DK138496B - Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.

Info

Publication number
DK138496B
DK138496B DK34572AA DK34572A DK138496B DK 138496 B DK138496 B DK 138496B DK 34572A A DK34572A A DK 34572AA DK 34572 A DK34572 A DK 34572A DK 138496 B DK138496 B DK 138496B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
imidazoline derivatives
analogous process
Prior art date
Application number
DK34572AA
Other languages
Danish (da)
English (en)
Other versions
DK138496C (de
Inventor
Fernand Binon
Alex Areschka
Original Assignee
Labaz
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Labaz filed Critical Labaz
Publication of DK138496B publication Critical patent/DK138496B/da
Application granted granted Critical
Publication of DK138496C publication Critical patent/DK138496C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK34572AA 1971-01-27 1972-01-26 Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. DK138496B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB332771 1971-01-27

Publications (2)

Publication Number Publication Date
DK138496B true DK138496B (da) 1978-09-18
DK138496C DK138496C (de) 1979-02-26

Family

ID=9756227

Family Applications (1)

Application Number Title Priority Date Filing Date
DK34572AA DK138496B (da) 1971-01-27 1972-01-26 Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.

Country Status (17)

Country Link
US (1) US3818035A (de)
JP (1) JPS4938273B1 (de)
AT (1) AT311336B (de)
BE (1) BE777689A (de)
CA (1) CA962273A (de)
CH (1) CH535254A (de)
DE (1) DE2203373C3 (de)
DK (1) DK138496B (de)
FI (1) FI55841C (de)
GB (1) GB1333471A (de)
HU (1) HU162823B (de)
NL (1) NL150454B (de)
NO (1) NO134115C (de)
SE (1) SE378426B (de)
SU (1) SU474145A3 (de)
YU (1) YU34694B (de)
ZA (1) ZA72286B (de)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3927023A (en) * 1974-05-24 1975-12-16 Warner Lambert Co Imidazolyl benzofurans
DE3049542A1 (de) * 1980-12-31 1982-07-29 Basf Ag, 6700 Ludwigshafen Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung
ZA825413B (en) * 1981-08-26 1983-06-29 Pfizer Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them
US4806663A (en) * 1987-04-06 1989-02-21 The University Of Tennessee Research Corporation Certain 3-substituted 2-alkyl benzofuran derivatives
US4851554A (en) * 1987-04-06 1989-07-25 University Of Tennessee Research Corporation Certain 3-substituted 2-alkyl benzofuran derivatives
US4831156A (en) * 1987-09-30 1989-05-16 The University Of Tennessee Research Corp. 3-substituted 2-alkyl indole derivatives
AU2003099A (en) * 1997-12-19 1999-07-12 Eli Lilly And Company Method for treating diabetes
US7777035B2 (en) * 2005-06-22 2010-08-17 Chemocentryx, Inc. Azaindazole compounds and methods of use
CA2637312A1 (en) * 2006-01-27 2007-08-02 F. Hoffmann-La Roche Ag Use of substituted 2-imidazole of imidazoline derivatives
EP2076496B1 (de) * 2006-10-19 2010-03-31 F. Hoffmann-Roche AG Aminomethyl-2-imidazole mit affinität zu mit dem trace-amin assoziierten rezeptoren
AU2007312390B2 (en) * 2006-10-19 2013-03-28 F. Hoffmann-La Roche Ag Aminomethyl-4-imidazoles
ATE533755T1 (de) * 2006-11-02 2011-12-15 Hoffmann La Roche Substituierte 2-imidazole als modulatoren der mit spurenaminen assoziierten rezeptoren
RU2456281C2 (ru) * 2006-11-16 2012-07-20 Ф. Хоффманн-Ля Рош Аг Замещенные 4-имидазолы, способ их получения и их применение
BRPI0720047A2 (pt) * 2006-12-13 2013-12-24 Hoffmann La Roche 2-imidazóis como ligantes para receptores associados a aminas de traço (taar)
US20080146523A1 (en) * 2006-12-18 2008-06-19 Guido Galley Imidazole derivatives
RU2473545C2 (ru) 2007-02-02 2013-01-27 Ф.Хоффманн-Ля Рош Аг Новые 2-аминооксазолины в качестве лигандов taar1 для заболеваний цнс
RU2460725C2 (ru) * 2007-02-15 2012-09-10 Ф. Хоффманн-Ля Рош Аг Новые 2-аминооксазолины в качестве лигандов taar1
JP2010531837A (ja) 2007-07-02 2010-09-30 エフ．ホフマン−ラ ロシュ アーゲー 微量アミン関連レセプター（ｔａａｒ）に対して良好な親和性を有する２−イミダゾリン
MX2009013745A (es) * 2007-07-03 2010-01-26 Hoffmann La Roche 4-imidazolinas y su uso como antidepresivos.
JP2010534701A (ja) * 2007-07-27 2010-11-11 エフ．ホフマン−ラ ロシュ アーゲー Ｔａａｒリガンドとしての２−アゼチジンメタンアミン及び２−ピロリジンメタンアミン
CN101765425A (zh) * 2007-08-02 2010-06-30 弗·哈夫曼-拉罗切有限公司 苯甲酰胺衍生物用于治疗cns障碍的用途
AU2008285795A1 (en) * 2007-08-03 2009-02-12 F. Hoffmann-La Roche Ag Pyridinecarboxamide and benzamide derivatives as TAAR1 ligands
ES2556633T3 (es) * 2008-07-24 2016-01-19 F. Hoffmann-La Roche Ag Derivados de 4,5-dihidro-oxazol-2-ilo
US8242153B2 (en) * 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
US20100311798A1 (en) * 2009-06-05 2010-12-09 Decoret Guillaume 2-aminooxazolines as taar1 ligands
US8354441B2 (en) * 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
MA53755A (fr) 2016-03-17 2021-08-04 Hoffmann La Roche Dérivé de 5-éthyl-4-méthyl-pyrazole-3-carboxamide ayant une activité comme agonist de taar

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1121054B (de) * 1960-11-23 1962-01-04 Merck Ag E Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen

Also Published As

Publication number Publication date
ZA72286B (en) 1972-09-27
DE2203373B2 (de) 1977-08-11
FI55841B (fi) 1979-06-29
NO134115C (de) 1976-08-18
YU34694B (en) 1979-12-31
HU162823B (de) 1973-04-28
NL7201121A (de) 1972-07-31
FI55841C (fi) 1979-10-10
NL150454B (nl) 1976-08-16
DE2203373C3 (de) 1978-04-13
AU3817772A (en) 1973-07-26
DE2203373A1 (de) 1972-08-17
JPS4938273B1 (de) 1974-10-16
CA962273A (en) 1975-02-04
SE378426B (de) 1975-09-01
NO134115B (de) 1976-05-10
SU474145A3 (ru) 1975-06-14
YU18172A (en) 1979-07-10
CH535254A (fr) 1973-03-31
US3818035A (en) 1974-06-18
GB1333471A (en) 1973-10-10
BE777689A (fr) 1972-07-05
AT311336B (de) 1973-11-12
DK138496C (de) 1979-02-26

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