DK153150C - Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater - Google Patents

Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater

Info

Publication number: DK153150C
Authority: DK; Denmark
Prior art keywords: pyridooe1; tetrahydro; oxo; derivatives; preparing
Prior art date: 1975-11-27

Application number

DK534076A

Other languages

Danish (da)

English (en)

Other versions

DK153150B (da

DK534076A (da

Inventor

Zoltan Meszaros

Jozsef Knoll

Peter Szentmiklosi

Istvan Hermecz

Agnes Horvath

Sandor Virag

Lelle Vasvari

Agoston David

Original Assignee

Chinoin Gyogyszer Es Vegyeszet

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1975-11-27

Filing date

1976-11-26

Publication date

1988-10-24

1976-11-26 Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet

1977-05-28 Publication of DK534076A publication Critical patent/DK534076A/da

1988-06-20 Publication of DK153150B publication Critical patent/DK153150B/da

1988-10-24 Application granted granted Critical

1988-10-24 Publication of DK153150C publication Critical patent/DK153150C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Diabetes (AREA)
Hematology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

DK534076A 1975-11-27 1976-11-26 Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater DK153150C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HUCI001623		1975-11-27
HU75CI1623A HU173438B (hu)	1975-11-27	1975-11-27	Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom

Publications (3)

Publication Number	Publication Date
DK534076A DK534076A (da)	1977-05-28
DK153150B DK153150B (da)	1988-06-20
DK153150C true DK153150C (da)	1988-10-24

Family

ID=10994587

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK534076A DK153150C (da)	1975-11-27	1976-11-26	Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater

Country Status (28)

Country	Link
US (2)	US4460771A (nl)
JP (1)	JPS5914033B2 (nl)
AT (1)	AT359506B (nl)
AU (1)	AU512256B2 (nl)
BE (1)	BE848868A (nl)
BG (1)	BG31226A4 (nl)
CA (1)	CA1088531A (nl)
CH (2)	CH630378A5 (nl)
CS (1)	CS203135B2 (nl)
DD (1)	DD130431A5 (nl)
DE (1)	DE2653257A1 (nl)
DK (1)	DK153150C (nl)
EG (1)	EG12495A (nl)
ES (1)	ES453690A1 (nl)
FI (1)	FI62085C (nl)
FR (1)	FR2332755A1 (nl)
GB (1)	GB1531963A (nl)
GR (1)	GR61820B (nl)
HU (1)	HU173438B (nl)
IL (1)	IL50930A (nl)
IN (1)	IN148945B (nl)
MX (1)	MX5178E (nl)
NL (1)	NL188948C (nl)
PL (1)	PL109657B1 (nl)
RO (2)	RO79705A (nl)
SE (1)	SE433353B (nl)
SU (2)	SU664565A3 (nl)
YU (2)	YU289076A (nl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU180701B (en) *	1977-12-29	1983-04-29	Chinoin Gyogyszer Es Vegyeszet	Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
US4192944A (en) *	1978-04-03	1980-03-11	Bristol-Myers Company	Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents
US4342870A (en) *	1980-03-28	1982-08-03	Janssen Pharmaceutica N.V.	Novel 3-(1-piperidinylalkyl)-4H-pyrido[1,2-a]pyrimidin-4-one derivatives
HU183408B (en) *	1981-04-28	1984-05-28	Chinoin Gyogyszer Es Vegyeszet	Process for producing oral ratard pharmaceutical compositions
HU186607B (en) *	1982-03-31	1985-08-28	Chinoin Gyogyszer Es Vegyeszet	Process for preparing pharmaceutical composition with synergetic antiinflammatory activity
NO162019C (no) *	1983-11-23	1989-10-25	Fujisawa Pharmaceutical Co	Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrimidoiskinolinderivater.
US4772475A (en) *	1985-03-08	1988-09-20	Yamanouchi Pharmaceutical Co., Ltd.	Controlled-release multiple units pharmaceutical formulation
HU201551B (en) *	1988-02-03	1990-11-28	Chinoin Gyogyszer Es Vegyeszet	Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
US5252572A (en) *	1988-02-03	1993-10-12	Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt.	Pyridopyrimidine derivatives, pharmaceutical compositions containing them and process for preparing same
MY125533A (en) *	1999-12-06	2006-08-30	Bristol Myers Squibb Co	Heterocyclic dihydropyrimidine compounds
RU2005103398A (ru) *	2002-07-09	2006-06-27	Актелион Фармасьютикалз Лтд. (Ch)	Производные 7,8,9,10-тетрагидро-6h-азепино-, 6,7,8,9-тетрагидропиридо-и 2,3-дигидро-2h-пирроло-[2,1-b]-хиназолинона
US7772232B2 (en) *	2004-04-15	2010-08-10	Bristol-Myers Squibb Company	Quinazolinyl compounds as inhibitors of potassium channel function
US20060111307A1 (en) *	2004-11-16	2006-05-25	Wendye Robbins	Methods and compositions for treating pain

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH538494A (de) *	1966-11-02	1973-06-30	Chinoin Gyogyszer Es Vegyeszet	Verfahren zur Herstellung neuer Homopyrimidazol-Derivate
US3642797A (en) *	1968-06-10	1972-02-15	Sterling Drug Inc	4h-pyrido(1 2-a)pyrimidin-4-ones
US4209622A (en) *	1973-03-30	1980-06-24	Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt.	3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
HU168014B (nl) *	1973-03-30	1976-02-28
HU168541B (nl) *	1973-11-24	1976-05-28
US4022897A (en) *	1974-03-04	1977-05-10	E. R. Squibb & Sons, Inc.	CNS active compounds
US3960863A (en) *	1974-06-25	1976-06-01	Sankyo Company Limited	Pyrido[1,2-a]pyrimidinone derivatives
US4066766A (en) *	1975-03-03	1978-01-03	Pfizer Inc.	1-Oxo-6-substituted pyrimido [1,2-a]quinoline-2-carboxylic acids and derivatives thereof and their use as antiallergy agents
HU174693B (hu) *	1976-02-12	1980-03-28	Chinoin Gyogyszer Es Vegyeszet	Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
US4122274A (en) *	1977-05-25	1978-10-24	Bristol-Myers Company	3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones
US4192944A (en) *	1978-04-03	1980-03-11	Bristol-Myers Company	Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents

1975
- 1975-11-27 HU HU75CI1623A patent/HU173438B/hu not_active IP Right Cessation
1976
- 1976-11-16 BG BG7636221A patent/BG31226A4/xx unknown
- 1976-11-17 IL IL50930A patent/IL50930A/xx unknown
- 1976-11-17 US US05/742,464 patent/US4460771A/en not_active Expired - Lifetime
- 1976-11-18 AU AU19759/76A patent/AU512256B2/en not_active Expired
- 1976-11-19 IN IN2075/CAL/76A patent/IN148945B/en unknown
- 1976-11-23 EG EG725/76A patent/EG12495A/xx active
- 1976-11-24 DE DE19762653257 patent/DE2653257A1/de active Granted
- 1976-11-24 SE SE7613140A patent/SE433353B/xx not_active IP Right Cessation
- 1976-11-25 GB GB49273/76A patent/GB1531963A/en not_active Expired
- 1976-11-25 RO RO76101145A patent/RO79705A/ro unknown
- 1976-11-25 NL NLAANVRAGE7613140,A patent/NL188948C/nl not_active IP Right Cessation
- 1976-11-25 RO RO7688555A patent/RO73522A/ro unknown
- 1976-11-25 DD DD7600195963A patent/DD130431A5/xx unknown
- 1976-11-25 FI FI763401A patent/FI62085C/fi not_active IP Right Cessation
- 1976-11-25 AT AT873576A patent/AT359506B/de not_active IP Right Cessation
- 1976-11-25 GR GR52262A patent/GR61820B/el unknown
- 1976-11-25 FR FR7635550A patent/FR2332755A1/fr active Granted
- 1976-11-26 CS CS767665A patent/CS203135B2/cs unknown
- 1976-11-26 CA CA266,711A patent/CA1088531A/en not_active Expired
- 1976-11-26 YU YU02890/76A patent/YU289076A/xx unknown
- 1976-11-26 SU SU762424104A patent/SU664565A3/ru active
- 1976-11-26 PL PL1976209750A patent/PL109657B1/pl unknown
- 1976-11-26 MX MX765170U patent/MX5178E/es unknown
- 1976-11-26 ES ES453690A patent/ES453690A1/es not_active Expired
- 1976-11-26 DK DK534076A patent/DK153150C/da not_active IP Right Cessation
- 1976-11-26 CH CH1493176A patent/CH630378A5/de not_active IP Right Cessation
- 1976-11-27 JP JP51141797A patent/JPS5914033B2/ja not_active Expired
- 1976-11-29 BE BE172806A patent/BE848868A/xx not_active IP Right Cessation
1977
- 1977-11-03 SU SU772537600A patent/SU698532A3/ru active
1979
- 1979-02-23 US US06/014,689 patent/US4472398A/en not_active Expired - Lifetime
1981
- 1981-01-21 CH CH38381A patent/CH630379A5/de not_active IP Right Cessation
1983
- 1983-07-08 YU YU01475/83A patent/YU147583A/xx unknown

Also Published As

Publication number	Publication date
YU147583A (en)	1986-06-30
ES453690A1 (es)	1977-12-01
GR61820B (en)	1979-01-22
SU698532A3 (ru)	1979-11-15
IN148945B (nl)	1981-07-25
PL109657B1 (en)	1980-06-30
DE2653257C2 (nl)	1989-04-20
US4472398A (en)	1984-09-18
DE2653257A1 (de)	1977-06-02
FR2332755A1 (fr)	1977-06-24
YU289076A (en)	1983-12-31
CA1088531A (en)	1980-10-28
ATA873576A (de)	1980-04-15
SU664565A3 (ru)	1979-05-25
DD130431A5 (de)	1978-03-29
AT359506B (de)	1980-11-10
NL188948C (nl)	1992-11-16
FR2332755B1 (nl)	1978-12-22
JPS5268198A (en)	1977-06-06
FI62085C (fi)	1982-11-10
NL7613140A (nl)	1977-06-01
AU1975976A (en)	1978-05-25
FI62085B (fi)	1982-07-30
BE848868A (fr)	1977-03-16
FI763401A (nl)	1977-05-28
CH630379A5 (de)	1982-06-15
SE433353B (sv)	1984-05-21
RO79705A (ro)	1982-08-17
GB1531963A (en)	1978-11-15
NL188948B (nl)	1992-06-16
IL50930A0 (en)	1977-01-31
CH630378A5 (de)	1982-06-15
EG12495A (en)	1980-12-31
SE7613140L (sv)	1977-05-28
HU173438B (hu)	1979-05-28
JPS5914033B2 (ja)	1984-04-02
AU512256B2 (en)	1980-10-02
RO73522A (ro)	1981-11-04
IL50930A (en)	1981-06-29
CS203135B2 (en)	1981-02-27
DK153150B (da)	1988-06-20
MX5178E (es)	1983-04-20
BG31226A4 (en)	1981-11-16
US4460771A (en)	1984-07-17
DK534076A (da)	1977-05-28

Legal Events

Date	Code	Title	Description
1995-07-24	PBP	Patent lapsed

Publication	Publication Date	Title
DK298176A (da)	1977-01-03	Fremgangsmade til fremstilling af 1,4-dihydropyrinderivater
SE429970B (sv)	1983-10-10	Forfarande for framstellning av glukopyranosido-1,6-mannit
DK149749C (da)	1987-03-02	Analogifremgangsmaade til fremstilling af n-alkyl-2-hydroxy-metyl-3,4,5-trihydroxy-piperidinderivater
DK494876A (da)	1977-05-08	Fremgangsmade til fremstilling af piperidinderivater
DK145228C (da)	1983-02-28	Analogifremgangsmaade til fremstilling af 3-amino-4-deoxo-4-iminorifamycinderivater
DK143708C (da)	1982-03-15	Analogifremgangsmaade til fremstilling af 17alfa-acyloxy-9alfa,21-dihalogen-11beta-hydroxy-6alfa-fluor-16alfa-methyl-pregna-1,4-dien-3,20-dion-forbindelser
DK147068C (da)	1984-09-10	Analogifremgangsmaade til fremstilling af 1-naphthylmethyl-cinnamyl-aminderivater
DK562376A (da)	1977-06-24	Fremgangsmade til fremstilling af ergolinderivater
DK462376A (da)	1977-04-17	Fremgangsmade til fremstilling af 5-halogenpyrimidinderivater
DK563377A (da)	1978-06-18	R fremgangsmaade til fremstilling af 1,4-dihydropyridinderivate
DK147855C (da)	1985-06-10	Analogifremgangsmaade til fremstilling af 3,4-dihydro-quinazolinderivatereller salte deraf
DK153150C (da)	1988-10-24	Analogifremgangsmaade til fremstilling af 4-oxo-1,6,7,8-tetrahydro-4h-pyridooe1,2aaapyrimidinderivater
DK139267B (da)	1979-01-22	Fremgangsmaade til fremstilling af 4-androsten3,17-dionderivater
DK159787C (da)	1991-04-22	Fremgangsmaade til fremstilling af 3',4'-dideoxykanamycin b
DK143757C (da)	1982-03-22	Analogifremgangsmaade til fremstilling af 16,16-disubstituerede 3-oxoandrostener
DK150299C (da)	1987-10-26	Analogifremgangsmaade til fremstilling af 8-aminoalkyl-tetracyclo(4,3,0,02,4,03,7)nonanderivater
DK219776A (da)	1976-11-22	Fremgangsmade til fremstilling af 1,2-benzothiazin-oxadiazolforbindelse
DK143346C (da)	1981-12-14	Fremgangsmaade til fremstilling af 0,0-dialkylthionophosphorsyrechlorider
DK150543C (da)	1987-09-28	Analogifremgangsmaade til fremstilling af 4-phenyl-3-oxo-1,2,4-oxadiazinderivater
DK146624C (da)	1984-05-07	Analogifremgangsmaade til fremstilling af 1-aminoalkyl-3,4-diphenyl-1h-pyrazoler
DK319276A (da)	1977-01-24	Fremgangsmade til femstilling af nitroquinolinderivater
DK280376A (da)	1976-12-24	Fremgangsmade til fremstilling af 1-acyl-1,2,3,4-tetrahydro-6-quinoliner
DK205676A (da)	1976-11-11	Fremgangsmade til fremstilling af 2-substituerede 1,4-benzodiazepinderivater
DK140576A (da)	1976-11-10	Fremgangsmade til fremstilling af 21-hydroxy-16-pregnen-20-on-derivater
DK146593C (da)	1984-04-30	Analogifremgangsmaade til fremstilling af fluorprostaglandiner