DK148596C - Analogifremgangsmaade til fremstilling af 3-aminosubstituerede pyridaziner eller farmaceutisk acceptable syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af 3-aminosubstituerede pyridaziner eller farmaceutisk acceptable syreadditionssalte deraf

Info

Publication number: DK148596C
Authority: DK; Denmark
Prior art keywords: analogue; amino; preparation; acid addition; addition salts
Prior art date: 1981-08-11

Application number

DK358782A

Other languages

English (en)

Other versions

DK358782A (da

DK148596B (da

Inventor

Camille Georges Wermuth

Jean-Pierre Chambon

Original Assignee

Sanofi Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-08-11

Filing date

1982-08-10

Publication date

1986-01-13

1982-08-10 Application filed by Sanofi Sa filed Critical Sanofi Sa

1983-02-12 Publication of DK358782A publication Critical patent/DK358782A/da

1985-08-12 Publication of DK148596B publication Critical patent/DK148596B/da

1986-01-13 Application granted granted Critical

1986-01-13 Publication of DK148596C publication Critical patent/DK148596C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
- C07D237/30—Phthalazines
- C07D237/34—Phthalazines with nitrogen atoms directly attached to carbon atoms of the nitrogen-containing ring, e.g. hydrazine radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D237/20—Nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Biomedical Technology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Neurosurgery (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

DK358782A 1981-08-11 1982-08-10 Analogifremgangsmaade til fremstilling af 3-aminosubstituerede pyridaziner eller farmaceutisk acceptable syreadditionssalte deraf DK148596C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8115546A FR2511366A1 (fr)	1981-08-11	1981-08-11	Nouveaux derives de la pyridazine, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent
FR8115546		1981-08-11

Publications (3)

Publication Number	Publication Date
DK358782A DK358782A (da)	1983-02-12
DK148596B DK148596B (da)	1985-08-12
DK148596C true DK148596C (da)	1986-01-13

Family

ID=9261385

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK358782A DK148596C (da)	1981-08-11	1982-08-10	Analogifremgangsmaade til fremstilling af 3-aminosubstituerede pyridaziner eller farmaceutisk acceptable syreadditionssalte deraf

Country Status (30)

Country	Link
US (1)	US4710499A (da)
EP (1)	EP0073161B1 (da)
JP (1)	JPS5838263A (da)
KR (1)	KR880002711B1 (da)
AR (1)	AR231537A1 (da)
AT (1)	ATE23042T1 (da)
AU (1)	AU579570B2 (da)
CA (1)	CA1179347A (da)
CS (1)	CS239929B2 (da)
DD (1)	DD202550A5 (da)
DE (1)	DE3273893D1 (da)
DK (1)	DK148596C (da)
EG (1)	EG15749A (da)
ES (1)	ES514887A0 (da)
FI (1)	FI72970C (da)
FR (1)	FR2511366A1 (da)
GR (1)	GR76236B (da)
HU (1)	HU189608B (da)
IE (1)	IE53493B1 (da)
IL (1)	IL66424A (da)
MA (1)	MA19559A1 (da)
NO (1)	NO158871C (da)
NZ (1)	NZ201553A (da)
OA (1)	OA07179A (da)
PH (1)	PH18921A (da)
PL (1)	PL137200B1 (da)
PT (1)	PT75372B (da)
SU (1)	SU1356960A3 (da)
YU (1)	YU171682A (da)
ZA (1)	ZA825515B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2539741A1 (fr) *	1983-01-21	1984-07-27	Sanofi Sa	Composes a noyau heterocyclique diazote, leur procede de preparation et les medicaments, actifs sur le systeme nerveux central, qui en contiennent
US5001125A (en) *	1984-03-26	1991-03-19	Janssen Pharmaceutica N.V.	Anti-virally active pyridazinamines
JPS60218377A (ja) *	1984-04-16	1985-11-01	Mitsubishi Yuka Yakuhin Kk	４−フエニルフタラジン誘導体及びそれを有効成分とする循環改善剤
EP0190563B1 (de) *	1985-01-14	1989-08-02	Boehringer Ingelheim Kg	Neue 12-Amino-pyridazino[4',5':3,4]pyrrolo-[2,1-a]isochinoline, Verfahren zu ihrer Herstellung und ihre Verwendung
US5106973A (en) *	1987-11-23	1992-04-21	Janssen Pharmaceutica N.V.	Pyridzainamine derivatives
DK0628550T3 (da) *	1993-06-08	1998-09-28	Vertex Pharma	Pyridazin som interleukin-1 beta-omdannede enzyminhibitorer
US20100210590A1 (en) *	1995-09-27	2010-08-19	Northwestern University	Compositions and treatments for seizure-related disorders
GB9707693D0 (en) *	1997-04-16	1997-06-04	Smithkline Beecham Plc	Novel method of treatment
EP1430033A4 (en) *	2001-08-31	2004-12-15	Univ Northwestern	PROTEIN KINASE ANTI-INFLAMMATORY AND INHIBITOR COMPOSITION AND METHOD OF USE
JP2008518955A (ja) *	2004-11-02	2008-06-05	ノースウェスタンユニバーシティ	ピリダジン化合物および方法
EP1812408B1 (en) *	2004-11-02	2013-10-09	Northwestern University	Pyridazine compounds, compositions and methods
WO2007127448A2 (en) *	2006-04-28	2007-11-08	Northwestern University	Salts of pyridazine compounds
CN101754762A (zh)	2006-04-28	2010-06-23	西北大学	用于治疗神经炎症性疾病的包含哒嗪化合物的制剂
CA2650711A1 (en) *	2006-04-28	2007-11-08	Northwestern University	Compositions and treatments using pyridazine compounds and cholinesterase inhibitors
JP2010520223A (ja) *	2007-03-02	2010-06-10	ノースウェスタンユニバーシティ	発作関連障害のための組成物および方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1345880A (en) *	1971-06-18	1974-02-06	Cepbepe	Pyridazine derivatives
FR2473522A1 (fr) *	1980-01-16	1981-07-17	Synthelabo	Nouveaux derives substitues de dihydro-2,3 imidazo(1,2-b)pyridazines et les medicaments, utiles notamment comme antidepresseurs, qui en contiennent

1981
- 1981-08-11 FR FR8115546A patent/FR2511366A1/fr active Granted
1982
- 1982-07-26 GR GR68872A patent/GR76236B/el unknown
- 1982-07-28 IE IE1822/82A patent/IE53493B1/en not_active IP Right Cessation
- 1982-07-29 IL IL66424A patent/IL66424A/xx unknown
- 1982-07-30 AT AT82401426T patent/ATE23042T1/de not_active IP Right Cessation
- 1982-07-30 ZA ZA825515A patent/ZA825515B/xx unknown
- 1982-07-30 EP EP82401426A patent/EP0073161B1/fr not_active Expired
- 1982-07-30 DE DE8282401426T patent/DE3273893D1/de not_active Expired
- 1982-08-02 MA MA19770A patent/MA19559A1/fr unknown
- 1982-08-03 PT PT75372A patent/PT75372B/pt not_active IP Right Cessation
- 1982-08-06 HU HU822546A patent/HU189608B/hu not_active IP Right Cessation
- 1982-08-06 YU YU01716/82A patent/YU171682A/xx unknown
- 1982-08-07 EG EG478/82A patent/EG15749A/xx active
- 1982-08-09 PL PL1982237836A patent/PL137200B1/pl unknown
- 1982-08-09 FI FI822768A patent/FI72970C/fi not_active IP Right Cessation
- 1982-08-09 CS CS825913A patent/CS239929B2/cs unknown
- 1982-08-10 AU AU87029/82A patent/AU579570B2/en not_active Ceased
- 1982-08-10 NZ NZ201553A patent/NZ201553A/en unknown
- 1982-08-10 NO NO822717A patent/NO158871C/no unknown
- 1982-08-10 PH PH27701A patent/PH18921A/en unknown
- 1982-08-10 DK DK358782A patent/DK148596C/da not_active IP Right Cessation
- 1982-08-10 AR AR290279A patent/AR231537A1/es active
- 1982-08-10 CA CA000409143A patent/CA1179347A/en not_active Expired
- 1982-08-10 OA OA57771A patent/OA07179A/xx unknown
- 1982-08-10 ES ES514887A patent/ES514887A0/es active Granted
- 1982-08-10 SU SU823475703A patent/SU1356960A3/ru active
- 1982-08-11 DD DD82242426A patent/DD202550A5/de unknown
- 1982-08-11 JP JP57138671A patent/JPS5838263A/ja active Granted
- 1982-08-11 KR KR8203609A patent/KR880002711B1/ko active
1984
- 1984-08-07 US US06/638,363 patent/US4710499A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
US4710499A (en)	1987-12-01
DD202550A5 (de)	1983-09-21
NO822717L (no)	1983-02-14
PH18921A (en)	1985-11-11
PT75372B (en)	1984-12-10
FI72970C (fi)	1987-08-10
IE821822L (en)	1983-02-11
KR880002711B1 (ko)	1988-12-26
HU189608B (en)	1986-07-28
FR2511366B1 (da)	1984-12-14
CS239929B2 (en)	1986-01-16
ATE23042T1 (de)	1986-11-15
ES8305736A1 (es)	1983-04-16
PL137200B1 (en)	1986-05-31
FR2511366A1 (fr)	1983-02-18
MA19559A1 (fr)	1983-04-01
YU171682A (en)	1985-03-20
JPS5838263A (ja)	1983-03-05
FI822768A0 (fi)	1982-08-09
PL237836A1 (en)	1983-02-28
IE53493B1 (en)	1988-11-23
DK358782A (da)	1983-02-12
ES514887A0 (es)	1983-04-16
PT75372A (en)	1982-09-01
IL66424A0 (en)	1982-11-30
FI72970B (fi)	1987-04-30
AR231537A1 (es)	1984-12-28
EP0073161B1 (fr)	1986-10-22
KR840001147A (ko)	1984-03-28
JPH0456032B2 (da)	1992-09-07
ZA825515B (en)	1983-06-29
DK148596B (da)	1985-08-12
GR76236B (da)	1984-08-04
OA07179A (fr)	1984-04-30
AU579570B2 (en)	1988-12-01
DE3273893D1 (en)	1986-11-27
AU8702982A (en)	1983-05-12
CA1179347A (en)	1984-12-11
EP0073161A1 (fr)	1983-03-02
EG15749A (en)	1986-09-30
FI822768L (fi)	1983-02-11
SU1356960A3 (ru)	1987-11-30
NZ201553A (en)	1985-08-16
NO158871C (no)	1988-11-09
IL66424A (en)	1985-10-31
NO158871B (no)	1988-08-01

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Legal Events

Date	Code	Title	Description
1994-04-25	PBP	Patent lapsed