DK150484C - ANALOGY PROCEDURE FOR PREPARING 4-AMINO-3-THIOPHENCARBOXYLIC ACID DERIVATIVES - Google Patents

ANALOGY PROCEDURE FOR PREPARING 4-AMINO-3-THIOPHENCARBOXYLIC ACID DERIVATIVES

Info

Publication number
DK150484C
DK150484C DK372177A DK372177A DK150484C DK 150484 C DK150484 C DK 150484C DK 372177 A DK372177 A DK 372177A DK 372177 A DK372177 A DK 372177A DK 150484 C DK150484 C DK 150484C
Authority
DK
Denmark
Prior art keywords
amino
preparing
acid derivatives
analogy procedure
thiophencarboxylic acid
Prior art date
Application number
DK372177A
Other languages
Danish (da)
Other versions
DK150484B (en
DK372177A (en
Inventor
Pasquale Nicholas Confalone
Giacomo Pizzolato
Marianne Rouge
Milan Radoje Uskokovic
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK372177A publication Critical patent/DK372177A/en
Publication of DK150484B publication Critical patent/DK150484B/en
Application granted granted Critical
Publication of DK150484C publication Critical patent/DK150484C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
DK372177A 1976-08-23 1977-08-22 ANALOGY PROCEDURE FOR PREPARING 4-AMINO-3-THIOPHENCARBOXYLIC ACID DERIVATIVES DK150484C (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US71685376A 1976-08-23 1976-08-23
US71685476A 1976-08-23 1976-08-23
US71685476 1976-08-23
US71685376 1976-08-23
US82052177A 1977-08-01 1977-08-01
US82052177 1977-08-01

Publications (3)

Publication Number Publication Date
DK372177A DK372177A (en) 1978-02-24
DK150484B DK150484B (en) 1987-03-09
DK150484C true DK150484C (en) 1987-10-05

Family

ID=27418961

Family Applications (1)

Application Number Title Priority Date Filing Date
DK372177A DK150484C (en) 1976-08-23 1977-08-22 ANALOGY PROCEDURE FOR PREPARING 4-AMINO-3-THIOPHENCARBOXYLIC ACID DERIVATIVES

Country Status (21)

Country Link
JP (1) JPS5340755A (en)
AR (1) AR222453A1 (en)
AT (1) AT359486B (en)
AU (1) AU509956B2 (en)
BE (1) BE858012A (en)
CH (1) CH628628A5 (en)
DE (1) DE2737738C2 (en)
DK (1) DK150484C (en)
ES (1) ES461796A1 (en)
FI (1) FI66859C (en)
FR (1) FR2365566A1 (en)
GB (1) GB1587084A (en)
HU (1) HU179484B (en)
IE (1) IE45470B1 (en)
IL (1) IL52792A (en)
IT (1) IT1143757B (en)
LU (1) LU78003A1 (en)
MC (1) MC1156A1 (en)
NL (1) NL7709246A (en)
NO (1) NO148673C (en)
NZ (1) NZ184981A (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6232765Y2 (en) * 1981-02-28 1987-08-21
US6515009B1 (en) 1991-09-27 2003-02-04 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US5811447A (en) 1993-01-28 1998-09-22 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US6251920B1 (en) 1993-05-13 2001-06-26 Neorx Corporation Prevention and treatment of cardiovascular pathologies
US6491938B2 (en) 1993-05-13 2002-12-10 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
DE69435137D1 (en) 1993-05-13 2008-10-16 Poniard Pharmaceuticals Inc PREVENTION AND TREATMENT OF PATHOLOGIES ASSOCIATED WITH AN ABNORMAL PROLIFERATION GLATTER MUSCLE CELLS
WO1998046588A2 (en) * 1997-04-11 1998-10-22 Neorx Corporation Compounds and therapies for the prevention of vascular and non-vascular pathologies
DE102004063191A1 (en) 2004-12-29 2006-07-13 Bayer Cropscience Ag Process for the preparation of substituted 2-alkoxycarbonyl-3-aminothiophenes
NZ587261A (en) 2008-02-29 2012-05-25 Nissan Chemical Ind Ltd Process for producing thiophene compound and intermediate thereof
WO2024079734A1 (en) 2022-10-14 2024-04-18 Adama Agan Ltd. Process for the preparation of substituted aminothiophene

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2502421A (en) * 1944-08-28 1950-04-04 Parke Davis & Co Tetrahydrothiophenes
US2502424A (en) * 1944-12-23 1950-04-04 Parke Davis & Co 3-acylamino-4-carboalkoxy-2-omega-ralkylthiophenes
US2502423A (en) * 1944-12-23 1950-04-04 Parke Davis & Co 4-carbalkoxy-3-keto-2-substituted tetrahydrothiophene oximes
US2443598A (en) * 1944-12-23 1948-06-22 Parke Davis & Co 3-amino-4-carbethoxy-2-alkyl derivatives of thiophene

Also Published As

Publication number Publication date
NO148673C (en) 1983-11-23
HU179484B (en) 1982-10-28
NO772917L (en) 1978-02-24
IE45470B1 (en) 1982-09-08
DE2737738C2 (en) 1987-01-29
NL7709246A (en) 1978-02-27
DK150484B (en) 1987-03-09
LU78003A1 (en) 1978-09-14
DK372177A (en) 1978-02-24
IT1143757B (en) 1986-10-22
IE45470L (en) 1978-02-23
AU509956B2 (en) 1980-06-05
JPS5340755A (en) 1978-04-13
AU2809277A (en) 1979-03-01
FR2365566B1 (en) 1980-12-26
FI66859B (en) 1984-08-31
AR222453A1 (en) 1981-05-29
ES461796A1 (en) 1978-12-16
JPS6121235B2 (en) 1986-05-26
IL52792A (en) 1981-06-29
BE858012A (en) 1978-02-22
FR2365566A1 (en) 1978-04-21
IL52792A0 (en) 1977-10-31
CH628628A5 (en) 1982-03-15
NZ184981A (en) 1980-08-26
AT359486B (en) 1980-11-10
ATA607477A (en) 1980-04-15
NO148673B (en) 1983-08-15
MC1156A1 (en) 1978-04-17
DE2737738A1 (en) 1978-03-09
FI66859C (en) 1984-12-10
GB1587084A (en) 1981-03-25
FI772494A (en) 1978-02-24

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