DK133382B - Analogifremgangsmåde til fremstilling af 6alfa,9alfa-diflour-11beta,17,21-trihydroxy-16beta-methylpregna-1,4-dien-3,20-dion-17,21-diacetat. - Google Patents

Analogifremgangsmåde til fremstilling af 6alfa,9alfa-diflour-11beta,17,21-trihydroxy-16beta-methylpregna-1,4-dien-3,20-dion-17,21-diacetat.

Info

Publication number: DK133382B
Authority: DK; Denmark
Prior art keywords: 16beta; 9alpha; 6alpha; methylpregna; 11beta
Prior art date: 1972-03-09

Application number

DK128173AA

Other languages

English (en)

Other versions

DK133382C (da

Inventor

Donald Emory Ayer

Carl Alvin Schlagel

Gordon Leonard Flynn

Original Assignee

Upjohn Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-03-09

Filing date

1973-03-08

Publication date

1976-05-10

1973-03-08 Application filed by Upjohn Co filed Critical Upjohn Co

1976-05-10 Publication of DK133382B publication Critical patent/DK133382B/da

1976-10-04 Application granted granted Critical

1976-10-04 Publication of DK133382C publication Critical patent/DK133382C/da

Links

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Rheumatology (AREA)
Chemical Kinetics & Catalysis (AREA)
Pain & Pain Management (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Epidemiology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK128173AA 1972-03-09 1973-03-08 Analogifremgangsmåde til fremstilling af 6alfa,9alfa-diflour-11beta,17,21-trihydroxy-16beta-methylpregna-1,4-dien-3,20-dion-17,21-diacetat. DK133382B (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US23333772A	1972-03-09	1972-03-09
US31697372A	1972-12-20	1972-12-20

Publications (2)

Publication Number	Publication Date
DK133382B true DK133382B (da)	1976-05-10
DK133382C DK133382C (da)	1976-10-04

Family

ID=26926821

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK128173AA DK133382B (da)	1972-03-09	1973-03-08	Analogifremgangsmåde til fremstilling af 6alfa,9alfa-diflour-11beta,17,21-trihydroxy-16beta-methylpregna-1,4-dien-3,20-dion-17,21-diacetat.

Country Status (13)

Country	Link
JP (3)	JPS5331156B2 (da)
AR (1)	AR197216A1 (da)
AU (1)	AU468257B2 (da)
CH (3)	CH580118A5 (da)
DE (1)	DE2365992C3 (da)
DK (1)	DK133382B (da)
ES (1)	ES412235A1 (da)
FR (1)	FR2181802B1 (da)
GB (1)	GB1403962A (da)
HK (1)	HK62680A (da)
NL (1)	NL165178C (da)
PH (1)	PH14703A (da)
SE (1)	SE396756B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1430223A (en) *	1973-10-25	1976-03-31	Upjohn Co	Anti-inflammatory composition comprising steroids
ZA77943B (en) *	1976-03-19	1977-12-28	Upjohn Co	Topical steroid clindamycin preparations
NL187577C (nl) *	1978-04-05	1991-11-18	Sibla Srl	3-acetoxy-9beta,11beta-epoxy-pregna-1,3,5-trienen, werkwijze voor de bereiding daarvan en werkwijze voor de bereiding van 6alfa-halogeen-pregna-1,4-dieen-3-onen.
DE3069074D1 (en)	1979-11-16	1984-10-04	Sterosynt Ltd	6-alpha-9-alpha-difluoro-16-beta-methyl-prednisolone-17,21 diesters and pharmaceutical compositions containing them
JPH0240957Y2 (da) *	1986-08-30	1990-10-31

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB933859A (da) *	1958-09-06	1963-08-14	Syntex S.A.

1973
- 1973-02-22 DE DE2365992A patent/DE2365992C3/de not_active Expired
- 1973-02-22 GB GB877373A patent/GB1403962A/en not_active Expired
- 1973-02-26 AU AU52579/73A patent/AU468257B2/en not_active Expired
- 1973-02-26 CH CH396076A patent/CH580118A5/xx not_active IP Right Cessation
- 1973-02-26 CH CH395976A patent/CH580117A5/xx not_active IP Right Cessation
- 1973-02-26 CH CH277073A patent/CH580116A5/xx not_active IP Right Cessation
- 1973-03-02 ES ES412235A patent/ES412235A1/es not_active Expired
- 1973-03-07 AR AR246918A patent/AR197216A1/es active
- 1973-03-07 JP JP2625073A patent/JPS5331156B2/ja not_active Expired
- 1973-03-08 SE SE7303287A patent/SE396756B/xx unknown
- 1973-03-08 DK DK128173AA patent/DK133382B/da unknown
- 1973-03-08 FR FR7308331A patent/FR2181802B1/fr not_active Expired
- 1973-03-08 NL NL7303262.A patent/NL165178C/xx not_active IP Right Cessation
1976
- 1976-05-06 PH PH18405A patent/PH14703A/en unknown
- 1976-09-09 JP JP51107346A patent/JPS5227760A/ja active Granted
- 1976-09-09 JP JP51107347A patent/JPS5227761A/ja active Granted
1980
- 1980-11-06 HK HK626/80A patent/HK62680A/xx unknown

Also Published As

Publication number	Publication date
AU468257B2 (en)	1976-01-08
DE2365992C3 (de)	1982-05-19
CH580116A5 (da)	1976-09-30
FR2181802A1 (da)	1973-12-07
JPS5227760A (en)	1977-03-02
GB1403962A (en)	1975-08-28
NL165178B (nl)	1980-10-15
JPS5344464B2 (da)	1978-11-29
SE396756B (sv)	1977-10-03
JPS5344465B2 (da)	1978-11-29
CH580117A5 (da)	1976-09-30
JPS5331156B2 (da)	1978-08-31
CH580118A5 (da)	1976-09-30
DE2365992A1 (de)	1977-05-18
DE2365992B2 (de)	1981-08-06
PH14703A (en)	1981-11-10
ES412235A1 (es)	1976-01-01
AU5257973A (en)	1974-08-29
AR197216A1 (es)	1974-03-22
HK62680A (en)	1980-11-14
NL165178C (nl)	1981-03-16
DK133382C (da)	1976-10-04
JPS4899157A (da)	1973-12-15
FR2181802B1 (da)	1976-10-22
JPS5227761A (en)	1977-03-02
NL7303262A (da)	1973-09-11

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