DK1592699T3 - Avermectin og avermectin-monosaccharidderivater substitueret i 4"- eller 4' -positionen, hvilke forbindelser har pesticidegenskaber - Google Patents

Avermectin og avermectin-monosaccharidderivater substitueret i 4"- eller 4' -positionen, hvilke forbindelser har pesticidegenskaber

Info

Publication number
DK1592699T3
DK1592699T3 DK04706638T DK04706638T DK1592699T3 DK 1592699 T3 DK1592699 T3 DK 1592699T3 DK 04706638 T DK04706638 T DK 04706638T DK 04706638 T DK04706638 T DK 04706638T DK 1592699 T3 DK1592699 T3 DK 1592699T3
Authority
DK
Denmark
Prior art keywords
avermectin
compounds
derivatives substituted
monosaccharide derivatives
pesticide properties
Prior art date
Application number
DK04706638T
Other languages
Danish (da)
English (en)
Inventor
Thomas Pitterna
Laura Quaranta
Pierre Jung
Kessabi Fiona Murphy
Peter Maienfisch
Jerome Cassayre
Original Assignee
Merial Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Ltd filed Critical Merial Ltd
Application granted granted Critical
Publication of DK1592699T3 publication Critical patent/DK1592699T3/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Pest Control & Pesticides (AREA)
  • Molecular Biology (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DK04706638T 2003-01-31 2004-01-30 Avermectin og avermectin-monosaccharidderivater substitueret i 4"- eller 4' -positionen, hvilke forbindelser har pesticidegenskaber DK1592699T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0302308.2A GB0302308D0 (en) 2003-01-31 2003-01-31 Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
PCT/EP2004/000890 WO2004067543A1 (en) 2003-01-31 2004-01-30 Avermectin and avermectin monosaccharide derivatives substituted in the 4”- or 4’-position having pesticidal properties

Publications (1)

Publication Number Publication Date
DK1592699T3 true DK1592699T3 (da) 2007-05-07

Family

ID=9952239

Family Applications (1)

Application Number Title Priority Date Filing Date
DK04706638T DK1592699T3 (da) 2003-01-31 2004-01-30 Avermectin og avermectin-monosaccharidderivater substitueret i 4"- eller 4' -positionen, hvilke forbindelser har pesticidegenskaber

Country Status (15)

Country Link
US (1) US7678740B2 (de)
EP (1) EP1592699B1 (de)
JP (1) JP2006516584A (de)
AR (1) AR042966A1 (de)
AT (1) ATE349457T1 (de)
CL (1) CL2004000148A1 (de)
CY (1) CY1108005T1 (de)
DE (1) DE602004003907T2 (de)
DK (1) DK1592699T3 (de)
ES (1) ES2280022T3 (de)
GB (1) GB0302308D0 (de)
PT (1) PT1592699E (de)
SI (1) SI1592699T1 (de)
TW (1) TW200510443A (de)
WO (1) WO2004067543A1 (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) * 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
GB0129267D0 (en) * 2001-12-06 2002-01-23 Syngenta Ltd Fungicides
TW200407330A (en) * 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0227554D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227558D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227556D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227555D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0302310D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0312863D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0312864D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively
AR081187A1 (es) 2010-05-12 2012-07-04 Merial Ltd Formulaciones inyectables parasiticidas de levamisol y lactonas macrociclicas. metodo de preparacion. metodo de tratamiento.
NZ627856A (en) 2010-12-07 2016-03-31 Merial Inc Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
CN109485683A (zh) * 2018-11-27 2019-03-19 齐鲁晟华制药有限公司 一种含氟系列阿维菌素衍生物及其制备方法
CN113150053A (zh) * 2020-01-22 2021-07-23 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用
CN115403644B (zh) * 2022-09-01 2024-04-05 石家庄学院 一种烟碱甲氨基或氨基阿维菌素B1a化合物及其制备方法和应用

Family Cites Families (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4206205A (en) 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4203976A (en) 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4427663A (en) 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4622313A (en) 1985-08-01 1986-11-11 Merck & Co., Inc. O-sulfate derivatives of avermectins and milbemycins having improved water solubility
US4662313A (en) * 1985-10-23 1987-05-05 Xerox Corporation Image density controller
US4886828A (en) 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
US4831016A (en) 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4874749A (en) 1987-07-31 1989-10-17 Merck & Co., Inc. 4"-Deoxy-4-N-methylamino avermectin Bla/Blb
US4895837A (en) 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
NZ228866A (en) 1988-05-02 1991-10-25 Merck & Co Inc Fluoro-substituted milbemycins and avermectins for combatting parasites and insects
US4873224A (en) 1988-05-23 1989-10-10 Merck & Co., Inc. Avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
US5057499A (en) 1989-06-02 1991-10-15 Merck & Co. Inc. Avermectin derivatives
US5023241A (en) 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
US5169839A (en) 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
IL98599A (en) 1990-06-28 1995-06-29 Merck & Co Inc Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them
US5192546A (en) 1991-01-15 1993-03-09 Mycogen Corporation Synergistic pesticidal compositions
US5346698A (en) 1991-01-15 1994-09-13 Mycogen Corporation Synergistic pesticidal compositions
US5208222A (en) 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
US5262400A (en) 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
GB9201505D0 (en) 1992-01-24 1992-03-11 Pfizer Ltd Antiparasitic agents
US5229415A (en) 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US6486195B1 (en) 1993-08-19 2002-11-26 Merck & Co., Inc. Thermodynamically stable crystal form of 4″-deoxy-4″-epi-methylamino avermectin B1a/B1b benzoic acid salt and processes for its preparation
US5362863A (en) 1993-09-29 1994-11-08 Merck & Co., Inc. Process for the preparation of 4"-amino avermectin compounds
US5981500A (en) 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
US5436355A (en) 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
US6875727B2 (en) 1997-12-23 2005-04-05 Syngenta Crop Protection, Inc. Use of macrolides in pest control
KR20010101819A (ko) 1999-02-09 2001-11-14 오무라 사토시 에바멕틴 유도체
WO2002012248A1 (fr) 2000-08-09 2002-02-14 The Kitasato Institute Derives d'avermectine
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR037938A1 (es) 2001-12-21 2004-12-22 Syngenta Participations Ag Derivados de avermectina b1 que tienen un substituyente de aminosulfoniloxilo en la posicion 4''
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302548D0 (en) 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

Also Published As

Publication number Publication date
ES2280022T3 (es) 2007-09-01
ATE349457T1 (de) 2007-01-15
US20060140997A1 (en) 2006-06-29
JP2006516584A (ja) 2006-07-06
SI1592699T1 (sl) 2007-08-31
DE602004003907D1 (de) 2007-02-08
AR042966A1 (es) 2005-07-13
TW200510443A (en) 2005-03-16
US7678740B2 (en) 2010-03-16
EP1592699B1 (de) 2006-12-27
EP1592699A1 (de) 2005-11-09
PT1592699E (pt) 2007-04-30
CY1108005T1 (el) 2013-09-04
GB0302308D0 (en) 2003-03-05
CL2004000148A1 (es) 2005-01-14
WO2004067543A1 (en) 2004-08-12
DE602004003907T2 (de) 2007-10-25

Similar Documents

Publication Publication Date Title
DK1592699T3 (da) Avermectin og avermectin-monosaccharidderivater substitueret i 4"- eller 4' -positionen, hvilke forbindelser har pesticidegenskaber
DE602005015835D1 (de) An der 4"- bzw. 4'-stellung substituiertes avermectin und avermectin-monosaccharid
IL169598A0 (en) Vermectin monosaccharide derivatives having pesticidal properties
DE602004006169D1 (de) Substituierte 8'-pyri(mi)dinyl-dihydrospiro-äcycloalkylaminü-pyrimidoä1,2aüpyrimidin-6-onderivate
NO20055568D0 (no) Substituerte 1,4-diazepiner og anvendelser derav
PT1373216E (pt) Derivados de 4,5-diidro-1h-pirazol que possuem actividade antagonista de cb1
DE60222494D1 (de) Stabilisatorstab
ATE516275T1 (de) Microbiozide (z.b. fungizide) 1,2,3- triazolderivate
DE602004024770D1 (de) Substituierte 8-perfluoro-6,7,8,9-tetrahydropyrimido-(1,2a) pyrimidin-4-on derivate
DE602004021572D1 (de) SUBSTITUIERTE 8-PERFLUORO-6,7,8,9-TETRAHYDROPYRIMIDOi1,2-A PYRIMIDIN-4-ON-DERIVATE
ATE483721T1 (de) In 4''- bzw. 4'-position substituierte avermectine mit pestiziden eigenschaften
DK1592700T3 (da) Avermectin-derivater og Avermectin-monosaccharidderivater der er substitueret i 4'' - eller 4' - stillingen, og som har pesticidegenskaber
MA26089A1 (fr) Avermectines substituees en position 4" ayant des proprietes pesticides.
DK1660510T3 (da) Avermectiner of avermectinmonosaccharider som er substitueret i 4' - og 4'' -positionen og som har pesticidegenskaber
BRPI0402574B1 (pt) combinada agrìcola.
ATE355060T1 (de) 2-methoxymethyl-3-(3,4-dichlorophenyl)-8- azabicyclo (3.2.1)octantartrat-salze
ITSS20050009A1 (it) Sistema di mobilita' individuale muscolare innovativo (acronimo smimi).
NO20044405L (no) Neurotensinaktive 2,3-diaryl-pyrazolidin derivater
DK1638984T3 (da) Avermectin B1-monosaccharidderivater
GB0302547D0 (en) Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
ES1050026Y (es) Disposicion de puerta ignifuga perfeccionada.
ES1049590Y (es) Cenicero ambientador perfeccionado.
ES1050843Y (es) Bisagra regulable para puertas.
ES1054113Y (es) Puerta de mueble reversible.
ITSV20030024A1 (it) Porta, portone sezionale o simili.