DE602004003907D1 - Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen - Google Patents

Avermectin- und avermectinmonosaccharidderivate, die in der 4'' - oder 4' -stellung substituiert sind und pestizide eigenschaften aufweisen

Info

Publication number
DE602004003907D1
DE602004003907D1 DE602004003907T DE602004003907T DE602004003907D1 DE 602004003907 D1 DE602004003907 D1 DE 602004003907D1 DE 602004003907 T DE602004003907 T DE 602004003907T DE 602004003907 T DE602004003907 T DE 602004003907T DE 602004003907 D1 DE602004003907 D1 DE 602004003907D1
Authority
DE
Germany
Prior art keywords
avermectinmonosaccharide
avermectin
derivatives substituted
pesticidal properties
pesticidal
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE602004003907T
Other languages
English (en)
Other versions
DE602004003907T2 (de
Inventor
Thomas Pitterna
Kessabi Fiona Murphy
Peter Maienfisch
Jerome Cassayre
Laura Quaranta
Pierre Jung
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merial Ltd
Original Assignee
Syngenta Participations AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations AG filed Critical Syngenta Participations AG
Publication of DE602004003907D1 publication Critical patent/DE602004003907D1/de
Application granted granted Critical
Publication of DE602004003907T2 publication Critical patent/DE602004003907T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Agronomy & Crop Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Environmental Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Biochemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
DE602004003907T 2003-01-31 2004-01-30 Avermectin- und avermectinmonosaccharidderivate, die in der 4''- oder 4 -stellung substituiert sind und pestizide eigenschaften aufweisen Expired - Lifetime DE602004003907T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0302308 2003-01-31
GBGB0302308.2A GB0302308D0 (en) 2003-01-31 2003-01-31 Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
PCT/EP2004/000890 WO2004067543A1 (en) 2003-01-31 2004-01-30 Avermectin and avermectin monosaccharide derivatives substituted in the 4”- or 4’-position having pesticidal properties

Publications (2)

Publication Number Publication Date
DE602004003907D1 true DE602004003907D1 (de) 2007-02-08
DE602004003907T2 DE602004003907T2 (de) 2007-10-25

Family

ID=9952239

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602004003907T Expired - Lifetime DE602004003907T2 (de) 2003-01-31 2004-01-30 Avermectin- und avermectinmonosaccharidderivate, die in der 4''- oder 4 -stellung substituiert sind und pestizide eigenschaften aufweisen

Country Status (15)

Country Link
US (1) US7678740B2 (de)
EP (1) EP1592699B1 (de)
JP (1) JP2006516584A (de)
AR (1) AR042966A1 (de)
AT (1) ATE349457T1 (de)
CL (1) CL2004000148A1 (de)
CY (1) CY1108005T1 (de)
DE (1) DE602004003907T2 (de)
DK (1) DK1592699T3 (de)
ES (1) ES2280022T3 (de)
GB (1) GB0302308D0 (de)
PT (1) PT1592699E (de)
SI (1) SI1592699T1 (de)
TW (1) TW200510443A (de)
WO (1) WO2004067543A1 (de)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CR6574A (es) * 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) * 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) * 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
GB0129267D0 (en) * 2001-12-06 2002-01-23 Syngenta Ltd Fungicides
AR040073A1 (es) * 2002-05-07 2005-03-16 Syngenta Participations Ag Derivados de 4''-desoxi-4''-(s)-amido avermectina y su uso como plaguicidas
GB0227555D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227558D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227556D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0227554D0 (en) * 2002-11-26 2002-12-31 Syngenta Ltd Fungicides
GB0302309D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302310D0 (en) * 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302547D0 (en) * 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties
GB0312864D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0312863D0 (en) * 2003-06-04 2003-07-09 Syngenta Ltd Fungicides
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively
EP2568980B1 (de) 2010-05-12 2015-11-11 Merial, Inc. Injizierbare parasitizide formulierungen aus levamisol und makrocyclischen lactonen
NZ612185A (en) 2010-12-07 2015-10-30 Merial Inc Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
CN109485683A (zh) * 2018-11-27 2019-03-19 齐鲁晟华制药有限公司 一种含氟系列阿维菌素衍生物及其制备方法
CN113150053A (zh) * 2020-01-22 2021-07-23 华东理工大学 偶氮苯类阿维菌素衍生物及其制备方法和应用
CN115403644B (zh) * 2022-09-01 2024-04-05 石家庄学院 一种烟碱甲氨基或氨基阿维菌素B1a化合物及其制备方法和应用

Family Cites Families (39)

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Publication number Priority date Publication date Assignee Title
US4206205A (en) 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4203976A (en) 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4427663A (en) 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4622313A (en) 1985-08-01 1986-11-11 Merck & Co., Inc. O-sulfate derivatives of avermectins and milbemycins having improved water solubility
US4662313A (en) * 1985-10-23 1987-05-05 Xerox Corporation Image density controller
US4886828A (en) 1986-09-12 1989-12-12 American Cyanamid Company Δ22 -derivatives of LL-F28249 compounds
US4831016A (en) 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives
US4874749A (en) 1987-07-31 1989-10-17 Merck & Co., Inc. 4"-Deoxy-4-N-methylamino avermectin Bla/Blb
US4895837A (en) 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
NZ228866A (en) 1988-05-02 1991-10-25 Merck & Co Inc Fluoro-substituted milbemycins and avermectins for combatting parasites and insects
US4873224A (en) * 1988-05-23 1989-10-10 Merck & Co., Inc. Avermectin derivatives
NZ231773A (en) * 1988-12-23 1992-09-25 Merck & Co Inc Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof
US5057499A (en) 1989-06-02 1991-10-15 Merck & Co. Inc. Avermectin derivatives
US5023241A (en) * 1989-07-31 1991-06-11 Merck & Co., Inc. Avermectin derivatives
US5169839A (en) 1990-05-11 1992-12-08 Merck & Co., Inc. Derivatives of 3'- and 3"-o-desmethyl avermectin compounds, compositions and methods of treating melmintic and parasitic infections
IL98599A (en) 1990-06-28 1995-06-29 Merck & Co Inc Stable salts of "4-deoxy-" 4-epi-methylamino abramectin and insecticides containing them
US5192546A (en) 1991-01-15 1993-03-09 Mycogen Corporation Synergistic pesticidal compositions
US5346698A (en) 1991-01-15 1994-09-13 Mycogen Corporation Synergistic pesticidal compositions
US5208222A (en) 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
US5262400A (en) 1991-06-20 1993-11-16 Merck & Co., Inc. 4α-substituted avermectin derivatives
GB9201505D0 (en) 1992-01-24 1992-03-11 Pfizer Ltd Antiparasitic agents
US5229415A (en) 1992-03-24 1993-07-20 Merck & Co., Inc. Alkylthio alkyl avermectins are active antiparasitic agents
US6486195B1 (en) 1993-08-19 2002-11-26 Merck & Co., Inc. Thermodynamically stable crystal form of 4″-deoxy-4″-epi-methylamino avermectin B1a/B1b benzoic acid salt and processes for its preparation
US5362863A (en) 1993-09-29 1994-11-08 Merck & Co., Inc. Process for the preparation of 4"-amino avermectin compounds
US5981500A (en) 1994-01-12 1999-11-09 Pfizer Inc. Antiparasitic agents related to the milbemycins and avermectins
US5436355A (en) 1994-02-03 1995-07-25 Merck & Co., Inc. Process for making avermectin/zein compositions
TW327125B (en) 1994-02-07 1998-02-21 Merck & Co Inc Composition and method for protecting against pine exhausted
US6875727B2 (en) 1997-12-23 2005-04-05 Syngenta Crop Protection, Inc. Use of macrolides in pest control
KR20010101819A (ko) 1999-02-09 2001-11-14 오무라 사토시 에바멕틴 유도체
US20040087519A1 (en) 2000-08-09 2004-05-06 Satoshi Omura Avermectin derivatives
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
AR037938A1 (es) 2001-12-21 2004-12-22 Syngenta Participations Ag Derivados de avermectina b1 que tienen un substituyente de aminosulfoniloxilo en la posicion 4''
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0302309D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties
GB0302548D0 (en) 2003-02-04 2003-03-12 Syngenta Participations Ag Avermectins substituted in the 4"- and 4' -positions having pesticidal properties
TW200538461A (en) * 2004-04-07 2005-12-01 Syngenta Participations Ag Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively

Also Published As

Publication number Publication date
US7678740B2 (en) 2010-03-16
AR042966A1 (es) 2005-07-13
JP2006516584A (ja) 2006-07-06
PT1592699E (pt) 2007-04-30
DK1592699T3 (da) 2007-05-07
WO2004067543A1 (en) 2004-08-12
TW200510443A (en) 2005-03-16
CL2004000148A1 (es) 2005-01-14
DE602004003907T2 (de) 2007-10-25
US20060140997A1 (en) 2006-06-29
ES2280022T3 (es) 2007-09-01
EP1592699A1 (de) 2005-11-09
EP1592699B1 (de) 2006-12-27
CY1108005T1 (el) 2013-09-04
SI1592699T1 (sl) 2007-08-31
ATE349457T1 (de) 2007-01-15
GB0302308D0 (en) 2003-03-05

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Legal Events

Date Code Title Description
8327 Change in the person/name/address of the patent owner

Owner name: MERIAL LTD., HARLOW, ESSEX, GB

8364 No opposition during term of opposition