DK1223933T3 - 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer - Google Patents

5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer

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Publication number
DK1223933T3
DK1223933T3 DK00967988T DK00967988T DK1223933T3 DK 1223933 T3 DK1223933 T3 DK 1223933T3 DK 00967988 T DK00967988 T DK 00967988T DK 00967988 T DK00967988 T DK 00967988T DK 1223933 T3 DK1223933 T3 DK 1223933T3
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Prior art keywords
heterocycles
monoamine oxidase
oxidase inhibitors
membered derivatives
membered
Prior art date
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DK00967988T
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English (en)
Inventor
De Lassauniere Pierre Chabrier
Jeremiah Harnett
Dennis Bigg
Jacques Pommier
Anne-Marie Liberatore
Christophe Thurieau
Jacques Lannoy
Original Assignee
Sod Conseils Rech Applic
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Priority claimed from FR9912643A external-priority patent/FR2799461B1/fr
Priority claimed from FR0010151A external-priority patent/FR2812546B1/fr
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Application granted granted Critical
Publication of DK1223933T3 publication Critical patent/DK1223933T3/da

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    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28Radicals substituted by nitrogen atoms
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
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    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
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DK00967988T 1999-10-11 2000-10-10 5-leddet derivater af heterocyklusser og deres anvendelse som monoaminoxidaseinhibitorer DK1223933T3 (da)

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FR9912643A FR2799461B1 (fr) 1999-10-11 1999-10-11 Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments
FR0010151A FR2812546B1 (fr) 2000-08-01 2000-08-01 Derives d'heterocycles a 5 chainons, leur preparation et leur application a titre de medicaments
FR0011169 2000-09-01

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DK05076749.0T DK1589007T3 (da) 1999-10-11 2000-10-10 Heterocyklusderivater med 5 led, fremstilling og anvendelse deraf som lægemidler

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PT1589007E (pt) 2015-10-12
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TWI283577B (en) 2007-07-11
EP1589007A3 (fr) 2009-04-29
PL215580B1 (pl) 2013-12-31
IL148896A0 (en) 2002-09-12
CZ20021292A3 (cs) 2002-10-16
CA2388505A1 (fr) 2001-04-19
IL185118A0 (en) 2007-12-03
JP2003511416A (ja) 2003-03-25
CA2388505C (fr) 2013-03-12
US7956075B2 (en) 2011-06-07
HU228254B1 (en) 2013-02-28
NZ533429A (en) 2004-09-24
JP4972263B2 (ja) 2012-07-11
MXPA02003665A (es) 2003-10-14
PT1223933E (pt) 2006-12-29
EP1228760A3 (fr) 2004-01-28
BR0014649A (pt) 2002-06-18
HUP0203841A2 (en) 2003-05-28
HK1049957A1 (en) 2003-06-06
NO20021689D0 (no) 2002-04-10
TW200509916A (en) 2005-03-16
TWI292316B (en) 2008-01-11
HK1049957B (zh) 2009-08-28
DE60030574T2 (de) 2007-09-20
EP1589007A2 (fr) 2005-10-26
US20070021390A1 (en) 2007-01-25
US20070179153A1 (en) 2007-08-02
US20110172434A1 (en) 2011-07-14
CY1106237T1 (el) 2011-06-08
WO2001026656A3 (fr) 2002-04-18
EP1223933A2 (fr) 2002-07-24
ATE338547T1 (de) 2006-09-15
DK1589007T3 (da) 2015-08-10
PL355147A1 (en) 2004-04-05
HUP0203841A3 (en) 2003-07-28
KR20070068491A (ko) 2007-06-29
ATE522213T1 (de) 2011-09-15
CN100488506C (zh) 2009-05-20
NZ518304A (en) 2004-07-30
AR029006A1 (es) 2003-06-04
EP1589007B1 (fr) 2015-06-03
KR20020060195A (ko) 2002-07-16
AU783129B2 (en) 2005-09-29
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AU7796500A (en) 2001-04-23
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CN1391474A (zh) 2003-01-15
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US8288560B2 (en) 2012-10-16
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US20080146627A1 (en) 2008-06-19
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