=36578246

Family Applications (1)

Application Number Title Priority Date Filing Date
DK05853429.8T DK1819670T3 (da) 2004-12-10 2005-12-08 12-Aryl-prostaglandinanaloger

Country Status (21)

Country Link
US (3) US7091231B2 (da)
EP (1) EP1819670B1 (da)
JP (1) JP5342142B2 (da)
KR (1) KR101367553B1 (da)
CN (1) CN101107225B (da)
AR (1) AR052264A1 (da)
AU (1) AU2005314000B2 (da)
BR (1) BRPI0518642A2 (da)
CA (1) CA2589864C (da)
DK (1) DK1819670T3 (da)
ES (1) ES2394838T3 (da)
HK (1) HK1114832A1 (da)
IL (1) IL183360A (da)
MX (1) MX2007006690A (da)
NO (1) NO20072662L (da)
NZ (1) NZ555352A (da)
PL (1) PL216197B1 (da)
RU (1) RU2439055C2 (da)
TW (1) TWI392666B (da)
WO (1) WO2006063179A1 (da)
ZA (1) ZA200704087B (da)

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US7993634B2 (en) 2004-04-30 2011-08-09 Allergan, Inc. Oil-in-oil emulsified polymeric implants containing a hypotensive lipid and related methods
US7799336B2 (en) 2004-04-30 2010-09-21 Allergan, Inc. Hypotensive lipid-containing biodegradable intraocular implants and related methods
US9498457B2 (en) 2004-04-30 2016-11-22 Allergan, Inc. Hypotensive prostamide-containing biodegradable intraocular implants and related implants
US7674786B2 (en) * 2005-05-06 2010-03-09 Allergan, Inc. Therapeutic β-lactams
WO2007005176A1 (en) * 2005-06-29 2007-01-11 Allergan, Inc. Pyrrolidinones for the treatment of glaucoma and ocular hypertension
US7585895B2 (en) * 2005-12-06 2009-09-08 Allergan, Inc. Therapeutic substituted cyclopentanes
US7427685B2 (en) * 2005-12-06 2008-09-23 Allergan, Inc. Therapeutic substituted cyclopentanes
US7592364B2 (en) * 2006-02-28 2009-09-22 Allergan, Inc. Substituted gamma lactams as therapeutic agents
ES2573323T3 (es) 2006-03-29 2016-06-07 Dignity Health Estímulo eléctrico de microrráfaga de nervios craneales para el tratamiento de afecciones médicas
US20090016981A1 (en) * 2006-05-03 2009-01-15 Allergan, Inc. Therapeutic compounds
US7491844B2 (en) * 2006-05-04 2009-02-17 Allergan, Inc. Therapeutic cyclopentane derivatives
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US20090062361A1 (en) * 2007-08-30 2009-03-05 Allergan, Inc. Therapeutic hydantoins
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US7956051B2 (en) * 2008-01-24 2011-06-07 Allergan, Inc. Therapeutic amides and related compounds
US8455547B2 (en) 2008-02-05 2013-06-04 Allergan, Inc. Substituted cyclopentanes having prostaglandin activity
US8633310B2 (en) * 2008-02-19 2014-01-21 Allergan, Inc. Therapeutic substituted lactams
US8440819B2 (en) * 2008-02-22 2013-05-14 Allergan, Inc. Therapeutic substituted beta-lactams
US8487091B2 (en) * 2008-03-04 2013-07-16 Allergan, Inc. Substituted cyclopentanes having prostaglandin activity
US7964596B2 (en) 2008-03-07 2011-06-21 Allergan, Inc. Therapeutic compounds
US20090233921A1 (en) * 2008-03-11 2009-09-17 Allergan, Inc. Therapeutic cyclopentane derivatives
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US7705001B2 (en) * 2008-03-18 2010-04-27 Allergan, Inc Therapeutic substituted gamma lactams
US7956055B2 (en) * 2008-03-25 2011-06-07 Allergan, Inc. Substituted gamma lactams as therapeutic agents
US20110152328A1 (en) * 2008-04-16 2011-06-23 Whitcup Scott M Combination Therapy For Glaucoma
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US8952051B2 (en) * 2009-11-05 2015-02-10 Allergan, Inc. Ophthalmic formulations containing substituted gamma lactams and methods for use thereof
US9090584B2 (en) * 2010-01-26 2015-07-28 Allergan, Inc. Therapeutic agents for treatment of ocular hypertension
US8299068B2 (en) 2010-01-29 2012-10-30 Allergan, Inc. Therapeutically active cyclopentanes
KR102304111B1 (ko) * 2012-08-27 2021-09-23 알레간 인코포레이티드 베타-클로로시클로펜탄의 친수성 에스테르 전구약물의 이용에 의한 감소된 중심 각막 비후
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Also Published As

Publication number Publication date
PL383422A1 (pl) 2008-03-17
IL183360A (en) 2010-12-30
CA2589864C (en) 2015-02-03
PL216197B1 (pl) 2014-03-31
AU2005314000B2 (en) 2012-06-14
RU2007120520A (ru) 2009-01-20
US8044092B2 (en) 2011-10-25
KR101367553B1 (ko) 2014-03-14
KR20070086001A (ko) 2007-08-27
AR052264A1 (es) 2007-03-07
TWI392666B (zh) 2013-04-11
RU2439055C2 (ru) 2012-01-10
NZ555352A (en) 2011-01-28
CN101107225A (zh) 2008-01-16
US7799821B2 (en) 2010-09-21
NO20072662L (no) 2007-09-04
TW200633966A (en) 2006-10-01
ZA200704087B (en) 2008-09-25
AU2005314000A1 (en) 2006-06-15
JP2008523088A (ja) 2008-07-03
IL183360A0 (en) 2007-09-20
ES2394838T3 (es) 2013-02-06
HK1114832A1 (en) 2008-11-14
CN101107225B (zh) 2012-11-28
JP5342142B2 (ja) 2013-11-13
EP1819670A1 (en) 2007-08-22
MX2007006690A (es) 2007-08-14
BRPI0518642A2 (pt) 2008-12-02
WO2006063179A1 (en) 2006-06-15
CA2589864A1 (en) 2006-06-15
US20060205800A1 (en) 2006-09-14
US7091231B2 (en) 2006-08-15
US20100317872A1 (en) 2010-12-16
EP1819670B1 (en) 2012-08-08
US20060148894A1 (en) 2006-07-06

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