AR222453A1 - PROCEDURE FOR PREPARING 3-AMINO-4-CARBOXY-THIOPHENES - Google Patents

PROCEDURE FOR PREPARING 3-AMINO-4-CARBOXY-THIOPHENES

Info

Publication number
AR222453A1
AR222453A1 AR268888A AR26888877A AR222453A1 AR 222453 A1 AR222453 A1 AR 222453A1 AR 268888 A AR268888 A AR 268888A AR 26888877 A AR26888877 A AR 26888877A AR 222453 A1 AR222453 A1 AR 222453A1
Authority
AR
Argentina
Prior art keywords
thiophenes
carboxy
amino
preparing
procedure
Prior art date
Application number
AR268888A
Other languages
Spanish (es)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR222453A1 publication Critical patent/AR222453A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
AR268888A 1976-08-23 1977-08-22 PROCEDURE FOR PREPARING 3-AMINO-4-CARBOXY-THIOPHENES AR222453A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US71685476A 1976-08-23 1976-08-23
US71685376A 1976-08-23 1976-08-23
US82052177A 1977-08-01 1977-08-01

Publications (1)

Publication Number Publication Date
AR222453A1 true AR222453A1 (en) 1981-05-29

Family

ID=27418961

Family Applications (1)

Application Number Title Priority Date Filing Date
AR268888A AR222453A1 (en) 1976-08-23 1977-08-22 PROCEDURE FOR PREPARING 3-AMINO-4-CARBOXY-THIOPHENES

Country Status (21)

Country Link
JP (1) JPS5340755A (en)
AR (1) AR222453A1 (en)
AT (1) AT359486B (en)
AU (1) AU509956B2 (en)
BE (1) BE858012A (en)
CH (1) CH628628A5 (en)
DE (1) DE2737738A1 (en)
DK (1) DK150484C (en)
ES (1) ES461796A1 (en)
FI (1) FI66859C (en)
FR (1) FR2365566A1 (en)
GB (1) GB1587084A (en)
HU (1) HU179484B (en)
IE (1) IE45470B1 (en)
IL (1) IL52792A (en)
IT (1) IT1143757B (en)
LU (1) LU78003A1 (en)
MC (1) MC1156A1 (en)
NL (1) NL7709246A (en)
NO (1) NO148673C (en)
NZ (1) NZ184981A (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6232765Y2 (en) * 1981-02-28 1987-08-21
US6515009B1 (en) 1991-09-27 2003-02-04 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US5811447A (en) 1993-01-28 1998-09-22 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
US6251920B1 (en) 1993-05-13 2001-06-26 Neorx Corporation Prevention and treatment of cardiovascular pathologies
US6491938B2 (en) 1993-05-13 2002-12-10 Neorx Corporation Therapeutic inhibitor of vascular smooth muscle cells
CA2162586C (en) 1993-05-13 2006-01-03 David J. Grainger Prevention and treatment of pathologies associated with abnormally proliferative smooth muscle cells
US6117911A (en) * 1997-04-11 2000-09-12 Neorx Corporation Compounds and therapies for the prevention of vascular and non-vascular pathologies
DE102004063191A1 (en) 2004-12-29 2006-07-13 Bayer Cropscience Ag Process for the preparation of substituted 2-alkoxycarbonyl-3-aminothiophenes
JP5440490B2 (en) 2008-02-29 2014-03-12 日産化学工業株式会社 Method for producing thiophene compound and intermediate thereof
WO2024079734A1 (en) 2022-10-14 2024-04-18 Adama Agan Ltd. Process for the preparation of substituted aminothiophene

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2502421A (en) * 1944-08-28 1950-04-04 Parke Davis & Co Tetrahydrothiophenes
US2502423A (en) * 1944-12-23 1950-04-04 Parke Davis & Co 4-carbalkoxy-3-keto-2-substituted tetrahydrothiophene oximes
US2443598A (en) * 1944-12-23 1948-06-22 Parke Davis & Co 3-amino-4-carbethoxy-2-alkyl derivatives of thiophene
US2502424A (en) * 1944-12-23 1950-04-04 Parke Davis & Co 3-acylamino-4-carboalkoxy-2-omega-ralkylthiophenes

Also Published As

Publication number Publication date
FI66859C (en) 1984-12-10
NO148673C (en) 1983-11-23
IL52792A (en) 1981-06-29
NO148673B (en) 1983-08-15
DE2737738A1 (en) 1978-03-09
AU509956B2 (en) 1980-06-05
DE2737738C2 (en) 1987-01-29
HU179484B (en) 1982-10-28
LU78003A1 (en) 1978-09-14
DK372177A (en) 1978-02-24
IT1143757B (en) 1986-10-22
IE45470B1 (en) 1982-09-08
ES461796A1 (en) 1978-12-16
NO772917L (en) 1978-02-24
AU2809277A (en) 1979-03-01
BE858012A (en) 1978-02-22
DK150484C (en) 1987-10-05
ATA607477A (en) 1980-04-15
FR2365566B1 (en) 1980-12-26
AT359486B (en) 1980-11-10
NZ184981A (en) 1980-08-26
MC1156A1 (en) 1978-04-17
FI772494A (en) 1978-02-24
GB1587084A (en) 1981-03-25
IL52792A0 (en) 1977-10-31
FR2365566A1 (en) 1978-04-21
FI66859B (en) 1984-08-31
JPS5340755A (en) 1978-04-13
CH628628A5 (en) 1982-03-15
DK150484B (en) 1987-03-09
JPS6121235B2 (en) 1986-05-26
IE45470L (en) 1978-02-23
NL7709246A (en) 1978-02-27

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